Page last updated: 2024-09-04

docetaxel anhydrous and disulfiram

docetaxel anhydrous has been researched along with disulfiram in 6 studies

Compound Research Comparison

Studies
(docetaxel anhydrous)
Trials
(docetaxel anhydrous)
Recent Studies (post-2010)
(docetaxel anhydrous)
Studies
(disulfiram)
Trials
(disulfiram)
Recent Studies (post-2010) (disulfiram)
12,1103,2166,9203,776175723

Protein Interaction Comparison

ProteinTaxonomydocetaxel anhydrous (IC50)disulfiram (IC50)
glucose-6-phosphate dehydrogenase-6-phosphogluconolactonasePlasmodium berghei10.1
Spike glycoproteinBetacoronavirus England 19.35
Replicase polyprotein 1abBetacoronavirus England 19.35
type-1 angiotensin II receptorHomo sapiens (human)6.637
perilipin-5Homo sapiens (human)1.622
perilipin-1Homo sapiens (human)6.959
apelin receptorHomo sapiens (human)2.63
1-acylglycerol-3-phosphate O-acyltransferase ABHD5 isoform aHomo sapiens (human)4.2905
bifunctional UDP-N-acetylglucosamine pyrophosphorylase/glucosamine-1-phosphate N-acetyltransferaseMycobacterium tuberculosis H37Rv85.03
Transmembrane protease serine 2Homo sapiens (human)9.35
Bile salt export pumpHomo sapiens (human)10
Carbamate kinaseGiardia intestinalis0.6
Retinal dehydrogenase 1Homo sapiens (human)0.13
Aldehyde dehydrogenase, mitochondrialHomo sapiens (human)3.4
Cytochrome P450 1A2Homo sapiens (human)4
Procathepsin LHomo sapiens (human)9.35
Alpha-2A adrenergic receptorHomo sapiens (human)4.904
Fructose-1,6-bisphosphatase 1Homo sapiens (human)1.3756
Replicase polyprotein 1aSevere acute respiratory syndrome-related coronavirus9.35
Replicase polyprotein 1abHuman coronavirus 229E9.35
Replicase polyprotein 1abSevere acute respiratory syndrome-related coronavirus9.35
Adenosine receptor A3Homo sapiens (human)0.356
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 26.9171
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.356
Alpha-2B adrenergic receptorHomo sapiens (human)3.218
D(1A) dopamine receptorHomo sapiens (human)2.158
D(4) dopamine receptorHomo sapiens (human)3.15
C-X-C chemokine receptor type 2Homo sapiens (human)6.013
Mitogen-activated protein kinase 3 Homo sapiens (human)1.51
Protein-lysine 6-oxidaseHomo sapiens (human)0.32
Lysine-specific demethylase 5AHomo sapiens (human)10
Caspase-1Homo sapiens (human)1.8
Mu-type opioid receptorHomo sapiens (human)3.511
D(3) dopamine receptorHomo sapiens (human)1.084
Kappa-type opioid receptorHomo sapiens (human)6.103
C-C chemokine receptor type 2Homo sapiens (human)2.468
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.356
C-C chemokine receptor type 4Homo sapiens (human)8.395
Gasdermin-DHomo sapiens (human)0.4
Lysyl oxidase homolog 3Homo sapiens (human)0.093
Spike glycoproteinSevere acute respiratory syndrome-related coronavirus9.35
Sodium-dependent dopamine transporter Homo sapiens (human)4.637
NACHT, LRR and PYD domains-containing protein 3 Mus musculus (house mouse)3
Lysyl oxidase homolog 4Homo sapiens (human)0.059
Histone-lysine N-methyltransferase EHMT2Homo sapiens (human)0.6
Monoglyceride lipaseHomo sapiens (human)0.8095
Angiotensin-converting enzyme 2 Homo sapiens (human)9.35
Gasdermin-DMus musculus (house mouse)0.4
Histone-lysine N-methyltransferase EHMT1Homo sapiens (human)1.6
Lysyl oxidase homolog 2Homo sapiens (human)0.15
large T antigenBetapolyomavirus macacae10.73

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (16.67)29.6817
2010's3 (50.00)24.3611
2020's2 (33.33)2.80

Authors

AuthorsStudies
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Budman, DR; Calabro, A1
Armesilla, AL; Brown, S; Darling, JL; Jiang, W; Kannappan, V; Kumar, IS; Liu, P; Tang, JZ; Tawari, PE; Wang, W1
Chowdhury, R; Roy, A; Sharma, S; Swetha, KL1
Biswas, S; Kumbham, S; Maravajjala, KS; Paul, M; Roy, A; Swetha, KL1

Reviews

1 review(s) available for docetaxel anhydrous and disulfiram

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

5 other study(ies) available for docetaxel anhydrous and disulfiram

ArticleYear
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
In vitro search for synergy and antagonism: evaluation of docetaxel combinations in breast cancer cell lines.
    Breast cancer research and treatment, 2002, Volume: 74, Issue:1

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Antineoplastic Agents, Phytogenic; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Disulfiram; Docetaxel; Drug Interactions; Drug Screening Assays, Antitumor; Enzyme Inhibitors; Epirubicin; Female; Humans; Paclitaxel; Razoxane; Taxoids; Tretinoin; Tumor Cells, Cultured; Vinblastine; Vinorelbine

2002
Disulfiram targets cancer stem-like cells and reverses resistance and cross-resistance in acquired paclitaxel-resistant triple-negative breast cancer cells.
    British journal of cancer, 2013, Oct-01, Volume: 109, Issue:7

    Topics: Antineoplastic Agents, Phytogenic; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Cisplatin; Disulfiram; Docetaxel; Doxorubicin; Drug Resistance, Neoplasm; Enzyme Inhibitors; ErbB Receptors; Female; Humans; Neoplastic Stem Cells; Paclitaxel; Receptors, Estrogen; Receptors, Progesterone; Taxoids

2013
Disulfiram potentiates docetaxel cytotoxicity in breast cancer cells through enhanced ROS and autophagy.
    Pharmacological reports : PR, 2020, Volume: 72, Issue:6

    Topics: Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Autophagy; Breast Neoplasms; Cell Line, Tumor; Disulfiram; Docetaxel; Drug Synergism; Female; Humans; MCF-7 Cells; Reactive Oxygen Species

2020
Overcoming drug resistance with a docetaxel and disulfiram loaded pH-sensitive nanoparticle.
    Journal of controlled release : official journal of the Controlled Release Society, 2023, Volume: 356

    Topics: Animals; Antineoplastic Agents; Cell Line, Tumor; Disulfiram; Docetaxel; Drug Resistance, Multiple; Hydrogen-Ion Concentration; Mice; Nanoparticles

2023