dimaprit has been researched along with sk&f 91488 in 29 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 8 (27.59) | 18.7374 |
1990's | 11 (37.93) | 18.2507 |
2000's | 6 (20.69) | 29.6817 |
2010's | 4 (13.79) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Beaven, MA; Shaff, RE | 1 |
Maeyama, K; Ohkawara, Y; Ohrui, T; Sasaki, H; Sasaki, M; Sekizawa, K; Takemura, M; Wada, H; Watanabe, T; Yamauchi, K | 1 |
Hannibal, T; Jørgensen, H; Knigge, U; Matzen, S; Warberg, J | 1 |
Gerges, E; Gertner, SB | 1 |
Donaldson, J; Hill, SJ | 1 |
Gertner, SB; Poulakos, JJ | 1 |
Jouvet, M; Lin, JS; Sakai, K | 1 |
Andersson, P; Bergstrand, H | 1 |
Rothschild, AM | 1 |
Gatti, PJ; Gertner, SB | 1 |
Gertner, SB; Klein, MC | 1 |
Katayose, D; Nakazawa, H; Ohkawara, Y; Ohtsu, H; Sekizawa, K; Shibahara, S; Suzuki, H; Takemura, M; Tamura, G; Yamauchi, K | 1 |
Sasaki, T; Satoh, M; Shimura, S; Takishima, T; Yamada, K; Yamauchi, K | 1 |
Maeyama, K; Morikawa, M; Nakazawa, H; Sasaki, H; Satoh, M; Sekizawa, K; Watanabe, T; Yamauchi, K | 1 |
Maeyama, K; Nakazawa, H; Ohkawara, Y; Ohrui, T; Sasaki, H; Sekizawa, K; Takishima, T; Watanabe, T; Yamauchi, K | 1 |
Maeyama, K; Morikawa, M; Nakazawa, H; Sasaki, H; Sekizawa, K; Watanabe, T; Yamauchi, K | 1 |
Chiyotani, A; Konno, K; Nakata, J; Takeyama, K; Tamaoki, J | 1 |
Bartolini, A; Ghelardini, C; Hänninen, J; Ipponi, A; Lamberti, C; Malmberg-Aiello, P | 1 |
Irokawa, T; Nagaki, M; Sasaki, T; Shimura, S; Shirato, K; Yamauchi, K; Yamaya, M | 1 |
Kitanaka, J; Kitanaka, N; Takemura, M; Terada, N; Tsujimura, T | 2 |
Jochem, J | 1 |
Akagi, M; Fukuishi, N; Imajo, N; Matsui, N; Matsui, S; Yasui, Y | 1 |
Kitanaka, J; Kitanaka, N; Morita, Y; Takemura, M; Tatsuta, T | 1 |
Cheng, YS; Huang, CC; Huang, CW; Yu, J | 1 |
Ambrose, RE; Dankoski, EC; Hashemi, P; Wightman, RM; Wood, KM | 1 |
Sanchez-Alavez, M; Sethi, J; Tabarean, IV | 1 |
Benetti, F; Izquierdo, I | 1 |
Benetti, F; da Silveira, CK; Izquierdo, I; Rosa, J | 1 |
29 other study(ies) available for dimaprit and sk&f 91488
Article | Year |
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Inhibition of histamine methylation in vivo by the dimaprit analog, SKF Compound 91488.
Topics: Amine Oxidase (Copper-Containing); Animals; Brain; Dimaprit; Guanidines; Histamine; Histamine N-Methyltransferase; Kidney; Male; Methylation; Methyltransferases; Mice; Rats; Thiourea | 1979 |
Histamine N-methyltransferase controls the contractile response of guinea pig trachea to histamine.
Topics: Animals; Dimaprit; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; Histamine; Histamine N-Methyltransferase; Male; Muscle Contraction; Muscle, Smooth; Thiourea; Trachea | 1992 |
Involvement of histamine in the mediation of the stress-induced release of alpha-melanocyte-stimulating hormone in male rats.
Topics: Adrenocorticotropic Hormone; alpha-MSH; Animals; Bromocriptine; Dimaprit; Histamine; Male; Methylhistidines; Propranolol; Rats; Rats, Inbred Strains; Stress, Physiological; Thiourea | 1991 |
Central cardiovascular responses of histamine and homodimaprit in normal and hypophysectomized rats.
Topics: Animals; Blood Pressure; Brain; Dimaprit; Hexamethonium; Hexamethonium Compounds; Histamine; Hypophysectomy; Kinetics; Male; Rats; Rats, Inbred Strains; Thiourea; Vasopressins | 1990 |
Selective enhancement of histamine H1-receptor responses in guinea-pig ileal smooth muscle by 1,4-dithiothreitol.
Topics: Acetylcholine; Animals; Dimaprit; Dithionitrobenzoic Acid; Dithiothreitol; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Thiourea | 1986 |
Studies on the desensitization of the central cardiovascular responses of histamine.
Topics: Animals; Blood Pressure; Brain; Cardiovascular System; Dimaprit; Heart Rate; Histamine; Imidazoles; Impromidine; Injections, Intraventricular; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1986 |
Evidence for histaminergic arousal mechanisms in the hypothalamus of cat.
Topics: Animals; Arousal; Cats; Dimaprit; Female; Histamine; Histamine Antagonists; Histidine Decarboxylase; Hypothalamus; Hypothalamus, Posterior; Injections; Injections, Intraperitoneal; Male; Methylhistidines; Pyrilamine; Thiourea | 1988 |
Changes in bronchial anaphylactic reactivity induced in guinea-pigs by long-term treatment with histamine H2-agents.
Topics: Anaphylaxis; Animals; Bronchi; Cimetidine; Dimaprit; Female; Guinea Pigs; Histamine H2 Antagonists; Histamine Release; Immunoglobulin E; Immunoglobulin G; In Vitro Techniques; Lung; Male; Ovalbumin; Passive Cutaneous Anaphylaxis; Respiratory Function Tests; Thiourea | 1984 |
Enhancement of histamine synthesis in mouse skin by epinephrine.
Topics: Animals; Dimaprit; Epinephrine; Guanidines; Histamine; Histamine Release; Kinetics; Male; Methylhistidines; Mice; Skin; Skin Physiological Phenomena; Thiourea | 1984 |
The effect of intrahypothalamic injection of homodimaprit on blood pressure.
Topics: Adrenal Medulla; Animals; Arginine Vasopressin; Blood Pressure; Body Temperature; Brain; Cerebrospinal Fluid; Dimaprit; Heart Rate; Hexamethonium Compounds; Histamine N-Methyltransferase; Hypothalamus; Male; Methyltransferases; Pulmonary Edema; Rats; Rats, Inbred Strains; Sympathectomy, Chemical; Thiourea | 1984 |
Evidence for a role of endogenous histamine in central cardiovascular regulation: inhibition of histamine-N-methyltransferase by SKF 91488.
Topics: Animals; Blood Pressure; Brain; Dimaprit; Heart Rate; Hemodynamics; Histamine; Histamine N-Methyltransferase; Male; Methyltransferases; Rats; Thiourea | 1981 |
Structure and function of human histamine N-methyltransferase: critical enzyme in histamine metabolism in airway.
Topics: Amino Acid Sequence; Animals; Base Sequence; Bronchi; Bronchoconstriction; Chromosome Mapping; Chromosomes, Human, Pair 1; Cloning, Molecular; Dimaprit; DNA, Complementary; Genes; Histamine; Histamine N-Methyltransferase; Humans; Molecular Sequence Data; Rats; RNA, Messenger; Structure-Activity Relationship | 1994 |
HMT regulates histamine-induced Cl- secretion across the canine tracheal epithelium.
Topics: Amiloride; Animals; Chlorides; Dimaprit; Dogs; Electrophysiology; Epithelium; Female; Histamine; Histamine N-Methyltransferase; Male; Trachea | 1994 |
Viral respiratory infection causes airway hyperresponsiveness and decreases histamine N-methyltransferase activity in guinea pigs.
Topics: Acetylcholine; Acetylcholinesterase; Airway Resistance; Animals; Bronchi; Bronchial Hyperreactivity; Bronchoconstriction; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine N-Methyltransferase; Lung; Male; Parainfluenza Virus 1, Human; Paramyxoviridae Infections; Respiratory Tract Infections; Trachea | 1994 |
Histamine N-methyltransferase modulates histamine- and antigen-induced bronchoconstriction in guinea pigs in vivo.
Topics: Aerosols; Animals; Antigens; Bronchial Provocation Tests; Bronchoconstriction; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine N-Methyltransferase; Immunization; Male; Ovalbumin; Tissue Distribution | 1993 |
Histamine N-methyltransferase inhibitor potentiates histamine- and antigen-induced airway microvascular leakage in guinea pigs.
Topics: Amine Oxidase (Copper-Containing); Animals; Antigens; Capillary Permeability; Dimaprit; Drug Synergism; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine N-Methyltransferase; Immunization; Male; Nasal Mucosa; Respiratory System | 1995 |
Histamine H2 receptor-mediated airway goblet cell secretion and its modulation by histamine-degrading enzymes.
Topics: Amine Oxidase (Copper-Containing); Animals; Asthma; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glycoproteins; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine N-Methyltransferase; Male; Methylhistamines; Mucus; Piperidines; Pyrilamine; Recombinant Proteins; Trachea | 1997 |
Effects of two histamine-N-methyltransferase inhibitors, SKF 91488 and BW 301 U, in rodent antinociception.
Topics: Analgesics; Animals; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Folic Acid Antagonists; Histamine Agonists; Histamine N-Methyltransferase; Injections, Intraventricular; Male; Methylhistamines; Mice; Muscle Contraction; Pain Measurement; Postural Balance; Psychomotor Performance; Pyrimidines; Rats; Rats, Wistar | 1997 |
HMT regulates histamine-induced glycoconjugate secretion from human airways in vitro.
Topics: Animals; Cats; Cimetidine; Dimaprit; Dinoprostone; Glycoconjugates; Glycoproteins; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine N-Methyltransferase; Humans; Indomethacin; Organ Culture Techniques; Phenothiazines; Receptors, Prostaglandin E; Trachea | 1997 |
Histamine N-methyltransferase regulates histamine-induced phosphoinositide hydrolysis in guinea pig cerebellum.
Topics: Animals; Cerebellum; Dimaprit; Dose-Response Relationship, Drug; Glycerol-3-Phosphate Dehydrogenase (NAD+); Glycerolphosphate Dehydrogenase; Guinea Pigs; Histamine; Histamine Antagonists; Histamine N-Methyltransferase; Hydrolysis; Male; Neurons; Oligonucleotide Probes; Organ Culture Techniques; Phosphatidylinositols; RNA; Synaptic Transmission; Tritium | 2001 |
Expression of diamine oxidase (histaminase) in guinea-pig tissues.
Topics: Amine Oxidase (Copper-Containing); Animals; Brain; Dimaprit; Dose-Response Relationship, Drug; Gastric Mucosa; Gene Expression Regulation, Enzymologic; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; In Situ Hybridization; In Vitro Techniques; Intestine, Small; Kidney; Liver; Male; Muscle Contraction; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Stomach | 2002 |
Endogenous central histamine-induced reversal of critical haemorrhagic hypotension in rats--studies with histamine N-methyltransferase inhibitor SKF 91488.
Topics: Animals; Blood Pressure; Brain Chemistry; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Heart Rate; Histamine; Histamine Antagonists; Histamine N-Methyltransferase; Hypotension; Injections, Intraventricular; Male; Rats; Rats, Wistar; Shock, Hemorrhagic; Survival | 2002 |
The protective effect of H2-receptor activation against the duration of myocardial hypoxia/reoxygenation-induced ventricular fibrillation in sensitized guinea-pig hearts.
Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Cytoplasmic Granules; Dimaprit; Electrocardiography; Enzyme Inhibitors; Female; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Histamine N-Methyltransferase; Histamine Release; Immunoglobulin E; In Vitro Techniques; Mast Cells; Myocardial Reperfusion Injury; Perfusion; Receptors, Histamine H2; Ventricular Fibrillation | 2005 |
Blockade of brain histamine metabolism alters methamphetamine-induced expression pattern of stereotypy in mice via histamine H1 receptors.
Topics: Analysis of Variance; Animals; Behavior, Animal; Brain; Dimaprit; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Histamine; Histamine Agents; Male; Maze Learning; Methamphetamine; Mice; Mice, Inbred ICR; Motor Activity; Receptors, Histamine H1; Stereotyped Behavior | 2007 |
Histamine metabolism influences blood vessel branching in zebrafish reg6 mutants.
Topics: Animals; Blood Vessels; Cell Movement; Dimaprit; Early Growth Response Protein 1; Embryo, Nonmammalian; Endothelium, Vascular; Histamine; Histamine N-Methyltransferase; Mutation; Neovascularization, Physiologic; Phenotype; Regeneration; Suppression, Genetic; Zebrafish | 2008 |
In vivo electrochemical evidence for simultaneous 5-HT and histamine release in the rat substantia nigra pars reticulata following medial forebrain bundle stimulation.
Topics: Animals; Dimaprit; Electric Stimulation; Electrochemistry; Histamine; Histamine Agonists; Histamine H3 Antagonists; Linear Models; Male; Medial Forebrain Bundle; Neural Pathways; Piperidines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Serotonin; Substantia Nigra | 2011 |
Loss of histaminergic modulation of thermoregulation and energy homeostasis in obese mice.
Topics: Adipose Tissue, Brown; Animals; Body Temperature Regulation; Dimaprit; Eating; Energy Metabolism; Histamine; Histamine Agonists; Homeostasis; Mice; Mice, Obese; Obesity; Preoptic Area; Receptors, Histamine | 2012 |
Histamine infused into basolateral amygdala enhances memory consolidation of inhibitory avoidance.
Topics: Amygdala; Analysis of Variance; Animals; Avoidance Learning; Dimaprit; Exploratory Behavior; Histamine; Histamine Agonists; Histamine Antagonists; Male; Maze Learning; Memory; Rats; Rats, Wistar; Reaction Time; Statistics, Nonparametric | 2013 |
Histamine acting on the basolateral amygdala reverts the impairment of aversive memory of rats submitted to neonatal maternal deprivation.
Topics: Analysis of Variance; Animals; Avoidance Learning; Basolateral Nuclear Complex; Dimaprit; Disease Models, Animal; Dose-Response Relationship, Drug; Exploratory Behavior; Female; Histamine; Histamine Agonists; Histamine Antagonists; Inhibition, Psychological; Male; Maternal Deprivation; Maze Learning; Memory Disorders; Pregnancy; Rats; Rats, Wistar | 2015 |