dimaprit and alpha-methylhistamine

dimaprit has been researched along with alpha-methylhistamine in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's13 (52.00)18.2507
2000's10 (40.00)29.6817
2010's2 (8.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bull, HA; Courtney, PF; Dowd, PM; Rustin, MH1
Kohno, S; Nabe, T; Nakao, S; Ogawa, K; Ohata, K; Yamamura, H1
Bynum, TE; Kronauge, JF; Morales, RE; Palitzsch, KD; Szabo, S1
Carson, CC; Davies, MG; Hagen, PO; Kim, YC; Lee, TH1
Luo, XX; Tan, YH1
Malinowska, B; Schlicker, E1
Blandina, P; Cecchi, M; Giorgetti, M; Giovannini, MG; Leurs, R; Timmerman, H1
Chiyotani, A; Konno, K; Nakata, J; Takeyama, K; Tamaoki, J1
Bartolini, A; Ghelardini, C; Hänninen, J; Ipponi, A; Lamberti, C; Malmberg-Aiello, P1
Ballabeni, V; Barocelli, E; Bordi, F; Caretta, A; Carrupt, PA; Crivori, P; Impicciatore, M; Mor, M; Plazzi, PV; Rivara, S; Silva, C; Testa, B1
Fu, LW; Longhurst, JC; Pan, HL1
Akaike, N; Ishibashi, H; Munakata, M; Sakata, T; Takeshita, Y; Watanabe, T1
Gao, C; Hu, Hz; Liu, S; Ren, J; Wood, JD; Xia, Y1
Kawarai, M; Koss, MC; Yu, Y1
Fox, JL; von der Weid, PY1
Bacon, KB; Center, DM; Cruikshank, WW; Gantner, F; Sakai, K; Tusche, MW1
Bocheva, A; Dobrinova, Y; Todorov, S; Zamfirova, R1
Korosteleva, AS; Potapieva, NN; Shteinikov, VY; Tikhonov, DB; Tikhonova, TB1
Timmerman, H1
Blevitt, J; Carruthers, N; Chai, W; Hofstra, CL; Jiang, X; Li, X; Liu, C; Lovenberg, TW; Ma, X; Pyati, J; Wilson, SJ1
Alston, J; Ames, RS; Bergsma, DJ; Boyce, R; Davenport, CM; Dytko, GM; Fitzgerald, LR; Herrity, NC; Hieble, JP; Li, X; Mannan, IJ; Michalovich, D; Sarau, HM; Tan, KB; Tierney, LA; Vawter, L; Wilson, S; Wu, H; Zhu, Y1
Anthes, JC; Bayne, M; Behan, J; Gonsiorek, W; Greene, J; Greenfeder, SA; Gustafson, EL; Hedrick, JA; Hipkin, RW; Laz, TM; Monsma, FJ; Morse, KL; Qiao, X; Shin, N; Umland, S; Wan, Y; Wang, S; West, RE1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Falus, A; Jelinek, I; Keseru, GM; Kiss, B; Kiss, R; Könczöl, A; László, V; Noszál, B; Szalai, F1
Buschauer, A; Dove, S; Igel, P1

Reviews

1 review(s) available for dimaprit and alpha-methylhistamine

ArticleYear
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship

1990

Other Studies

24 other study(ies) available for dimaprit and alpha-methylhistamine

ArticleYear
Characterization of histamine receptor sub-types regulating prostacyclin release from human endothelial cells.
    British journal of pharmacology, 1992, Volume: 107, Issue:2

    Topics: Cells, Cultured; Dimaprit; Endothelium, Vascular; Epoprostenol; Histamine; Histamine Agonists; Humans; Impromidine; Methylhistamines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Thiazoles; Umbilical Veins

1992
Possible participation of histamine H3-receptors in the regulation of anaphylactic histamine release from isolated rat peritoneal mast cells.
    Japanese journal of pharmacology, 1994, Volume: 66, Issue:2

    Topics: Anaphylaxis; Animals; Anticonvulsants; Chromatography, High Pressure Liquid; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Histamine; Histamine Agonists; Histamine Antagonists; Histamine Release; In Vitro Techniques; L-Lactate Dehydrogenase; Male; Mast Cells; Methylhistamines; p-Methoxy-N-methylphenethylamine; Peritoneal Cavity; Peritoneum; Piperidines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H3

1994
Effect of histamine on haemorrhagic mucosal lesions is related to vascular permeability in rats: studies with histamine, H1-, H2- and H3-agonists and bradykinin.
    European journal of gastroenterology & hepatology, 1995, Volume: 7, Issue:5

    Topics: Absorption; Animals; Betahistine; Bradykinin; Capillary Permeability; Dimaprit; Dose-Response Relationship, Drug; Ethanol; Female; Gastric Mucosa; Gastrointestinal Hemorrhage; Histamine; Histamine Agonists; Injections, Subcutaneous; Intubation, Gastrointestinal; Methylhistamines; Organotechnetium Compounds; Rats; Rats, Sprague-Dawley; Stomach Diseases; Sugar Acids

1995
Characterization and function of histamine receptors in corpus cavernosum.
    The Journal of urology, 1995, Volume: 153, Issue:2

    Topics: Acetylcholine; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Papaverine; Penis; Piperidines; Pyrilamine; Rabbits; Receptors, Histamine; Thiazoles

1995
Presynaptic histamine H1- and H3-receptors modulate sympathetic neurotransmission in isolated guinea pig vas deferens.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1994, Volume: 15, Issue:1

    Topics: Animals; Chlorpheniramine; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; Piperidines; Ranitidine; Sympathetic Nervous System; Synaptic Transmission; Vas Deferens

1994
Identification of endothelial H1, vascular H2 and cardiac presynaptic H3 receptors in the pithed rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1993, Volume: 347, Issue:1

    Topics: Animals; Blood Pressure; Blood Vessels; Cardiovascular System; Dimaprit; Electric Stimulation; Endothelium, Vascular; Heart Rate; Histamine Agonists; Male; Methylhistamines; Myocardium; Rats; Rats, Wistar; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Thiazoles

1993
Histamine H3 receptor inhibition of K(+)-evoked release of acetylcholine from rat cortex in vivo.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1996, Volume: 45 Suppl 1

    Topics: Acetylcholine; Analysis of Variance; Animals; Chromatography, High Pressure Liquid; Dimaprit; Histamine; Histamine Agonists; Histamine Antagonists; Male; Methylhistamines; Microdialysis; Neurons; Parietal Lobe; Piperidines; Potassium; Rats; Rats, Wistar; Receptors, Histamine H3; Thiazoles

1996
Histamine H2 receptor-mediated airway goblet cell secretion and its modulation by histamine-degrading enzymes.
    The Journal of allergy and clinical immunology, 1997, Volume: 99, Issue:2

    Topics: Amine Oxidase (Copper-Containing); Animals; Asthma; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glycoproteins; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine N-Methyltransferase; Male; Methylhistamines; Mucus; Piperidines; Pyrilamine; Recombinant Proteins; Trachea

1997
Effects of two histamine-N-methyltransferase inhibitors, SKF 91488 and BW 301 U, in rodent antinociception.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 355, Issue:3

    Topics: Analgesics; Animals; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Folic Acid Antagonists; Histamine Agonists; Histamine N-Methyltransferase; Injections, Intraventricular; Male; Methylhistamines; Mice; Muscle Contraction; Pain Measurement; Postural Balance; Psychomotor Performance; Pyrimidines; Rats; Rats, Wistar

1997
H3-receptor antagonists: synthesis and structure-activity relationships of para- and meta-substituted 4(5)-phenyl-2-[[2-[4(5)-imidazolyl]ethyl]thio]imidazoles.
    Journal of medicinal chemistry, 1997, Aug-01, Volume: 40, Issue:16

    Topics: Animals; Binding, Competitive; Cerebral Cortex; Dimaprit; Electric Stimulation; Evoked Potentials; Guinea Pigs; Histamine Antagonists; Ileum; Imidazoles; Methylhistamines; Rats; Rats, Wistar; Receptors, Histamine H3; Structure-Activity Relationship

1997
Endogenous histamine stimulates ischemically sensitive abdominal visceral afferents through H1 receptors.
    The American journal of physiology, 1997, Volume: 273, Issue:6

    Topics: Abdomen; Afferent Pathways; Animals; Bile Ducts; Blood Pressure; Cats; Chlorpheniramine; Dimaprit; Duodenum; Female; Gallbladder; Histamine; Histamine H1 Antagonists; Indomethacin; Ischemia; Male; Methylhistamines; Nerve Fibers; Neural Conduction; Pancreas; Pyrilamine; Receptors, Histamine H1

1997
Histamine modulates high-voltage-activated calcium channels in neurons dissociated from the rat tuberomammillary nucleus.
    Neuroscience, 1998, Volume: 87, Issue:4

    Topics: Animals; Calcium; Calcium Channels; Calcium Channels, N-Type; Depression, Chemical; Dimaprit; Histamine; Histamine Agonists; Histamine Antagonists; Ion Channel Gating; Mammillary Bodies; Methylhistamines; Nerve Tissue Proteins; Neurons; Nicardipine; omega-Agatoxin IVA; omega-Conotoxin GVIA; omega-Conotoxins; Patch-Clamp Techniques; Peptides; Pertussis Toxin; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; Spider Venoms; Tuber Cinereum; Virulence Factors, Bordetella

1998
Histamine H3 receptor-mediated suppression of inhibitory synaptic transmission in the submucous plexus of guinea-pig small intestine.
    European journal of pharmacology, 2000, May-26, Volume: 397, Issue:1

    Topics: Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Intestine, Small; Male; Methylhistamines; Norepinephrine; Phentolamine; Piperidines; Receptors, Histamine H3; Submucous Plexus; Synaptic Transmission

2000
Histamine H3 receptor-mediated inhibition of sympathetically evoked mydriasis in rats.
    European journal of pharmacology, 2001, May-04, Volume: 419, Issue:1

    Topics: Animals; Chlorpheniramine; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Male; Methylhistamines; Mydriasis; Pupil; Rats; Rats, Sprague-Dawley; Sympathetic Nervous System; Thiourea

2001
Effects of histamine on the contractile and electrical activity in isolated lymphatic vessels of the guinea-pig mesentery.
    British journal of pharmacology, 2002, Volume: 136, Issue:8

    Topics: Animals; Dimaprit; Dose-Response Relationship, Drug; Endothelium, Lymphatic; Female; Guinea Pigs; Histamine; Histamine Agonists; In Vitro Techniques; Lymphatic System; Male; Membrane Potentials; Mesentery; Methylhistamines; Muscle Contraction; Muscle, Smooth; Nitric Oxide; Nitroarginine; Receptors, Histamine H2; Receptors, Histamine H3

2002
Histamine h(4) and h(2) receptors control histamine-induced interleukin-16 release from human CD8(+) T cells.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 303, Issue:1

    Topics: Base Sequence; CD4-Positive T-Lymphocytes; CD8-Positive T-Lymphocytes; Cells, Cultured; Cimetidine; Dimaprit; DNA Primers; Female; Gene Expression Regulation; Histamine; Humans; Interleukin-16; Male; Methylhistamines; Polymerase Chain Reaction; Pyrilamine; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H2; Receptors, Histamine H4

2002
Study on the antinociceptive action of Tyr-K-MIF-1, a peptide from the MIF family.
    Autonomic & autacoid pharmacology, 2007, Volume: 27, Issue:2

    Topics: Analgesics; Animals; Dimaprit; Diphenhydramine; Famotidine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; MSH Release-Inhibiting Hormone; Naloxone; Narcotic Antagonists; Pain Measurement; Pain Threshold; Rats; Rats, Wistar

2007
Ligands of histamine receptors modulate acid-sensing ion channels.
    Biochemical and biophysical research communications, 2017, 09-02, Volume: 490, Issue:4

    Topics: Acid Sensing Ion Channels; Animals; CHO Cells; Cricetulus; Dimaprit; Gene Expression Regulation; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Hydrogen-Ion Concentration; Ligands; Methylhistamines; Patch-Clamp Techniques; Piperidines; Receptors, Histamine; Recombinant Proteins; Signal Transduction

2017
Cloning and pharmacological characterization of a fourth histamine receptor (H(4)) expressed in bone marrow.
    Molecular pharmacology, 2001, Volume: 59, Issue:3

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Bone Marrow; Cloning, Molecular; Histamine; Humans; Methylhistamines; Molecular Sequence Data; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; RNA, Messenger; Sequence Homology, Amino Acid; Tissue Distribution; Tritium

2001
Cloning, expression, and pharmacological characterization of a novel human histamine receptor.
    Molecular pharmacology, 2001, Volume: 59, Issue:3

    Topics: Amino Acid Sequence; Animals; Calcium; Cloning, Molecular; Dose-Response Relationship, Drug; Gene Expression; Genes, Reporter; Histamine; Humans; Luciferases; Mice; Molecular Sequence Data; Radioligand Assay; Receptors, Histamine; Receptors, Histamine H3; Sequence Homology, Amino Acid; Tissue Distribution; Tritium

2001
Cloning and characterization of a novel human histamine receptor.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 296, Issue:3

    Topics: Amino Acid Sequence; Cells, Cultured; Cloning, Molecular; Histamine; Histamine Agonists; Humans; Imidazoles; Molecular Sequence Data; Radioligand Assay; Receptors, Histamine; Receptors, Histamine H3; RNA, Messenger; Sequence Homology, Amino Acid; Thiourea; Tissue Distribution; Transfection

2001
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Discovery of novel human histamine H4 receptor ligands by large-scale structure-based virtual screening.
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Binding, Competitive; Cell Line, Tumor; Databases, Factual; Histamine Antagonists; Humans; Ligands; Models, Molecular; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Structure-Activity Relationship

2008
Histamine H4 receptor agonists.
    Bioorganic & medicinal chemistry letters, 2010, Dec-15, Volume: 20, Issue:24

    Topics: Animals; Benzimidazoles; Binding Sites; Clozapine; Guanidines; Humans; Ligands; Mice; Oximes; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Structure-Activity Relationship

2010