diminazene has been researched along with adenosine in 10 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 3 (30.00) | 18.2507 |
2000's | 4 (40.00) | 29.6817 |
2010's | 2 (20.00) | 24.3611 |
2020's | 1 (10.00) | 2.80 |
Authors | Studies |
---|---|
Caljon, G; Campagnaro, GD; de Koning, HP; Hulpia, F; Maes, L; Scortichini, M; Van Calenbergh, S; Van Hecke, K | 1 |
Alfayez, IA; Bouton, J; Caljon, G; Campagnaro, GD; de Koning, HP; Hulpia, F; Mabille, D; Maes, L; Van Calenbergh, S | 1 |
Baltz, T; Barrett, MP; Denise, H; Giroud, C; Zhang, ZQ | 1 |
Scott, AG; Tait, A; Turner, CM | 1 |
Alonso, C; González, VM; Pérez, JM | 1 |
Martin, RJ; Ross, CA; Suswam, EA; Taylor, DW | 1 |
Barrett, MP; Brun, R; Burchmore, RJ; de Koning, HP; Enyaru, JC; Geiser, F; Kaminsky, R; Mäser, P; Matovu, E; Seebeck, T; Stewart, ML; Wallace, LJ | 1 |
Martin, RJ; Ross, CA; Suswam, EA | 1 |
Anderson, LF; Barrett, MP; Burchmore, RJ; de Koning, HP; Stewart, M; Wallace, LJ | 1 |
Idaka, N; Iguchi, A; Ohta, H; Otsuguro, K; Takiguchi, M; Uchida, N; Watanabe, N; Yamamori, T; Yamasaki, M | 1 |
10 other study(ies) available for diminazene and adenosine
Article | Year |
---|---|
Revisiting tubercidin against kinetoplastid parasites: Aromatic substitutions at position 7 improve activity and reduce toxicity.
Topics: Animals; Biological Transport; Kinetoplastida; Mice; Nucleoside Transport Proteins; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei; Tubercidin | 2019 |
C6-O-alkylated 7-deazainosine nucleoside analogues: Discovery of potent and selective anti-sleeping sickness agents.
Topics: Alkylation; Cell Line; Cell Survival; Dose-Response Relationship, Drug; Drug Discovery; Humans; Inosine; Molecular Structure; Nucleosides; Parasitic Sensitivity Tests; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei | 2020 |
A diamidine-resistant Trypanosoma equiperdum clone contains a P2 purine transporter with reduced substrate affinity.
Topics: Adenosine; Animals; Arsenicals; Biological Transport, Active; Carrier Proteins; Diminazene; Drug Resistance; Kinetics; Pentamidine; Receptors, Purinergic P2; Trypanocidal Agents; Trypanosoma | 1995 |
Trypanosoma brucei: lack of cross-resistance to melarsoprol in vitro by cymelarsan-resistant parasites.
Topics: Adenine; Adenosine; Animals; Arsenicals; Diminazene; Dose-Response Relationship, Drug; Drug Resistance; Enzyme Inhibitors; Female; Inosine; Melarsoprol; Mice; Pentamidine; Trypanocidal Agents; Trypanosoma brucei brucei | 1997 |
The berenil ligand directs the DNA binding of the cytotoxic drug Pt-berenil.
Topics: Adenosine; Antineoplastic Agents; Binding Sites; Cisplatin; Deoxyribonuclease BamHI; Deoxyribonuclease HindIII; Deoxyribonuclease I; Diminazene; DNA; DNA Footprinting; Enzyme Inhibitors; Guanosine; Intercalating Agents; Magnetic Resonance Spectroscopy; Organoplatinum Compounds | 1997 |
Changes in properties of adenosine transporters in Trypanosoma evansi and modes of selection of resistance to the melaminophenyl arsenical drug, Mel Cy.
Topics: Adenine; Adenosine; Animals; Arsenicals; Biological Transport; Biomarkers; Carrier Proteins; Diminazene; Dose-Response Relationship, Drug; Drug Resistance; Inosine; Membrane Transport Proteins; Nucleoside Transport Proteins; Parasitic Sensitivity Tests; Trypanocidal Agents; Trypanosoma | 2001 |
Mechanisms of arsenical and diamidine uptake and resistance in Trypanosoma brucei.
Topics: Adenine; Adenosine; Animals; Arsenicals; Benzamidines; Cell Death; Cell Division; Diminazene; Drug Resistance; Female; Gene Silencing; Hypoxanthine; Inhibitory Concentration 50; Inosine; Melarsoprol; Mice; Mutation; Nucleoside Transport Proteins; Pentamidine; Stilbamidines; Trypanosoma brucei brucei | 2003 |
Changes in adenosine transport associated with melaminophenyl arsenical (Mel CY) resistance in Trypanosoma evansi: down-regulation and affinity changes of the P2 transporter.
Topics: Adenine; Adenosine; Animals; Arsenicals; Diminazene; Down-Regulation; Drug Resistance; Inosine; Kinetics; Nucleoside Transport Proteins; Trypanocidal Agents; Trypanosoma | 2003 |
The trypanocide diminazene aceturate is accumulated predominantly through the TbAT1 purine transporter: additional insights on diamidine resistance in african trypanosomes.
Topics: Adenosine; Animals; Biological Transport, Active; Diminazene; Drug Resistance; Female; Kinetics; Mutation; Nucleoside Transport Proteins; Rats; Rats, Wistar; Saccharomyces cerevisiae; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 2004 |
Intracellular diminazene aceturate content and adenosine incorporation in diminazene aceturate-resistant Babesia gibsoni isolate in vitro.
Topics: Adenosine; Animals; Babesia; Babesiosis; Blood Glucose; Chromatography, High Pressure Liquid; Diminazene; Dog Diseases; Dogs; Drug Resistance; Erythrocyte Count; Erythrocytes; Hypoxanthine; Male; Parasitemia; Potassium; Sodium | 2017 |