dimaprit has been researched along with histamine in 249 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 118 (47.39) | 18.7374 |
| 1990's | 80 (32.13) | 18.2507 |
| 2000's | 37 (14.86) | 29.6817 |
| 2010's | 12 (4.82) | 24.3611 |
| 2020's | 2 (0.80) | 2.80 |
| Authors | Studies |
|---|---|
| Eriks, JC; Sterk, GJ; Timmerman, H; van der Goot, H | 1 |
| Timmerman, H | 1 |
| Chou, YL; Erhardt, PW; Greenberg, SS; Hanna, RG; Ingebretsen, WR; Lampe, JW; Lumma, WC; Marshall, DC; Piscitelli, TA; Wiggins, J | 1 |
| Blevitt, J; Carruthers, N; Chai, W; Hofstra, CL; Jiang, X; Li, X; Liu, C; Lovenberg, TW; Ma, X; Pyati, J; Wilson, SJ | 1 |
| Alston, J; Ames, RS; Bergsma, DJ; Boyce, R; Davenport, CM; Dytko, GM; Fitzgerald, LR; Herrity, NC; Hieble, JP; Li, X; Mannan, IJ; Michalovich, D; Sarau, HM; Tan, KB; Tierney, LA; Vawter, L; Wilson, S; Wu, H; Zhu, Y | 1 |
| Anthes, JC; Bayne, M; Behan, J; Gonsiorek, W; Greene, J; Greenfeder, SA; Gustafson, EL; Hedrick, JA; Hipkin, RW; Laz, TM; Monsma, FJ; Morse, KL; Qiao, X; Shin, N; Umland, S; Wan, Y; Wang, S; West, RE | 1 |
| Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM | 1 |
| Falus, A; Jelinek, I; Keseru, GM; Kiss, B; Kiss, R; Könczöl, A; László, V; Noszál, B; Szalai, F | 1 |
| Buschauer, A; Dove, S; Igel, P | 1 |
| Beaven, MA; Shaff, RE | 1 |
| Aksulu, HE; Ercan, ZS; Türker, RK | 1 |
| Bull, HA; Courtney, PF; Dowd, PM; Rustin, MH | 1 |
| Buschauer, A; Höer, A; Schwaner, I; Seifert, R | 1 |
| Donné-Op den Kelder, GM; Haaksma, EE; Timmerman, H; Vernooijs, P | 1 |
| Barker, LA; Petropoulos, AC; Winbery, SL | 1 |
| Brink, C; Gorenne, I; Labat, C; Norel, X; Ortiz, JL; Verley, J | 1 |
| Maeyama, K; Ohkawara, Y; Ohrui, T; Sasaki, H; Sasaki, M; Sekizawa, K; Takemura, M; Wada, H; Watanabe, T; Yamauchi, K | 1 |
| Bast, A; Brozius, MM; Leurs, R; Smit, MJ; Timmerman, H | 1 |
| Donné- op den Kelder, GM; Haaksma, EE; Timmerman, H; Weinstein, H | 1 |
| Hannibal, T; Jørgensen, H; Knigge, U; Matzen, S; Warberg, J | 1 |
| Nowak, JZ; Sek, B | 2 |
| Krielaart, MJ; van Buuren, KJ; Veenstra, DM | 1 |
| Benedito, S; Nyborg, NC; Prieto, D | 1 |
| Benedito, S; Nielsen, PJ; Nyborg, NC; Prieto, D | 1 |
| Bermejo, E; Egozcue, J; Gimeno, M; Lazzari, MA; Maugeri, N; Serpente, N | 1 |
| Matsumoto, M; Nishio, A; Obi, T | 1 |
| Chediak, AD; Csete, ME; Elsasser, S; Gazeroglu, H; Wanner, A | 1 |
| Mutafova-Yambolieva, V; Staneva-Stoytcheva, D; Todorov, S; Vassilev, P | 1 |
| Dy, M; Piquet-Pellorce, C; Schneider, E | 2 |
| Chiba, S; Tsukada, M | 2 |
| Campillo, M; Giraldo, J; Martín, M; Pardo, L | 1 |
| Dolata, J; Lindberg, S; Mercke, U | 1 |
| Amerini, S; Cerbai, E; Mugelli, A | 1 |
| Gerges, E; Gertner, SB | 1 |
| Almeida, L; Figueiredo, A; Gonçalo, M; Poiares-Baptista, A; Ribeiro, CA; Teixeira, F | 1 |
| Cooke, HJ; Wang, YZ | 2 |
| Młynarska, MS | 1 |
| Matsuki, T; Ohhashi, T | 1 |
| Asea, A; Hellstrand, K; Hermodsson, S | 1 |
| Clark, MA; Egan, RW; Shih, NY; Siegel, MI; West, RE; Zweig, A | 1 |
| Borchard, U; Hafner, D; Hirth, C | 1 |
| Borchard, U; Hafner, D | 1 |
| Donné-Op den Kelder, GM; Haaksma, EE; Ravenek, W; Timmerman, H; Vernooijs, P | 1 |
| Hashimoto, K; Motomura, S | 1 |
| Bugajski, J; Gadek-Michalska, A | 1 |
| Cortijo, J; Esplugues, J; Morcillo, EJ; Orón, JD; Ortiz, JL; Perpiñá, M; Sanz, C | 1 |
| Bueno, L; Fargeas, MJ; Fioramonti, J | 1 |
| Abboud, HE; Sedor, JR | 1 |
| Gannon, MN; Hough, LB | 1 |
| Girard, A; Marche, P | 1 |
| Batzri, S; Thompson, WF; Toles, R | 1 |
| Bertaccini, G; Coruzzi, G; Poli, E | 1 |
| Mieda, M; Sakuma, H; Shiratsuchi, K; Tarutani, M | 1 |
| Rising, TJ; Steward, A | 1 |
| Sterk, GJ; Timmerman, H; van der Goot, H | 1 |
| Hutchison, VH; Spriestersbach, KK | 1 |
| Knigge, U; Matzen, S; Warberg, J | 2 |
| Coruzzi, G; Noci, MT | 1 |
| Boucher, M; Duchene-Marullaz, P; Li, JH | 1 |
| Blandina, P; Brunelleschi, S; Fantozzi, R; Giannella, E; Mannaioni, PF; Masini, E | 1 |
| Bertaccini, G; Coruzzi, G | 1 |
| Salonen, RO; Webber, SE; Widdicombe, JG | 1 |
| Akahori, H; Kamei, C; Kitazumi, K; Tasaka, K | 1 |
| Ledgard, SE; Nieves, AL; Woodward, DF | 1 |
| Beaudoin, J; Beaulieu, L; Hébert, J; Jobin, M | 1 |
| Barker, LA; Winbery, SL | 1 |
| Donaldson, J; Hill, SJ | 1 |
| Bordi, F; Chiavarini, M; Impicciatore, M; Morini, G; Plazzi, PV; Vitali, F | 2 |
| Adami, M; Bertaccini, G; Coruzzi, G | 1 |
| Fan, HX; Wen, R | 1 |
| Kim, LE; Oudart, N; Sercombe, R; Teste, JF | 1 |
| Gertner, SB; Poulakos, JJ | 1 |
| Holstein, B | 1 |
| Granata, AR; Reis, DJ | 1 |
| Hayashi, S; Miichi, H; Tanaka, H; Umemoto, M | 1 |
| Jouvet, M; Lin, JS; Sakai, K | 1 |
| Chiba, S; Nakane, T | 1 |
| Nishiwaki, H; Okabe, S; Okada, M; Takeuchi, K | 1 |
| Knigge, U; Matzen, S; Sleimann, I; Warberg, J | 1 |
| Fromm, D; Furukawa, T; Olender, EJ; Woods, DJ | 1 |
| Altman, CB; Bassett, AL; Cameron, JS; Cuevas, J; Gaide, MS; Goad, PL; Myerburg, RJ | 1 |
| Faanes, R; French, S; Susskind, B; Walker, M | 1 |
| Leff, P; Trist, DG | 1 |
| Batzri, S | 1 |
| Kume, S; Ohashi, T; Ozaki, Y | 1 |
| Gerber, JG; Nies, AS | 2 |
| Gristwood, RW; Lincoln, JC; Owen, DA | 1 |
| Daniel, D; Owen, DA; Poy, E; Woodward, DF | 1 |
| Askenase, PW; Gershon, RK; Schwartz, A | 1 |
| Cho, CH; Pfeiffer, CJ | 1 |
| Fondacaro, JD; Jacobson, ED; Walus, KM | 1 |
| Eyre, P; Norris, AA | 1 |
| Colboc, O; Costentin, J; Protais, P | 1 |
| Oriowo, MA | 1 |
| Ooi, YM | 1 |
| Clineschmidt, BV; Cook, PG; Hanson, CA; Pendleton, RG; Torchiana, ML | 1 |
| Birkett, DH; La Morte, WW; Schoetz, DJ; Williams, LF; Wise, WE | 1 |
| Fletcher, MP; Gallin, JI; Seligmann, BE | 1 |
| Heldsinger, AA; Skoglund, ML; Vinik, AI | 1 |
| Donoso, AO; Zárate, MB | 1 |
| Guldvog, I; Linnestad, P; Schrumpf, E | 1 |
| Nemeth, PR; Ort, CA; Wood, JD | 1 |
| Tsai, BS; Yellin, TO | 1 |
| Burtin, C; Lebel, B; Soubrane, C | 1 |
| Bielkiewicz, B; Kordecka, A; Lebrecht, U; Maslinski, C; Nowak, JZ | 1 |
| Rothschild, AM | 1 |
| Johnson, CL; Kalinyak, K; Sawutz, DG; Whitsett, JA | 1 |
| Birkett, DH; Gaca, JM; LaMorte, WW; Schoetz, DJ; Williams, LF; Wise, WE | 1 |
| Christiansen, VJ; Horst, MA; Robinson, CP | 1 |
| Eyre, P; Mirbahar, KB | 1 |
| Ganellin, CR; Martin, D; Milliner, K; Vickers, MR | 1 |
| Sykes, KJ; Vickers, MR | 1 |
| Horowitz, GP; Isaacson, RL; O'Callaghan, M | 1 |
| Badger, AM; Poste, G; Young, J | 1 |
| Bertaccini, G; Bezzi, E; Potenzoni, D; Zappia, L | 1 |
| Salvati, P; Whittle, BJ | 1 |
| Bugajski, J; Gadek, A | 1 |
| Bugajski, J; Janusz, Z | 1 |
| Brooks, HL; Christensen, CW; Gross, GJ; Hardman, HF; Warltier, DC | 1 |
| Owen, DA; Pipkin, MA; Woodward, DF | 1 |
| Clark, KE; Harrington, DJ; Mills, EG | 1 |
| Jespersen, LT; Mikkelsen, E; Sakr, AM | 1 |
| Cooke, HJ; Nemeth, PR; Wood, JD | 1 |
| Christiansen, VJ; Horst, MA; Robinson, C | 1 |
| Dale, MM; Ladd, R | 1 |
| Horst, MA; Robinson, CP | 1 |
| Cheret, AM; Lewin, MJ; Mangeat, P; Marchis-Mouren, G | 1 |
| Brown, EM | 1 |
| Baumann, G; Blömer, H; Erhardt, WD; Felix, SB; Heidecke, CD; Loher, U; Ludwig, L; Riess, G; Schrader, J; Sebening, F | 1 |
| Nishibori, M | 1 |
| Daly, MJ; Humphray, JM; Stables, R | 1 |
| Batzri, S; Harmon, JW; Thompson, WF | 1 |
| Eckel, L; Gristwood, RW; Nawrath, H; Owen, DA; Satter, P | 1 |
| Bonnet, M; Burtin, C; Lespinats, G | 1 |
| Del Soldato, P | 1 |
| Hughes, MJ | 1 |
| Birkett, DH; Gaca, JM; LaMorte, WW; Williams, LF; Wise, WE | 1 |
| Anderson, C; Busse, WW; Cooper, W | 1 |
| Eriksson, L; Tuomisto, L | 1 |
| Davies, MG; Greaves, MW | 1 |
| Gertner, SB; Klein, MC | 1 |
| Hingston, SJ; La Morte, WW; Wise, WE | 1 |
| Harvey, CA; Owen, DA; Quinn, EH | 1 |
| Philippu, A; Wiedemann, K | 2 |
| Pang, PK; Tenner, TE; Yang, MC | 1 |
| Bielkiewicz, B; Nowak, JZ | 1 |
| Tenner, TE | 1 |
| Di Donato, M; Mantovani, P; Santicioli, P | 1 |
| Nunoki, K; Shimizu, T; Taira, N | 1 |
| Gross, PM; Harper, AM; Teasdale, GM | 1 |
| Baker, AP; Chakrin, LW; Holden, DA; Smith, WJ; Sung, CP | 1 |
| Brink, C; Douglas, JS; Duncan, PG | 1 |
| Kawai, Y; Ohhashi, T | 1 |
| Bochner, BS; Galli, SJ; Guo, CB; Kagey-Sobotka, A; Lichtenstein, LM; Liu, MC | 1 |
| Kohno, S; Nabe, T; Nakao, S; Ogawa, K; Ohata, K; Yamamura, H | 1 |
| Bynum, TE; Kronauge, JF; Morales, RE; Palitzsch, KD; Szabo, S | 1 |
| Bast, A; Leurs, R; Shukrula, SR; Smit, MJ; Timmerman, H | 1 |
| Carson, CC; Davies, MG; Hagen, PO; Kim, YC; Lee, TH | 1 |
| Elezoglou, V; Kokolis, N; Kounenis, G; Koutsoviti-Papadopoulou, M | 1 |
| Iinuma, K; Onodera, K; Watanabe, T; Yokoyama, H | 1 |
| Fujimoto, M; Kimata, H | 1 |
| Katayose, D; Nakazawa, H; Ohkawara, Y; Ohtsu, H; Sekizawa, K; Shibahara, S; Suzuki, H; Takemura, M; Tamura, G; Yamauchi, K | 1 |
| Prior, T; Rangachari, PK | 1 |
| Borycz, J; Bugajski, J; Gadek-Michalska, A | 2 |
| Fechner, GA; Jacobs, JJ; Parsons, PG | 1 |
| Braga, PC; Guidobono, F; Netti, C; Pecile, A; Sibilia, V; Villani, P | 1 |
| Chiba, S; Fujiwara, T | 1 |
| Sasaki, T; Satoh, M; Shimura, S; Takishima, T; Yamada, K; Yamauchi, K | 1 |
| Sako, J; Yasuda, Y | 1 |
| Bertaccini, G; Coruzzi, G; Poli, E; Pozzoli, C; Timmerman, H | 1 |
| Maeyama, K; Morikawa, M; Nakazawa, H; Sasaki, H; Satoh, M; Sekizawa, K; Watanabe, T; Yamauchi, K | 1 |
| Honda, K; Ito, H; Kamato, T; Miyata, K; Nishida, A; Takeda, M; Yuki, H | 1 |
| Maeyama, K; Nakazawa, H; Ohkawara, Y; Ohrui, T; Sasaki, H; Sekizawa, K; Takishima, T; Watanabe, T; Yamauchi, K | 1 |
| Maeyama, K; Morikawa, M; Nakazawa, H; Sasaki, H; Sekizawa, K; Watanabe, T; Yamauchi, K | 1 |
| Davison, JS; Jennings, LJ; Lea, RW; Pozo, MJ; Salido, GM; Sharkey, KA; Singh, J | 1 |
| Blandina, P; Cecchi, M; Giorgetti, M; Giovannini, MG; Leurs, R; Timmerman, H | 1 |
| Benvenuti, S; Brandi, ML; Frediani, U; Masi, L; Tanini, AL | 1 |
| Chiyotani, A; Konno, K; Nakata, J; Takeyama, K; Tamaoki, J | 1 |
| Bello, MG; Di Bello, MG; Mannaioni, PF; Masini, E; Schunack, W | 1 |
| Kitazawa, T; Sato, T; Shishido, H; Taneike, T | 1 |
| Baldi, A; Brodsky, A; Davio, C; Legnazzi, BL; Mladovan, AG; Rivera, E; Shayo, C | 1 |
| Irokawa, T; Nagaki, M; Sasaki, T; Shimura, S; Shirato, K; Yamauchi, K; Yamaya, M | 1 |
| Fu, LW; Longhurst, JC; Pan, HL | 1 |
| Easton, AS; Fraser, PA; Sarker, MH | 1 |
| Moody, MW; Nguyen, TD; Okolo, CN | 1 |
| Nakano, K; Takamatsu, S | 1 |
| Chrousos, GP; Elenkov, IJ; Fleisher, TA; Papanicolaou, DA; Webster, E; Wilder, RL | 1 |
| Grundy, D; Haupt, W; Kirkup, AJ; Kreis, ME | 1 |
| Akaike, N; Ishibashi, H; Munakata, M; Sakata, T; Takeshita, Y; Watanabe, T | 1 |
| Coupar, IM; Hemedah, M; Mitchelson, FJ | 1 |
| Capasso, F; Costa, M; Izzo, AA; Mascolo, N | 1 |
| Philippu, A; Prast, H; Tran, MH | 1 |
| Arebi, N; Bliss, PW; Calam, J; Healey, ZV | 1 |
| Chen, Z; Fujii, Y; Kamei, C; Sugimoto, Y; Suzuki, G | 1 |
| Arai, M; Chiba, S | 1 |
| Gao, C; Hu, Hz; Liu, S; Ren, J; Wood, JD; Xia, Y | 1 |
| Starodub, AM; Wood, JD | 1 |
| Firth, TA; Guarraci, FA; Hemming, JM; Jennings, LJ; Mawe, GM; Nelson, MT | 1 |
| Attarzadeh, M; Farzin, D | 1 |
| Ezeamuzie, CI; Philips, E | 1 |
| Annunziato, L; Gentile, M; Granata, F; Marone, G; Oriente, A; Secondo, A; Taglialatela, M; Triggiani, M | 1 |
| Kitanaka, J; Kitanaka, N; Takemura, M; Terada, N; Tsujimura, T | 2 |
| Azuma, Y; Hidaka, A; Ohura, K; Shinohara, M; Wang, PL | 1 |
| Fraser, PA; Sarker, MH | 1 |
| Ghosh, AK; Hirasawa, N; Ohtsu, H; Ohuchi, K; Watanabe, T | 1 |
| Brandão, ML; Husto, JP; Santos, NR | 1 |
| Fox, JL; von der Weid, PY | 1 |
| Bacon, KB; Center, DM; Cruikshank, WW; Gantner, F; Sakai, K; Tusche, MW | 1 |
| Li, HZ; Shen, B; Wang, JJ | 1 |
| Jochem, J | 1 |
| Gil Marqués, M; Martínez-Mir, I; Morales-Olivas, FJ; Rubio-Gomis, E | 1 |
| Esbenshade, TA; Hancock, AA; Kang, CH; Krueger, KM; Masters, JN; Miller, TR; Roch, JM; Witte, DG | 1 |
| Brandão, ML; Huston, JP; Santos, NR | 1 |
| Nakamura, T; Ueno, K; Yamaura, K; Yano, S; Yonekawa, T | 1 |
| Akagi, T; Iwagaki, H; Kubo, S; Mori, S; Morichika, T; Nishibori, M; Takahashi, HK; Tamura, R; Tanaka, N; Yoshino, T | 1 |
| Bello, MG; Mannaioni, PF; Marzocca, C; Masini, E; Pierpaoli, S; Schunack, W | 1 |
| Kuramasu, A; Mobarakeh, JI; Nunoki, K; Sukegawa, J; Suzuki, H; Watanabe, H; Watanabe, T; Yanagisawa, T; Yanai, K | 1 |
| Akagi, M; Fukuishi, N; Imajo, N; Matsui, N; Matsui, S; Yasui, Y | 1 |
| Blanks, AM; Lee, K; Renaud, LP; Spanswick, D; Whyment, AD | 1 |
| Dube, PH; Handley, SA; Miller, VL | 1 |
| Adachi, N; Arai, T; Liu, K; Motoki, A; Nishibori, M | 1 |
| Kitanaka, J; Kitanaka, N; Morita, Y; Takemura, M; Tatsuta, T | 1 |
| Bastaki, SM; Chandranath, IS; Singh, J | 1 |
| Adachi, N; Arai, T; Liu, K; Motoki, A; Nagaro, T; Nishibori, M; Takahashi, HK; Yorozuya, T | 1 |
| Cheng, YS; Huang, CC; Huang, CW; Yu, J | 1 |
| Alhaj, M; Bozarov, A; Christofi, FL; Cooke, HJ; Grants, I; Hassanain, HH; Ren, T; Wang, YZ; Wunderlich, J; Yu, JG | 1 |
| Ambrose, RE; Dankoski, EC; Hashemi, P; Wightman, RM; Wood, KM | 1 |
| Li, B; Ma, SH; Peng, YP; Qin, YT; Qiu, YH; Wang, JJ; Zhuang, QX | 1 |
| Behrens, CJ; Caliskan, G; Fano, S; Heinemann, U | 1 |
| Chan, YS; Han, XH; Wang, JJ; Wu, GY; Yung, WH; Zhang, J; Zhu, JN; Zhuang, QX | 1 |
| Sanchez-Alavez, M; Sethi, J; Tabarean, IV | 1 |
| Wang, JJ; Wu, GY; Wu, YH; Zhu, JN; Zhuang, QX | 1 |
| Benetti, F; Izquierdo, I | 1 |
| Ciz, M; Jancinova, V; Lojek, A; Nosal, R; Vasicek, O | 1 |
| Benetti, F; da Silveira, CK; Izquierdo, I; Rosa, J | 1 |
| Korosteleva, AS; Potapieva, NN; Shteinikov, VY; Tikhonov, DB; Tikhonova, TB | 1 |
| Chen, Z; Ji, MJ; Peng, XC; Wang, JJ; Yu, L; Zhang, XY; Zhang, YX; Zhu, JN | 1 |
| Gergs, U; Griethe, K; Kirchhefer, U; Mißlinger, N; Neumann, J; Weisgut, J | 1 |
| Awane, H; Ezaki, M; Hishinuma, S; Inazuki, N; Michinaga, S; Mizuguchi, H; Shimizu, K; Sonoda, K | 1 |
1 review(s) available for dimaprit and histamine
| Article | Year |
|---|---|
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship | 1990 |
1 trial(s) available for dimaprit and histamine
| Article | Year |
|---|---|
Sensory responses of human skin to synthetic histamine analogues and histamine.
Topics: Adult; Chlorpheniramine; Dimaprit; Female; Histamine; Humans; Male; Methylhistamines; Pruritus; Receptors, Histamine H1; Receptors, Histamine H2; Skin; Thiourea | 1980 |
247 other study(ies) available for dimaprit and histamine
| Article | Year |
|---|---|
Histamine H2-receptor agonists. Synthesis, in vitro pharmacology, and qualitative structure-activity relationships of substituted 4- and 5-(2-aminoethyl)thiazoles.
Topics: Animals; Atrial Function; Chemical Phenomena; Chemistry, Physical; Electrochemistry; Guinea Pigs; Heart Atria; Histamine; Ileum; Molecular Structure; Muscle Contraction; Receptors, Histamine H2; Structure-Activity Relationship; Thiazoles | 1992 |
Cardiotonic agents. 6. Histamine analogues as potential cardiovascular selective H2 agonists.
Topics: Animals; Cardiotonic Agents; Drug Design; Ferrets; Gastric Acid; Guinea Pigs; Heart Rate; Histamine; In Vitro Techniques; Male; Muscle Contraction; Myocardial Contraction; Rats; Receptors, Histamine H2 | 1990 |
Cloning and pharmacological characterization of a fourth histamine receptor (H(4)) expressed in bone marrow.
Topics: Adenylyl Cyclases; Amino Acid Sequence; Bone Marrow; Cloning, Molecular; Histamine; Humans; Methylhistamines; Molecular Sequence Data; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; RNA, Messenger; Sequence Homology, Amino Acid; Tissue Distribution; Tritium | 2001 |
Cloning, expression, and pharmacological characterization of a novel human histamine receptor.
Topics: Amino Acid Sequence; Animals; Calcium; Cloning, Molecular; Dose-Response Relationship, Drug; Gene Expression; Genes, Reporter; Histamine; Humans; Luciferases; Mice; Molecular Sequence Data; Radioligand Assay; Receptors, Histamine; Receptors, Histamine H3; Sequence Homology, Amino Acid; Tissue Distribution; Tritium | 2001 |
Cloning and characterization of a novel human histamine receptor.
Topics: Amino Acid Sequence; Cells, Cultured; Cloning, Molecular; Histamine; Histamine Agonists; Humans; Imidazoles; Molecular Sequence Data; Radioligand Assay; Receptors, Histamine; Receptors, Histamine H3; RNA, Messenger; Sequence Homology, Amino Acid; Thiourea; Tissue Distribution; Transfection | 2001 |
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4 | 2005 |
Discovery of novel human histamine H4 receptor ligands by large-scale structure-based virtual screening.
Topics: Binding, Competitive; Cell Line, Tumor; Databases, Factual; Histamine Antagonists; Humans; Ligands; Models, Molecular; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Structure-Activity Relationship | 2008 |
Histamine H4 receptor agonists.
Topics: Animals; Benzimidazoles; Binding Sites; Clozapine; Guanidines; Humans; Ligands; Mice; Oximes; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Structure-Activity Relationship | 2010 |
Inhibition of histamine methylation in vivo by the dimaprit analog, SKF Compound 91488.
Topics: Amine Oxidase (Copper-Containing); Animals; Brain; Dimaprit; Guanidines; Histamine; Histamine N-Methyltransferase; Kidney; Male; Methylation; Methyltransferases; Mice; Rats; Thiourea | 1979 |
A comparative study with impromidine (SKF 92676), a potent agonist for histamine H2-receptors.
Topics: Airway Resistance; Animals; Blood Pressure; Cats; Dimaprit; Diuresis; Drug Interactions; Female; Guanidines; Guinea Pigs; Histamine; Imidazoles; Impromidine; In Vitro Techniques; Kidney; Lung; Male; Metiamide; Rabbits; Receptors, Histamine; Receptors, Histamine H2; Tachyphylaxis; Thiourea; Trachea | 1979 |
Characterization of histamine receptor sub-types regulating prostacyclin release from human endothelial cells.
Topics: Cells, Cultured; Dimaprit; Endothelium, Vascular; Epoprostenol; Histamine; Histamine Agonists; Humans; Impromidine; Methylhistamines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Thiazoles; Umbilical Veins | 1992 |
Histamine increases cytosolic Ca2+ in HL-60 promyelocytes predominantly via H2 receptors with an unique agonist/antagonist profile and induces functional differentiation.
Topics: Adenosine Triphosphate; Calcium; Cations; Cell Differentiation; Cyclic AMP; Cytosol; Dimaprit; Famotidine; Guanidines; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Impromidine; Ion Channels; Leukemia, Experimental; Leukemia, Promyelocytic, Acute; Phosphatidylinositols; Receptors, Histamine H2; Stimulation, Chemical; Thiourea; Tumor Cells, Cultured | 1992 |
A theoretical study concerning the mode of interaction of the histamine H2-agonist dimaprit.
Topics: Computer Simulation; Dimaprit; Electrophysiology; Histamine; Methylation; Models, Molecular; Molecular Conformation; Receptors, Histamine H2; Thiourea | 1992 |
Effect of short-term treatment with gastrin and related peptides on gastrointestinal histamine H2-receptors.
Topics: Adenylyl Cyclases; Animals; Cimetidine; Digestive System; Dimaprit; Gastrins; Guinea Pigs; Histamine; In Vitro Techniques; Male; Pentagastrin; Receptors, Histamine H2; Sincalide; Thiourea | 1992 |
Histamine receptors on human isolated pulmonary arterial muscle preparations: effects of endothelial cell removal and nitric oxide inhibitors.
Topics: Arginine; Burimamide; Chlorpheniramine; Cimetidine; Dimaprit; Endothelium, Vascular; Histamine; Humans; In Vitro Techniques; Indomethacin; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Nitroarginine; omega-N-Methylarginine; Pulmonary Artery; Receptors, Histamine; Serotonin; Tetraethylammonium; Tetraethylammonium Compounds; Thiourea | 1992 |
Histamine N-methyltransferase controls the contractile response of guinea pig trachea to histamine.
Topics: Animals; Dimaprit; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; Histamine; Histamine N-Methyltransferase; Male; Muscle Contraction; Muscle, Smooth; Thiourea; Trachea | 1992 |
Effects of histamine H1-, H2- and H3-receptor selective drugs on the mechanical activity of guinea-pig small and large intestine.
Topics: Animals; Atropine; Dimaprit; Electric Stimulation; Guanidines; Guinea Pigs; Histamine; In Vitro Techniques; Intestine, Large; Intestine, Small; Male; Methacholine Compounds; Muscle Contraction; Muscle, Smooth; Pinacidil; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Stereoisomerism; Tetraethylammonium Compounds; Thiourea | 1991 |
Theoretical analysis of the activity of dimaprit derivatives on the H2-receptor.
Topics: Chemical Phenomena; Chemistry, Physical; Dimaprit; Electrochemistry; Histamine; Models, Molecular; Protons; Receptors, Histamine H2; Software; Thermodynamics; Thiourea | 1991 |
Involvement of histamine in the mediation of the stress-induced release of alpha-melanocyte-stimulating hormone in male rats.
Topics: Adrenocorticotropic Hormone; alpha-MSH; Animals; Bromocriptine; Dimaprit; Histamine; Male; Methylhistidines; Propranolol; Rats; Rats, Inbred Strains; Stress, Physiological; Thiourea | 1991 |
Cyclic AMP generating systems in vertebrate retina: effects of histamine and an established retinal modulator, dopamine.
Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Chickens; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dopamine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Retina; Thiazoles; Thiourea | 1991 |
Mechanism of action of H2-antagonists on histamine- or dimaprit-stimulated H2-receptors of spontaneously beating guinea-pig atrium.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cimetidine; Dimaprit; Famotidine; Female; Guinea Pigs; Heart; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Radioligand Assay; Ranitidine; Receptors, Histamine H2; Thiourea | 1990 |
Influence of the endothelium on histamine-induced relaxation of rat middle cerebral arteries in vitro.
Topics: Animals; Cerebral Arteries; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Histamine; Histamine H2 Antagonists; Kinetics; Male; Methylhistamines; Muscle Relaxation; Muscle, Smooth, Vascular; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H2; Receptors, Histamine H3; Thiourea | 1991 |
Histamine induces endothelium-dependent relaxation of bovine retinal arteries.
Topics: Acetylcholine; Animals; Cattle; Cimetidine; Dimaprit; Endothelium, Vascular; Histamine; Muscle Relaxation; Pyridines; Pyrilamine; Receptors, Histamine; Retinal Artery; Tachyphylaxis; Thiourea | 1991 |
Effect of histamine on human lymphocyte aggregation.
Topics: Adult; Arachidonic Acid; Arachidonic Acids; Cell Aggregation; Dimaprit; Endothelium, Vascular; Histamine; Humans; In Vitro Techniques; Receptors, Histamine; T-Lymphocytes; Thiourea | 1991 |
Vasomotor effect of histamine on pig and cattle coronary artery in vitro.
Topics: Animals; Cattle; Cimetidine; Coronary Vessels; Dimaprit; Diphenhydramine; Endothelium, Vascular; Histamine; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Swine; Thiourea | 1991 |
Effect of histamine on tracheal mucosal perfusion, water content and airway smooth muscle in sheep.
Topics: Animals; Atropine; Chlorpheniramine; Dimaprit; Female; Histamine; Lung Volume Measurements; Metiamide; Mucous Membrane; Muscle, Smooth; Receptors, Cholinergic; Receptors, Histamine H1; Receptors, Histamine H2; Regional Blood Flow; Sheep; Thiourea; Trachea; Water | 1991 |
Involvement of calcium ions in the modulation of electrically-induced rat vas deferens contractions by histaminergic drugs.
Topics: Animals; Calcium; Cimetidine; Dimaprit; Diphenhydramine; Electric Stimulation; Histamine; In Vitro Techniques; Male; Muscle Contraction; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea; Vas Deferens; Verapamil | 1991 |
GM-CSF in association with IL-1 triggers day-8 CFU-S into cell cycle: role of histamine.
Topics: Animals; Bone Marrow Cells; Cell Cycle; Cells, Cultured; Dimaprit; Female; Granulocyte-Macrophage Colony-Stimulating Factor; Hematopoietic Stem Cells; Histamine; Interleukin-1; Male; Mice; Mice, Inbred C57BL; S Phase; Spleen; Thiourea | 1991 |
Histamine-induced vasodilations mediated by H1- and H2-receptors in isolated rat common carotid arteries.
Topics: Acetylcholine; Animals; Carotid Arteries; Cimetidine; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Female; Histamine; In Vitro Techniques; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Saponins; Thiourea; Vasodilation | 1991 |
Theoretical studies on the histamine H2 receptor: construction of a receptor model based on the structural properties of dimaprit and N alpha-guanylhistamine.
Topics: Computer Simulation; Dimaprit; Histamine; Kinetics; Models, Chemical; Models, Molecular; Receptors, Histamine H2; Thiourea | 1991 |
New role for histamine in interleukin-3-induced proliferation of hematopoietic stem cells.
Topics: Animals; Bone Marrow Cells; Cell Division; Cetirizine; Colony-Forming Units Assay; Dimaprit; Hematopoiesis; Hematopoietic Stem Cells; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Hydroxyzine; Imidazoles; In Vitro Techniques; Interleukin-3; Methylhistidines; Mice; Mice, Inbred C57BL; Thiourea | 1990 |
Histamine stimulation of mucociliary activity in the rabbit maxillary sinus.
Topics: Animals; Atropine; Cilia; Cimetidine; Dimaprit; Female; Histamine; Histamine H2 Antagonists; Male; Maxillary Sinus; Mucociliary Clearance; Pyrilamine; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Muscarinic; Thiourea | 1990 |
Histamine and abnormal automaticity in barium- and strophanthidin-treated sheep Purkinje fibers.
Topics: Animals; Barium; Dimaprit; Electrophysiology; Heart; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Membrane Potentials; Methylhistamines; Purkinje Fibers; Sheep; Strophanthidin; Thiourea | 1990 |
Central cardiovascular responses of histamine and homodimaprit in normal and hypophysectomized rats.
Topics: Animals; Blood Pressure; Brain; Dimaprit; Hexamethonium; Hexamethonium Compounds; Histamine; Hypophysectomy; Kinetics; Male; Rats; Rats, Inbred Strains; Thiourea; Vasopressins | 1990 |
Mechanism of action of doxepin in the treatment of chronic urticaria.
Topics: Adult; Aged; Animals; Atropine; Carbachol; Chronic Disease; Dimaprit; Doxepin; Female; Gastric Juice; Guinea Pigs; Heart; Histamine; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Pylorus; Pyrilamine; Rats; Thiourea; Urticaria | 1990 |
H2 receptors mediate cyclical chloride secretion in guinea pig distal colon.
Topics: Animals; Bumetanide; Chlorides; Cimetidine; Colon; Dimaprit; Guinea Pigs; Histamine; In Vitro Techniques; Intestinal Mucosa; Kinetics; Male; Muscle, Smooth; Pyrilamine; Receptors, Histamine H2; Tetrodotoxin; Thiourea | 1990 |
Antagonistic effect of naloxone on the hypertensive response of intraventricularly administered histamine.
Topics: Animals; Blood Pressure; Cimetidine; Dimaprit; Hemodynamics; Histamine; In Vitro Techniques; Injections, Intraventricular; Male; Naloxone; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Thiourea | 1990 |
Endothelium and mechanical responses of isolated monkey pulmonary veins to histamine.
Topics: Animals; Dimaprit; Endothelium, Vascular; Famotidine; Hemoglobins; Histamine; In Vitro Techniques; Macaca; Methylene Blue; Pulmonary Veins; Pyridines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Vasoconstriction; Vasodilation | 1990 |
Role of histamine in natural killer cell-mediated resistance against tumor cells.
Topics: Animals; Cytotoxicity, Immunologic; Dimaprit; Histamine; Immunity, Cellular; Interleukin-2; Killer Cells, Natural; Lung Neoplasms; Melanoma, Experimental; Mice; Mice, Inbred Strains; Neoplasm Metastasis; Neoplasms, Experimental; Ranitidine; Receptors, Histamine H2; Thiourea | 1990 |
Identification of two H3-histamine receptor subtypes.
Topics: Animals; Binding Sites; Binding, Competitive; Brain Chemistry; Burimamide; Dimaprit; Guanidines; Guanosine 5'-O-(3-Thiotriphosphate); Histamine; Imidazoles; Impromidine; Male; Methylhistamines; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H3; Thiourea; Tritium | 1990 |
Electrophysiological actions of histamine and H1-, H2-receptor antagonists in cardiac tissue.
Topics: 1-Methyl-3-isobutylxanthine; Action Potentials; Animals; Atrioventricular Node; Dimaprit; Guinea Pigs; Heart; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Male; Rabbits; Thiourea | 1986 |
Electrophysiological characterization of histamine receptor subtypes in mammalian heart preparations.
Topics: 1-Methyl-3-isobutylxanthine; Action Potentials; Animals; Atrioventricular Node; Cimetidine; Dimaprit; Dimethindene; Guinea Pigs; Heart; Histamine; Histamine H1 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Male; Myocardial Contraction; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1986 |
Comparison of the interaction of the histamine H2-agonists [correction of H2-antagonists] histamine and dimaprit.
Topics: Computer Simulation; Dimaprit; Electrochemistry; Histamine; Models, Molecular; Molecular Conformation; Receptors, Histamine H2; Thiourea | 1989 |
Histamine H2-receptor mediated positive dromotropic effect in the canine atrioventricular node.
Topics: Animals; Atenolol; Atrioventricular Node; Cimetidine; Dimaprit; Diphenhydramine; Dogs; Female; Heart Conduction System; Histamine; Male; Norepinephrine; Receptors, Histamine H2; Stimulation, Chemical; Thiourea | 1989 |
Antagonistic action of naloxone on central histamine receptors-stimulated corticosterone secretion in rats under stress.
Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Histamine; Male; Methylhistamines; Naloxone; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Restraint, Physical; Stress, Physiological; Thiourea | 1989 |
Responses to histamine and selective H2-receptor agonists in lung parenchymal strips from normal and sensitized guinea-pigs.
Topics: Animals; Benzimidazoles; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; Histamine; Imidazoles; Impromidine; Isoproterenol; Lung; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; Receptors, Histamine H2; Thiourea | 1989 |
Involvement of different receptors in the central and peripheral effects of histamine on intestinal motility in the rat.
Topics: Animals; Chlorpheniramine; Dimaprit; Gastrointestinal Motility; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Injections, Intraperitoneal; Injections, Intraventricular; Male; Methylhistamines; Rats; Rats, Inbred Strains; Receptors, Histamine; Thiourea | 1989 |
Histamine modulates contraction and cyclic nucleotides in cultured rat mesangial cells. Differential effects mediated by histamine H1 and H2 receptors.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Cell Movement; Cells, Cultured; Cyclic AMP; Cyclic GMP; Dimaprit; Glomerular Mesangium; Histamine; Kidney Glomerulus; Male; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1985 |
Histamine receptors coupled to [3H]cAMP accumulation in brain: pharmacological characterization in a vesicular preparation of guinea pig cortex.
Topics: Adenosine Deaminase; Animals; Cerebral Cortex; Chlorpheniramine; Cimetidine; Cyclic AMP; Dimaprit; Egtazic Acid; Guinea Pigs; Histamine; In Vitro Techniques; Receptors, Histamine; Subcellular Fractions; Thiourea | 1988 |
Phosphoinositides and cicletanine.
Topics: Angiotensin II; Animals; Antihypertensive Agents; Aorta, Thoracic; Cells, Cultured; Dimaprit; Diuretics; Guinea Pigs; Histamine; Male; Muscle, Smooth, Vascular; Phenylephrine; Phosphatidylinositols; Pyridines; Pyrilamine; Thiourea | 1988 |
Distortion of H2-antagonist equilibrium constants by uptake in rabbit gastric mucosal cells.
Topics: Aminopyrine; Animals; Cimetidine; Cyclic AMP; Dimaprit; Gastric Acid; Gastric Mucosa; Guanidines; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Pyrimidinones; Rabbits; Radioisotopes; Rubidium; Thiadiazoles; Thiourea | 1985 |
Histamine H2 receptor antagonists may modify dog intestinal motility independently of their primary action on the H2 receptors.
Topics: Acetylcholine; Animals; Blood Pressure; Ceruletide; Cimetidine; Dimaprit; Dogs; Female; Gastrointestinal Motility; Histamine; Histamine H2 Antagonists; Ileum; Imidazoles; Impromidine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Physalaemin; Ranitidine; Receptors, Histamine; Receptors, Histamine H2; Thiourea | 1985 |
Histamine H2-receptor antagonistic action of N-(3-[3-(1-piperidinylmethyl)phenoxy]propyl)acetoxyacetamide hydrochloride (TZU-0460).
Topics: Animals; Cimetidine; Dimaprit; Dogs; Female; Gastric Acid; Guinea Pigs; Heart Atria; Heart Rate; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Male; Muscle Relaxation; Piperidines; Rats; Thiourea; Uterus | 1985 |
The determination of receptor constants for histamine H2-agonists in the guinea-pig isolated right atrium using an irreversible H2-antagonist.
Topics: Animals; Dimaprit; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; Heart Rate; Histamine; Histamine H2 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Male; Methylhistamines; Receptors, Adrenergic, beta; Receptors, Histamine; Receptors, Histamine H2; Thiazoles; Thiourea | 1986 |
Studies on histaminergic compounds, III. Synthesis and histamine H2-activity of a series of corresponding histamine and dimaprit analogues.
Topics: Animals; Dimaprit; Female; Guinea Pigs; Histamine; Histamine H2 Antagonists; Male; Structure-Activity Relationship; Thiourea | 1986 |
Histamine and histamine receptors: behavioral thermoregulation in the salamander Necturus maculosus.
Topics: Animals; Body Temperature Regulation; Cimetidine; Dimaprit; Histamine; Histidine; Necturus; Pyridines; Pyrilamine; Receptors, Histamine; Thiourea | 1986 |
Histaminergic stimulation of prolactin secretion mediated via H1- or H2-receptors: dependence on routes of administration.
Topics: Animals; Cimetidine; Dimaprit; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Pituitary Gland, Anterior; Prolactin; Pyrilamine; Pyrimidinones; Rats; Receptors, Histamine; Thiazoles; Thiourea | 1986 |
[Effect of a new H2 receptor antagonist, famotidine, on gastric secretion].
Topics: Animals; Cats; Dimaprit; Dose-Response Relationship, Drug; Famotidine; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Ranitidine; Rats; Thiazoles; Thiourea | 1986 |
Chronotropic cardiac effects of histamine in the conscious dog with chronic atrioventricular block: interactions with the autonomic nervous system.
Topics: Adrenergic beta-Antagonists; Animals; Atrioventricular Node; Autonomic Nervous System; Blood Pressure; Dimaprit; Dogs; Drug Interactions; Electrocardiography; Female; Heart Block; Heart Conduction System; Heart Rate; Histamine; Male; Parasympatholytics; Thiourea | 1986 |
The antianaphylactic action of histamine H2-receptor agonists in the guinea-pig isolated heart.
Topics: Anaphylaxis; Animals; Cimetidine; Dimaprit; Female; Guinea Pigs; Heart; Heart Rate; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Male; Myocardial Contraction; Pyridines; Thiourea | 1987 |
Famotidine and ranitidine: any difference in the duration of action?
Topics: Animals; Cats; Dimaprit; Famotidine; Gastric Acid; Gastric Juice; Histamine; Histamine H2 Antagonists; Ranitidine; Rats; Thiazoles; Thiourea; Time Factors | 1987 |
H1- and H2-receptor characterization in the tracheal circulation of sheep.
Topics: Animals; Dimaprit; Female; Histamine; Histamine H2 Antagonists; Male; Muscle Tonus; Receptors, Histamine H2; Regional Blood Flow; Sheep; Thiourea; Trachea; Vagotomy; Vascular Resistance | 1988 |
The effects of histamine and some related compounds on conditioned avoidance response in rats.
Topics: Acetylcholine; Animals; Avoidance Learning; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Hypothalamus; Injections, Intraventricular; Kinetics; Male; Methylhistamines; Pyrilamine; Rats; Rats, Inbred Strains; Scopolamine; Thiazoles; Thiourea | 1985 |
Conjunctival immediate hypersensitivity: re-evaluation of histamine involvement in the vasopermeability response.
Topics: Albumins; Animals; Capillary Permeability; Cimetidine; Conjunctiva; Dimaprit; Dose-Response Relationship, Drug; Drug Combinations; Eyelids; Guinea Pigs; Histamine; Histamine Antagonists; Hypersensitivity, Immediate; Imidazoles; Impromidine; Male; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1986 |
Effects of H1 and H2 receptor agonists on nonspecific proliferative response of human peripheral blood lymphocytes.
Topics: Cimetidine; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Humans; Immunosuppressive Agents; Lymphocyte Activation; Methylhistamines; Phytohemagglutinins; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1986 |
Metronidazole and 5-aminosalicylic acid enhance the contractile activity of histaminergic agonists on the guinea-pig isolated ileum.
Topics: Aminosalicylic Acids; Animals; Cimetidine; Computers; Dimaprit; Dose-Response Relationship, Drug; Drug Synergism; Duodenum; Female; Guinea Pigs; Heart; Histamine; Ileum; In Vitro Techniques; Jejunum; Male; Mesalamine; Metronidazole; Muscle Contraction; Myenteric Plexus; Pyrilamine; Receptors, Histamine; Scopolamine; Tetrodotoxin; Thiourea | 1986 |
Selective enhancement of histamine H1-receptor responses in guinea-pig ileal smooth muscle by 1,4-dithiothreitol.
Topics: Acetylcholine; Animals; Dimaprit; Dithionitrobenzoic Acid; Dithiothreitol; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Thiourea | 1986 |
Pharmacological activities of two new histamine analogs.
Topics: Animals; Cats; Dimaprit; Dose-Response Relationship, Drug; Gastric Acid; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Methylhistamines; Muscle Contraction; Receptors, Histamine H1; Structure-Activity Relationship; Thiourea | 1986 |
Effects of Ca2+ ions on gastric acid secretion by the rat isolated stomach.
Topics: Adenylyl Cyclases; Animals; Calcium; Dimaprit; Dose-Response Relationship, Drug; Gastric Acid; Histamine; In Vitro Techniques; Male; Rats; Receptors, Histamine; Theophylline; Thiourea | 1986 |
[Miosis induced by histamine injected into the anterior chamber of isolated pig eyes].
Topics: Animals; Anterior Chamber; Chlorpheniramine; Cimetidine; Dimaprit; Female; Histamine; In Vitro Techniques; Male; Pupil; Receptors, Histamine H2; Swine; Thiourea | 1986 |
Participation of vascular H1-receptors in histaminergic relaxation of rabbit middle cerebral artery in vitro.
Topics: Animals; Cerebral Arteries; Cimetidine; Dimaprit; Drug Interactions; Histamine; In Vitro Techniques; Methylhistamines; Muscle Relaxation; Muscle, Smooth, Vascular; Phenethylamines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Thiourea | 1986 |
Studies on the desensitization of the central cardiovascular responses of histamine.
Topics: Animals; Blood Pressure; Brain; Cardiovascular System; Dimaprit; Heart Rate; Histamine; Imidazoles; Impromidine; Injections, Intraventricular; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1986 |
Characterization with agonists of the histamine receptors mediating stimulation of gastric acid secretion in the Atlantic cod, Gadus morhua.
Topics: Animals; Cimetidine; Dimaprit; Female; Fishes; Gastric Acid; Histamine; Imidazoles; Impromidine; Male; Methylhistamines; Receptors, Histamine H2; Thiourea | 1986 |
Hypotension and bradycardia elicited by histamine into the C1 area of the rostral ventrolateral medulla.
Topics: Animals; Blood Pressure; Dimaprit; Heart Rate; Hemodynamics; Histamine; Injections; Male; Medulla Oblongata; Metiamide; Naphazoline; Phenoxybenzamine; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Thiourea | 1987 |
Histamine receptors on rat ocular surface.
Topics: Animals; Capillary Permeability; Chlorpheniramine; Cimetidine; Conjunctiva; Dimaprit; Dose-Response Relationship, Drug; Drug Combinations; Histamine; Male; Rats; Rats, Inbred Strains; Receptors, Histamine; Thiourea | 1987 |
Evidence for histaminergic arousal mechanisms in the hypothalamus of cat.
Topics: Animals; Arousal; Cats; Dimaprit; Female; Histamine; Histamine Antagonists; Histidine Decarboxylase; Hypothalamus; Hypothalamus, Posterior; Injections; Injections, Intraperitoneal; Male; Methylhistidines; Pyrilamine; Thiourea | 1988 |
Characteristics of histamine receptors in the isolated and perfused canine coronary arteries.
Topics: Animals; Chlorpheniramine; Cimetidine; Coronary Vessels; Dimaprit; Dogs; Endothelium, Vascular; Female; Histamine; In Vitro Techniques; Male; Pyridines; Receptors, Histamine; Saponins; Thiourea; Vasoconstriction; Vasodilation | 1987 |
Mucosal protective action of histamine against gastric lesions induced by HCl in rats: importance of antigastric motor activity mediated by H2-receptors.
Topics: Animals; Cimetidine; Dimaprit; Gastric Acid; Gastric Mucosa; Gastrointestinal Motility; Histamine; Hydrochloric Acid; Indomethacin; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Tripelennamine | 1988 |
Histaminergic regulation of prolactin secretion: involvement of tuberoinfundibular dopaminergic neurons.
Topics: Animals; Cerebral Ventricles; Dimaprit; Dopamine; Histamine; Infusions, Intra-Arterial; Injections, Intraventricular; Male; Neurons; Prolactin; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Reference Values; Thiazoles; Thiourea | 1988 |
Histaminergic regulation of prolactin secretion: involvement of serotoninergic neurons.
Topics: Dimaprit; Histamine; Ketanserin; Methysergide; Neurons; Prolactin; Receptors, Dopamine; Receptors, Serotonin; Serotonin; Thiourea | 1988 |
Histamine receptor effects on dissipation of an intracellular proton gradient of isolated gastric mucosal surface cells.
Topics: Animals; Bicarbonates; Chlorides; Cimetidine; Dimaprit; Diphenhydramine; Gastric Acid; Gastric Mucosa; Histamine; Protons; Pyridines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Sodium; Thiourea | 1987 |
Enhanced adverse electrophysiologic effects of histamine after myocardial infarction in guinea pigs.
Topics: Action Potentials; Animals; Arrhythmias, Cardiac; Chlorpheniramine; Dimaprit; Electrophysiology; Guinea Pigs; Heart; Heart Rate; Histamine; Male; Myocardial Infarction; Thiourea | 1985 |
Modulation of in vitro cellular immune response by histamine agonists or antagonists in murine species.
Topics: Animals; Cell Line; Cell Survival; Chlorpheniramine; Chromium Radioisotopes; Cimetidine; Dimaprit; Diphenhydramine; Histamine; Histamine Antagonists; Imidazoles; Immunity, Cellular; Impromidine; Kinetics; Male; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Ranitidine; T-Lymphocytes, Cytotoxic; T-Lymphocytes, Regulatory; Thiourea | 1985 |
Quantification of H2-agonism by clonidine and dimaprit in an adenylate cyclase assay.
Topics: Adenylyl Cyclases; Animals; Cimetidine; Clonidine; Dimaprit; Guinea Pigs; Histamine; In Vitro Techniques; Myocardium; Receptors, Histamine; Receptors, Histamine H2; Thiourea | 1985 |
Action of tricyclic antidepressants on cyclic AMP in mucosal cells from guinea pig stomach.
Topics: Alprostadil; Amitriptyline; Animals; Antidepressive Agents, Tricyclic; Brain; Cyclic AMP; Dimaprit; Gastric Mucosa; Guinea Pigs; Histamine; In Vitro Techniques; Oxygen Consumption; Prostaglandins E; Receptors, Histamine; Theophylline; Thiourea | 1984 |
Effects of histamine agonists and antagonists on luminol-dependent chemiluminescence of granulocytes.
Topics: Cimetidine; Dimaprit; Granulocytes; Histamine; Histamine Antagonists; Humans; In Vitro Techniques; Luminescent Measurements; Luminol; Pyridazines; Pyridines; Pyrilamine; Ranitidine; Thiourea | 1984 |
The role of prostaglandins in histamine-induced gastric vasodilation in the dog.
Topics: Acetazolamide; Animals; Anti-Inflammatory Agents; Arachidonic Acids; Dimaprit; Dogs; Drug Interactions; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Hydroxyzine; Male; Pharmaceutical Vehicles; Prostaglandins; Pyridines; Receptors, Histamine H1; Receptors, Histamine H2; Stomach; Thiourea; Time Factors; Vasodilation | 1980 |
Effects of histamine on human isolated heart muscle: comparison with effects of noradrenaline.
Topics: Cimetidine; Dimaprit; Heart; Histamine; Humans; In Vitro Techniques; Myocardial Contraction; Norepinephrine; Propranolol; Pyrilamine; Receptors, Histamine H2; Thiourea | 1980 |
Evaluation of the role of Histamine H1- and H2-receptors in cutaneous inflammation in the guinea-pig produced by histamine and mast cell degranulation.
Topics: Animals; Cimetidine; Dimaprit; Guinea Pigs; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Inflammation; Male; Mast Cells; Mathematics; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Skin; Thiourea; Vasodilation | 1980 |
Histamine inhibition of the in vitro induction of cytotoxic T-cell responses.
Topics: Animals; Cytotoxicity, Immunologic; Dimaprit; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Lymphocyte Culture Test, Mixed; Mice; T-Lymphocytes; Thiourea | 1980 |
Gastrointestinal ulceration in the guinea pig in response to dimaprit, histamine, and H1- and H2-blocking agents.
Topics: Animals; Cimetidine; Dimaprit; Diphenhydramine; Duodenal Ulcer; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Injections, Intramuscular; Injections, Intraperitoneal; Male; Receptors, Histamine H1; Receptors, Histamine H2; Stomach Ulcer; Thiourea | 1981 |
Mesenteric vascular reactivity to histamine receptor agonists and antagonists.
Topics: Adrenergic Agonists; Animals; Blood Flow Velocity; Dimaprit; Dogs; Dose-Response Relationship, Drug; Female; Furans; Hemodynamics; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Infusions, Intra-Arterial; Male; Mesentery; Oxygen Consumption; Ranitidine; Receptors, Histamine; Receptors, Histamine H1; Regional Blood Flow; Thiourea; Tripelennamine | 1981 |
Impairment of pharmacological modulation of airways smooth muscle by a respiratory pathogen.
Topics: Airway Resistance; Animals; Bacterial Vaccines; Carbachol; Dimaprit; Haemophilus; Histamine; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Rats; Respiratory Tract Infections; Thiourea; Trachea | 1981 |
Histamine-induced rise in core temperature of chloral-anaesthetized rats: mediation by H2-receptors located in the preopticus area of hypothalamus.
Topics: Animals; Body Temperature; Chloral Hydrate; Dimaprit; Guanidines; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Hypothalamus; Imidazoles; Impromidine; Male; Preoptic Area; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H2; Thiourea | 1982 |
An inhibitory effect of histamine on the rat anococcygeus muscle.
Topics: Acetylcholine; Animals; Carbachol; Cimetidine; Dimaprit; Drug Interactions; Guanidines; Histamine; Imidazoles; Impromidine; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Pyrilamine; Rats; Thiourea | 1982 |
Histamine suppresses in vitro synthesis of precursor (pro-C5) of the fifth complement component (C5) by mouse peritoneal macrophages.
Topics: Animals; Antigens; Bucladesine; Cimetidine; Complement C5; Complement Inactivator Proteins; Dimaprit; Guinea Pigs; Hemolysis; Histamine; Histamine H2 Antagonists; Humans; Macrophages; Male; Mice; Mice, Inbred C57BL; Protein Precursors; Receptors, Histamine H2; Thiourea; Tripelennamine | 1982 |
Apparent irreversible H2-receptor blocking and prolonged gastric antisecretory activities of 3-N-(3-[3-(1-piperidinomethyl)phenoxy]propyl) amino-4-amino-1,2,5-thiadiazole-1-oxide (L-643, 441).
Topics: Animals; Cimetidine; Dimaprit; Dogs; Female; Furans; Gastric Juice; Guinea Pigs; Heart Rate; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Male; Ranitidine; Thiadiazoles; Thiourea | 1983 |
Histamine receptors in primate gallbladder.
Topics: Animals; Dimaprit; Dose-Response Relationship, Drug; Female; Gallbladder; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Papio; Pressure; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1983 |
Histamine modulation of human neutrophil oxidative metabolism, locomotion, degranulation, and membrane potential changes.
Topics: Carbocyanines; Chemotaxis, Leukocyte; Cytoplasmic Granules; Dimaprit; Glucuronidase; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Hydrogen Peroxide; Membrane Potentials; Muramidase; Neutrophils; Oxygen Consumption; Receptors, Histamine H1; Receptors, Histamine H2; Superoxides; Thiourea | 1983 |
Evidence for histamine H1 and H2 receptors in guinea-pig oxyntic cells.
Topics: Animals; Carbonic Anhydrases; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Methylhistamines; Parietal Cells, Gastric; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1983 |
Release of prolactin and luteinizing hormone by histamine agonists in ovariectomized, steroid-treated rats under ether anesthesia.
Topics: Animals; Castration; Dimaprit; Female; Histamine; Histamine H1 Antagonists; Luteinizing Hormone; Methylhistamines; Metiamide; Pituitary Gland, Anterior; Prolactin; Pyridines; Pyrilamine; Rats; Thiourea | 1983 |
The effect of histamine, H1 and H2 agonists, and H1 and H2 antagonists on postprandial pancreatic polypeptide release in dogs.
Topics: Animals; Cimetidine; Dimaprit; Dogs; Food; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Pancreatic Polypeptide; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Secretory Rate; Thiazoles; Thiourea | 1983 |
Intracellular study of effects of histamine on electrical behaviour of myenteric neurones in guinea-pig small intestine.
Topics: Action Potentials; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine Antagonists; In Vitro Techniques; Intestine, Small; Membrane Potentials; Myenteric Plexus; Neurons; Neurotransmitter Agents; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Serotonin; Thiourea | 1984 |
Differences in the interaction of histamine H2 receptor antagonists and tricyclic antidepressants with adenylate cyclase from guinea pig gastric mucosa.
Topics: Adenylyl Cyclases; Animals; Antidepressive Agents, Tricyclic; Cell Membrane; Dimaprit; Gastric Fundus; Gastric Mucosa; Guinea Pigs; Histamine; Histamine H2 Antagonists; Iprindole; Kinetics; Receptors, Histamine H2; Thiourea | 1984 |
Influence of histamine or dimaprit on histamine release induced by anti-ige from human whole blood.
Topics: Antibodies; Dimaprit; Histamine; Histamine Release; Humans; Immunoglobulin E; Receptors, Histamine; Receptors, Histamine H2; Thiourea | 1980 |
Effects of the histamine H2-receptor agonists dimaprit and 4-methylhistamine on the central noradrenaline and serotonin system.
Topics: Animals; Behavior, Animal; Brain; Dimaprit; Female; Histamine; Hydroxyindoleacetic Acid; Methoxyhydroxyphenylglycol; Methylhistamines; Norepinephrine; Rats; Receptors, Histamine; Receptors, Histamine H2; Serotonin; Thiourea; Tranylcypromine | 1980 |
Enhancement of histamine synthesis in mouse skin by epinephrine.
Topics: Animals; Dimaprit; Epinephrine; Guanidines; Histamine; Histamine Release; Kinetics; Male; Methylhistidines; Mice; Skin; Skin Physiological Phenomena; Thiourea | 1984 |
Histamine H2 receptor desensitization in HL-60 human promyelocytic leukemia cells.
Topics: 1-Methyl-3-isobutylxanthine; Cell Differentiation; Cell Line; Cimetidine; Cyclic AMP; Dimaprit; Dinoprostone; Dose-Response Relationship, Drug; Histamine; Humans; Leukemia, Myeloid, Acute; Prostaglandins E; Receptors, Histamine; Receptors, Histamine H2; Thiocarbamates; Thiourea | 1984 |
Reciprocal H1- and H2-histamine receptors in guinea pig gallbladder.
Topics: Animals; Dimaprit; Female; Gallbladder; Guinea Pigs; Histamine; Male; Muscle Contraction; Muscle, Smooth; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1982 |
Rabbit mesenteric artery receptors formed by cold exposure mediating increased histamine-induced relaxation.
Topics: Animals; Cold Temperature; Dimaprit; Histamine; In Vitro Techniques; Mesenteric Arteries; Metiamide; Muscle, Smooth, Vascular; Phenylephrine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Reserpine; Thiourea; Tripelennamine; Vasodilation | 1982 |
Autacoid and autonomic reactivity of bovine and ovine bronchus: modifications by antigenic sensitization.
Topics: Animals; Bronchi; Carbachol; Cattle; Dimaprit; Dose-Response Relationship, Drug; Epinephrine; Histamine; In Vitro Techniques; Isoproterenol; Muscle Contraction; Phenylephrine; Serotonin; Sheep; Thiourea | 1982 |
Histamine-induced inhibition of lymphocyte proliferation and lysosomal enzyme release from polymorphs may not be mediated via H1- or H2-receptors.
Topics: Dimaprit; Histamine; Humans; Lymphocyte Activation; Lysosomes; Metiamide; Phytohemagglutinins; Polymorphism, Genetic; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1982 |
The effect of histamine on the development of adjuvant arthritis in the rat.
Topics: Animals; Arthritis; Arthritis, Experimental; Dimaprit; Dose-Response Relationship, Drug; Female; Histamine; Metiamide; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Time Factors | 1982 |
An investigation of the involvement of histaminergic systems in novelty-induced grooming in the mouse.
Topics: Animals; Arousal; Cimetidine; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Grooming; Histamine; Male; Mice; Pyridines; Receptors, Histamine; Thiourea | 1982 |
Inhibition of phytohaemagglutinin-induced proliferation of human peripheral blood lymphocytes by histamine and histamine H1 and H2 agonists.
Topics: Cell Division; Cells, Cultured; Dimaprit; Dose-Response Relationship, Drug; Histamine; Humans; Imidazoles; Impromidine; Lymphocytes; Methylhistamines; Phytohemagglutinins; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea | 1983 |
Histamine receptors in the human ureter.
Topics: Chlorpheniramine; Dimaprit; Histamine; Humans; In Vitro Techniques; Metiamide; Muscle Contraction; Muscle, Smooth; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Ureter | 1983 |
Vascular responses of the isolated perfused stomach of rabbit and rat to histamine.
Topics: Animals; Dimaprit; Histamine; Histamine Antagonists; Male; Muscle, Smooth, Vascular; Rabbits; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Species Specificity; Stomach; Thiourea; Vasodilator Agents | 1983 |
The role of histamine receptors in the release of renin.
Topics: Animals; Dimaprit; Dogs; Female; Histamine; Kidney; Male; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Renal Circulation; Renin; Sodium Chloride; Thiourea | 1983 |
Central H1- and H2-histaminergic stimulation of pituitary-adrenocortical response under stress in rats.
Topics: Animals; Corticosterone; Dimaprit; Histamine; Histamine Antagonists; Male; Methylhistamines; Pituitary-Adrenal System; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Stress, Physiological; Thiourea | 1983 |
Central histaminergic stimulation of pituitary--adrenocortical response in the rat.
Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Dose-Response Relationship, Drug; Histamine; Imidazoles; Impromidine; Male; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1983 |
Effects of histamine receptor stimulation on regional myocardial blood flow.
Topics: Animals; Blood Pressure; Cimetidine; Coronary Circulation; Dimaprit; Diphenhydramine; Dogs; Female; Heart Rate; Histamine; Male; Microspheres; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea | 1983 |
Studies on cutaneous vascular permeability in the rat: increases caused by histamine and histamine-like agents.
Topics: Animals; Capillary Permeability; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Histamine; Microcirculation; Pyrilamine; Rats; Regional Blood Flow; Skin; Thiourea | 1984 |
Effect of histamine receptor agonists and antagonists on the uterine vasculature.
Topics: Animals; Dimaprit; Female; Histamine; p-Methoxy-N-methylphenethylamine; Pyridines; Receptors, Histamine H1; Receptors, Histamine H2; Regional Blood Flow; Sheep; Thiourea; Uterus | 1984 |
Studies on the effect of histamine in isolated human pulmonary arteries and veins.
Topics: Aged; Dimaprit; Female; Histamine; Humans; In Vitro Techniques; Male; Methylhistamines; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phentolamine; Potassium; Pulmonary Artery; Pulmonary Veins; Pyrilamine; Thiourea | 1984 |
Histamine action on guinea pig ileal mucosa.
Topics: Animals; Bicarbonates; Biological Transport, Active; Chlorides; Dimaprit; Electric Conductivity; Female; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Intestinal Mucosa; Male; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1984 |
Dibenamine enhancement of histamine-induced relaxation of the rabbit mesenteric artery.
Topics: Animals; Cold Temperature; Dibenzylchlorethamine; Dimaprit; Drug Synergism; Histamine; Mesenteric Arteries; Muscle Contraction; Muscle Relaxation; Papaverine; Rabbits; Receptors, Histamine; Thiourea | 1983 |
[Imidazolic H2-agonists: importance of 2-amino substitution for pharmacological activity].
Topics: Animals; Biological Assay; Cats; Dimaprit; Gastric Acid; Guinea Pigs; Histamine; Methylhistamines; Muscle Relaxation; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Structure-Activity Relationship; Thiourea; Urinary Bladder | 1984 |
A comparison of dimaprit, nordimaprit, methylamine and chloroquine as inhibitors of mitogen-induced lymphocyte activation.
Topics: Cells, Cultured; Chloroquine; Chromium Radioisotopes; Concanavalin A; Dimaprit; Histamine; Humans; Lymphocyte Activation; Lymphocytes; Methylamines; Mitogens; Phytohemagglutinins; Thiourea; Thymidine | 1984 |
Lack of an effect of drugs acting at histamine receptors on norepinephrine-induced relaxation of porcine coronary arteries.
Topics: Animals; Coronary Vessels; Dimaprit; Histamine; In Vitro Techniques; Muscle Relaxation; Muscle, Smooth, Vascular; Myocardial Contraction; Norepinephrine; Phenethylamines; Receptors, Histamine; Swine; Thiourea | 1984 |
Specific activation of cyclic AMP-dependent protein kinase(s) by H2-histamine agonists in isolated gastric mucosal cells from guinea-pig.
Topics: Animals; Cimetidine; Cyclic AMP; Dimaprit; Diphenhydramine; Enzyme Activation; Gastric Mucosa; Guanidines; Guinea Pigs; Histamine; Imidazoles; Impromidine; In Vitro Techniques; Protein Kinases; Pyridines; Receptors, Histamine; Receptors, Histamine H2; Thiourea | 1980 |
Histamine receptors on dispersed parathyroid cells from pathological human parathyroid tissue.
Topics: Cyclic AMP; Dimaprit; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Humans; Hyperparathyroidism; In Vitro Techniques; Parathyroid Glands; Parathyroid Hormone; Receptors, Histamine H2; Thiourea | 1980 |
Cardiac contractile and metabolic effects mediated via the myocardial H2-receptor adenylate cyclase system. Characterization of two new specific H2-receptor agonists, impromidine and dimaprit, in the guinea pig and human myocardium.
Topics: Adenylyl Cyclases; Animals; Cimetidine; Cyclic AMP; Dimaprit; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; Histamine; Humans; Imidazoles; Impromidine; Isoproterenol; Metoprolol; Myocardial Contraction; Myocardial Infarction; Myocardium; Phosphoric Diester Hydrolases; Receptors, Histamine; Receptors, Histamine H2; Thiourea; Tyramine | 1981 |
Cyclic AMP increase in canine parotid gland mediated by histamine H2-receptors.
Topics: Animals; Cyclic AMP; Dimaprit; Dogs; Female; Histamine; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Parotid Gland; Pyridines; Receptors, Histamine; Receptors, Histamine H2; Thiourea | 1981 |
Pharmacological interactions between ranitidine, cimetidine, metiamide and tiotidine at histamine H2-receptor sites in guinea-pig atria.
Topics: Animals; Cimetidine; Dimaprit; Drug Interactions; Furans; Guanidines; Guinea Pigs; Heart; Heart Rate; Histamine; In Vitro Techniques; Metiamide; Ranitidine; Receptors, Histamine; Receptors, Histamine H2; Thiazoles; Thiourea | 1982 |
Interaction of histamine with gastric mucosal cells. Effect of histamine agonists on binding and biological response.
Topics: Animals; Chemical Phenomena; Chemistry; Cyclic AMP; Dimaprit; Gastric Mucosa; Guinea Pigs; Histamine; In Vitro Techniques; Inosine Monophosphate; Kinetics; Male; Receptors, Histamine; Thiourea | 1982 |
Inotropic and electrophysiological effects of histamine on human ventricular heart muscle.
Topics: Action Potentials; Adolescent; Adult; Aged; Animals; Child; Child, Preschool; Cyclic AMP; Dimaprit; Female; Guinea Pigs; Heart Ventricles; Histamine; Humans; Isoproterenol; Male; Middle Aged; Myocardial Contraction; Norepinephrine; Papillary Muscles; Receptors, Histamine H2; Stimulation, Chemical; Thionucleotides; Thiourea | 1982 |
Histamine and serotonin suppression of lymphocyte response to phytohemagglutinin and allogeneic cells.
Topics: Animals; Cimetidine; Dimaprit; Drug Antagonism; Female; Histamine; Lymphocyte Activation; Lymphocyte Culture Test, Mixed; Male; Metiamide; Mice; Mice, Inbred Strains; Phytohemagglutinins; Ranitidine; Serotonin; Thiourea | 1984 |
Studies with specific agonists and antagonists of the role of histamine H1- and H2-receptor activation in the pathogenesis of gastric lesions in rats.
Topics: Aminopyridines; Animals; Atropine; Dimaprit; Drug Interactions; Female; Histamine; Pyridines; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Stomach Ulcer; Thiourea | 1984 |
A question of the specificity of rabbit atrial chronotropic histamine receptors and agents which affect their activity.
Topics: Animals; Dimaprit; Female; Guinea Pigs; Heart Rate; Histamine; Male; Methylhistamines; Pyridines; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Time Factors | 1980 |
Choledochal sphincter relaxation in response to histamine in the primate.
Topics: Animals; Cholecystokinin; Dimaprit; Female; Gallbladder; Haplorhini; Histamine; Muscle, Smooth; Papio; Pressure; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1980 |
Dimaprit inhibition of zymosan-stimulated beta-glucuronidase release from human granulocytes.
Topics: Adult; Dimaprit; Glucuronidase; Granulocytes; Histamine; Humans; In Vitro Techniques; Lysosomes; Metiamide; Neutrophils; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Zymosan | 1980 |
Cardiovascular and behavioural changes after i.c.v. infusions of histamine and agonists in conscious goat.
Topics: Animals; Behavior, Animal; Dimaprit; Female; Goats; Hemodynamics; Histamine; Injections, Intraventricular; Pyridines; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1980 |
Evidence for a role of endogenous histamine in central cardiovascular regulation: inhibition of histamine-N-methyltransferase by SKF 91488.
Topics: Animals; Blood Pressure; Brain; Dimaprit; Heart Rate; Hemodynamics; Histamine; Histamine N-Methyltransferase; Male; Methyltransferases; Rats; Thiourea | 1981 |
pH-dependent activity of H1- and H2-histamine receptors in guinea-pig gallbladder.
Topics: Acetylcholine; Animals; Dimaprit; Female; Gallbladder; Guinea Pigs; Histamine; Hydrogen-Ion Concentration; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Potassium Chloride; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1981 |
Vascular studies with histamine in vitro.
Topics: Animals; Blood Vessels; Cimetidine; Dimaprit; Hindlimb; Histamine; Histamine Antagonists; Male; Rats; Regional Blood Flow; Thiourea; Vasodilator Agents | 1981 |
Hypothalamic superfusion with histamine agonists and antagonists modifies the pressor response to hypothalamic stimulation.
Topics: Animals; Blood Pressure; Cats; Dimaprit; Electric Stimulation; Histamine; Histamine Antagonists; Hypothalamus; Thiourea | 1981 |
Lack of histamine involvement in parathyroid hormone hypotensive action.
Topics: Animals; Blood Pressure; Cimetidine; Dimaprit; Female; Histamine; Hypotension; Male; p-Methoxy-N-methylphenethylamine; Parathyroid Hormone; Peptide Fragments; Promethazine; Propranolol; Pyridines; Rats; Thiourea | 1981 |
Effect of histamine H1- and H2-receptor agonists on gamma-aminobutyric acid (GABA) content in hypothalamus and striatum of the rat brain.
Topics: Animals; Brain Chemistry; Corpus Striatum; Dimaprit; Female; gamma-Aminobutyric Acid; Histamine; Hypothalamus; Methylhistamines; Rats; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1980 |
Comparison of H2 receptor agonists in rabbit atria and aorta.
Topics: Animals; Aorta; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Guanidines; Heart Atria; Heart Rate; Histamine; Imidazoles; Impromidine; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Rabbits; Receptors, Histamine; Receptors, Histamine H2; Thiourea | 1981 |
Further experiments on the pharmacological actions of ergometrine.
Topics: Animals; Cattle; Cimetidine; Coronary Vessels; Dimaprit; Ergonovine; Gastric Acid; Guinea Pigs; Histamine; Muscle Contraction; Pyrilamine; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1981 |
Characterization of neuronal and vascular histamine receptors mediating the salivary and vasodilator responses to histamine of the dog submandibular gland.
Topics: Animals; Dimaprit; Dogs; Female; Histamine; Male; Pyridines; Receptors, Histamine; Regional Blood Flow; Salivation; Submandibular Gland; Thiourea; Vasodilation | 1981 |
Cerebral circulation and histamine: 1. Participation of vascular H1- and H2-receptors in vasodilatory responses to carotid arterial infusion.
Topics: Animals; Blood-Brain Barrier; Carotid Artery, Internal; Cerebrovascular Circulation; Dimaprit; Glucose; Histamine; Injections, Intra-Arterial; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Urea; Vasodilation | 1981 |
Effect of histamine agonists and antagonists on the production of murine reaginic antibodies.
Topics: Animals; Antibody Formation; Dimaprit; Histamine; Histamine Antagonists; Immunoglobulin E; Male; Methylhistamines; Metiamide; Mice; Reagins; Receptors, Histamine; Thiourea | 1981 |
Changes in the response of guinea-pig airways in vivo and in vitro to cimetidine and propranolol during development.
Topics: Aging; Airway Resistance; Animals; Bronchi; Cimetidine; Dimaprit; Female; Guanidines; Guinea Pigs; Histamine; In Vitro Techniques; Methylhistamines; Muscle Contraction; Propranolol; Receptors, Histamine; Receptors, Histamine H2; Thiourea; Trachea | 1982 |
Hypothalamic superfusion with histamine agonists and antagonists modifies the pressor response to hypothalamic stimulation.
Topics: Animals; Blood Pressure; Cats; Dimaprit; Electric Stimulation; Female; Histamine; Histamine Antagonists; Hypothalamus; Male; Methylhistamines; Metiamide; Sympathomimetics; Thiourea; Time Factors | 1981 |
Histamine H2 receptor-mediated endothelium-dependent relaxation in canine spinal artery.
Topics: Animals; Arteries; Dimaprit; Dogs; Endothelium, Vascular; Female; Histamine; In Vitro Techniques; Male; Receptors, Histamine H2; Spinal Cord; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents | 1995 |
Identification of IgE-bearing cells in the late-phase response to antigen in the lung as basophils.
Topics: Alcian Blue; Allergens; Antibodies, Anti-Idiotypic; Antigens, Surface; Basophils; Bronchoalveolar Lavage Fluid; Dimaprit; Histamine; Histamine Release; Humans; Hypersensitivity; Immunoglobulin E; Lung; Mast Cells; N-Formylmethionine Leucyl-Phenylalanine; Tetradecanoylphorbol Acetate | 1994 |
Stimulatory effect of histamine on cyclic AMP formation in chick pineal gland.
Topics: 1-Methyl-3-isobutylxanthine; Adenine; Analysis of Variance; Animals; Carbon Radioisotopes; Chickens; Colforsin; Cyclic AMP; Dimaprit; Guinea Pigs; Hippocampus; Histamine; Histamine Agonists; In Vitro Techniques; Kinetics; Male; Methylhistamines; Pineal Gland; Ranitidine; Rats; Rats, Wistar; Thiazoles; Tritium | 1994 |
Possible participation of histamine H3-receptors in the regulation of anaphylactic histamine release from isolated rat peritoneal mast cells.
Topics: Anaphylaxis; Animals; Anticonvulsants; Chromatography, High Pressure Liquid; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Histamine; Histamine Agonists; Histamine Antagonists; Histamine Release; In Vitro Techniques; L-Lactate Dehydrogenase; Male; Mast Cells; Methylhistamines; p-Methoxy-N-methylphenethylamine; Peritoneal Cavity; Peritoneum; Piperidines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H3 | 1994 |
Effect of histamine on haemorrhagic mucosal lesions is related to vascular permeability in rats: studies with histamine, H1-, H2- and H3-agonists and bradykinin.
Topics: Absorption; Animals; Betahistine; Bradykinin; Capillary Permeability; Dimaprit; Dose-Response Relationship, Drug; Ethanol; Female; Gastric Mucosa; Gastrointestinal Hemorrhage; Histamine; Histamine Agonists; Injections, Subcutaneous; Intubation, Gastrointestinal; Methylhistamines; Organotechnetium Compounds; Rats; Rats, Sprague-Dawley; Stomach Diseases; Sugar Acids | 1995 |
Rapid desensitization of the histamine H2 receptor on the human monocytic cell line U937.
Topics: Cells, Cultured; Cyclic AMP; Dimaprit; Dose-Response Relationship, Drug; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Leukemia, Monocytic, Acute; Monocytes; Receptors, Histamine H2; Tumor Cells, Cultured | 1994 |
Characterization and function of histamine receptors in corpus cavernosum.
Topics: Acetylcholine; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Papaverine; Penis; Piperidines; Pyrilamine; Rabbits; Receptors, Histamine; Thiazoles | 1995 |
H3 receptors: modulation of histamine-stimulated neural pathways influencing electrogenic ion transport in the guinea pig colon.
Topics: Animals; Chloride Channels; Colon; Dimaprit; Electrophysiology; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Membrane Potentials; Neural Pathways; Receptors, Histamine H2; Receptors, Histamine H3 | 1994 |
Effect of cimetidine on the histamine and dimaprit induced responses on the guinea pig ileum during development.
Topics: Aging; Animals; Animals, Newborn; Cimetidine; Dimaprit; Female; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; Ileum; In Vitro Techniques; Male; Muscle Development; Muscle, Smooth | 1993 |
2-Thiazolylethylamine, a selective histamine H1 agonist, decreases seizure susceptibility in mice.
Topics: Animals; Anticonvulsants; Dimaprit; Dose-Response Relationship, Drug; Electroshock; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Injections, Intraventricular; Male; Mice; Mice, Inbred Strains; Pentylenetetrazole; Receptors, Histamine H1; Seizures; Thiazoles | 1994 |
Histamine inhibits immunoglobulin production via histamine H2 receptors without affecting cell growth in human B cells.
Topics: B-Lymphocytes; Cell Division; Cell Line; Dimaprit; Histamine; Histamine H2 Antagonists; Humans; Immunoglobulins; Kinetics; Receptors, Histamine H2 | 1994 |
Structure and function of human histamine N-methyltransferase: critical enzyme in histamine metabolism in airway.
Topics: Amino Acid Sequence; Animals; Base Sequence; Bronchi; Bronchoconstriction; Chromosome Mapping; Chromosomes, Human, Pair 1; Cloning, Molecular; Dimaprit; DNA, Complementary; Genes; Histamine; Histamine N-Methyltransferase; Humans; Molecular Sequence Data; Rats; RNA, Messenger; Structure-Activity Relationship | 1994 |
Functional subtyping of histamine receptors on the canine proximal colonic mucosa.
Topics: Animals; Chlorides; Colon; Dimaprit; Dogs; Dose-Response Relationship, Drug; Female; Histamine; In Vitro Techniques; Intestinal Mucosa; Male; Pyridines; Receptors, Histamine; Sodium | 1994 |
Effect of social isolation on corticosterone secretion elicited by histaminergic stimulation.
Topics: Animals; Biogenic Monoamines; Corticosterone; Dimaprit; Histamine; Histamine Agonists; Hypothalamus; Injections, Intraventricular; Male; Pyridines; Rats; Rats, Wistar; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Social Isolation; Stress, Psychological | 1994 |
Pituitary-adrenocortical responsiveness to histaminergic stimulation during social stress of crowding in rats.
Topics: Animals; Corticosterone; Crowding; Dimaprit; Histamine; Histamine Agonists; Injections, Intraventricular; Male; Pituitary-Adrenal System; Pyridines; Rats; Rats, Wistar; Receptors, Histamine; Stress, Psychological | 1994 |
Dimaprit analogues inhibit tyrosinase via a disulphide breakdown product independently of the histamine H2 receptor.
Topics: Biotransformation; Cell Line; Dimaprit; Disulfides; Histamine; Humans; Kinetics; Melanoma; Monophenol Monooxygenase; Receptors, Histamine H2; Sulfhydryl Compounds; Tumor Cells, Cultured | 1994 |
Evidence for an inhibitory role of central histamine on carrageenin-induced hyperalgesia.
Topics: Animals; Carrageenan; Central Nervous System; Dimaprit; Histamine; Histamine Agonists; Hyperalgesia; Male; Methylhistamines; Rats; Rats, Sprague-Dawley | 1994 |
Mechanisms of augmented vascular responses to histamine in atherosclerotic rabbit common carotid arteries.
Topics: Animals; Arteriosclerosis; Carotid Artery, Common; Dimaprit; Dose-Response Relationship, Drug; Histamine; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Pyridines; Rabbits; Receptors, Histamine H2; Vasoconstriction; Vasodilation | 1994 |
HMT regulates histamine-induced Cl- secretion across the canine tracheal epithelium.
Topics: Amiloride; Animals; Chlorides; Dimaprit; Dogs; Electrophysiology; Epithelium; Female; Histamine; Histamine N-Methyltransferase; Male; Trachea | 1994 |
[The effect of intravenous cimetidine and histamine on splanchnic circulation in the dogs].
Topics: Animals; Blood Pressure; Cimetidine; Dimaprit; Dogs; Hepatic Artery; Histamine; Histamine H2 Antagonists; Infusions, Intravenous; Maleates; Mesenteric Arteries; Receptors, Histamine H1; Splanchnic Circulation; Vascular Resistance; Vasoconstriction; Vasodilation | 1993 |
In vitro cardiac pharmacology of the new histamine H2-receptor agonist amthamine: comparisons with histamine and dimaprit.
Topics: Animals; Atrial Function; Dimaprit; Electric Stimulation; Guinea Pigs; Heart; Heart Atria; Histamine; Histamine Agonists; Humans; In Vitro Techniques; Myocardial Contraction; Papillary Muscles; Rabbits; Ranitidine; Thiazoles | 1993 |
Viral respiratory infection causes airway hyperresponsiveness and decreases histamine N-methyltransferase activity in guinea pigs.
Topics: Acetylcholine; Acetylcholinesterase; Airway Resistance; Animals; Bronchi; Bronchial Hyperreactivity; Bronchoconstriction; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine N-Methyltransferase; Lung; Male; Parainfluenza Virus 1, Human; Paramyxoviridae Infections; Respiratory Tract Infections; Trachea | 1994 |
Histamine H2-receptor plays only a minor role in histamine-induced wheal response in the squirrel monkey and guinea pig.
Topics: Animals; Chlorpheniramine; Dimaprit; Dose-Response Relationship, Drug; Famotidine; Female; Guinea Pigs; Histamine; Histamine Agonists; Injections, Intradermal; Male; Pyridines; Ranitidine; Receptors, Histamine H2; Saimiri; Urticaria | 1993 |
Histamine N-methyltransferase modulates histamine- and antigen-induced bronchoconstriction in guinea pigs in vivo.
Topics: Aerosols; Animals; Antigens; Bronchial Provocation Tests; Bronchoconstriction; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine N-Methyltransferase; Immunization; Male; Ovalbumin; Tissue Distribution | 1993 |
Histamine N-methyltransferase inhibitor potentiates histamine- and antigen-induced airway microvascular leakage in guinea pigs.
Topics: Amine Oxidase (Copper-Containing); Animals; Antigens; Capillary Permeability; Dimaprit; Drug Synergism; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine N-Methyltransferase; Immunization; Male; Nasal Mucosa; Respiratory System | 1995 |
The source and action of histamine in the isolated guinea-pig gallbladder.
Topics: Animals; Dimaprit; Electric Stimulation; Female; Gallbladder; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; Immunohistochemistry; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Ranitidine; Receptors, Histamine H3; Thiazoles | 1995 |
Histamine H3 receptor inhibition of K(+)-evoked release of acetylcholine from rat cortex in vivo.
Topics: Acetylcholine; Analysis of Variance; Animals; Chromatography, High Pressure Liquid; Dimaprit; Histamine; Histamine Agonists; Histamine Antagonists; Male; Methylhistamines; Microdialysis; Neurons; Parietal Lobe; Piperidines; Potassium; Rats; Rats, Wistar; Receptors, Histamine H3; Thiazoles | 1996 |
Histamine receptors and bioeffects on clonal parathyroid endothelial cells.
Topics: Animals; Cattle; Cell Line; Cell Membrane; Cyclic AMP; Dimaprit; DNA; Endothelium; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Iodine Radioisotopes; Kinetics; Parathyroid Glands; Receptors, Histamine H2 | 1996 |
Histamine H2 receptor-mediated airway goblet cell secretion and its modulation by histamine-degrading enzymes.
Topics: Amine Oxidase (Copper-Containing); Animals; Asthma; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glycoproteins; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine N-Methyltransferase; Male; Methylhistamines; Mucus; Piperidines; Pyrilamine; Recombinant Proteins; Trachea | 1997 |
Histamine up-regulates the generation of nitric oxide, and nitric oxide down-regulates the release of histamine in cardiovascular preparations.
Topics: Animals; Cardiovascular Physiological Phenomena; Cardiovascular System; Cattle; Cells, Cultured; Coronary Circulation; Dimaprit; Enzyme Inhibitors; Guinea Pigs; Histamine; Histamine Agonists; Histamine Release; Male; Muscle, Smooth, Vascular; Nitric Oxide; Nitric Oxide Synthase; omega-N-Methylarginine | 1997 |
Histamine mediates the muscle layer-specific responses in the isolated swine myometrium.
Topics: Animals; Dimaprit; Female; Histamine; Histamine Agonists; Histamine H1 Antagonists; Muscle, Smooth; Myometrium; Pyrilamine; Receptors, Histamine; Swine; Uterine Contraction | 1997 |
Histamine modulates the expression of c-fos through cyclic AMP production via the H2 receptor in the human promonocytic cell line U937.
Topics: Cell Differentiation; Cell Division; Cell Line; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dimaprit; Enzyme Activation; Gene Expression; Gene Expression Regulation; Genes, fos; Genes, myc; Histamine; Histamine Agonists; Humans; Kinetics; Monocytes; Proto-Oncogene Mas; Proto-Oncogene Proteins c-fos; Proto-Oncogene Proteins c-myc; Receptors, Histamine H2; RNA, Messenger; Stimulation, Chemical; Substrate Specificity | 1997 |
Mechanisms for histamine H1 receptor-mediated vasodilation in isolated canine lingual arteries.
Topics: Animals; Arteries; Cimetidine; Dimaprit; Diphenhydramine; Dogs; Female; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Pyridines; Receptors, Histamine H1; Tongue; Vasodilation | 1997 |
HMT regulates histamine-induced glycoconjugate secretion from human airways in vitro.
Topics: Animals; Cats; Cimetidine; Dimaprit; Dinoprostone; Glycoconjugates; Glycoproteins; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine N-Methyltransferase; Humans; Indomethacin; Organ Culture Techniques; Phenothiazines; Receptors, Prostaglandin E; Trachea | 1997 |
Endogenous histamine stimulates ischemically sensitive abdominal visceral afferents through H1 receptors.
Topics: Abdomen; Afferent Pathways; Animals; Bile Ducts; Blood Pressure; Cats; Chlorpheniramine; Dimaprit; Duodenum; Female; Gallbladder; Histamine; Histamine H1 Antagonists; Indomethacin; Ischemia; Male; Methylhistamines; Nerve Fibers; Neural Conduction; Pancreas; Pyrilamine; Receptors, Histamine H1 | 1997 |
Regulation of cerebral microvascular permeability by histamine in the anaesthetized rat.
Topics: Anesthesia, General; Animals; Capillary Permeability; Cerebrovascular Circulation; Cimetidine; Dimaprit; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Muscle, Smooth, Vascular; Pia Mater; Pyrilamine; Rats; Venules | 1998 |
Histamine stimulates ion transport by dog pancreatic duct epithelial cells through H1 receptors.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Calcium; Calcium Channel Blockers; Cells, Cultured; Chelating Agents; Chlorides; Cimetidine; Dimaprit; Diphenhydramine; Dogs; Egtazic Acid; Epithelial Cells; Histamine; Iodides; Iodine Radioisotopes; Kinetics; Nitrobenzoates; ortho-Aminobenzoates; Pancreatic Ducts; Receptors, Histamine H1 | 1998 |
Regulation of interleukin-6, and macrophage colony-stimulating factor mRNA levels by histamine in stromal cell line (MC3T3-G2/PA6).
Topics: Animals; Blotting, Northern; Bone Marrow Cells; Cell Line; Dimaprit; Gene Expression Regulation; Histamine; Histamine Agonists; Interleukin-6; Macrophage Colony-Stimulating Factor; Mice; Pyridines; RNA, Messenger; Stromal Cells | 1998 |
Histamine potently suppresses human IL-12 and stimulates IL-10 production via H2 receptors.
Topics: Adult; Cells, Cultured; Cimetidine; Cyclic AMP; Dimaprit; Drug Synergism; Female; Histamine; Histamine Agonists; Histamine H2 Antagonists; Humans; Interleukin-10; Interleukin-12; Lipopolysaccharides; Male; Monocytes; Receptors, Histamine H2; Th1 Cells; Th2 Cells | 1998 |
Histamine sensitivity of mesenteric afferent nerves in the rat jejunum.
Topics: Afferent Pathways; Animals; Blood Pressure; Dimaprit; Histamine; Histamine Agonists; Histamine Antagonists; Jejunum; Muscle, Smooth; Nifedipine; Piperidines; Pyrilamine; Ranitidine; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Splanchnic Circulation | 1998 |
Histamine modulates high-voltage-activated calcium channels in neurons dissociated from the rat tuberomammillary nucleus.
Topics: Animals; Calcium; Calcium Channels; Calcium Channels, N-Type; Depression, Chemical; Dimaprit; Histamine; Histamine Agonists; Histamine Antagonists; Ion Channel Gating; Mammillary Bodies; Methylhistamines; Nerve Tissue Proteins; Neurons; Nicardipine; omega-Agatoxin IVA; omega-Conotoxin GVIA; omega-Conotoxins; Patch-Clamp Techniques; Peptides; Pertussis Toxin; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; Spider Venoms; Tuber Cinereum; Virulence Factors, Bordetella | 1998 |
Evidence of H3 receptor inhibition by iodoaminopotentidine in the guinea pig ileum.
Topics: Animals; Cholinergic Fibers; Dimaprit; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; Ileum; In Vitro Techniques; Methylhistamines; Muscle, Smooth; Ranitidine; Receptors, Histamine H3; Synaptic Transmission | 1998 |
The role of histamine H1, H2 and H3 receptors on enteric ascending synaptic transmission in the guinea pig ileum.
Topics: Animals; Cimetidine; Dimaprit; Electric Stimulation; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Ileum; Male; Motor Neurons; Muscle Contraction; Muscle, Smooth; Pyrilamine; Receptors, Histamine; Synaptic Transmission | 1998 |
Histaminergic H2 receptor ligands modulate acetylcholine release in the ventral striatum.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Corpus Striatum; Dimaprit; Dopamine; Dopamine Agonists; Dopamine Antagonists; Famotidine; gamma-Aminobutyric Acid; Histamine; Histamine H2 Antagonists; Male; Neurons; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Histamine H2 | 1999 |
Nalpha-methyl histamine and histamine stimulate gastrin release from rabbit G-cells via histamine H2-receptors.
Topics: Animals; Antibodies, Monoclonal; Cells, Cultured; Chlorpheniramine; Dimaprit; Dose-Response Relationship, Drug; Drug Interactions; Gastrin-Secreting Cells; Gastrins; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H2 Antagonists; Piperidines; Pyloric Antrum; Rabbits; Ranitidine; Receptors, Histamine | 1999 |
Effects of histamine and related compounds on regional cerebral blood flow in rats.
Topics: Animals; Benzothiazoles; Blood Pressure; Brain Chemistry; Dimaprit; Diphenhydramine; Drug Interactions; Hippocampus; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Male; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Wistar; Regional Blood Flow; Thiazoles; Time Factors | 1999 |
Endothelium-dependent vasodilatation mechanisms by histamine in simian but not in canine femoral arterial branches.
Topics: Animals; Dimaprit; Diphenhydramine; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Endothelium, Vascular; Female; Femoral Artery; Histamine; Histamine Agonists; Histamine H1 Antagonists; Macaca; Male; Muscle, Smooth, Vascular; Pyridines; Saponins; Species Specificity; Vasoconstriction; Vasodilation | 1999 |
Histamine H3 receptor-mediated suppression of inhibitory synaptic transmission in the submucous plexus of guinea-pig small intestine.
Topics: Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Intestine, Small; Male; Methylhistamines; Norepinephrine; Phentolamine; Piperidines; Receptors, Histamine H3; Submucous Plexus; Synaptic Transmission | 2000 |
Histamine suppresses A-type potassium current in myenteric neurons from guinea pig small intestine.
Topics: Animals; Cimetidine; Cyclic AMP; Dimaprit; Drug Interactions; Excitatory Postsynaptic Potentials; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Intestine, Small; Male; Membrane Potentials; Myenteric Plexus; Neurons; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Receptors, Histamine H2 | 2000 |
Actions of histamine on muscle and ganglia of the guinea pig gallbladder.
Topics: Adenosine Triphosphate; Animals; Dimaprit; Excitatory Postsynaptic Potentials; Female; Gallbladder; Gallbladder Emptying; Ganglia, Autonomic; Guinea Pigs; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Mast Cells; Membrane Potentials; Muscle, Smooth; p-Methoxy-N-methylphenethylamine; Patch-Clamp Techniques; Potassium Channels; Pyrilamine; Ranitidine; Receptors, Histamine H1; Receptors, Histamine H2 | 2000 |
Influence of different histamine receptor agonists and antagonists on apomorphine-induced licking behavior in rat.
Topics: Animals; Apomorphine; Chlorpheniramine; Dimaprit; Diphenhydramine; Dopamine Agonists; Drug Interactions; Famotidine; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Piperidines; Ranitidine; Rats; Rats, Sprague-Dawley; Stereotyped Behavior; Thiourea; Toluidines | 2000 |
Histamine H(2) receptors mediate the inhibitory effect of histamine on human eosinophil degranulation.
Topics: Adenylyl Cyclases; Cell Degranulation; Complement C5a; Cyclic AMP; Dimaprit; Eosinophil Peroxidase; Eosinophils; Histamine; Histamine Agonists; Histamine Antagonists; Humans; In Vitro Techniques; Molecular Mimicry; Peroxidases; Receptors, Histamine H2 | 2000 |
Histamine induces exocytosis and IL-6 production from human lung macrophages through interaction with H1 receptors.
Topics: Calcium; Cytosol; Dimaprit; Dose-Response Relationship, Immunologic; Exocytosis; Glucuronidase; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Interleukin-6; Lung; Macrophages, Alveolar; Receptors, Histamine H1; RNA, Messenger; Toluidines; Up-Regulation | 2001 |
Histamine N-methyltransferase regulates histamine-induced phosphoinositide hydrolysis in guinea pig cerebellum.
Topics: Animals; Cerebellum; Dimaprit; Dose-Response Relationship, Drug; Glycerol-3-Phosphate Dehydrogenase (NAD+); Glycerolphosphate Dehydrogenase; Guinea Pigs; Histamine; Histamine Antagonists; Histamine N-Methyltransferase; Hydrolysis; Male; Neurons; Oligonucleotide Probes; Organ Culture Techniques; Phosphatidylinositols; RNA; Synaptic Transmission; Tritium | 2001 |
Histamine inhibits chemotaxis, phagocytosis, superoxide anion production, and the production of TNFalpha and IL-12 by macrophages via H2-receptors.
Topics: Animals; Chemotaxis, Leukocyte; Cytokines; Dimaprit; Histamine; Histamine Agonists; Immunity, Cellular; In Vitro Techniques; Interleukin-12; Macrophages, Peritoneal; Male; Mice; Phagocytosis; Rats; Rats, Wistar; Receptors, Histamine H2; Superoxides; Tumor Necrosis Factor-alpha | 2001 |
Expression of diamine oxidase (histaminase) in guinea-pig tissues.
Topics: Amine Oxidase (Copper-Containing); Animals; Brain; Dimaprit; Dose-Response Relationship, Drug; Gastric Mucosa; Gene Expression Regulation, Enzymologic; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; In Situ Hybridization; In Vitro Techniques; Intestine, Small; Kidney; Liver; Male; Muscle Contraction; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Stomach | 2002 |
The role of guanylyl cyclases in the permeability response to inflammatory mediators in pial venular capillaries in the rat.
Topics: Animals; Atrial Natriuretic Factor; Blood-Brain Barrier; Bradykinin; Brain Edema; Capillaries; Capillary Permeability; Cyclic GMP; Dimaprit; Female; Guanylate Cyclase; Histamine; Histamine Agonists; Inflammation Mediators; Male; Nitric Oxide; Pia Mater; Rats; Rats, Wistar; Receptor, Bradykinin B2; Receptors, Bradykinin; Receptors, Cytoplasmic and Nuclear; Receptors, Histamine H2; Soluble Guanylyl Cyclase; Venules | 2002 |
Defective angiogenesis in the inflammatory granulation tissue in histidine decarboxylase-deficient mice but not in mast cell-deficient mice.
Topics: Animals; Dimaprit; Endothelial Growth Factors; Gossypium; Granulation Tissue; Histamine; Histamine Agonists; Histidine Decarboxylase; Lymphokines; Male; Mast Cells; Mice; Mice, Inbred Strains; Mice, Knockout; Neovascularization, Pathologic; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors | 2002 |
Further evidence for the involvement of histamine H2 receptors in the control of defensive behaviour generated in the midbrain tectum.
Topics: Animals; Arousal; Brain Mapping; Dimaprit; Escape Reaction; Fear; Histamine; Inferior Colliculi; Male; Microinjections; Periaqueductal Gray; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine H2 | 2002 |
Effects of histamine on the contractile and electrical activity in isolated lymphatic vessels of the guinea-pig mesentery.
Topics: Animals; Dimaprit; Dose-Response Relationship, Drug; Endothelium, Lymphatic; Female; Guinea Pigs; Histamine; Histamine Agonists; In Vitro Techniques; Lymphatic System; Male; Membrane Potentials; Mesentery; Methylhistamines; Muscle Contraction; Muscle, Smooth; Nitric Oxide; Nitroarginine; Receptors, Histamine H2; Receptors, Histamine H3 | 2002 |
Histamine h(4) and h(2) receptors control histamine-induced interleukin-16 release from human CD8(+) T cells.
Topics: Base Sequence; CD4-Positive T-Lymphocytes; CD8-Positive T-Lymphocytes; Cells, Cultured; Cimetidine; Dimaprit; DNA Primers; Female; Gene Expression Regulation; Histamine; Humans; Interleukin-16; Male; Methylhistamines; Polymerase Chain Reaction; Pyrilamine; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H2; Receptors, Histamine H4 | 2002 |
Excitatory effects of histamine on cerebellar interpositus nuclear cells of rats through H(2) receptors in vitro.
Topics: Animals; Cerebellar Nuclei; Dimaprit; Dose-Response Relationship, Drug; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Neurons; Ranitidine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H1; Receptors, Histamine H2; Triprolidine | 2002 |
Endogenous central histamine-induced reversal of critical haemorrhagic hypotension in rats--studies with histamine N-methyltransferase inhibitor SKF 91488.
Topics: Animals; Blood Pressure; Brain Chemistry; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Heart Rate; Histamine; Histamine Antagonists; Histamine N-Methyltransferase; Hypotension; Injections, Intraventricular; Male; Rats; Rats, Wistar; Shock, Hemorrhagic; Survival | 2002 |
Characteristics of histamine tachyphylaxis in rat uterine smooth muscle.
Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Cyclic AMP; Dimaprit; Dose-Response Relationship, Drug; Epinephrine; Estrogens; Female; Histamine; Histamine Agonists; In Vitro Techniques; Isotonic Contraction; Muscle Relaxation; Rats; Rats, Wistar; Tachyphylaxis; Uterine Contraction; Uterus | 2002 |
Differential activation of dual signaling responses by human H1 and H2 histamine receptors.
Topics: Calcium Signaling; Cell Line; Colforsin; Cyclic AMP; Dimaprit; Histamine; Histamine Agonists; Humans; Kinetics; Receptors, Histamine H1; Receptors, Histamine H2; Recombinant Proteins; Signal Transduction; Transfection | 2003 |
Blockade of histamine H2 receptors of the periaqueductal gray and inferior colliculus induces fear-like behaviors.
Topics: Animals; Behavior, Animal; Dimaprit; Exploratory Behavior; Fear; Histamine; Histamine Agonists; Histamine H2 Antagonists; Inferior Colliculi; Male; Mesencephalon; Microinjections; Periaqueductal Gray; Ranitidine; Rats; Rats, Wistar | 2003 |
The histamine H2-receptor antagonist, cimetidine, inhibits the articular osteopenia in rats with adjuvant-induced arthritis by suppressing the osteoclast differentiation induced by histamine.
Topics: Animals; Arthritis, Experimental; Bone Density; Bone Resorption; Cartilage, Articular; Cell Differentiation; Cimetidine; Dimaprit; Female; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Osteoclasts; Pyrilamine; Rats; Rats, Inbred Lew | 2003 |
Histamine downregulates CD14 expression via H2 receptors on human monocytes.
Topics: Cells, Cultured; Dimaprit; Down-Regulation; Histamine; Histamine Agonists; Histamine H2 Antagonists; Humans; Leukocytes, Mononuclear; Lipopolysaccharide Receptors; Lipopolysaccharides; Methylhistamines; Monocytes; Receptors, Histamine H2; Time Factors; Tumor Necrosis Factor-alpha | 2003 |
Histaminergic receptors modulate the coronary vascular response in isolated guinea pig hearts. Role of nitric oxide.
Topics: Animals; Bradykinin; Coronary Circulation; Coronary Vessels; Dimaprit; Guinea Pigs; Heart; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Myocardium; Nitrates; Nitric Oxide; Nitric Oxide Synthase; Perfusion; Receptors, Histamine | 2003 |
Effects of activation of central nervous histamine receptors in cardiovascular regulation; studies in H(1) and H(2) receptor gene knockout mice.
Topics: Animals; Blood Pressure; Central Nervous System; Dimaprit; Heart Rate; Histamine; Histamine Agonists; Imidazoles; Injections, Spinal; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Piperidines; Receptors, Histamine | 2005 |
The protective effect of H2-receptor activation against the duration of myocardial hypoxia/reoxygenation-induced ventricular fibrillation in sensitized guinea-pig hearts.
Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Cytoplasmic Granules; Dimaprit; Electrocardiography; Enzyme Inhibitors; Female; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Histamine N-Methyltransferase; Histamine Release; Immunoglobulin E; In Vitro Techniques; Mast Cells; Myocardial Reperfusion Injury; Perfusion; Receptors, Histamine H2; Ventricular Fibrillation | 2005 |
Histamine excites neonatal rat sympathetic preganglionic neurons in vitro via activation of H1 receptors.
Topics: Action Potentials; Animals; Animals, Newborn; Autonomic Fibers, Preganglionic; Barium; Dimaprit; Female; Ganglia, Sympathetic; Histamine; Histamine Agonists; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Potassium; Rats; Rats, Inbred WKY; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiourea; Triprolidine | 2006 |
Histamine signaling through the H(2) receptor in the Peyer's patch is important for controlling Yersinia enterocolitica infection.
Topics: Animals; Anti-Allergic Agents; Anti-Ulcer Agents; Cimetidine; Dimaprit; Female; Gene Expression Profiling; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine Decarboxylase; Mice; Mice, Inbred C57BL; Oligonucleotide Array Sequence Analysis; Omeprazole; Peyer's Patches; Pyrilamine; Receptors, Histamine H2; Signal Transduction; Survival Rate; Yersinia enterocolitica; Yersinia Infections | 2006 |
Suppression of ischemia/reperfusion liver injury by histamine H4 receptor stimulation in rats.
Topics: Alanine Transaminase; Animals; Aspartate Aminotransferases; Clozapine; Dimaprit; Dose-Response Relationship, Drug; Histamine; Ischemia; Liver; Male; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Reperfusion Injury; Time Factors | 2006 |
Blockade of brain histamine metabolism alters methamphetamine-induced expression pattern of stereotypy in mice via histamine H1 receptors.
Topics: Analysis of Variance; Animals; Behavior, Animal; Brain; Dimaprit; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Histamine; Histamine Agents; Male; Maze Learning; Methamphetamine; Mice; Mice, Inbred ICR; Motor Activity; Receptors, Histamine H1; Stereotyped Behavior | 2007 |
The anti-secretory and anti-ulcer activities of esomeprazole in comparison with omeprazole in the stomach of rats and rabbits.
Topics: Aminopyrine; Animals; Anti-Ulcer Agents; Bucladesine; Carbon Isotopes; Dimaprit; Dinoprostone; Esomeprazole; Female; Gastric Acid; Gastric Mucosa; Histamine; Indomethacin; Inhibitory Concentration 50; Male; Omeprazole; Rabbits; Rats; Rats, Wistar; Stomach | 2008 |
Suppression of ischaemia-induced cytokine release by dimaprit and amelioration of liver injury in rats.
Topics: Adenosine Triphosphate; Alanine Transaminase; Animals; Aspartate Aminotransferases; Cytokines; Dimaprit; Disease Models, Animal; Down-Regulation; Hepatic Artery; Histamine; Histamine Agonists; Interleukin-12; Ischemia; Ligation; Liver; Male; Portal Vein; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H2; Receptors, Histamine H4; Reperfusion Injury; Severity of Illness Index; Time Factors | 2008 |
Histamine metabolism influences blood vessel branching in zebrafish reg6 mutants.
Topics: Animals; Blood Vessels; Cell Movement; Dimaprit; Early Growth Response Protein 1; Embryo, Nonmammalian; Endothelium, Vascular; Histamine; Histamine N-Methyltransferase; Mutation; Neovascularization, Physiologic; Phenotype; Regeneration; Suppression, Genetic; Zebrafish | 2008 |
Activation of adenosine low-affinity A3 receptors inhibits the enteric short interplexus neural circuit triggered by histamine.
Topics: Adenosine; Animals; Chlorides; Cimetidine; Colon; Dihydropyridines; Dimaprit; Dose-Response Relationship, Drug; Enteric Nervous System; Gastrointestinal Motility; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; In Vitro Techniques; Intestinal Secretions; Male; Mecamylamine; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Neural Inhibition; Neurogenic Bowel; Neurokinin-1 Receptor Antagonists; Nicotinic Antagonists; Piperidines; Propane; Receptor, Adenosine A1; Receptor, Adenosine A3; Receptors, Histamine H2; Receptors, Neurokinin-1; Reflex; Theophylline; Xanthines | 2009 |
In vivo electrochemical evidence for simultaneous 5-HT and histamine release in the rat substantia nigra pars reticulata following medial forebrain bundle stimulation.
Topics: Animals; Dimaprit; Electric Stimulation; Electrochemistry; Histamine; Histamine Agonists; Histamine H3 Antagonists; Linear Models; Male; Medial Forebrain Bundle; Neural Pathways; Piperidines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Serotonin; Substantia Nigra | 2011 |
Histamine evokes excitatory response of neurons in the cerebellar dentate nucleus via H2 receptors.
Topics: Animals; Cell Movement; Cerebellar Nuclei; Dimaprit; Excitatory Postsynaptic Potentials; Histamine; Histamine Agonists; Hypothalamic Area, Lateral; Neural Pathways; Neurons; Organ Culture Techniques; Rats; Rats, Sprague-Dawley; Receptors, Histamine H2 | 2011 |
Histaminergic modulation of acetylcholine-induced γ oscillations in rat hippocampus.
Topics: Acetylcholine; Animals; Attention; Cholinesterase Inhibitors; Cimetidine; Dimaprit; Electroencephalography; Hippocampus; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine Release; Hypoxia, Brain; In Vitro Techniques; Male; Microelectrodes; Physostigmine; Pyramidal Tracts; Rats; Rats, Wistar; Terfenadine | 2011 |
Excitatory effect of histamine on rat spinal motoneurons by activation of both H₁ and H₂ receptors in vitro.
Topics: Action Potentials; Analysis of Variance; Animals; Animals, Newborn; Biophysics; Calcium Channel Blockers; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine H2 Antagonists; In Vitro Techniques; Motor Neurons; Patch-Clamp Techniques; Pyridines; Ranitidine; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Spinal Cord; Tetrodotoxin | 2012 |
Loss of histaminergic modulation of thermoregulation and energy homeostasis in obese mice.
Topics: Adipose Tissue, Brown; Animals; Body Temperature Regulation; Dimaprit; Eating; Energy Metabolism; Histamine; Histamine Agonists; Homeostasis; Mice; Mice, Obese; Obesity; Preoptic Area; Receptors, Histamine | 2012 |
Histamine excites rat superior vestibular nuclear neurons via postsynaptic H1 and H2 receptors in vitro.
Topics: Action Potentials; Animals; Dimaprit; Female; Histamine; Histamine Agonists; Male; Neurons; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Histamine H1; Receptors, Histamine H2; Vestibular Nuclei | 2013 |
Histamine infused into basolateral amygdala enhances memory consolidation of inhibitory avoidance.
Topics: Amygdala; Analysis of Variance; Animals; Avoidance Learning; Dimaprit; Exploratory Behavior; Histamine; Histamine Agonists; Histamine Antagonists; Male; Maze Learning; Memory; Rats; Rats, Wistar; Reaction Time; Statistics, Nonparametric | 2013 |
Role of histamine receptors in the effects of histamine on the production of reactive oxygen species by whole blood phagocytes.
Topics: Benzimidazoles; Dimaprit; Guanidines; Histamine; Histamine Agonists; Humans; Male; Methylhistamines; Phagocytes; Reactive Oxygen Species; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H2; Receptors, Histamine H4; Thiourea | 2014 |
Histamine acting on the basolateral amygdala reverts the impairment of aversive memory of rats submitted to neonatal maternal deprivation.
Topics: Analysis of Variance; Animals; Avoidance Learning; Basolateral Nuclear Complex; Dimaprit; Disease Models, Animal; Dose-Response Relationship, Drug; Exploratory Behavior; Female; Histamine; Histamine Agonists; Histamine Antagonists; Inhibition, Psychological; Male; Maternal Deprivation; Maze Learning; Memory Disorders; Pregnancy; Rats; Rats, Wistar | 2015 |
Ligands of histamine receptors modulate acid-sensing ion channels.
Topics: Acid Sensing Ion Channels; Animals; CHO Cells; Cricetulus; Dimaprit; Gene Expression Regulation; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Hydrogen-Ion Concentration; Ligands; Methylhistamines; Patch-Clamp Techniques; Piperidines; Receptors, Histamine; Recombinant Proteins; Signal Transduction | 2017 |
Histamine Excites Rat GABAergic Ventral Pallidum Neurons via Co-activation of H1 and H2 Receptors.
Topics: Action Potentials; Animals; Basal Forebrain; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Female; GABAergic Neurons; gamma-Aminobutyric Acid; Histamine; Histamine Agonists; Lysine; Male; Patch-Clamp Techniques; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Histamine H1; Receptors, Histamine H2; Sodium Channel Blockers; Tetrodotoxin | 2018 |
Human histamine H
Topics: Animals; Arrhythmias, Cardiac; Cimetidine; Dimaprit; Disease Models, Animal; Heart Atria; Heart Ventricles; Histamine; Humans; Mice; Mice, Transgenic; Receptors, Histamine H2; Signal Transduction | 2021 |
Selective histamine H
Topics: Angiopoietin-1; Animals; Blood-Brain Barrier; Brain Injuries, Traumatic; Dimaprit; Endothelial Cells; Evans Blue; Hedgehog Proteins; Histamine; Histamine Agonists; Male; Mice; Protective Factors; Ranitidine; Receptors, Histamine H2; RNA, Messenger; Thiazoles | 2022 |