dilazep has been researched along with adenosine in 80 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 41 (51.25) | 18.7374 |
1990's | 28 (35.00) | 18.2507 |
2000's | 7 (8.75) | 29.6817 |
2010's | 3 (3.75) | 24.3611 |
2020's | 1 (1.25) | 2.80 |
Authors | Studies |
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Heitman, LH; IJzerman, AP; Vlachodimou, A | 1 |
Nakanishi, H; Ohtaki, Y; Ueda, J | 1 |
Kolassa, N; Stengg, R; Turnheim, K | 1 |
Blum, KU; Merkel, R | 1 |
Hori, H; Kondo, S; Shirasawa, Y; Tamura, H | 1 |
Coleman, RA | 1 |
Cass, CE; Janowska-Wieczorek, A; King, KM; Montaño, JT | 1 |
Cushing, DJ; Makujina, SR; Mustafa, SJ; Sabouni, MH | 1 |
Lautt, WW; Zhang, Y | 2 |
Gero, AM; Wood, AM | 1 |
Van Belle, H; Ver Donck, KL; Verheyen, WJ | 1 |
Baer, HP; Moorji, A; Serignese, V; Van Belle, H | 1 |
Geiger, JD; Lautt, WW; Legare, DJ; Zhang, Y | 2 |
al-Jaser, MH; Baer, HP; Ogbunude, PO | 1 |
Baer, HP; el-Soofi, A; Haq, A; Paterson, AR; Serignese, V | 1 |
Baer, HP; Ogbunude, PO | 1 |
Baer, HP; Moorji, A | 1 |
Franklin, PH; Murray, TF; Zhang, G | 1 |
Barraco, RA; DeLong, RE; Phillis, JW; Washington, DO | 1 |
Barrett, J; Beechey, RB; Harris, DI; Linstead, D | 1 |
Clark, M; Dar, MS | 2 |
Meghji, P; Rubio, R; Tuttle, JB | 1 |
Gero, AM | 1 |
Agarwal, KC; Maitra, RS; Zielinski, BA | 1 |
Gustafsson, LE | 1 |
Agarwal, KC; Buckley, RS; Parks, RE | 1 |
Berne, RM; Meghji, P; Rubio, R | 1 |
Geiger, JD; Johnston, ME | 1 |
Agarwal, KC; Dawicki, DD; Parks, RE | 3 |
Gudenzi, M; Mustafa, SJ; Nakagawa, Y | 3 |
Mustafa, SJ; Nakagawa, Y | 1 |
Hassall, CJ; Meghji, P; Middleton, K; Newby, AC; Phillips, MI | 1 |
Burnstock, G; Centelles, JJ; Franco, R; Hoyle, CH | 1 |
Geiger, JD; Johnston, ME; Yago, V | 1 |
Plagemann, PG | 1 |
Cha, S; el Kouni, MH | 1 |
Cha, S; el Kouni, MH; Messier, NJ | 1 |
Uchida, Y; Yoshinaka, Y | 1 |
Acampora, R; Filippelli, A; Iarussi, D; Lampa, E; Marmo, E; Matera, C; Soreca, S; Tortora, G | 1 |
Sanderson, G; Scholfield, CN | 1 |
Fredholm, BB; Hedqvist, P; Lindström, K; Wennmalm, M | 1 |
D'Angelo, L; Manzo, L; Marcoli, M; Onori, L; Perucca, E; Saltarelli, P; Tonini, M | 1 |
Kobayashi, A; Ogawa, K; Yamazaki, N | 1 |
Cass, CE; Harley, ER; Paterson, AR | 1 |
Haraoka, S; Kusachi, S; Nagashima, H; Saito, D | 1 |
Fredholm, BB; Lerner, U | 1 |
Fredholm, BB; Sollevi, A | 2 |
Fujita, S; Ishida, Y; Izumi, K; Moritoki, H; Ohara, M; Takei, M | 1 |
Delander, GE; Keil, GJ | 1 |
Gero, AM; Upston, JM | 1 |
Sasvari-Szekely, M; Solymossy, M; Staub, M; Szikla, K | 1 |
Foga, IO; Geiger, JD; Gu, JG; Parkinson, FE | 1 |
Lautt, WW; Zhang, YL | 1 |
Geiger, JD; Gu, JG; Kala, G | 1 |
Cass, CE; Fang, X; Mowles, DA; Parkinson, FE; Young, JD | 1 |
Geiger, JD; Gu, JG; Nath, A | 1 |
Geiger, JD; Mukherjee, K; Parkinson, FE | 1 |
Abiko, Y; Hara, A; Hashizume, H | 1 |
Guo, X; Kulkarni, JS; Palmer, KC; Przywara, DA; Wakade, AR; Wakade, TD | 1 |
Deguchi, H; Gabazza, EC; Hayashi, N; Suzuki, K; Takeya, H; Urano, H; Wada, H | 1 |
Delaney, SM; Geiger, JD | 1 |
Funaya, H; Hori, M; Kitakaze, M; Komamura, K; Koretsune, Y; Kuzuya, T; Minamino, T; Node, K | 1 |
Camarasa, J; Camins, A; Escubedo, E; Jiménez, A; Lladó, S; Pallàs, M; Pubill, D | 1 |
Bilan, PJ; Coe, IR; Shuralyova, I; Sweeney, G; Tajmir, P | 1 |
Endres, CJ; Sengupta, DJ; Unadkat, JD | 1 |
Day, A; Lawrence, AJ; Ledent, C; Snell, BJ | 1 |
Baldwin, SA; Cass, CE; Raborn, RT; Visser, F; Young, JD; Zhang, J | 1 |
Baldwin, SA; Cass, CE; Damaraju, V; Peng, Y; Robins, MJ; Sun, L; Tackaberry, T; Visser, F; Young, JD | 1 |
Baldwin, SA; Cass, CE; Damaraju, V; Paproski, RJ; Tackaberry, T; Visser, F; Young, JD; Zhang, J | 1 |
Glaumann, C; Grishina, VA; Gustafsson, LE; Nilsson, KF | 1 |
Lee, SY; Wright, NJ | 1 |
Fasching, A; Palm, F; Persson, P; Pihl, L | 1 |
1 trial(s) available for dilazep and adenosine
Article | Year |
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Elevation of plasma adenosine levels may attenuate the severity of chronic heart failure.
Topics: Adenosine; Adult; Aged; Cardiac Output, Low; Chronic Disease; Dilazep; Dipyridamole; Humans; Middle Aged; Prognosis; Vasodilator Agents | 1998 |
79 other study(ies) available for dilazep and adenosine
Article | Year |
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Label-free detection of transporter activity via GPCR signalling in living cells: A case for SLC29A1, the equilibrative nucleoside transporter 1.
Topics: Cell Line, Tumor; Equilibrative Nucleoside Transporter 1; Humans; Ligands; Membrane Transport Proteins; Osteosarcoma; Receptors, G-Protein-Coupled; Receptors, Purinergic P1; Signal Transduction | 2019 |
[Effects of adenosine compounds of the vascular bed and effects of dilazep, theophylline, and indomethacin on blood flow changes of the postocclusive renal vessels].
Topics: Adenine Nucleotides; Adenosine; Angiotensin II; Animals; Azepines; Blood Flow Velocity; Blood Vessels; Dilazep; Dogs; Drug Synergism; Female; Femoral Artery; Indomethacin; Kidney; Ligation; Male; Mesenteric Arteries; Norepinephrine; Renal Artery; Theophylline | 1977 |
Influence of hexobendine, dipyridamole, dilazep, lidoflazine, inosine and purine riboside on adenosine uptake by the isolated epithelium of guinea pig jejunum.
Topics: Adenosine; Animals; Dilazep; Dipyridamole; Epithelium; Guinea Pigs; Hexobendine; Inosine; Intestinal Absorption; Jejunum; Lidoflazine; Piperazines; Purines; Vasodilator Agents | 1978 |
[Adenosine degradation in human erythrocytes in the presence of dilazep].
Topics: Adenosine; Adenosine Deaminase; Azepines; Dilazep; Erythrocytes; Humans; Methylene Blue; Oxygen Consumption | 1976 |
[Effects of 1, 4-bis-(3-(3, 4, 5-trimethoxy benzoyl oxy)-propyl) perhydro-1, 4-diazepine (dilazep) on the isolated smooth muscles].
Topics: Adenine Nucleotides; Adenosine; Animals; Aorta; Calcium; Dilazep; Dogs; Dose-Response Relationship, Drug; Female; Guinea Pigs; In Vitro Techniques; Intestines; Male; Muscle Contraction; Muscle, Smooth; Papaverine; Potassium; Rabbits; Rats; Uterus; Vas Deferens | 1975 |
Effects of some purine derivatives on the guinea-pig trachea and their interaction with drugs that block adenosine uptake.
Topics: Adenosine; Adenosine Triphosphate; Animals; Depression, Chemical; Dilazep; Dipyridamole; Drug Interactions; Guinea Pigs; Hexobendine; In Vitro Techniques; Parasympatholytics; Propranolol; Purine Nucleosides; Trachea | 1976 |
A comparison of the abilities of nitrobenzylthioinosine, dilazep, and dipyridamole to protect human hematopoietic cells from 7-deazaadenosine (tubercidin).
Topics: Adenosine; Colony-Forming Units Assay; Dilazep; Dipyridamole; Hematopoietic Stem Cells; Humans; Leukemia, Promyelocytic, Acute; Thioinosine; Tubercidin; Tumor Cells, Cultured | 1992 |
Inhibition of adenylate cyclase attenuates adenosine receptor-mediated relaxation in coronary artery.
Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclase Inhibitors; Animals; Colforsin; Coronary Vessels; Cyclic AMP; Dideoxyadenosine; Dilazep; Guanosine Triphosphate; In Vitro Techniques; Muscle Relaxation; Receptors, Purinergic; Sodium Fluoride; Swine; Vasodilator Agents | 1991 |
Dilazep increases plasma adenosine levels during adenosine infusion in the anesthetized cat.
Topics: Adenosine; Anesthesia; Animals; Cats; Dilazep; Female; Infusions, Intravenous; Male | 1991 |
New nucleoside transport pathways induced in the host erythrocyte membrane of malaria and Babesia infected cells.
Topics: Adenosine; Animals; Babesia bovis; Babesiosis; Biological Transport; Cattle; Cattle Diseases; Dilazep; Drug Therapy, Combination; Erythrocyte Membrane; Erythrocytes; Malaria; Malaria, Falciparum; Mice; Plasmodium falciparum; Pyrimidine Nucleosides; Thioinosine; Thionucleotides; Tubercidin | 1991 |
Nucleoside transport inhibition and fMLP-stimulated whole blood luminescence.
Topics: Adenosine; Biological Transport; Dilazep; Dipyridamole; Humans; Luminescent Measurements; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Piperazines; Respiratory Burst | 1991 |
In vivo effectiveness of several nucleoside transport inhibitors in mice and hamsters.
Topics: Adenosine; Administration, Oral; Animals; Biological Transport; Cardiovascular Agents; Cricetinae; Dilazep; Injections, Intraperitoneal; Mesocricetus; Mice; Mice, Inbred BALB C; Piperazines; Species Specificity; Thioinosine | 1991 |
Dilazep potentiation of adenosine-mediated superior mesenteric arterial vasodilation.
Topics: Adenosine; Animals; Cats; Dilazep; Dose-Response Relationship, Drug; Drug Synergism; Female; Male; Mesenteric Arteries; Receptors, Purinergic; Theophylline; Vasodilator Agents | 1991 |
Leishmania donovani: characteristics of adenosine and inosine transporters in promastigotes of two different strains.
Topics: Adenosine; Animals; Biological Transport; Diffusion; Dilazep; Inosine; Kinetics; Leishmania donovani; Nucleosides; Thioinosine; Thymidine; Uridine | 1991 |
Dilazep-induced vasodilation is mediated through adenosine receptors.
Topics: Adenosine; Animals; Blood Flow Velocity; Blood Pressure; Cats; Chromatography, High Pressure Liquid; Dilazep; Female; Homeostasis; Male; Mesenteric Arteries; Receptors, Purinergic; Theophylline; Vasodilation | 1991 |
Potencies of mioflazine and its derivatives as inhibitors of adenosine transport in isolated erythrocytes from different species.
Topics: Adenosine; Animals; Cricetinae; Dilazep; Dimethyl Sulfoxide; Erythrocytes; Humans; In Vitro Techniques; Male; Mesocricetus; Mice; Mice, Inbred BALB C; Papio; Piperazines; Rabbits; Species Specificity; Thioinosine | 1990 |
Competition of nucleoside transport inhibitors with binding of 6-[(4-nitrobenzyl)-mercapto]purine ribonucleoside to intact erythrocytes and ghost membranes from different species.
Topics: Adenosine; Animals; Binding, Competitive; Carrier Proteins; Cricetinae; Dilazep; Erythrocyte Membrane; Erythrocytes; Hot Temperature; Humans; Hydrogen-Ion Concentration; Inosine; Membrane Proteins; Mice; Nucleoside Transport Proteins; Piperazines; Rats; Thioinosine | 1990 |
Sodium-dependent and inhibitor-insensitive uptake of adenosine by mouse peritoneal exudate cells.
Topics: Adenosine; Animals; Biological Transport, Active; Cell Adhesion; Dilazep; Erythrocytes; In Vitro Techniques; Macrophages; Mice; Mice, Inbred BALB C; Peritoneal Cavity; Sodium; Thioinosine; Time Factors | 1990 |
Anticonvulsant effect of N-ethylcarboxamidoadenosine against kainic acid-induced behavioral seizures in the rat prepiriform cortex.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Dilazep; Kainic Acid; Limbic System; Male; Rats; Rats, Inbred Strains; Seizures; Theophylline | 1990 |
Behavioral characteristics of centrally administered adenosine analogs.
Topics: 1-Methyl-3-isobutylxanthine; Adenosine; Adenosine Deaminase Inhibitors; Animals; Caffeine; Dilazep; Dipyridamole; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Motor Activity | 1986 |
Nucleoside uptake by Trichomonas vaginalis.
Topics: Adenosine; Animals; Binding, Competitive; Biological Transport; Carrier Proteins; Cytidine; Dilazep; DNA; Guanosine; Inosine; Kinetics; Nucleosides; RNA; Thioinosine; Thionucleosides; Thymidine; Trichomonas vaginalis; Uridine | 1988 |
Effect of acute ethanol on uptake of [3H]adenosine by rat cerebellar synaptosomes.
Topics: Adenosine; Alcohol Drinking; Animals; Cerebellum; Dilazep; Dose-Response Relationship, Drug; Ethanol; Male; Rats; Rats, Inbred Strains; Synaptic Transmission; Synaptosomes | 1989 |
Adenosine formation and release by embryonic chick neurons and glia in cell culture.
Topics: 5'-Nucleotidase; Adenine Nucleotides; Adenosine; Adenosine Monophosphate; Animals; Cells, Cultured; Chick Embryo; Deoxyglucose; Dilazep; Dipyridamole; Hexobendine; Inosine Monophosphate; Neuroglia; Neurons; Oligomycins; Purines | 1989 |
Induction of nucleoside transport sites into the host cell membrane of Babesia bovis infected erythrocytes.
Topics: Adenosine; Animals; Babesia; Binding Sites; Biological Transport; Cattle; Dilazep; Dipyridamole; Erythrocyte Membrane; Erythrocytes; Guanosine; Humans; Kinetics; Phloretin; Phlorhizin; Thioinosine; Thionucleosides; Verapamil | 1989 |
Significance of plasma adenosine in the antiplatelet activity of forskolin: potentiation by dipyridamole and dilazep.
Topics: Adenosine; Adenosine Deaminase; Animals; Azepines; Colforsin; Dilazep; Dipyridamole; Drug Synergism; Humans; In Vitro Techniques; Male; Platelet Aggregation Inhibitors; Rats | 1989 |
Mechanisms involved in the action of prostaglandins as modulators of neurotransmission.
Topics: Acetylcholine; Adenosine; Animals; Blood Pressure; Dilazep; Electric Stimulation; Female; Heart Rate; In Vitro Techniques; Indomethacin; Kidney; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Prostaglandins; Rabbits; Theophylline; Xanthines | 1989 |
Role of plasma adenosine in the antiplatelet action of HL 725, a potent inhibitor of cAMP phosphodiesterase: species differences.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenosine; Adenosine Deaminase; Animals; Blood Platelets; Dilazep; Dipyridamole; Drug Synergism; Humans; Isoquinolines; Male; Mopidamol; Platelet Aggregation; Pyrimidines; Rats; Rats, Inbred Strains; Species Specificity; Tetrahydroisoquinolines | 1987 |
Intracellular adenosine formation and its carrier-mediated release in cultured embryonic chick heart cells.
Topics: 5'-Nucleotidase; Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Biological Transport; Carrier Proteins; Cells, Cultured; Chick Embryo; Deoxyglucose; Dilazep; Dipyridamole; Heart; Hexobendine; Membrane Proteins; Myocardium; Nucleoside Transport Proteins; Nucleotidases; Nucleotides; Oligomycins; Oxygen | 1988 |
Sodium-dependent uptake of nucleosides by dissociated brain cells from the rat.
Topics: Adenosine; Animals; Brain; Dilazep; Dipyridamole; Kinetics; Male; Nucleosides; Ouabain; Rats; Rats, Inbred Strains; Sodium; Thioinosine; Uridine | 1989 |
Potentiation of the antiplatelet action of adenosine in whole blood by dipyridamole or dilazep and the cAMP phosphodiesterase inhibitor, RA 233.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenosine; Azepines; Biological Transport, Active; Blood Platelets; Cyclic AMP; Dilazep; Dipyridamole; Drug Synergism; Humans; In Vitro Techniques; Mopidamol; Nucleosides; Platelet Aggregation; Pyrimidines | 1986 |
Calcium entry blocking activity of dilazep in dog coronary artery.
Topics: Adenine; Adenosine; Adenosine Deaminase; Animals; Arteries; Azepines; Calcium; Calcium Channel Blockers; Coronary Vessels; Dilazep; Diltiazem; Dipyridamole; Dogs; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Lidoflazine; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Potassium; Receptors, Cell Surface; Receptors, Purinergic; Theophylline | 1986 |
Mediation of acute ethanol-induced motor disturbances by cerebellar adenosine in rats.
Topics: Adenosine; Animals; Cerebellum; Dilazep; Dose-Response Relationship, Drug; Ethanol; Male; Motor Activity; Motor Skills; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Theophylline | 1988 |
Relaxing effects of dilazep and lidoflazine in dog cerebral and renal arteries independent of adenosine.
Topics: Adenosine; Adenosine Deaminase; Animals; Azepines; Cerebral Arteries; Dilazep; Dinoprost; Dogs; Female; In Vitro Techniques; Isometric Contraction; Lidoflazine; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Piperazines; Potassium; Renal Artery; Serotonin | 1988 |
Evidence for extracellular deamination of adenosine in the rat heart.
Topics: Adenosine; Adenosine Deaminase; Animals; Cytosol; Deamination; Dilazep; Immunohistochemistry; Male; Myocardium; Perfusion; Rats | 1988 |
Degradation of adenosine by extracellular adenosine deaminase in the rat duodenum.
Topics: Adenosine; Adenosine Deaminase; Adenosine Deaminase Inhibitors; Animals; Coformycin; Dilazep; Duodenum; In Vitro Techniques; Male; Muscle Contraction; Nucleoside Deaminases; Pentostatin; Rats; Rats, Inbred Strains | 1988 |
Adenosine metabolism in human whole blood. Effects of nucleoside transport inhibitors and phosphate concentration.
Topics: Adenosine; Adenosine Deaminase; Adenosine Kinase; Biological Transport; Dilazep; Dipyridamole; Humans; Phosphates; Thioinosine | 1988 |
Pharmacological characterization of rapidly accumulated adenosine by dissociated brain cells from adult rat.
Topics: Adenosine; Adenosine Monophosphate; Animals; Binding, Competitive; Brain; Dilazep; Dipyridamole; Inosine; Kinetics; Male; Rats; Rats, Inbred Strains; Serum Albumin, Bovine; Thioinosine; Uridine | 1988 |
Transport and metabolism of adenosine in human erythrocytes: effect of transport inhibitors and regulation by phosphate.
Topics: Adenine Phosphoribosyltransferase; Adenosine; Adenosine Kinase; Biological Transport; Coformycin; Dilazep; Dipyridamole; Erythrocytes; Humans; Pentostatin; Phosphates; Phosphorylation; Thioinosine | 1986 |
Metabolism of adenosine analogues by Schistosoma mansoni and the effect of nucleoside transport inhibitors.
Topics: Adenosine; Animals; Biological Transport; Dilazep; Dipyridamole; Kinetics; Nucleosides; Schistosoma mansoni; Structure-Activity Relationship; Thioinosine; Thionucleotides; Uracil | 1987 |
Treatment of schistosomiasis by purine nucleoside analogues in combination with nucleoside transport inhibitors.
Topics: Adenosine; Animals; Biological Transport; Dilazep; Dipyridamole; Drug Therapy, Combination; Female; Mice; Purine Nucleosides; Ribonucleosides; Schistosoma mansoni; Schistosomiasis; Thioinosine; Thionucleotides; Toyocamycin; Tubercidin; Uracil | 1987 |
Calcium entry blocking activity of adenosine potentiating compounds in guinea pig taenia coli.
Topics: Adenosine; Animals; Calcium Channel Blockers; Colon; Dilazep; Diltiazem; Dipyridamole; Drug Synergism; Guinea Pigs; In Vitro Techniques; Lidoflazine; Male; Muscle, Smooth; Nifedipine; Potassium; Vasodilator Agents; Verapamil | 1986 |
Inhibition of 3,4-diaminopyridine-induced coronary oscillation by adenyl compounds.
Topics: 4-Aminopyridine; Adenine Nucleotides; Adenosine; Amifampridine; Aminophylline; Aminopyridines; Animals; Coronary Vessels; Dilazep; Dogs; Drug Interactions; In Vitro Techniques; Indomethacin; Membrane Potentials; Muscle, Smooth, Vascular | 1986 |
Experimental documentation of presence of purinergic receptors at human atria.
Topics: Adenosine; Adenosine Triphosphate; Aminophylline; Atrial Function; Dilazep; Dipyridamole; Heart; Heart Atria; Heart Rate; Humans; Kinetics; Myocardial Contraction; Organ Culture Techniques; Quinidine; Receptors, Purinergic | 1986 |
Effects of adenosine uptake blockers and adenosine on evoked potentials of guinea-pig olfactory cortex.
Topics: Adenosine; Adenosine Deaminase; Animals; Diazepam; Dilazep; Dipyridamole; Evoked Potentials; Flurazepam; Guanosine; Guinea Pigs; Hexobendine; In Vitro Techniques; Limbic System; Olfactory Pathways; Thioinosine; Thionucleosides | 1986 |
Calcium entry blocking activity of dilazep and other adenosine potentiating compounds in guinea-pig atria.
Topics: Adenosine; Adenosine Deaminase; Animals; Azepines; Calcium; Calcium Channel Blockers; Dilazep; Dipyridamole; Dose-Response Relationship, Drug; Guinea Pigs; Heart; Heart Atria; Isoproterenol; Lidoflazine; Myocardial Contraction; Theophylline | 1986 |
Role of adenosine uptake and metabolism by blood cells in the antiplatelet actions of dipyridamole, dilazep and nitrobenzylthioinosine.
Topics: Adenosine; Azepines; Blood Platelets; Dilazep; Dipyridamole; Erythrocytes; Humans; In Vitro Techniques; Inosine; Mopidamol; Platelet Aggregation; Thioinosine | 1985 |
Release of nucleosides and nucleotides from the rabbit heart by sympathetic nerve stimulation.
Topics: Adenosine; Adenosine Deaminase; Adenosine Monophosphate; Adrenergic beta-Antagonists; Animals; Dilazep; Dipyridamole; Electric Stimulation; Heart; Hypoxanthines; Inosine; Myocardium; Norepinephrine; Nucleosides; Nucleotides; Phentolamine; Propranolol; Rabbits; Sympathetic Nervous System | 1982 |
Dilazep: an inhibitor of adenosine uptake with intrinsic calcium antagonistic properties.
Topics: Adenosine; Animals; Azepines; Calcium Channel Blockers; Dilazep; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Rabbits | 1983 |
The effects of dilazep and SG 75 on cyclic nucleotides in the coronary artery.
Topics: Adenosine; Animals; Arteries; Azepines; Coronary Circulation; Coronary Vessels; Cyclic AMP; Cyclic GMP; Dilazep; Dogs; Muscle Contraction; Myocardium; Niacinamide; Nicorandil; Nitrates; Vasodilator Agents | 1980 |
Inward fluxes of adenosine in erythrocytes and cultured cells measured by a quenched-flow method.
Topics: Adenosine; Animals; Biological Transport; Cells, Cultured; Dilazep; Erythrocytes; Humans; Kinetics; Methods; Mice; Tubercidin | 1984 |
Enhancement of myocardial reactive hyperemia and adenosine-induced coronary vasodilation by dilazep, a new adenosine potentiator.
Topics: Adenosine; Animals; Azepines; Coronary Circulation; Dilazep; Dogs; Drug Interactions; Hyperemia; Infusions, Parenteral; Myocardium | 1982 |
Metabolism of adenosine and 2'-deoxy-adenosine by fetal mouse calvaria in culture.
Topics: Adenine; Adenosine; Animals; Bone and Bones; Culture Media; Deoxyadenosines; Dilazep; Dipyridamole; Hypoxanthine; Hypoxanthines; Inosine; Mice; Organ Culture Techniques | 1982 |
Role of adenosine in adipose tissue circulation.
Topics: Adenine; Adenosine; Adipose Tissue; Animals; Capillary Permeability; Dilazep; Dipyridamole; Dogs; Female; Inosine; Vascular Resistance; Vasodilator Agents | 1981 |
The antilipolytic effect of endogenous and exogenous adenosine in canine adipose tissue in situ.
Topics: 2-Chloroadenosine; Adenine; Adenosine; Adipose Tissue; Animals; Dilazep; Dipyridamole; Dogs; Female; Lipolysis | 1981 |
Potentiation by dilazep on the negative inotropic effect of adenosine on guinea-pig atria.
Topics: Adenosine; Adenosine Deaminase; Animals; Azepines; Calcium; Dilazep; Drug Synergism; Female; Male; Mice; Muscle Contraction; Myocardial Contraction; Time Factors | 1980 |
Time-dependent antinociceptive interactions between opioids and nucleoside transport inhibitors.
Topics: Adenosine; Analgesics; Animals; Biological Transport; Dilazep; Dipyridamole; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Male; Mice; Narcotics; Nucleosides; Receptors, Opioid; Thioinosine; Time Factors | 1995 |
Altered purine nucleoside transport as a target for malaria chemotherapy.
Topics: Adenosine; Affinity Labels; Alkaloids; Animals; Antimalarials; Benzodioxoles; Benzoquinones; Biological Transport; Ciona intestinalis; Crithidia; Dilazep; Erythrocytes; Furosemide; HeLa Cells; Humans; Malaria, Falciparum; Phlorhizin; Piperidines; Plasmodium falciparum; Polyunsaturated Alkamides; Stereoisomerism; Thioinosine; Trichomonas vaginalis | 1994 |
Nucleoside transport and metabolism in lymphocytes, polymorphonuclear cells and cerebral synaptosomes.
Topics: Adenosine; Animals; Biological Transport; Cerebral Cortex; Child; Deoxycytidine; Dilazep; Dipyridamole; DNA; Humans; Kinetics; Lymphocytes; Neutrophils; Nucleosides; Palatine Tonsil; Papaverine; Rats; Synaptosomes; Thioinosine; Thymidine; Uridine | 1994 |
Involvement of bidirectional adenosine transporters in the release of L-[3H]adenosine from rat brain synaptosomal preparations.
Topics: Adenosine; Animals; Biological Transport; Brain; Carrier Proteins; Dilazep; Dipyridamole; Kinetics; Male; Membrane Proteins; Nucleoside Transport Proteins; Potassium Chloride; Rats; Rats, Sprague-Dawley; Synaptosomes; Thioinosine; Tritium | 1995 |
Release and regulation of endogenous adenosine during hemorrhage.
Topics: Adenine; Adenosine; Adenosine Deaminase Inhibitors; Animals; Blood Pressure; Cats; Chromatography, High Pressure Liquid; Dilazep; Drug Interactions; Female; Hemorrhage; Male | 1994 |
Effects of the liver on circulating adenosine in blood.
Topics: Adenosine; Animals; Blood Pressure; Cats; Chromatography, High Pressure Liquid; Dilazep; Female; Infusions, Intravenous; Liver; Male; Spectrometry, Fluorescence | 1993 |
[3H]adenosine transport in synaptoneurosomes of postmortem human brain.
Topics: Adenine; Adenosine; Aged; Biological Transport; Cadaver; Cerebral Cortex; Dilazep; Dipyridamole; Female; Humans; Kinetics; Male; Synaptosomes; Time Factors; Tritium; Tubercidin | 1993 |
Functional characterization of a recombinant sodium-dependent nucleoside transporter with selectivity for pyrimidine nucleosides (cNT1rat) by transient expression in cultured mammalian cells.
Topics: Adenosine; Amino Acid Sequence; Animals; Base Sequence; Biological Transport; Carrier Proteins; Cells, Cultured; Dilazep; Dipyridamole; Genes, myc; Guanosine; Haplorhini; Intestines; Kidney; Membrane Transport Proteins; Molecular Sequence Data; Nucleosides; Pyrimidine Nucleosides; Rats; Recombinant Proteins; Thioinosine; Transfection; Uridine | 1996 |
Characterization of inhibitor-sensitive and -resistant adenosine transporters in cultured human fetal astrocytes.
Topics: Adenine; Adenosine; Affinity Labels; Astrocytes; Biological Transport; Carrier Proteins; Cells, Cultured; Dilazep; Dipyridamole; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fetus; Humans; Kinetics; Membrane Proteins; Nucleoside Transport Proteins; Thioinosine; Tritium; Tubercidin; Vasodilator Agents | 1996 |
[3H]adenosine transport in DDT1 MF-2 smooth muscle cells: inhibition by metabolites of propentofylline.
Topics: Adenosine; Animals; Binding Sites; Biological Transport; Cricetinae; Dilazep; Dipyridamole; Genital Neoplasms, Male; Kinetics; Leiomyosarcoma; Leukemia L1210; Male; Mesocricetus; Muscle, Smooth; Rats; Thioinosine; Tumor Cells, Cultured; Vas Deferens; Xanthines | 1996 |
Dilazep and its derivative, K-7259, attenuate mechanical derangement induced by palmitoyl-L-carnitine in the isolated, perfused rat heart.
Topics: Adenosine; Animals; Calcium; Dilazep; Heart; Male; Palmitoylcarnitine; Perfusion; Rats; Rats, Sprague-Dawley; Vasodilator Agents | 1996 |
2'-deoxyadenosine induces apoptosis in rat chromaffin cells.
Topics: Adenosine; Adenosine Deaminase; Adenosine Triphosphate; Adrenergic alpha-Agonists; Animals; Apoptosis; Chromaffin Cells; Deoxyadenosines; Dilazep; Enzyme Inhibitors; Epinephrine; Mutagens; Norepinephrine; Phosphorylation; Rats; Rats, Sprague-Dawley; Sensitivity and Specificity; Thioinosine; Tubercidin; Vasodilator Agents | 1996 |
Dilazep, an antiplatelet agent, inhibits tissue factor expression in endothelial cells and monocytes.
Topics: Adenosine; Dilazep; Endothelium, Vascular; Gene Expression; Humans; Monocytes; Platelet Aggregation Inhibitors; Purinergic P1 Receptor Agonists; Tetradecanoylphorbol Acetate; Theophylline; Thrombin; Thromboplastin; Tumor Necrosis Factor-alpha | 1997 |
Levels of endogenous adenosine in rat striatum. II. Regulation of basal and N-methyl-D-aspartate-induced levels by inhibitors of adenosine transport and metabolism.
Topics: 5'-Nucleotidase; Adenosine; Adenosine Deaminase Inhibitors; Animals; Biological Transport; Corpus Striatum; Dilazep; Male; N-Methylaspartate; Pentostatin; Rats; Rats, Sprague-Dawley | 1998 |
Further characterization of an adenosine transport system in the mitochondrial fraction of rat testis.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Benzodiazepinones; Biological Transport; Dilazep; Dipyridamole; Dose-Response Relationship, Drug; Guanosine; Hexobendine; Hydrogen-Ion Concentration; Inosine; Isoquinolines; Kinetics; Male; Mitochondria; Osmolar Concentration; Phenylisopropyladenosine; Rats; Rats, Sprague-Dawley; Sodium; Subcellular Fractions; Temperature; Testis; Thioinosine; Thionucleosides; Time Factors; Tritium; Uridine | 2000 |
Inhibition of glucose uptake in murine cardiomyocyte cell line HL-1 by cardioprotective drugs dilazep and dipyridamole.
Topics: Adenosine; Animals; Biological Transport; Cardiotonic Agents; Cell Line; Deoxyglucose; Dilazep; Dipyridamole; Glucose; Glucose Transporter Type 1; Glucose Transporter Type 4; Kinetics; Mice; Monosaccharide Transport Proteins; Muscle Proteins; Myocytes, Cardiac; Thioinosine | 2004 |
Mutation of leucine-92 selectively reduces the apparent affinity of inosine, guanosine, NBMPR [S6-(4-nitrobenzyl)-mercaptopurine riboside] and dilazep for the human equilibrative nucleoside transporter, hENT1.
Topics: Adenosine; Amino Acid Substitution; Biological Transport; Dilazep; Dipyridamole; Drug Resistance; Equilibrative Nucleoside Transporter 1; Guanosine; Humans; Inhibitory Concentration 50; Inosine; Leucine; Mutagenesis; Mutation, Missense; Point Mutation; Recombinant Fusion Proteins; Saccharomyces cerevisiae; Structure-Activity Relationship; Thioinosine | 2004 |
[(3)H]Adenosine uptake in brainstem membranes of CD-1 mice lacking the adenosine A(2a) receptor.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Autoradiography; Brain Stem; Carrier Proteins; Dilazep; Dipyridamole; Membrane Transport Proteins; Membranes; Mice; Mice, Knockout; Nucleoside Transport Proteins; Receptors, Adenosine A2; Time Factors; Tritium | 2004 |
Residue 33 of human equilibrative nucleoside transporter 2 is a functionally important component of both the dipyridamole and nucleoside binding sites.
Topics: Adenosine; Binding Sites; Biological Transport; Dilazep; Dipyridamole; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Humans; Nucleosides; Structure-Activity Relationship; Uridine | 2005 |
Residues 334 and 338 in transmembrane segment 8 of human equilibrative nucleoside transporter 1 are important determinants of inhibitor sensitivity, protein folding, and catalytic turnover.
Topics: Adenosine; Amino Acid Sequence; Biological Transport; Dilazep; Equilibrative Nucleoside Transporter 1; Genetic Complementation Test; Heterocyclic Compounds; Humans; Membrane Proteins; Molecular Sequence Data; Mutagenesis; Mutation; Nucleosides; Protein Conformation; Protein Folding; Saccharomyces cerevisiae; Sequence Homology, Amino Acid; Thioinosine | 2007 |
Mutation of Trp29 of human equilibrative nucleoside transporter 1 alters affinity for coronary vasodilator drugs and nucleoside selectivity.
Topics: Adenosine; Biological Transport; Dilazep; Dipyridamole; Enzyme Activation; Equilibrative Nucleoside Transporter 1; Humans; Kinetics; Models, Biological; Mutation; Nucleosides; Piperazines; Protein Binding; Thioinosine; Tryptophan; Vasodilator Agents | 2008 |
Estimation of endogenous adenosine activity at adenosine receptors in guinea-pig ileum using a new pharmacological method.
Topics: 2-Chloroadenosine; Adenosine; Animals; Dilazep; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; Male; Muscle Contraction; Receptors, Purinergic P1; Synaptic Transmission; Theophylline; Vasodilator Agents | 2010 |
Structures of human ENT1 in complex with adenosine reuptake inhibitors.
Topics: Adenosine; Crystallography, X-Ray; Dilazep; Equilibrative Nucleoside Transporter 1; Humans; Models, Molecular; Protein Conformation; Thioinosine | 2019 |
Adenosine reuptake inhibition reduces diabetes-induced glomerular hyperfiltration via the adenosine A2
Topics: Adenosine; Animals; Diabetes Mellitus; Dilazep; Glomerular Filtration Rate; Kidney; Kidney Diseases; Kidney Glomerulus; Male; Rats; Rats, Sprague-Dawley | 2023 |