Page last updated: 2024-09-02

dihydrokainate and sym 2081

dihydrokainate has been researched along with sym 2081 in 2 studies

Compound Research Comparison

Studies
(dihydrokainate)
Trials
(dihydrokainate)
Recent Studies (post-2010)
(dihydrokainate)
Studies
(sym 2081)
Trials
(sym 2081)
Recent Studies (post-2010) (sym 2081)
180046903

Protein Interaction Comparison

ProteinTaxonomydihydrokainate (IC50)sym 2081 (IC50)
Metabotropic glutamate receptor 6Homo sapiens (human)4
Glutamate receptor ionotropic, kainate 1Rattus norvegicus (Norway rat)0.035
Glutamate receptor ionotropic, kainate 2Rattus norvegicus (Norway rat)0.035
Glutamate receptor ionotropic, kainate 3Rattus norvegicus (Norway rat)0.035
Glutamate receptor ionotropic, kainate 4Rattus norvegicus (Norway rat)0.035
Glutamate receptor ionotropic, kainate 5Rattus norvegicus (Norway rat)0.035

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bolte, J; Bunch, L; Chapelet, M; Gefflaut, T; Nielsen, B; Pickering, DS; Pu, X; Sagot, E; Stensbøl, TB; Umberti, M1
Amir, A; Brindisi, M; Butini, S; Campiani, G; Coccone, SS; Frydenvang, K; Gemma, S; Guarino, E; Kastrup, JS; Kumar, V; Maramai, S; Novellino, E; Pickering, DS; Valadés, EA; Valenti, S; Venskutonyte, R1

Other Studies

2 other study(ies) available for dihydrokainate and sym 2081

ArticleYear
Chemo-enzymatic synthesis of a series of 2,4-syn-functionalized (S)-glutamate analogues: new insight into the structure-activity relation of ionotropic glutamate receptor subtypes 5, 6, and 7.
    Journal of medicinal chemistry, 2008, Jul-24, Volume: 51, Issue:14

    Topics: Amination; Animals; Glutamic Acid; Magnetic Resonance Spectroscopy; Mass Spectrometry; Rats; Receptors, Glutamate; Spectrophotometry, Infrared; Structure-Activity Relationship; Synaptosomes

2008
Selective kainate receptor (GluK1) ligands structurally based upon 1H-cyclopentapyrimidin-2,4(1H,3H)-dione: synthesis, molecular modeling, and pharmacological and biostructural characterization.
    Journal of medicinal chemistry, 2011, Jul-14, Volume: 54, Issue:13

    Topics: Animals; Cell Line; Cricetinae; Crystallography, X-Ray; Female; Ligands; Models, Molecular; Oocytes; Patch-Clamp Techniques; Protein Conformation; Pyrimidines; Rats; Receptors, Kainic Acid; Recombinant Proteins; Stereoisomerism; Structure-Activity Relationship; Thiophenes; Xenopus laevis

2011