dimaprit and pyrilamine

dimaprit has been researched along with pyrilamine in 55 studies

Research

Studies (55)

TimeframeStudies, this research(%)All Research%
pre-199032 (58.18)18.7374
1990's18 (32.73)18.2507
2000's5 (9.09)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Timmerman, H1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Nowak, JZ; Sek, B1
Benedito, S; Nielsen, PJ; Nyborg, NC; Prieto, D1
Dolata, J; Lindberg, S; Mercke, U1
Almeida, L; Figueiredo, A; Gonçalo, M; Poiares-Baptista, A; Ribeiro, CA; Teixeira, F1
Cooke, HJ; Wang, YZ1
Młynarska, MS1
Matsuki, T; Ohhashi, T1
Bugajski, J; Gadek-Michalska, A1
Girard, A; Marche, P1
Hutchison, VH; Spriestersbach, KK1
Knigge, U; Matzen, S; Warberg, J1
Akahori, H; Kamei, C; Kitazumi, K; Tasaka, K1
Ledgard, SE; Nieves, AL; Woodward, DF1
Barker, LA; Winbery, SL1
Donaldson, J; Hill, SJ1
Kim, LE; Oudart, N; Sercombe, R; Teste, JF1
Bugajski, J; Gadek, A1
Jouvet, M; Lin, JS; Sakai, K1
Fromm, D; Furukawa, T; Olender, EJ; Woods, DJ1
Kume, S; Ohashi, T; Ozaki, Y1
Gristwood, RW; Lincoln, JC; Owen, DA1
Daniel, D; Owen, DA; Poy, E; Woodward, DF1
Oriowo, MA1
Heldsinger, AA; Skoglund, ML; Vinik, AI1
Donoso, AO; Zárate, MB1
Guldvog, I; Linnestad, P; Schrumpf, E1
Nemeth, PR; Ort, CA; Wood, JD1
Bugajski, J; Janusz, Z1
Owen, DA; Pipkin, MA; Woodward, DF1
Bottomley, KM; Lewis, S; Rising, TJ; Steward, A1
Jespersen, LT; Mikkelsen, E; Sakr, AM1
Cooke, HJ; Nemeth, PR; Wood, JD1
Bordi, F; Chiavarini, M; Impicciatore, M; Morini, G; Plazzi, PV; Vitali, F1
Binderup, L1
Chand, N; DeRoth, L1
Del Soldato, P1
Harvey, CA; Owen, DA; Shaw, KD1
Di Donato, M; Mantovani, P; Santicioli, P1
Duchemin, AM; Quach, TT; Rose, C; Schwartz, JC1
Kohno, S; Nabe, T; Nakao, S; Ogawa, K; Ohata, K; Yamamura, H1
Kohno, S; Nabe, T; Ogawa, K; Ohata, K; Yamamura, H1
Carson, CC; Davies, MG; Hagen, PO; Kim, YC; Lee, TH1
Chiyotani, A; Konno, K; Nakata, J; Takeyama, K; Tamaoki, J1
Kitazawa, T; Sato, T; Shishido, H; Taneike, T1
Fu, LW; Longhurst, JC; Pan, HL1
Easton, AS; Fraser, PA; Sarker, MH1
Grundy, D; Haupt, W; Kirkup, AJ; Kreis, ME1
Capasso, F; Costa, M; Izzo, AA; Mascolo, N1
Chen, Z; Fujii, Y; Kamei, C; Sugimoto, Y; Suzuki, G1
Firth, TA; Guarraci, FA; Hemming, JM; Jennings, LJ; Mawe, GM; Nelson, MT1
Bacon, KB; Center, DM; Cruikshank, WW; Gantner, F; Sakai, K; Tusche, MW1
Nakamura, T; Ueno, K; Yamaura, K; Yano, S; Yonekawa, T1
Dube, PH; Handley, SA; Miller, VL1

Reviews

1 review(s) available for dimaprit and pyrilamine

ArticleYear
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship

1990

Other Studies

54 other study(ies) available for dimaprit and pyrilamine

ArticleYear
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Cyclic AMP generating systems in vertebrate retina: effects of histamine and an established retinal modulator, dopamine.
    Agents and actions, 1991, Volume: 33, Issue:1-2

    Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Chickens; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dopamine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Retina; Thiazoles; Thiourea

1991
Histamine induces endothelium-dependent relaxation of bovine retinal arteries.
    Investigative ophthalmology & visual science, 1991, Volume: 32, Issue:1

    Topics: Acetylcholine; Animals; Cattle; Cimetidine; Dimaprit; Endothelium, Vascular; Histamine; Muscle Relaxation; Pyridines; Pyrilamine; Receptors, Histamine; Retinal Artery; Tachyphylaxis; Thiourea

1991
Histamine stimulation of mucociliary activity in the rabbit maxillary sinus.
    The Annals of otology, rhinology, and laryngology, 1990, Volume: 99, Issue:8

    Topics: Animals; Atropine; Cilia; Cimetidine; Dimaprit; Female; Histamine; Histamine H2 Antagonists; Male; Maxillary Sinus; Mucociliary Clearance; Pyrilamine; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Muscarinic; Thiourea

1990
Mechanism of action of doxepin in the treatment of chronic urticaria.
    Fundamental & clinical pharmacology, 1990, Volume: 4, Issue:2

    Topics: Adult; Aged; Animals; Atropine; Carbachol; Chronic Disease; Dimaprit; Doxepin; Female; Gastric Juice; Guinea Pigs; Heart; Histamine; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Pylorus; Pyrilamine; Rats; Thiourea; Urticaria

1990
H2 receptors mediate cyclical chloride secretion in guinea pig distal colon.
    The American journal of physiology, 1990, Volume: 258, Issue:6 Pt 1

    Topics: Animals; Bumetanide; Chlorides; Cimetidine; Colon; Dimaprit; Guinea Pigs; Histamine; In Vitro Techniques; Intestinal Mucosa; Kinetics; Male; Muscle, Smooth; Pyrilamine; Receptors, Histamine H2; Tetrodotoxin; Thiourea

1990
Antagonistic effect of naloxone on the hypertensive response of intraventricularly administered histamine.
    Agents and actions, 1990, Volume: 30, Issue:1-2

    Topics: Animals; Blood Pressure; Cimetidine; Dimaprit; Hemodynamics; Histamine; In Vitro Techniques; Injections, Intraventricular; Male; Naloxone; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Thiourea

1990
Endothelium and mechanical responses of isolated monkey pulmonary veins to histamine.
    The American journal of physiology, 1990, Volume: 259, Issue:4 Pt 2

    Topics: Animals; Dimaprit; Endothelium, Vascular; Famotidine; Hemoglobins; Histamine; In Vitro Techniques; Macaca; Methylene Blue; Pulmonary Veins; Pyridines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Vasoconstriction; Vasodilation

1990
Antagonistic action of naloxone on central histamine receptors-stimulated corticosterone secretion in rats under stress.
    Agents and actions, 1989, Volume: 28, Issue:3-4

    Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Histamine; Male; Methylhistamines; Naloxone; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Restraint, Physical; Stress, Physiological; Thiourea

1989
Phosphoinositides and cicletanine.
    Drugs under experimental and clinical research, 1988, Volume: 14, Issue:2-3

    Topics: Angiotensin II; Animals; Antihypertensive Agents; Aorta, Thoracic; Cells, Cultured; Dimaprit; Diuretics; Guinea Pigs; Histamine; Male; Muscle, Smooth, Vascular; Phenylephrine; Phosphatidylinositols; Pyridines; Pyrilamine; Thiourea

1988
Histamine and histamine receptors: behavioral thermoregulation in the salamander Necturus maculosus.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1986, Volume: 85, Issue:1

    Topics: Animals; Body Temperature Regulation; Cimetidine; Dimaprit; Histamine; Histidine; Necturus; Pyridines; Pyrilamine; Receptors, Histamine; Thiourea

1986
Histaminergic stimulation of prolactin secretion mediated via H1- or H2-receptors: dependence on routes of administration.
    Neuroendocrinology, 1986, Volume: 44, Issue:1

    Topics: Animals; Cimetidine; Dimaprit; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Pituitary Gland, Anterior; Prolactin; Pyrilamine; Pyrimidinones; Rats; Receptors, Histamine; Thiazoles; Thiourea

1986
The effects of histamine and some related compounds on conditioned avoidance response in rats.
    Life sciences, 1985, Nov-25, Volume: 37, Issue:21

    Topics: Acetylcholine; Animals; Avoidance Learning; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Hypothalamus; Injections, Intraventricular; Kinetics; Male; Methylhistamines; Pyrilamine; Rats; Rats, Inbred Strains; Scopolamine; Thiazoles; Thiourea

1985
Conjunctival immediate hypersensitivity: re-evaluation of histamine involvement in the vasopermeability response.
    Investigative ophthalmology & visual science, 1986, Volume: 27, Issue:1

    Topics: Albumins; Animals; Capillary Permeability; Cimetidine; Conjunctiva; Dimaprit; Dose-Response Relationship, Drug; Drug Combinations; Eyelids; Guinea Pigs; Histamine; Histamine Antagonists; Hypersensitivity, Immediate; Imidazoles; Impromidine; Male; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1986
Metronidazole and 5-aminosalicylic acid enhance the contractile activity of histaminergic agonists on the guinea-pig isolated ileum.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 236, Issue:3

    Topics: Aminosalicylic Acids; Animals; Cimetidine; Computers; Dimaprit; Dose-Response Relationship, Drug; Drug Synergism; Duodenum; Female; Guinea Pigs; Heart; Histamine; Ileum; In Vitro Techniques; Jejunum; Male; Mesalamine; Metronidazole; Muscle Contraction; Myenteric Plexus; Pyrilamine; Receptors, Histamine; Scopolamine; Tetrodotoxin; Thiourea

1986
Selective enhancement of histamine H1-receptor responses in guinea-pig ileal smooth muscle by 1,4-dithiothreitol.
    British journal of pharmacology, 1986, Volume: 87, Issue:1

    Topics: Acetylcholine; Animals; Dimaprit; Dithionitrobenzoic Acid; Dithiothreitol; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Thiourea

1986
Participation of vascular H1-receptors in histaminergic relaxation of rabbit middle cerebral artery in vitro.
    Archives internationales de pharmacodynamie et de therapie, 1986, Volume: 283, Issue:2

    Topics: Animals; Cerebral Arteries; Cimetidine; Dimaprit; Drug Interactions; Histamine; In Vitro Techniques; Methylhistamines; Muscle Relaxation; Muscle, Smooth, Vascular; Phenethylamines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Thiourea

1986
Hyperlipemic responses induced by centrally administered histamine H1- and H2-receptor agonists in rats.
    Agents and actions, 1987, Volume: 20, Issue:3-4

    Topics: Animals; Brain; Cimetidine; Dimaprit; Fatty Acids, Nonesterified; Hyperlipidemias; Imidazoles; Impromidine; Injections, Intraventricular; Male; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Thiourea

1987
Evidence for histaminergic arousal mechanisms in the hypothalamus of cat.
    Neuropharmacology, 1988, Volume: 27, Issue:2

    Topics: Animals; Arousal; Cats; Dimaprit; Female; Histamine; Histamine Antagonists; Histidine Decarboxylase; Hypothalamus; Hypothalamus, Posterior; Injections; Injections, Intraperitoneal; Male; Methylhistidines; Pyrilamine; Thiourea

1988
Histamine receptor effects on dissipation of an intracellular proton gradient of isolated gastric mucosal surface cells.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1987, Volume: 185, Issue:4

    Topics: Animals; Bicarbonates; Chlorides; Cimetidine; Dimaprit; Diphenhydramine; Gastric Acid; Gastric Mucosa; Histamine; Protons; Pyridines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Sodium; Thiourea

1987
Effects of histamine agonists and antagonists on luminol-dependent chemiluminescence of granulocytes.
    Agents and actions, 1984, Volume: 15, Issue:3-4

    Topics: Cimetidine; Dimaprit; Granulocytes; Histamine; Histamine Antagonists; Humans; In Vitro Techniques; Luminescent Measurements; Luminol; Pyridazines; Pyridines; Pyrilamine; Ranitidine; Thiourea

1984
Effects of histamine on human isolated heart muscle: comparison with effects of noradrenaline.
    The Journal of pharmacy and pharmacology, 1980, Volume: 32, Issue:2

    Topics: Cimetidine; Dimaprit; Heart; Histamine; Humans; In Vitro Techniques; Myocardial Contraction; Norepinephrine; Propranolol; Pyrilamine; Receptors, Histamine H2; Thiourea

1980
Evaluation of the role of Histamine H1- and H2-receptors in cutaneous inflammation in the guinea-pig produced by histamine and mast cell degranulation.
    British journal of pharmacology, 1980, Volume: 69, Issue:4

    Topics: Animals; Cimetidine; Dimaprit; Guinea Pigs; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Inflammation; Male; Mast Cells; Mathematics; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Skin; Thiourea; Vasodilation

1980
An inhibitory effect of histamine on the rat anococcygeus muscle.
    The Journal of pharmacy and pharmacology, 1982, Volume: 34, Issue:3

    Topics: Acetylcholine; Animals; Carbachol; Cimetidine; Dimaprit; Drug Interactions; Guanidines; Histamine; Imidazoles; Impromidine; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Pyrilamine; Rats; Thiourea

1982
Evidence for histamine H1 and H2 receptors in guinea-pig oxyntic cells.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:1

    Topics: Animals; Carbonic Anhydrases; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Methylhistamines; Parietal Cells, Gastric; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1983
Release of prolactin and luteinizing hormone by histamine agonists in ovariectomized, steroid-treated rats under ether anesthesia.
    Experimental brain research, 1983, Volume: 52, Issue:2

    Topics: Animals; Castration; Dimaprit; Female; Histamine; Histamine H1 Antagonists; Luteinizing Hormone; Methylhistamines; Metiamide; Pituitary Gland, Anterior; Prolactin; Pyridines; Pyrilamine; Rats; Thiourea

1983
The effect of histamine, H1 and H2 agonists, and H1 and H2 antagonists on postprandial pancreatic polypeptide release in dogs.
    Scandinavian journal of gastroenterology, 1983, Volume: 18, Issue:2

    Topics: Animals; Cimetidine; Dimaprit; Dogs; Food; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Pancreatic Polypeptide; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Secretory Rate; Thiazoles; Thiourea

1983
Intracellular study of effects of histamine on electrical behaviour of myenteric neurones in guinea-pig small intestine.
    The Journal of physiology, 1984, Volume: 355

    Topics: Action Potentials; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine Antagonists; In Vitro Techniques; Intestine, Small; Membrane Potentials; Myenteric Plexus; Neurons; Neurotransmitter Agents; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Serotonin; Thiourea

1984
Central histaminergic stimulation of pituitary--adrenocortical response in the rat.
    Life sciences, 1983, Sep-19, Volume: 33, Issue:12

    Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Dose-Response Relationship, Drug; Histamine; Imidazoles; Impromidine; Male; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1983
Studies on cutaneous vascular permeability in the rat: increases caused by histamine and histamine-like agents.
    Agents and actions, 1984, Volume: 14, Issue:1

    Topics: Animals; Capillary Permeability; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Histamine; Microcirculation; Pyrilamine; Rats; Regional Blood Flow; Skin; Thiourea

1984
A new in vivo method for the measurement of repetitive anaphylactic responses in the guinea-pig.
    British journal of pharmacology, 1984, Volume: 81, Issue:1

    Topics: Albuterol; Anaphylaxis; Animals; Antibodies; Cromolyn Sodium; Dimaprit; Guinea Pigs; Male; Pyrilamine; Theophylline; Thiourea

1984
Studies on the effect of histamine in isolated human pulmonary arteries and veins.
    Acta pharmacologica et toxicologica, 1984, Volume: 54, Issue:2

    Topics: Aged; Dimaprit; Female; Histamine; Humans; In Vitro Techniques; Male; Methylhistamines; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phentolamine; Potassium; Pulmonary Artery; Pulmonary Veins; Pyrilamine; Thiourea

1984
Histamine action on guinea pig ileal mucosa.
    The American journal of physiology, 1984, Volume: 246, Issue:4 Pt 1

    Topics: Animals; Bicarbonates; Biological Transport, Active; Chlorides; Dimaprit; Electric Conductivity; Female; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Intestinal Mucosa; Male; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1984
[Imidazolic H2-agonists: importance of 2-amino substitution for pharmacological activity].
    Bollettino della Societa italiana di biologia sperimentale, 1984, Apr-30, Volume: 60, Issue:4

    Topics: Animals; Biological Assay; Cats; Dimaprit; Gastric Acid; Guinea Pigs; Histamine; Methylhistamines; Muscle Relaxation; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Structure-Activity Relationship; Thiourea; Urinary Bladder

1984
Effects of the H2-receptor agonist dimaprit on lymphocyte responsiveness in vitro.
    Agents and actions, 1984, Volume: 15, Issue:3-4

    Topics: Animals; Cells, Cultured; Cimetidine; Dimaprit; Ephedrine; Female; Glucosamine; In Vitro Techniques; Lymphocyte Activation; Lymphocytes; Metoprolol; Phagocytosis; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H2; T-Lymphocytes; T-Lymphocytes, Regulatory; Thiourea; Thymidine

1984
Acute systemic anaphylaxis in adult domestic fowl: evidence for the protective role of H2-histaminergic and beta 2-adrenergic receptors.
    American journal of veterinary research, 1980, Volume: 41, Issue:1

    Topics: Anaphylaxis; Animals; Blood Pressure; Carotid Arteries; Chickens; Chromones; Cimetidine; Dimaprit; Ethers; Heart Rate; Metiamide; Poultry Diseases; Propranolol; Pyrilamine; Receptors, Adrenergic; Receptors, Adrenergic, beta; Receptors, Histamine; Receptors, Histamine H2; Terbutaline; Thiourea

1980
Studies with specific agonists and antagonists of the role of histamine H1- and H2-receptor activation in the pathogenesis of gastric lesions in rats.
    Agents and actions, 1984, Volume: 14, Issue:2

    Topics: Aminopyridines; Animals; Atropine; Dimaprit; Drug Interactions; Female; Histamine; Pyridines; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Stomach Ulcer; Thiourea

1984
Evidence for both histamine H1- and H2-receptors in the gastric vasculature of the cat.
    British journal of pharmacology, 1980, Volume: 69, Issue:1

    Topics: Animals; Cats; Celiac Artery; Dimaprit; Gastric Juice; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Regional Blood Flow; Stomach; Thiourea; Time Factors

1980
Further experiments on the pharmacological actions of ergometrine.
    Bollettino della Societa italiana di biologia sperimentale, 1981, Jun-30, Volume: 57, Issue:12

    Topics: Animals; Cattle; Cimetidine; Coronary Vessels; Dimaprit; Ergonovine; Gastric Acid; Guinea Pigs; Histamine; Muscle Contraction; Pyrilamine; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1981
Specific desensitization of histamine H1 receptor-mediated [3H]glycogen hydrolysis in brain slices.
    Molecular pharmacology, 1981, Volume: 20, Issue:2

    Topics: Adult; Animals; Brain; Cerebral Cortex; Cycloheximide; Dimaprit; Glycogen; Humans; Hydrolysis; In Vitro Techniques; Kinetics; Male; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Thiourea

1981
Possible participation of histamine H3-receptors in the regulation of anaphylactic histamine release from isolated rat peritoneal mast cells.
    Japanese journal of pharmacology, 1994, Volume: 66, Issue:2

    Topics: Anaphylaxis; Animals; Anticonvulsants; Chromatography, High Pressure Liquid; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Histamine; Histamine Agonists; Histamine Antagonists; Histamine Release; In Vitro Techniques; L-Lactate Dehydrogenase; Male; Mast Cells; Methylhistamines; p-Methoxy-N-methylphenethylamine; Peritoneal Cavity; Peritoneum; Piperidines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H3

1994
Dimaprit, a histamine H2-agonist, inhibits anaphylactic histamine release from mast cells and the decreased release is restored by thioperamide (H3-antagonist), but not by cimetidine (H2-antagonist).
    Japanese journal of pharmacology, 1993, Volume: 62, Issue:1

    Topics: Anaphylaxis; Animals; Anticonvulsants; Betahistine; Cimetidine; Dimaprit; Histamine H2 Antagonists; Histamine Release; In Vitro Techniques; Indicators and Reagents; Male; Mast Cells; Piperidines; Pyrilamine; Rats; Rats, Wistar

1993
Characterization and function of histamine receptors in corpus cavernosum.
    The Journal of urology, 1995, Volume: 153, Issue:2

    Topics: Acetylcholine; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Papaverine; Penis; Piperidines; Pyrilamine; Rabbits; Receptors, Histamine; Thiazoles

1995
Histamine H2 receptor-mediated airway goblet cell secretion and its modulation by histamine-degrading enzymes.
    The Journal of allergy and clinical immunology, 1997, Volume: 99, Issue:2

    Topics: Amine Oxidase (Copper-Containing); Animals; Asthma; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glycoproteins; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine N-Methyltransferase; Male; Methylhistamines; Mucus; Piperidines; Pyrilamine; Recombinant Proteins; Trachea

1997
Histamine mediates the muscle layer-specific responses in the isolated swine myometrium.
    Journal of veterinary pharmacology and therapeutics, 1997, Volume: 20, Issue:3

    Topics: Animals; Dimaprit; Female; Histamine; Histamine Agonists; Histamine H1 Antagonists; Muscle, Smooth; Myometrium; Pyrilamine; Receptors, Histamine; Swine; Uterine Contraction

1997
Endogenous histamine stimulates ischemically sensitive abdominal visceral afferents through H1 receptors.
    The American journal of physiology, 1997, Volume: 273, Issue:6

    Topics: Abdomen; Afferent Pathways; Animals; Bile Ducts; Blood Pressure; Cats; Chlorpheniramine; Dimaprit; Duodenum; Female; Gallbladder; Histamine; Histamine H1 Antagonists; Indomethacin; Ischemia; Male; Methylhistamines; Nerve Fibers; Neural Conduction; Pancreas; Pyrilamine; Receptors, Histamine H1

1997
Regulation of cerebral microvascular permeability by histamine in the anaesthetized rat.
    The Journal of physiology, 1998, Mar-15, Volume: 507 ( Pt 3)

    Topics: Anesthesia, General; Animals; Capillary Permeability; Cerebrovascular Circulation; Cimetidine; Dimaprit; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Muscle, Smooth, Vascular; Pia Mater; Pyrilamine; Rats; Venules

1998
Histamine sensitivity of mesenteric afferent nerves in the rat jejunum.
    The American journal of physiology, 1998, Volume: 275, Issue:4

    Topics: Afferent Pathways; Animals; Blood Pressure; Dimaprit; Histamine; Histamine Agonists; Histamine Antagonists; Jejunum; Muscle, Smooth; Nifedipine; Piperidines; Pyrilamine; Ranitidine; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Splanchnic Circulation

1998
The role of histamine H1, H2 and H3 receptors on enteric ascending synaptic transmission in the guinea pig ileum.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 287, Issue:3

    Topics: Animals; Cimetidine; Dimaprit; Electric Stimulation; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Ileum; Male; Motor Neurons; Muscle Contraction; Muscle, Smooth; Pyrilamine; Receptors, Histamine; Synaptic Transmission

1998
Effects of histamine and related compounds on regional cerebral blood flow in rats.
    Methods and findings in experimental and clinical pharmacology, 1999, Volume: 21, Issue:9

    Topics: Animals; Benzothiazoles; Blood Pressure; Brain Chemistry; Dimaprit; Diphenhydramine; Drug Interactions; Hippocampus; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Male; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Wistar; Regional Blood Flow; Thiazoles; Time Factors

1999
Actions of histamine on muscle and ganglia of the guinea pig gallbladder.
    American journal of physiology. Gastrointestinal and liver physiology, 2000, Volume: 279, Issue:3

    Topics: Adenosine Triphosphate; Animals; Dimaprit; Excitatory Postsynaptic Potentials; Female; Gallbladder; Gallbladder Emptying; Ganglia, Autonomic; Guinea Pigs; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Mast Cells; Membrane Potentials; Muscle, Smooth; p-Methoxy-N-methylphenethylamine; Patch-Clamp Techniques; Potassium Channels; Pyrilamine; Ranitidine; Receptors, Histamine H1; Receptors, Histamine H2

2000
Histamine h(4) and h(2) receptors control histamine-induced interleukin-16 release from human CD8(+) T cells.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 303, Issue:1

    Topics: Base Sequence; CD4-Positive T-Lymphocytes; CD8-Positive T-Lymphocytes; Cells, Cultured; Cimetidine; Dimaprit; DNA Primers; Female; Gene Expression Regulation; Histamine; Humans; Interleukin-16; Male; Methylhistamines; Polymerase Chain Reaction; Pyrilamine; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H2; Receptors, Histamine H4

2002
The histamine H2-receptor antagonist, cimetidine, inhibits the articular osteopenia in rats with adjuvant-induced arthritis by suppressing the osteoclast differentiation induced by histamine.
    Journal of pharmacological sciences, 2003, Volume: 92, Issue:1

    Topics: Animals; Arthritis, Experimental; Bone Density; Bone Resorption; Cartilage, Articular; Cell Differentiation; Cimetidine; Dimaprit; Female; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Osteoclasts; Pyrilamine; Rats; Rats, Inbred Lew

2003
Histamine signaling through the H(2) receptor in the Peyer's patch is important for controlling Yersinia enterocolitica infection.
    Proceedings of the National Academy of Sciences of the United States of America, 2006, Jun-13, Volume: 103, Issue:24

    Topics: Animals; Anti-Allergic Agents; Anti-Ulcer Agents; Cimetidine; Dimaprit; Female; Gene Expression Profiling; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine Decarboxylase; Mice; Mice, Inbred C57BL; Oligonucleotide Array Sequence Analysis; Omeprazole; Peyer's Patches; Pyrilamine; Receptors, Histamine H2; Signal Transduction; Survival Rate; Yersinia enterocolitica; Yersinia Infections

2006