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dihydrotestosterone 17-bromoacetate and dihydrotestosterone

dihydrotestosterone 17-bromoacetate has been researched along with dihydrotestosterone in 13 studies

Compound Research Comparison

Studies
(dihydrotestosterone 17-bromoacetate)
Trials
(dihydrotestosterone 17-bromoacetate)
Recent Studies (post-2010)
(dihydrotestosterone 17-bromoacetate)
Studies
(dihydrotestosterone)
Trials
(dihydrotestosterone)
Recent Studies (post-2010) (dihydrotestosterone)
13009,3253071,517

Protein Interaction Comparison

ProteinTaxonomydihydrotestosterone 17-bromoacetate (IC50)dihydrotestosterone (IC50)
Plasma kallikreinHomo sapiens (human)0.0031
Glucocorticoid receptorHomo sapiens (human)0.54
Sex hormone-binding globulinHomo sapiens (human)0.0038
Progesterone receptorOryctolagus cuniculus (rabbit)0.44
Progesterone receptorHomo sapiens (human)7.3
Mineralocorticoid receptor Homo sapiens (human)0.36
Sex hormone-binding globulinRattus norvegicus (Norway rat)0.023
Androgen receptorHomo sapiens (human)0.0048
Androgen receptorRattus norvegicus (Norway rat)0.4041
Androgen receptorMus musculus (house mouse)0.001
Mineralocorticoid receptorRattus norvegicus (Norway rat)2.1
Testosterone 17-beta-dehydrogenase 3Homo sapiens (human)0.0026

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19909 (69.23)18.7374
1990's4 (30.77)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kumar, S; Namkung, PC; Petra, PH; Walsh, KA1
Khan, MS; Rosner, W1
Penning, TM; Ricigliano, JW1
Danzo, BJ; Ellis, DL1
Belsham, DD; Faber, LE; Kovacs, WJ; Pereira, FA; Rosenmann, E; Turney, MK; Williams, SG; Wrogemann, K1
Anthony, CT; Kovacs, WJ; Skinner, MK1
Kovacs, WJ; Skinner, MK; Turney, MK1
Charbonneau, H; Griffin, PR; Hunt, DF; Namkung, PC; Petra, PH; Que, BG; Ross, JB; Shabanowitz, J; Walsh, KA1
Kovacs, WJ; Turney, MK1
Chang, CH; Lobl, TJ; Rowley, DR; Tindall, DJ2
Samant, BR; Sweet, F1
Kovacs, WJ; McCammon, DK; McPhaul, MJ; Turney, MK; Zhou, P1

Other Studies

13 other study(ies) available for dihydrotestosterone 17-bromoacetate and dihydrotestosterone

ArticleYear
Identification of lysine 134 in the steroid-binding site of the sex steroid-binding protein of human plasma.
    The Journal of biological chemistry, 1990, Oct-25, Volume: 265, Issue:30

    Topics: Affinity Labels; Alkylating Agents; Amino Acid Sequence; Binding Sites; Dihydrotestosterone; Humans; Hydrogen-Ion Concentration; Lysine; Molecular Sequence Data; Molecular Structure; Peptide Mapping; Sex Hormone-Binding Globulin; Structure-Activity Relationship

1990
Histidine 235 of human sex hormone-binding globulin is the covalent site of attachment of the nucleophilic steroid derivative, 17 beta-bromoacetoxydihydrotestosterone.
    The Journal of biological chemistry, 1990, May-25, Volume: 265, Issue:15

    Topics: Affinity Labels; Amino Acid Sequence; Binding Sites; Binding, Competitive; Chromatography, High Pressure Liquid; Dihydrotestosterone; Female; Histidine; Humans; Kinetics; Molecular Sequence Data; Peptide Fragments; Peptide Mapping; Pregnancy; Sex Hormone-Binding Globulin; Trypsin

1990
Evidence that enzyme-generated aromatic Michael acceptors covalently modify the nucleotide-binding site of 3 alpha-hydroxysteroid dehydrogenase.
    The Biochemical journal, 1990, Aug-01, Volume: 269, Issue:3

    Topics: 3-alpha-Hydroxysteroid Dehydrogenase (B-Specific); 3-Hydroxysteroid Dehydrogenases; Animals; Binding Sites; Chemical Phenomena; Chemistry; Chromatography, Affinity; Dihydrotestosterone; Kinetics; Male; Mercaptoethanol; NAD; NADP; Nitrobenzenes; Nucleotides; Oxidation-Reduction; Protein Synthesis Inhibitors; Rats; Rats, Inbred Strains; Triazines

1990
Identification of an androgen receptor in the adult chicken oviduct.
    Journal of steroid biochemistry, 1989, Volume: 33, Issue:6

    Topics: Affinity Labels; Animals; Binding, Competitive; Chickens; Cytosol; Dihydrotestosterone; Electrophoresis, Polyacrylamide Gel; Female; Oviducts; Receptors, Androgen; Spectrometry, Fluorescence; Substrate Specificity

1989
The 56 kDa protein of human genital skin fibroblasts is identical to that radiolabelled by [3H]dihydrotestosterone 17 beta-bromoacetate.
    Journal of steroid biochemistry, 1989, Volume: 33, Issue:3

    Topics: Affinity Labels; Antibodies, Monoclonal; Cells, Cultured; Dihydrotestosterone; Electrophoresis, Gel, Two-Dimensional; Fibroblasts; Genitalia; Humans; Immunoblotting; Immunochemistry; Molecular Weight; Photochemistry; Photofluorography; Proteins; Radioligand Assay; Receptors, Androgen; Skin

1989
Analysis of the androgen receptor in isolated testicular cell types with a microassay that uses an affinity ligand.
    Endocrinology, 1989, Volume: 125, Issue:5

    Topics: Affinity Labels; Animals; Cells, Cultured; Dihydrotestosterone; Fibroblasts; Humans; Kinetics; Leydig Cells; Male; Organ Specificity; Rats; Receptors, Androgen; Sertoli Cells; Skin; Testis

1989
Biochemical characterization of the protein affinity labeled by dihydrotestosterone 17 beta-bromoacetate: comparison with the human androgen receptor.
    Endocrinology, 1989, Volume: 124, Issue:3

    Topics: Affinity Labels; Centrifugation, Density Gradient; Chemical Phenomena; Chemistry, Physical; Cytosol; Dihydrotestosterone; Electrophoresis, Polyacrylamide Gel; Fibroblasts; Genitalia, Male; Isoelectric Point; Male; Molecular Weight; Protein Precursors; Proteins; Receptors, Androgen; Skin

1989
Affinity labeling, molecular cloning, and comparative amino acid sequence analyses of sex steroid-binding protein of plasma. A multidisciplinary approach for understanding steroid-protein interaction and its physiological role.
    Annals of the New York Academy of Sciences, 1988, Volume: 538

    Topics: Affinity Labels; Amino Acid Sequence; Androgen-Binding Protein; Animals; Dihydrotestosterone; Equilenin; Humans; Molecular Sequence Data; Photochemistry; Rats; Sex Hormone-Binding Globulin; Testosterone

1988
High efficiency covalent radiolabeling of the human androgen receptor. Studies in cultured fibroblasts using dihydrotestosterone 17 beta-bromoacetate.
    The Journal of clinical investigation, 1988, Volume: 81, Issue:2

    Topics: Affinity Labels; Cells, Cultured; Cytosol; Dihydrotestosterone; Fibroblasts; Humans; Kinetics; Molecular Weight; Receptors, Androgen

1988
Affinity labeling of the androgen receptor in rat prostate cytosol with 17 beta-[(bromoacetyl)oxy]-5 alpha-androstan-3-one.
    Biochemistry, 1984, May-22, Volume: 23, Issue:11

    Topics: Affinity Labels; Animals; Binding, Competitive; Cytosol; Dihydrotestosterone; Indicators and Reagents; Kinetics; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Prostate; Rats; Rats, Inbred Strains; Receptors, Androgen; Receptors, Steroid; Spectrophotometry

1984
Molecular properties of the androgen receptor in rat ventral prostate.
    Annals of the New York Academy of Sciences, 1984, Volume: 438

    Topics: Affinity Labels; Animals; Binding Sites; Dihydrotestosterone; Male; Molecular Weight; Prostate; Rats; Receptors, Androgen; Receptors, Steroid

1984
Bifunctional enzyme activity at the same active site: study of 3 alpha and 20 beta activity by affinity alkylation of 3 alpha, 20 beta-hydroxysteroid dehydrogenase with 17-(bromoacetoxy)steroids.
    Biochemistry, 1980, Mar-04, Volume: 19, Issue:5

    Topics: 20-Hydroxysteroid Dehydrogenases; Affinity Labels; Alkylation; Binding Sites; Cortisone Reductase; Dihydrotestosterone; Hydroxyprogesterones; Kinetics; Methods; Protein Binding; Streptomyces; Substrate Specificity

1980
An androgenic affinity ligand covalently binds to cytosolic aldehyde dehydrogenase from human genital skin fibroblasts.
    Molecular and cellular endocrinology, 1993, Volume: 91, Issue:1-2

    Topics: Affinity Labels; Aldehyde Dehydrogenase; Androgens; Animals; Base Sequence; Binding Sites; Binding, Competitive; CHO Cells; Cricetinae; Dihydrotestosterone; DNA; Fibroblasts; Genitalia; Humans; Molecular Sequence Data; Polymerase Chain Reaction; Protein Biosynthesis; Transfection

1993