dimaprit and burimamide

dimaprit has been researched along with burimamide in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19901 (16.67)18.7374
1990's3 (50.00)18.2507
2000's1 (16.67)29.6817
2010's1 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Timmerman, H1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Buschauer, A; Dove, S; Igel, P1
Brink, C; Gorenne, I; Labat, C; Norel, X; Ortiz, JL; Verley, J1
Clark, MA; Egan, RW; Shih, NY; Siegel, MI; West, RE; Zweig, A1
Bianucci, AM; Da Settimo, A; Martinelli, A1

Reviews

1 review(s) available for dimaprit and burimamide

ArticleYear
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship

1990

Other Studies

5 other study(ies) available for dimaprit and burimamide

ArticleYear
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Histamine H4 receptor agonists.
    Bioorganic & medicinal chemistry letters, 2010, Dec-15, Volume: 20, Issue:24

    Topics: Animals; Benzimidazoles; Binding Sites; Clozapine; Guanidines; Humans; Ligands; Mice; Oximes; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Structure-Activity Relationship

2010
Histamine receptors on human isolated pulmonary arterial muscle preparations: effects of endothelial cell removal and nitric oxide inhibitors.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:2

    Topics: Arginine; Burimamide; Chlorpheniramine; Cimetidine; Dimaprit; Endothelium, Vascular; Histamine; Humans; In Vitro Techniques; Indomethacin; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Nitroarginine; omega-N-Methylarginine; Pulmonary Artery; Receptors, Histamine; Serotonin; Tetraethylammonium; Tetraethylammonium Compounds; Thiourea

1992
Identification of two H3-histamine receptor subtypes.
    Molecular pharmacology, 1990, Volume: 38, Issue:5

    Topics: Animals; Binding Sites; Binding, Competitive; Brain Chemistry; Burimamide; Dimaprit; Guanidines; Guanosine 5'-O-(3-Thiotriphosphate); Histamine; Imidazoles; Impromidine; Male; Methylhistamines; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H3; Thiourea; Tritium

1990
A conformational approach to histamine H2-receptor antagonists.
    Il Farmaco; edizione scientifica, 1984, Volume: 39, Issue:8

    Topics: Animals; Burimamide; Cimetidine; Dimaprit; Guinea Pigs; Histamine H2 Antagonists; Hydrogen-Ion Concentration; Metiamide; Molecular Conformation; Structure-Activity Relationship; Thiourea

1984