dimaprit and sk&f 91488

dimaprit has been researched along with sk&f 91488 in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-19908 (27.59)18.7374
1990's11 (37.93)18.2507
2000's6 (20.69)29.6817
2010's4 (13.79)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Beaven, MA; Shaff, RE1
Maeyama, K; Ohkawara, Y; Ohrui, T; Sasaki, H; Sasaki, M; Sekizawa, K; Takemura, M; Wada, H; Watanabe, T; Yamauchi, K1
Hannibal, T; Jørgensen, H; Knigge, U; Matzen, S; Warberg, J1
Gerges, E; Gertner, SB1
Donaldson, J; Hill, SJ1
Gertner, SB; Poulakos, JJ1
Jouvet, M; Lin, JS; Sakai, K1
Andersson, P; Bergstrand, H1
Rothschild, AM1
Gatti, PJ; Gertner, SB1
Gertner, SB; Klein, MC1
Katayose, D; Nakazawa, H; Ohkawara, Y; Ohtsu, H; Sekizawa, K; Shibahara, S; Suzuki, H; Takemura, M; Tamura, G; Yamauchi, K1
Sasaki, T; Satoh, M; Shimura, S; Takishima, T; Yamada, K; Yamauchi, K1
Maeyama, K; Morikawa, M; Nakazawa, H; Sasaki, H; Satoh, M; Sekizawa, K; Watanabe, T; Yamauchi, K1
Maeyama, K; Nakazawa, H; Ohkawara, Y; Ohrui, T; Sasaki, H; Sekizawa, K; Takishima, T; Watanabe, T; Yamauchi, K1
Maeyama, K; Morikawa, M; Nakazawa, H; Sasaki, H; Sekizawa, K; Watanabe, T; Yamauchi, K1
Chiyotani, A; Konno, K; Nakata, J; Takeyama, K; Tamaoki, J1
Bartolini, A; Ghelardini, C; Hänninen, J; Ipponi, A; Lamberti, C; Malmberg-Aiello, P1
Irokawa, T; Nagaki, M; Sasaki, T; Shimura, S; Shirato, K; Yamauchi, K; Yamaya, M1
Kitanaka, J; Kitanaka, N; Takemura, M; Terada, N; Tsujimura, T2
Jochem, J1
Akagi, M; Fukuishi, N; Imajo, N; Matsui, N; Matsui, S; Yasui, Y1
Kitanaka, J; Kitanaka, N; Morita, Y; Takemura, M; Tatsuta, T1
Cheng, YS; Huang, CC; Huang, CW; Yu, J1
Ambrose, RE; Dankoski, EC; Hashemi, P; Wightman, RM; Wood, KM1
Sanchez-Alavez, M; Sethi, J; Tabarean, IV1
Benetti, F; Izquierdo, I1
Benetti, F; da Silveira, CK; Izquierdo, I; Rosa, J1

Other Studies

29 other study(ies) available for dimaprit and sk&f 91488

ArticleYear
Inhibition of histamine methylation in vivo by the dimaprit analog, SKF Compound 91488.
    Agents and actions, 1979, Volume: 9, Issue:5-6

    Topics: Amine Oxidase (Copper-Containing); Animals; Brain; Dimaprit; Guanidines; Histamine; Histamine N-Methyltransferase; Kidney; Male; Methylation; Methyltransferases; Mice; Rats; Thiourea

1979
Histamine N-methyltransferase controls the contractile response of guinea pig trachea to histamine.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:3

    Topics: Animals; Dimaprit; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; Histamine; Histamine N-Methyltransferase; Male; Muscle Contraction; Muscle, Smooth; Thiourea; Trachea

1992
Involvement of histamine in the mediation of the stress-induced release of alpha-melanocyte-stimulating hormone in male rats.
    Neuroendocrinology, 1991, Volume: 54, Issue:6

    Topics: Adrenocorticotropic Hormone; alpha-MSH; Animals; Bromocriptine; Dimaprit; Histamine; Male; Methylhistidines; Propranolol; Rats; Rats, Inbred Strains; Stress, Physiological; Thiourea

1991
Central cardiovascular responses of histamine and homodimaprit in normal and hypophysectomized rats.
    Agents and actions, 1990, Volume: 31, Issue:3-4

    Topics: Animals; Blood Pressure; Brain; Dimaprit; Hexamethonium; Hexamethonium Compounds; Histamine; Hypophysectomy; Kinetics; Male; Rats; Rats, Inbred Strains; Thiourea; Vasopressins

1990
Selective enhancement of histamine H1-receptor responses in guinea-pig ileal smooth muscle by 1,4-dithiothreitol.
    British journal of pharmacology, 1986, Volume: 87, Issue:1

    Topics: Acetylcholine; Animals; Dimaprit; Dithionitrobenzoic Acid; Dithiothreitol; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Thiourea

1986
Studies on the desensitization of the central cardiovascular responses of histamine.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:3

    Topics: Animals; Blood Pressure; Brain; Cardiovascular System; Dimaprit; Heart Rate; Histamine; Imidazoles; Impromidine; Injections, Intraventricular; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1986
Evidence for histaminergic arousal mechanisms in the hypothalamus of cat.
    Neuropharmacology, 1988, Volume: 27, Issue:2

    Topics: Animals; Arousal; Cats; Dimaprit; Female; Histamine; Histamine Antagonists; Histidine Decarboxylase; Hypothalamus; Hypothalamus, Posterior; Injections; Injections, Intraperitoneal; Male; Methylhistidines; Pyrilamine; Thiourea

1988
Changes in bronchial anaphylactic reactivity induced in guinea-pigs by long-term treatment with histamine H2-agents.
    British journal of pharmacology, 1984, Volume: 82, Issue:1

    Topics: Anaphylaxis; Animals; Bronchi; Cimetidine; Dimaprit; Female; Guinea Pigs; Histamine H2 Antagonists; Histamine Release; Immunoglobulin E; Immunoglobulin G; In Vitro Techniques; Lung; Male; Ovalbumin; Passive Cutaneous Anaphylaxis; Respiratory Function Tests; Thiourea

1984
Enhancement of histamine synthesis in mouse skin by epinephrine.
    Life sciences, 1984, Oct-15, Volume: 35, Issue:16

    Topics: Animals; Dimaprit; Epinephrine; Guanidines; Histamine; Histamine Release; Kinetics; Male; Methylhistidines; Mice; Skin; Skin Physiological Phenomena; Thiourea

1984
The effect of intrahypothalamic injection of homodimaprit on blood pressure.
    Neuropharmacology, 1984, Volume: 23, Issue:6

    Topics: Adrenal Medulla; Animals; Arginine Vasopressin; Blood Pressure; Body Temperature; Brain; Cerebrospinal Fluid; Dimaprit; Heart Rate; Hexamethonium Compounds; Histamine N-Methyltransferase; Hypothalamus; Male; Methyltransferases; Pulmonary Edema; Rats; Rats, Inbred Strains; Sympathectomy, Chemical; Thiourea

1984
Evidence for a role of endogenous histamine in central cardiovascular regulation: inhibition of histamine-N-methyltransferase by SKF 91488.
    The Journal of pharmacology and experimental therapeutics, 1981, Volume: 216, Issue:2

    Topics: Animals; Blood Pressure; Brain; Dimaprit; Heart Rate; Hemodynamics; Histamine; Histamine N-Methyltransferase; Male; Methyltransferases; Rats; Thiourea

1981
Structure and function of human histamine N-methyltransferase: critical enzyme in histamine metabolism in airway.
    The American journal of physiology, 1994, Volume: 267, Issue:3 Pt 1

    Topics: Amino Acid Sequence; Animals; Base Sequence; Bronchi; Bronchoconstriction; Chromosome Mapping; Chromosomes, Human, Pair 1; Cloning, Molecular; Dimaprit; DNA, Complementary; Genes; Histamine; Histamine N-Methyltransferase; Humans; Molecular Sequence Data; Rats; RNA, Messenger; Structure-Activity Relationship

1994
HMT regulates histamine-induced Cl- secretion across the canine tracheal epithelium.
    Respiration physiology, 1994, Volume: 97, Issue:1

    Topics: Amiloride; Animals; Chlorides; Dimaprit; Dogs; Electrophysiology; Epithelium; Female; Histamine; Histamine N-Methyltransferase; Male; Trachea

1994
Viral respiratory infection causes airway hyperresponsiveness and decreases histamine N-methyltransferase activity in guinea pigs.
    American journal of respiratory and critical care medicine, 1994, Volume: 149, Issue:5

    Topics: Acetylcholine; Acetylcholinesterase; Airway Resistance; Animals; Bronchi; Bronchial Hyperreactivity; Bronchoconstriction; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine N-Methyltransferase; Lung; Male; Parainfluenza Virus 1, Human; Paramyxoviridae Infections; Respiratory Tract Infections; Trachea

1994
Histamine N-methyltransferase modulates histamine- and antigen-induced bronchoconstriction in guinea pigs in vivo.
    The American review of respiratory disease, 1993, Volume: 147, Issue:1

    Topics: Aerosols; Animals; Antigens; Bronchial Provocation Tests; Bronchoconstriction; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine N-Methyltransferase; Immunization; Male; Ovalbumin; Tissue Distribution

1993
Histamine N-methyltransferase inhibitor potentiates histamine- and antigen-induced airway microvascular leakage in guinea pigs.
    The Journal of allergy and clinical immunology, 1995, Volume: 96, Issue:6 Pt 1

    Topics: Amine Oxidase (Copper-Containing); Animals; Antigens; Capillary Permeability; Dimaprit; Drug Synergism; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine N-Methyltransferase; Immunization; Male; Nasal Mucosa; Respiratory System

1995
Histamine H2 receptor-mediated airway goblet cell secretion and its modulation by histamine-degrading enzymes.
    The Journal of allergy and clinical immunology, 1997, Volume: 99, Issue:2

    Topics: Amine Oxidase (Copper-Containing); Animals; Asthma; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glycoproteins; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine N-Methyltransferase; Male; Methylhistamines; Mucus; Piperidines; Pyrilamine; Recombinant Proteins; Trachea

1997
Effects of two histamine-N-methyltransferase inhibitors, SKF 91488 and BW 301 U, in rodent antinociception.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 355, Issue:3

    Topics: Analgesics; Animals; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Folic Acid Antagonists; Histamine Agonists; Histamine N-Methyltransferase; Injections, Intraventricular; Male; Methylhistamines; Mice; Muscle Contraction; Pain Measurement; Postural Balance; Psychomotor Performance; Pyrimidines; Rats; Rats, Wistar

1997
HMT regulates histamine-induced glycoconjugate secretion from human airways in vitro.
    Respiration physiology, 1997, Volume: 108, Issue:3

    Topics: Animals; Cats; Cimetidine; Dimaprit; Dinoprostone; Glycoconjugates; Glycoproteins; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine N-Methyltransferase; Humans; Indomethacin; Organ Culture Techniques; Phenothiazines; Receptors, Prostaglandin E; Trachea

1997
Histamine N-methyltransferase regulates histamine-induced phosphoinositide hydrolysis in guinea pig cerebellum.
    Neuroscience letters, 2001, Jul-27, Volume: 308, Issue:1

    Topics: Animals; Cerebellum; Dimaprit; Dose-Response Relationship, Drug; Glycerol-3-Phosphate Dehydrogenase (NAD+); Glycerolphosphate Dehydrogenase; Guinea Pigs; Histamine; Histamine Antagonists; Histamine N-Methyltransferase; Hydrolysis; Male; Neurons; Oligonucleotide Probes; Organ Culture Techniques; Phosphatidylinositols; RNA; Synaptic Transmission; Tritium

2001
Expression of diamine oxidase (histaminase) in guinea-pig tissues.
    European journal of pharmacology, 2002, Feb-22, Volume: 437, Issue:3

    Topics: Amine Oxidase (Copper-Containing); Animals; Brain; Dimaprit; Dose-Response Relationship, Drug; Gastric Mucosa; Gene Expression Regulation, Enzymologic; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; In Situ Hybridization; In Vitro Techniques; Intestine, Small; Kidney; Liver; Male; Muscle Contraction; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Stomach

2002
Endogenous central histamine-induced reversal of critical haemorrhagic hypotension in rats--studies with histamine N-methyltransferase inhibitor SKF 91488.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 2002, Volume: 51, Issue:11

    Topics: Animals; Blood Pressure; Brain Chemistry; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Heart Rate; Histamine; Histamine Antagonists; Histamine N-Methyltransferase; Hypotension; Injections, Intraventricular; Male; Rats; Rats, Wistar; Shock, Hemorrhagic; Survival

2002
The protective effect of H2-receptor activation against the duration of myocardial hypoxia/reoxygenation-induced ventricular fibrillation in sensitized guinea-pig hearts.
    Journal of pharmacological sciences, 2005, Volume: 99, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Cytoplasmic Granules; Dimaprit; Electrocardiography; Enzyme Inhibitors; Female; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Histamine N-Methyltransferase; Histamine Release; Immunoglobulin E; In Vitro Techniques; Mast Cells; Myocardial Reperfusion Injury; Perfusion; Receptors, Histamine H2; Ventricular Fibrillation

2005
Blockade of brain histamine metabolism alters methamphetamine-induced expression pattern of stereotypy in mice via histamine H1 receptors.
    Neuroscience, 2007, Jul-13, Volume: 147, Issue:3

    Topics: Analysis of Variance; Animals; Behavior, Animal; Brain; Dimaprit; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Histamine; Histamine Agents; Male; Maze Learning; Methamphetamine; Mice; Mice, Inbred ICR; Motor Activity; Receptors, Histamine H1; Stereotyped Behavior

2007
Histamine metabolism influences blood vessel branching in zebrafish reg6 mutants.
    BMC developmental biology, 2008, Mar-25, Volume: 8

    Topics: Animals; Blood Vessels; Cell Movement; Dimaprit; Early Growth Response Protein 1; Embryo, Nonmammalian; Endothelium, Vascular; Histamine; Histamine N-Methyltransferase; Mutation; Neovascularization, Physiologic; Phenotype; Regeneration; Suppression, Genetic; Zebrafish

2008
In vivo electrochemical evidence for simultaneous 5-HT and histamine release in the rat substantia nigra pars reticulata following medial forebrain bundle stimulation.
    Journal of neurochemistry, 2011, Volume: 118, Issue:5

    Topics: Animals; Dimaprit; Electric Stimulation; Electrochemistry; Histamine; Histamine Agonists; Histamine H3 Antagonists; Linear Models; Male; Medial Forebrain Bundle; Neural Pathways; Piperidines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Serotonin; Substantia Nigra

2011
Loss of histaminergic modulation of thermoregulation and energy homeostasis in obese mice.
    Neuroscience, 2012, Aug-16, Volume: 217

    Topics: Adipose Tissue, Brown; Animals; Body Temperature Regulation; Dimaprit; Eating; Energy Metabolism; Histamine; Histamine Agonists; Homeostasis; Mice; Mice, Obese; Obesity; Preoptic Area; Receptors, Histamine

2012
Histamine infused into basolateral amygdala enhances memory consolidation of inhibitory avoidance.
    The international journal of neuropsychopharmacology, 2013, Volume: 16, Issue:7

    Topics: Amygdala; Analysis of Variance; Animals; Avoidance Learning; Dimaprit; Exploratory Behavior; Histamine; Histamine Agonists; Histamine Antagonists; Male; Maze Learning; Memory; Rats; Rats, Wistar; Reaction Time; Statistics, Nonparametric

2013
Histamine acting on the basolateral amygdala reverts the impairment of aversive memory of rats submitted to neonatal maternal deprivation.
    Behavioural brain research, 2015, Feb-01, Volume: 278

    Topics: Analysis of Variance; Animals; Avoidance Learning; Basolateral Nuclear Complex; Dimaprit; Disease Models, Animal; Dose-Response Relationship, Drug; Exploratory Behavior; Female; Histamine; Histamine Agonists; Histamine Antagonists; Inhibition, Psychological; Male; Maternal Deprivation; Maze Learning; Memory Disorders; Pregnancy; Rats; Rats, Wistar

2015