Page last updated: 2024-08-21

diphenylamine and pyrimidinones

diphenylamine has been researched along with pyrimidinones in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (11.11)29.6817
2010's7 (77.78)24.3611
2020's1 (11.11)2.80

Authors

AuthorsStudies
Akyel, KG; Albert, R; Beerli, C; Bruns, C; Francotte, E; Luyten, M; MacKenzie, D; Nuninger, F; Oberer, L; Schaefer, M; Streiff, MB; Thoma, G; Wagner, T; Walter, H; Weckbecker, G; Zerwes, HG1
Hantani, Y; Kakegawa, J; Nakamura, M; Okajima, N; Sakai, T; Watanabe, Y; Yamaguchi, T; Yoshida, T1
Fellmann, C; Gadal, S; Ishii, N; Joseph, E; Kastenhuber, E; Lito, P; Lowe, S; Lukacs, C; Miura, T; Morikami, K; Ohara, K; Rosen, N; Saborowski, A; Saborowski, M; Solomon, M; Yue, J1
Banks, AS; Beausoleil, SA; Everley, RA; Gygi, SP; McAllister, FE; Paulo, JA1
Kim, MS1
Kiessling, MK; Rogler, G1
Banno, E; Chiba, M; De Velasco, MA; Fujita, Y; Hayashi, H; Mitsudomi, T; Mizuuchi, H; Nakamura, Y; Nishio, K; Sakai, K; Terashima, M; Togashi, Y; Tomida, S1
Bago-Horvath, Z; Fece de la Cruz, F; Haura, EB; Katz, AM; Kerzendorfer, C; Konopka, T; Loizou, JI; Mair, B; Mazouzi, A; Muellner, MK; Nagy-Bojarszky, K; Nijman, SM; Paz, K; Smida, M; Suchankova, T; Uras, IZ1
Mergener, S; Peña-Llopis, S; Siveke, JT1

Reviews

1 review(s) available for diphenylamine and pyrimidinones

ArticleYear
Targeting the RAS pathway by mitogen-activated protein kinase inhibitors.
    Swiss medical weekly, 2015, Volume: 145

    Topics: Animals; Azetidines; Benzamides; Benzimidazoles; Diphenylamine; Genes, ras; GTP Phosphohydrolases; Humans; Membrane Proteins; Mice; Mitogen-Activated Protein Kinases; Mutation; Neoplasms; Niacinamide; Piperidines; Protein Kinase Inhibitors; Proto-Oncogene Proteins B-raf; Proto-Oncogene Proteins p21(ras); Pyridones; Pyrimidinones; Signal Transduction; Sulfonamides

2015

Other Studies

8 other study(ies) available for diphenylamine and pyrimidinones

ArticleYear
Orally bioavailable competitive CCR5 antagonists.
    Journal of medicinal chemistry, 2004, Apr-08, Volume: 47, Issue:8

    Topics: Administration, Oral; Animals; Biological Availability; Calcium; CCR5 Receptor Antagonists; Cell Line; Chemotaxis, Leukocyte; Cricetinae; Crystallography, X-Ray; Cyclic N-Oxides; Diphenylamine; Humans; In Vitro Techniques; Lymphocytes; Macaca fascicularis; Mice; Molecular Structure; Piperidines; Pyrimidines; Pyrimidinones; Radioligand Assay; Rats; Structure-Activity Relationship

2004
Identification and characterization of a novel chemotype MEK inhibitor able to alter the phosphorylation state of MEK1/2.
    Oncotarget, 2012, Volume: 3, Issue:12

    Topics: Allosteric Regulation; Antineoplastic Agents; Benzamides; Butadienes; Chromatography, Affinity; Diphenylamine; Dose-Response Relationship, Drug; HEK293 Cells; HT29 Cells; Humans; Kinetics; MAP Kinase Kinase 1; MAP Kinase Kinase 2; Molecular Structure; Molecular Targeted Therapy; Neoplasms; Nitriles; Phosphorylation; Protein Binding; Protein Kinase Inhibitors; Pyridones; Pyrimidinones; Signal Transduction

2012
Disruption of CRAF-mediated MEK activation is required for effective MEK inhibition in KRAS mutant tumors.
    Cancer cell, 2014, May-12, Volume: 25, Issue:5

    Topics: Animals; Benzamides; Cell Line; Coumarins; Diphenylamine; Drug Resistance, Neoplasm; Extracellular Signal-Regulated MAP Kinases; HEK293 Cells; Humans; Indoles; MAP Kinase Kinase 1; MAP Kinase Signaling System; Melanoma; Mice; Mice, Nude; Phosphorylation; Protein Kinase Inhibitors; Proto-Oncogene Proteins; Proto-Oncogene Proteins B-raf; Proto-Oncogene Proteins p21(ras); Pyridones; Pyrimidinones; raf Kinases; ras Proteins; RNA Interference; RNA, Small Interfering; Sulfonamides; Surface Plasmon Resonance; TNF Receptor-Associated Factor 3; Vemurafenib

2014
Effects of MEK inhibitors GSK1120212 and PD0325901 in vivo using 10-plex quantitative proteomics and phosphoproteomics.
    Proteomics, 2015, Volume: 15, Issue:2-3

    Topics: Amino Acid Sequence; Animals; Benzamides; Diphenylamine; Humans; Kidney; Liver; MAP Kinase Signaling System; Mice; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Molecular Sequence Data; Pancreas; Phosphopeptides; Phosphorylation; Protein Kinase Inhibitors; Proteome; Proteomics; Pyridones; Pyrimidinones; Tandem Mass Spectrometry

2015
Proteomics equipped with multiplexing toward ultra high throughput.
    Proteomics, 2015, Volume: 15, Issue:2-3

    Topics: Animals; Benzamides; Diphenylamine; Humans; Mitogen-Activated Protein Kinase Kinases; Phosphopeptides; Protein Kinase Inhibitors; Proteome; Pyridones; Pyrimidinones

2015
MEK inhibitors against MET-amplified non-small cell lung cancer.
    International journal of oncology, 2016, Volume: 49, Issue:6

    Topics: A549 Cells; Antineoplastic Agents; Benzamides; Carcinoma, Non-Small-Cell Lung; Cell Line, Tumor; Crizotinib; Diphenylamine; ErbB Receptors; Humans; Lung Neoplasms; MAP Kinase Kinase 1; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-met; Pyrazoles; Pyridines; Pyridones; Pyrimidinones

2016
MEK inhibitors block growth of lung tumours with mutations in ataxia-telangiectasia mutated.
    Nature communications, 2016, 12-06, Volume: 7

    Topics: Animals; Ataxia Telangiectasia Mutated Proteins; Benzamides; Cell Line, Tumor; Cell Proliferation; Diphenylamine; Humans; Lung Neoplasms; Mice, Nude; Mutation; Protein Kinase Inhibitors; Proto-Oncogene Proteins B-raf; Pyridones; Pyrimidinones; ras Proteins; RNA Interference; Thiophenes; Urea; Xenograft Model Antitumor Assays

2016
Monosomy 3 Is Linked to Resistance to MEK Inhibitors in Uveal Melanoma.
    International journal of molecular sciences, 2021, Jun-23, Volume: 22, Issue:13

    Topics: Cell Line, Tumor; Chromosomes, Human, Pair 3; Diphenylamine; DNA Copy Number Variations; Drug Resistance, Neoplasm; Eukaryotic Initiation Factor-2; Gene Expression Regulation, Neoplastic; Humans; MAP Kinase Signaling System; Melanoma; Mitogen-Activated Protein Kinase Kinases; Monosomy; Protein Kinase Inhibitors; Pyridones; Pyrimidinones; Sulfonamides; Survival Analysis; Tumor Suppressor Proteins; Ubiquitin Thiolesterase; Uveal Neoplasms

2021