Page last updated: 2024-09-04

diquafosol and denufosol tetrasodium

diquafosol has been researched along with denufosol tetrasodium in 9 studies

Compound Research Comparison

Studies
(diquafosol)
Trials
(diquafosol)
Recent Studies (post-2010)
(diquafosol)
Studies
(denufosol tetrasodium)
Trials
(denufosol tetrasodium)
Recent Studies (post-2010) (denufosol tetrasodium)
1263892600
12638922668

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's7 (77.78)29.6817
2010's2 (22.22)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dougherty, RW; Douglass, JG; Pendergast, W; Redick, CC; Rideout, JL; Shaver, SR; Sims, IF; Yerxa, BR1
Besada, P; Calenbergh, SV; Costanzi, S; Cosyn, L; Fricks, I; Harden, TK; Ivanov, AA; Jacobson, KA; Ko, H; Maddileti, S1
Besada, P; Cappellacci, L; Carter, RL; Cosyn, L; de Castro, S; Franchetti, P; Grifantini, M; Harden, TK; Jacobson, KA; Ko, H; Petrelli, R; Van Calenbergh, S; Zhou, Y1
Fischer, B; Ginsburg-Shmuel, T; Haas, M; Kalid, O; Reiser, G; Schumann, M; Stern, N1
Abraham, WM; Boucher, RC; Boyer, J; Cowlen, M; Davis, CW; Dougherty, R; Jones, AC; Lang-Furr, M; Picher, M; Sabater, JR; Stutts, MJ; Yerxa, BR1
Evans, R; Kellerman, D; Mathews, D; Shaffer, C1
Amar, T; Caillaud, T; Douglass, JG; Edick, C; Elena, PP; Peterson, WM; Yerxa, BR1
Engels, J; Gorden, J; Kellerman, D; Rossi Mospan, A; Schaberg, A; Smiley, L1
Appy, L; Chardet, C; Peyrottes, S; Roy, B1

Reviews

3 review(s) available for diquafosol and denufosol tetrasodium

ArticleYear
Inhaled P2Y2 receptor agonists as a treatment for patients with Cystic Fibrosis lung disease.
    Advanced drug delivery reviews, 2002, Dec-05, Volume: 54, Issue:11

    Topics: Administration, Inhalation; Animals; Clinical Trials as Topic; Cystic Fibrosis; Deoxycytosine Nucleotides; Epithelium; Humans; Mucociliary Clearance; Ophthalmic Solutions; Polyphosphates; Purinergic P2 Receptor Agonists; Receptors, Purinergic P2Y2; Uracil Nucleotides; Uridine

2002
Denufosol: a review of studies with inhaled P2Y(2) agonists that led to Phase 3.
    Pulmonary pharmacology & therapeutics, 2008, Volume: 21, Issue:4

    Topics: Administration, Inhalation; Clinical Trials, Phase I as Topic; Clinical Trials, Phase II as Topic; Cystic Fibrosis; Deoxycytosine Nucleotides; Female; Forced Expiratory Volume; Humans; Male; Polyphosphates; Purinergic P2 Receptor Agonists; Receptors, Purinergic P2Y2; Uracil Nucleotides; Uridine

2008
Synthetic Strategies for Dinucleotides Synthesis.
    Molecules (Basel, Switzerland), 2019, Nov-27, Volume: 24, Issue:23

    Topics: Deoxycytosine Nucleotides; Dinucleoside Phosphates; Dry Eye Syndromes; Green Chemistry Technology; Humans; Ophthalmic Solutions; Phosphorylation; Polyphosphates; Purinergic P2Y Receptor Agonists; Receptors, Purinergic; Uracil Nucleotides; Uridine

2019

Other Studies

6 other study(ies) available for diquafosol and denufosol tetrasodium

ArticleYear
Synthesis and P2Y receptor activity of a series of uridine dinucleoside 5'-polyphosphates.
    Bioorganic & medicinal chemistry letters, 2001, Jan-22, Volume: 11, Issue:2

    Topics: Calcium; Dinucleoside Phosphates; Humans; Protein Binding; Purinergic P2 Receptor Agonists; Receptors, Purinergic P2; Spectrometry, Fluorescence; Structure-Activity Relationship; Transduction, Genetic; Tumor Cells, Cultured; Uracil Nucleotides

2001
Molecular modeling of the human P2Y2 receptor and design of a selective agonist, 2'-amino-2'-deoxy-2-thiouridine 5'-triphosphate.
    Journal of medicinal chemistry, 2007, Mar-22, Volume: 50, Issue:6

    Topics: Adenosine Triphosphate; Binding Sites; Cell Line, Tumor; Drug Design; Humans; Models, Molecular; Monte Carlo Method; Protein Conformation; Purinergic P2 Receptor Agonists; Quantitative Structure-Activity Relationship; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; Uridine Triphosphate

2007
Synthesis and potency of novel uracil nucleotides and derivatives as P2Y2 and P2Y6 receptor agonists.
    Bioorganic & medicinal chemistry, 2008, Jun-15, Volume: 16, Issue:12

    Topics: Humans; Purinergic P2 Receptor Agonists; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; Structure-Activity Relationship; Uracil Nucleotides

2008
5-OMe-UDP is a potent and selective P2Y(6)-receptor agonist.
    Journal of medicinal chemistry, 2010, Feb-25, Volume: 53, Issue:4

    Topics: Calcium; Cell Line, Tumor; Humans; Ligands; Magnetic Resonance Spectroscopy; Molecular Conformation; Purinergic P2 Receptor Agonists; Receptors, Purinergic P2; Structure-Activity Relationship; Transfection; Uridine Diphosphate

2010
Pharmacology of INS37217 [P(1)-(uridine 5')-P(4)- (2'-deoxycytidine 5')tetraphosphate, tetrasodium salt], a next-generation P2Y(2) receptor agonist for the treatment of cystic fibrosis.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 302, Issue:3

    Topics: Animals; Astrocytoma; Brain Neoplasms; Calcium; Chlorides; Cilia; Cystic Fibrosis; Deoxycytosine Nucleotides; Epithelial Cells; Humans; In Situ Hybridization; In Vitro Techniques; Indicators and Reagents; Macaca mulatta; Mucins; Mucociliary Clearance; Ophthalmic Solutions; Polyphosphates; Purinergic P2 Receptor Agonists; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; Reverse Transcriptase Polymerase Chain Reaction; Sheep; Tumor Cells, Cultured; Uracil Nucleotides; Uridine

2002
Potency and duration of action of synthetic P2Y2 receptor agonists on Schirmer scores in rabbits.
    Advances in experimental medicine and biology, 2002, Volume: 506, Issue:Pt A

    Topics: Animals; Deoxycytosine Nucleotides; Eye; Male; Ophthalmic Solutions; Polyphosphates; Purinergic P2 Receptor Agonists; Rabbits; Tears; Uracil Nucleotides; Uridine

2002