Page last updated: 2024-09-03

dn 1417 and reserpine

dn 1417 has been researched along with reserpine in 3 studies

Compound Research Comparison

Studies
(dn 1417)
Trials
(dn 1417)
Recent Studies (post-2010)
(dn 1417)
Studies
(reserpine)
Trials
(reserpine)
Recent Studies (post-2010) (reserpine)
942015,546223436

Protein Interaction Comparison

ProteinTaxonomydn 1417 (IC50)reserpine (IC50)
Bile salt export pumpHomo sapiens (human)8.7875
ATP-dependent translocase ABCB1Homo sapiens (human)3.2092
Quinolone resistance protein NorAStaphylococcus aureus8.5429
Mu-type opioid receptorHomo sapiens (human)4.152
Chromaffin granule amine transporterHomo sapiens (human)0.05
Synaptic vesicular amine transporterRattus norvegicus (Norway rat)0.0034
Synaptic vesicular amine transporterHomo sapiens (human)0.0147

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19903 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Nagai, Y; Nagawa, Y; Narumi, S; Saji, Y2
Fukuda, N; Miyamoto, M; Nagai, Y; Nagawa, Y; Narumi, S; Saji, Y1

Other Studies

3 other study(ies) available for dn 1417 and reserpine

ArticleYear
[A TRH analog (DN-1417). Anti-reserpine action in electroconvulsive threshold and involvement of serotonergic (5-HT) mechanism in mice].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1985, Volume: 85, Issue:4

    Topics: 5-Hydroxytryptophan; Animals; Anticonvulsants; Biogenic Amines; Brain Chemistry; Drug Interactions; Electroshock; Levodopa; Male; Mice; Mice, Inbred ICR; Reserpine; Seizures; Serotonin; Thyrotropin-Releasing Hormone

1985
[A TRH analog (DN-1417). Antagonistic effects on reserpine-induced decreases in local cerebral glucose utilization and cerebral monoamine levels].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1985, Volume: 85, Issue:5

    Topics: Acid-Base Equilibrium; Animals; Anticonvulsants; Brain; Carbon Dioxide; Glucose; Male; Mice; Mice, Inbred ICR; Motor Activity; Oxygen; Rats; Rats, Inbred Strains; Reserpine; Thyrotropin-Releasing Hormone

1985
Gamma-butyrolactone-gamma-carbonyl-histidyl-prolinamide citrate (DN-1417): a novel TRH analog with potent effects on the central nervous system.
    Life sciences, 1981, Feb-23, Volume: 28, Issue:8

    Topics: Animals; Arousal; Behavior, Animal; Central Nervous System Agents; Hypothermia, Induced; Male; Mice; Motor Activity; Pentobarbital; Reserpine; Sleep; Structure-Activity Relationship; Thyrotropin-Releasing Hormone; Unconsciousness

1981