Page last updated: 2024-09-04

docetaxel anhydrous and palbociclib

docetaxel anhydrous has been researched along with palbociclib in 6 studies

Compound Research Comparison

Studies
(docetaxel anhydrous)
Trials
(docetaxel anhydrous)
Recent Studies (post-2010)
(docetaxel anhydrous)
Studies
(palbociclib)
Trials
(palbociclib)
Recent Studies (post-2010) (palbociclib)
12,1103,2166,920911126864

Protein Interaction Comparison

ProteinTaxonomydocetaxel anhydrous (IC50)palbociclib (IC50)
Chain B, Cell division protein kinase 6Homo sapiens (human)0.015
Chain B, Cell division protein kinase 6Homo sapiens (human)0.015
Cyclin-T1Homo sapiens (human)1.5085
Cyclin-KHomo sapiens (human)1.207
Cyclin-dependent kinase 1Homo sapiens (human)9.8
Cyclin-dependent kinase 4Homo sapiens (human)0.0109
G2/mitotic-specific cyclin-B1Homo sapiens (human)9.8
Cyclin-A2Homo sapiens (human)2.2042
AcetylcholinesteraseMus musculus (house mouse)0.021
G1/S-specific cyclin-D1Homo sapiens (human)0.0115
G1/S-specific cyclin-E1Homo sapiens (human)9.15
Cyclin-dependent kinase 2Homo sapiens (human)4.1887
G1/S-specific cyclin-D2Homo sapiens (human)0.0127
G1/S-specific cyclin-D3Homo sapiens (human)0.0194
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)3.48
Cyclin-dependent kinase 9Homo sapiens (human)1.1821
Tyrosine-protein kinase JAK3Homo sapiens (human)0.0631
Cyclin-dependent kinase 6Homo sapiens (human)0.018

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (16.67)29.6817
2010's4 (66.67)24.3611
2020's1 (16.67)2.80

Authors

AuthorsStudies
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1
Ajenjo, N; Albarrán, MI; Bischoff, JR; Blanco-Aparicio, C; Cebriá, A; Cebrián, D; Cuadrado-Urbano, M; García, AB; García-Serelde, B; Gómez de la Oliva, CA; Gómez-Casero, E; González Cantalapiedra, E; Hernández, AI; Klett, J; Martínez-González, S; Oyarzabal, J; Pastor, J; Rabal, O; Rodríguez-Arístegui, S; Varela, C1
Afratis, K; Gavras, H; Karamanos, NK; Koutsakis, C; Leonardi, S; Papaioannou, D; Piperigkou, Z; Rassias, G; Rigopoulou, D; Vachlioti, E1
Anderes, K; Arango, ME; Painter, CL; Yan, Z; Zhang, C1
Bagante, F; Connolly, R; Pawlik, TM; Spolverato, G; Vitale, A1
Brunken, L; Hassan, N; Jackson, J; Mellor, C; Mitchell, E; Ng'andu, K; O'Brien, A; Paus, R; Purba, TS; Shahmalak, A; Smart, E1

Other Studies

6 other study(ies) available for docetaxel anhydrous and palbociclib

ArticleYear
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013
Discovery of novel triazolo[4,3-b]pyridazin-3-yl-quinoline derivatives as PIM inhibitors.
    European journal of medicinal chemistry, 2019, Apr-15, Volume: 168

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Discovery; Drug Screening Assays, Antitumor; Humans; Molecular Structure; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-pim-1; Pyridazines; Quinolines; Structure-Activity Relationship; Triazoles

2019
Potent antiproliferative activity of bradykinin B2 receptor selective agonist FR-190997 and analogue structures thereof: A paradox resolved?
    European journal of medicinal chemistry, 2021, Jan-15, Volume: 210

    Topics: Anti-Bacterial Agents; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Female; Humans; MCF-7 Cells; Quinolines; Receptor, Bradykinin B2

2021
Advancing bioluminescence imaging technology for the evaluation of anticancer agents in the MDA-MB-435-HAL-Luc mammary fat pad and subrenal capsule tumor models.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2009, Jan-01, Volume: 15, Issue:1

    Topics: Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Bevacizumab; Cell Line, Tumor; Docetaxel; Female; Humans; Kidney; Luminescent Proteins; Lung Neoplasms; Mammary Glands, Human; Mice; Mice, Nude; Mice, SCID; Neoplasm Transplantation; Neoplasms, Experimental; Piperazines; Pyridines; Taxoids; Xenograft Model Antitumor Assays

2009
Liver Resection for Breast Cancer Liver Metastases: A Cost-utility Analysis.
    Annals of surgery, 2017, Volume: 265, Issue:4

    Topics: Antibodies, Monoclonal, Humanized; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Chemotherapy, Adjuvant; Cost-Benefit Analysis; Disease-Free Survival; Docetaxel; Female; Hepatectomy; Humans; Letrozole; Liver Neoplasms; Male; Markov Chains; Neoplasm Invasiveness; Neoplasm Staging; Nitriles; Piperazines; Pyridines; Quality-Adjusted Life Years; Survival Rate; Taxoids; Triazoles

2017
CDK4/6 inhibition mitigates stem cell damage in a novel model for taxane-induced alopecia.
    EMBO molecular medicine, 2019, Volume: 11, Issue:10

    Topics: Alopecia; Antineoplastic Agents; Bridged-Ring Compounds; Cyclin-Dependent Kinase 4; Cyclin-Dependent Kinase 6; Docetaxel; Humans; Keratinocytes; Models, Theoretical; Organ Culture Techniques; Paclitaxel; Piperazines; Protein Kinase Inhibitors; Pyridines; Stem Cells; Taxoids

2019