diphenhydramine and triprolidine

diphenhydramine has been researched along with triprolidine in 24 studies

Research

Studies (24)

TimeframeStudies, this research(%)All Research%
pre-199012 (50.00)18.7374
1990's6 (25.00)18.2507
2000's3 (12.50)29.6817
2010's3 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carrupt, PA; Jolliet, P; Morin, C; Morin, D; Pagliara, A; Rihoux, JP; Testa, B; Tillement, JP; Urien, S1
Booth, RG; Brown, RL; Bucholtz, EC; Tropsha, A; Wyrick, SD1
Bakker, RA; Booth, RG; Choksi, NY; Leurs, R; Moniri, NH; Nix, WB; Timmerman, H1
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
Bellman, K; Knegtel, RM; Settimo, L1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Champion, LA; Luddy, RE; Schindler, S; Schwartz, AD1
Chuang, DM; Dillon-Carter, O1
Fleisch, JH; Haisch, KD; Rinkema, LE; Whitesitt, CA1
Cohen, AF; Hamilton, MJ; Peck, AW1
Aselton, P; Jick, H1
Grimshaw, JJ; Jaffe, GV1
Kano, K; Kasukawa, R; Yoshida, H; Yoshida, T1
Harada, M; Katagiri, K; Takeuchi, M1
Fukao, T; Takagi, K1
Brody, TM; Commarato, MA; McNeill, JH1
Brody, TM; McNeill, JH1
Cook, DA; Kenakin, TP1
O'Hanlon, JF; Ramaekers, JG2
Muntjewerff, ND; O'Hanlon, JF; Sanders, RL; van Veggel, LM; Vuurman, EF1
Cruze, CA; Robinson, MK1
Katz, JL; Kopajtic, TA; Tanda, G1
Beebe, MR; Rider, ME; Semin, DJ; Shaw, BJ1

Reviews

1 review(s) available for diphenhydramine and triprolidine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

6 trial(s) available for diphenhydramine and triprolidine

ArticleYear
The effects of four commonly used drugs on platelet function.
    The Journal of pediatrics, 1976, Volume: 89, Issue:4

    Topics: Adenosine Diphosphate; Adult; Aspirin; Blood Coagulation; Blood Platelets; Diphenhydramine; Guaifenesin; Humans; In Vitro Techniques; Platelet Aggregation; Pyridines; Triprolidine

1976
The effects of acrivastine (BW825C), diphenhydramine and terfenadine in combination with alcohol on human CNS performance.
    European journal of clinical pharmacology, 1987, Volume: 32, Issue:3

    Topics: Adolescent; Adult; Benzhydryl Compounds; Brain; Diphenhydramine; Double-Blind Method; Drug Synergism; Ethanol; Eye Movements; Female; Histamine H1 Antagonists; Humans; Male; Middle Aged; Psychomotor Performance; Pyridines; Reaction Time; Terfenadine; Triprolidine

1987
Benylin expectorant versus actifed expectorant in the treatment of acute cough.
    The British journal of clinical practice, 1985, Volume: 39, Issue:6

    Topics: Adult; Consumer Behavior; Cough; Diphenhydramine; Drug Combinations; Ephedrine; Expectorants; Female; Humans; Male; Middle Aged; Patient Compliance; Pseudoephedrine; Pyridines; Triprolidine

1985
Antihistamine effects on actual driving performance in a standard test: a summary of Dutch experience, 1989-94.
    Allergy, 1995, Volume: 50, Issue:3

    Topics: Automobile Driving; Benzimidazoles; Butyrophenones; Cetirizine; Clemastine; Diphenhydramine; Dose-Response Relationship, Drug; Histamine H1 Antagonists; Humans; Loratadine; Netherlands; Piperidines; Psychomotor Performance; Terfenadine; Triprolidine

1995
Acrivastine, terfenadine and diphenhydramine effects on driving performance as a function of dose and time after dosing.
    European journal of clinical pharmacology, 1994, Volume: 47, Issue:3

    Topics: Administration, Oral; Adult; Automobile Driving; Cross-Over Studies; Diphenhydramine; Dose-Response Relationship, Drug; Drug Interactions; Drug Therapy, Combination; Ephedrine; Female; Humans; Infant, Newborn; Middle Aged; Single-Blind Method; Terfenadine; Triprolidine

1994
Effects of semprex-D and diphenhydramine on learning in young adults with seasonal allergic rhinitis.
    Annals of allergy, asthma & immunology : official publication of the American College of Allergy, Asthma, & Immunology, 1996, Volume: 76, Issue:3

    Topics: Adolescent; Adult; Diphenhydramine; Double-Blind Method; Drug Combinations; Ephedrine; Female; Histamine H1 Antagonists; Humans; Learning; Learning Disabilities; Male; Memory; Rhinitis, Allergic, Seasonal; Triprolidine

1996

Other Studies

17 other study(ies) available for diphenhydramine and triprolidine

ArticleYear
Molecular properties and pharmacokinetic behavior of cetirizine, a zwitterionic H1-receptor antagonist.
    Journal of medicinal chemistry, 1998, Mar-12, Volume: 41, Issue:6

    Topics: Alkanes; Animals; Biological Transport; Blood Proteins; Brain; Cetirizine; Histamine H1 Antagonists; Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydroxyzine; Isomerism; Models, Molecular; Molecular Conformation; Octanols; Rats; Water

1998
Synthesis, evaluation, and comparative molecular field analysis of 1-phenyl-3-amino-1,2,3,4-tetrahydronaphthalenes as ligands for histamine H(1) receptors.
    Journal of medicinal chemistry, 1999, Aug-12, Volume: 42, Issue:16

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ligands; Models, Molecular; Pyrilamine; Radioligand Assay; Structure-Activity Relationship; Tetrahydronaphthalenes

1999
A novel phenylaminotetralin radioligand reveals a subpopulation of histamine H(1) receptors.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 302, Issue:1

    Topics: Animals; Binding, Competitive; Cell Membrane; Chlorocebus aethiops; CHO Cells; COS Cells; Cricetinae; DNA, Complementary; Guinea Pigs; Histamine; Histamine Agonists; Humans; Ileum; Inositol Phosphates; Ligands; NF-kappa B; Pyrilamine; Radiopharmaceuticals; Receptors, Histamine H1; Tetrahydronaphthalenes; Thermodynamics; Transfection; Type C Phospholipases

2002
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
Comparison of the accuracy of experimental and predicted pKa values of basic and acidic compounds.
    Pharmaceutical research, 2014, Volume: 31, Issue:4

    Topics: Chemistry, Pharmaceutical; Forecasting; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Random Allocation

2014
Characterization of bradykinin-induced phosphoinositide turnover in neurohybrid NCB-20 cells.
    Journal of neurochemistry, 1988, Volume: 51, Issue:2

    Topics: Animals; Bradykinin; Cell Line; Diphenhydramine; GTP-Binding Proteins; Kinetics; Lithium; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phorbols; Phosphatidylinositols; Triprolidine; Type C Phospholipases

1988
Pharmacologic analysis of LY188695 (KB-2413), 1-(2-ethoxyethyl)-2-(4-methyl-1-homopiperazinyl)-benzimidazole difumarate, a potent histamine1 receptor antagonist.
    Agents and actions, 1987, Volume: 20, Issue:1-2

    Topics: Animals; Benzhydryl Compounds; Benzimidazoles; Bronchial Provocation Tests; Chlorpheniramine; Diphenhydramine; Guinea Pigs; Histamine H1 Antagonists; Lung; Male; Muscle, Smooth; Promethazine; Pyrilamine; Terfenadine; Triprolidine

1987
Re: Pyloric stenosis and maternal antihistamine exposure at group health cooperative.
    American journal of epidemiology, 1985, Volume: 122, Issue:1

    Topics: Diphenhydramine; Drug Combinations; Ephedrine; Female; Humans; Infant, Newborn; Maternal-Fetal Exchange; Pregnancy; Pseudoephedrine; Pyloric Stenosis; Pyridines; Triprolidine

1985
Skin reactions induced by sera of patients with monoclonal IgG gammapathy.
    International archives of allergy and applied immunology, 1973, Volume: 45, Issue:4

    Topics: Acetamides; Animals; Bence Jones Protein; Blood Protein Disorders; Blood Protein Electrophoresis; Capillary Permeability; Chromatography, DEAE-Cellulose; Complement System Proteins; Diphenhydramine; Hot Temperature; Humans; Immune Sera; Immune System Diseases; Immunodiffusion; Immunoelectrophoresis; Immunoglobulin A; Immunoglobulin Fc Fragments; Immunoglobulin G; Immunoglobulin M; Isoflurophate; Mercaptoethanol; Rabbits; Skin; Skin Tests; Triprolidine; Trypsin Inhibitors

1973
[Quantitative determination of passive cutaneous anaphylaxis and effects of anti-histaminics on anaphylaxis in guinea pigs].
    Arerugi = [Allergy], 1966, Volume: 15, Issue:1

    Topics: Anaphylaxis; Animals; Capillary Permeability; Diphenhydramine; Guinea Pigs; Histamine H1 Antagonists; Injections, Intradermal; Injections, Intraperitoneal; Male; Passive Cutaneous Anaphylaxis; Promethazine; Triprolidine

1966
Effects of some drugs on capillary permeability in the anaphylaxis of the mouse.
    Japanese journal of pharmacology, 1971, Volume: 21, Issue:4

    Topics: Aminopyrine; Anaphylaxis; Animals; Anti-Inflammatory Agents; Antilymphocyte Serum; Aprotinin; Aspirin; Body Temperature; Capillary Permeability; Chloroquine; Chlorpromazine; Cortisone; Cyclizine; Depression, Chemical; Desensitization, Immunologic; Diphenhydramine; Epinephrine; Female; Glycyrrhiza; Histamine H1 Antagonists; Indomethacin; Mice; Oxyphenbutazone; Phenylbutazone; Plants, Medicinal; Promethazine; Rectum; Reserpine; Splenectomy; Triprolidine

1971
Further studies on the effect of various drugs on the uptake of tyramine-3H and formation of octopamine-3H in the rat heart.
    Canadian journal of physiology and pharmacology, 1969, Volume: 47, Issue:6

    Topics: Amitriptyline; Animals; Cocaine; Desipramine; Diphenhydramine; Female; Glucosyltransferases; Methylphenidate; Myocardium; Neurons; Norepinephrine; Octopamine; Pyridines; Rats; Sympathetic Nervous System; Triprolidine; Tritium; Tyramine

1969
The effect of various drug pretreatments on amine-induced phosphorylase activation and amine uptake.
    The Journal of pharmacology and experimental therapeutics, 1968, Volume: 162, Issue:1

    Topics: Amitriptyline; Animals; Carbon Isotopes; Depression, Chemical; Desipramine; Diphenhydramine; Drug Synergism; Female; Glucosyltransferases; Heart; Imipramine; Isoproterenol; Methylphenidate; Myocardium; Norepinephrine; Promethazine; Propranolol; Rats; Stimulation, Chemical; Tranylcypromine; Triprolidine; Tritium; Tyramine

1968
N,N-Diethyl-2-(1-pyridyl)ethylamine, a partial agonist for the histamine receptor in guinea pig ileum.
    Canadian journal of physiology and pharmacology, 1980, Volume: 58, Issue:11

    Topics: Animals; Diphenhydramine; Ethylamines; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Receptors, Histamine; Receptors, Histamine H1; Triprolidine

1980
Preclinical skin sensitization testing of antihistamines: guinea pig and local lymph node assay responses.
    Food and chemical toxicology : an international journal published for the British Industrial Biological Research Association, 1996, Volume: 34, Issue:5

    Topics: Animals; Chlorpheniramine; Dermatitis, Allergic Contact; Diphenhydramine; Evaluation Studies as Topic; Guinea Pigs; Histamine H1 Antagonists; Immunologic Tests; Lymph Nodes; Mice; Mice, Inbred BALB C; Mice, Inbred ICR; Promethazine; Sensitivity and Specificity; Skin; Toxicity Tests; Triprolidine

1996
Cocaine-like neurochemical effects of antihistaminic medications.
    Journal of neurochemistry, 2008, Volume: 106, Issue:1

    Topics: Animals; Central Nervous System Stimulants; Chlorpheniramine; Cocaine; Diphenhydramine; Dopamine; Dopamine Agonists; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Histamine H1 Antagonists; Male; Nucleus Accumbens; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Reward; Serotonin Plasma Membrane Transport Proteins; Stereoisomerism; Substance-Related Disorders; Synaptic Transmission; Synaptosomes; Triprolidine

2008
Applicability of total reflection X-ray fluorescence (TXRF) as a screening platform for pharmaceutical inorganic impurity analysis.
    Journal of pharmaceutical and biomedical analysis, 2012, Apr-07, Volume: 63

    Topics: Calibration; Catalysis; Chemistry, Pharmaceutical; Chlorpheniramine; Diphenhydramine; Drug Contamination; Ephedrine; Palladium; Pharmaceutical Preparations; Pseudoephedrine; Scopolamine; Spectrometry, X-Ray Emission; Technology, Pharmaceutical; Triprolidine

2012