dihydroalprenolol has been researched along with isoproterenol in 343 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 281 (81.92) | 18.7374 |
1990's | 46 (13.41) | 18.2507 |
2000's | 14 (4.08) | 29.6817 |
2010's | 2 (0.58) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Aué, GH; Bultsma, T; IJzerman, AP; Linschoten, MR; Timmerman, H | 1 |
Lefkowitz, RJ; Mullikin, D; Wessels, MR | 1 |
Bockaert, J; Dolphin, A; Hamont, M | 1 |
Enna, SJ; U'Prichard, DC | 1 |
Cote, T; Kebabian, J; Munemura, M | 1 |
DeLean, A; Hickey, AR; Lefkowitz, RJ; Limbird, LE; Pike, LJ | 1 |
Agli, B; Giudicelli, Y; Lacasa, D | 4 |
Cabelli, RJ; Malbon, CC | 1 |
Limas, CJ | 1 |
Gillespie, DD; Manier, DH; Sulser, F | 2 |
Billon, MC; Geynet, P; Hanoune, J; Houssin, D; Munnich, A; Schmelck, PH | 1 |
Arnett, CD; Davis, JN | 1 |
Brunswick, DJ; Frazer, A; Greenberg, LH; Mendels, J; Moyer, JA; Weiss, B | 1 |
Chen, FM; Roeske, WR; Yamamura, HI | 1 |
Howlett, DR; Nahorski, SR; Redgrave, P | 1 |
Lefkowitz, RJ; Stadel, JM | 1 |
Caron, MG; Lefkowitz, RJ; Limbird, LE | 1 |
Extein, I; Goodwin, FK; Smith, CC; Tallman, J | 1 |
Azuma, H; Oshima, H; Tsujii, T; Yamaguchi, T | 1 |
Kato, T; Kokubu, N; Satoh, M; Takayanagi, I | 1 |
Austin, CE; Chess-Williams, R | 2 |
Grishin, AV; Kuznetzova, LA; Panchenko, MP; Pertseva, MN; Plesneva, SA | 1 |
Kinuya, M; Mamiya, G; Ohtakeno, S; Watanabe, H; Watanabe, M | 1 |
Allo, S; Punna, S; Schaffer, SW; White, T | 1 |
Moon, TW; Perry, SF; Reid, SD | 1 |
Adderholt, JG; Dwyer, TM; Farley, JM | 1 |
Latifpour, J; Marian, MJ; Nishimoto, T; Weiss, RM; Yoshida, M | 1 |
Kishi, M; Kuriyama, K; Ma, FH; Ohkuma, S | 1 |
Gousse, A; Latifpour, J; Weiss, RM; Yoshida, M | 1 |
Irie, M; Kajinuma, H; Suzuki, K; Watanabe, K | 1 |
Drímal, J; Drímalová, L; Knézl, V; Magna, D; Tokárová, J | 1 |
Higashijima, T; Kameyama, K; Parker, EM; Ross, EM | 1 |
Areso, P; Frazer, A; Gambarana, C; Hensler, JG; Ordway, GA | 1 |
Nakamura, T; Nomura, J; Tsujimura, R | 1 |
Agrawal, DK; Bergren, DR; Byorth, PJ; Townley, RG | 1 |
Adham, N; Blue, DR; Bond, RA; Clarke, DE; Delmendo, R; Eglen, RM; Michel, AD; Whiting, RL | 1 |
Pilc, A; Vetulani, J | 1 |
Donta, ST; Shanley, JD | 1 |
Abe, K; Matsuki, N; Nagata, K; Saito, H; Wang, CH | 1 |
Abrahamsson, T; Nerme, V; Vauquelin, G | 1 |
Lefebvre, J; Revillion, F; Vandewalle, B | 1 |
Shigenobu, K; Tanaka, H | 1 |
Kawano, K; Koike, K; Takayanagi, I | 1 |
Nedvídková, J; Pacák, K; Schreiber, V; Stolba, P | 1 |
Ganguly, PK; Lee, SL; Waghray, G | 1 |
Cheng, KW; Ghahary, A | 1 |
Fukunaga, H; Saito, K; Tanaka, H | 1 |
Hansel-Bessey, S; Ratge, D; Wisser, H | 1 |
Amann, FW; Bühler, FR; Landmann, R; van Brummelen, P | 1 |
Barnes, PJ; Gold, WM; Phillips, MJ | 1 |
Braquet, P; Dausse, JP; Garay, R; Hannaert, P; Rosati, C | 1 |
Cantor, E; Greenberg, S; Paul, J | 1 |
Limas, C; Limas, CJ | 3 |
Moises, HC; Smith, CB | 1 |
Creese, I; Riva, MA | 1 |
Camilion de Hurtado, MC; Gende, OA | 1 |
Pascual, J; Sterin-Borda, L; Wald, M | 1 |
Burkard, WP; Eigenmann, R; Goodman, M; Holck, M; Märki, HP; Melmon, KL; Osterrieder, W | 1 |
Irie, M; Kajinuma, H; Sato, N; Suzuki, K | 1 |
Dunlap, CE; Gould, RJ; Murphy, KM; Snyder, SH; Strandhoy, JW | 1 |
Grobecker, H; Schrader, E | 1 |
LaBella, FS; Nukina, I | 1 |
Enna, SJ; Nomura, S; Pilc, A; Vetulani, J | 1 |
Hui, KK; Yu, JL | 1 |
Cheetham, SC; Crompton, MR; De Paermentier, F; Horton, RW | 1 |
Berlan, M; Lafontan, M; Montastruc, P; Taouis, M | 1 |
Broadley, KJ; Chess-Williams, RG; Sheridan, DJ | 2 |
Banerjee, SP; Fan, TH; Kawashima, S; Liang, CS | 1 |
Engels, F; Folkerts, G; Nijkamp, FP; van Heuven-Nolsen, D | 1 |
Dan'ura, T; Ishibashi, S; Kurokawa, T; Yamashita, A; Yanagiuchi, H | 1 |
Andersson, RG; Johansson, SR; Salomonsson, I | 1 |
Humphreys-Beher, M; Schneyer, CA | 1 |
Borda, E; Cremaschi, G; Podestá, EJ; Sánchez, ML; Solano, AR; Sterin-Borda, L | 1 |
Jazayeri, A; Meyer, WJ | 2 |
Crooke, ST; Stadel, JM | 1 |
Bukantz, SC; Krzanowski, JJ; Lockey, RF; Lowitt, S; Polson, JB; Szentivanyi, A | 1 |
Kellar, KJ; Stockmeier, CA | 1 |
Legrand, C; Maltier, JP | 1 |
Bockaert, J; Bouhelal, R; Gozlan, H; Homburger, V; Lucas, M | 1 |
Koike, K; Takayanagi, I | 3 |
Clegg, RA; Mullaney, I | 1 |
De Blasi, A; Fratelli, M; Insel, PA; Lipartiti, M; Motulsky, HJ | 1 |
Camilión de Hurtado, MC; Cingolani, HE; Gende, OA | 1 |
Fujita, H; Goto, J; Hashizume, K; Kase, H; Kubo, K; Nakamura, J; Shuto, K | 1 |
Baker, SP; Muther, TF; Nelson, CA; Pitha, J | 1 |
Kitada, Y; Kosasa, T; Miyauchi, T; Satoh, S | 1 |
Ikezawa, H; Nakajima, M; Taguchi, R | 1 |
Ijzerman, A; Nerme, V; Severne, Y; Timmerman, H; Vauquelin, G | 1 |
Cheng, HY; Crooke, ST; Hwang, SM; Wong, A | 1 |
Lyles, GA; Neilson, DG; Ogg, GD; Stevenson, IH | 1 |
Drímal, J; Knezl, V; Magna, D; Strízová, K | 1 |
Cambray-Deakin, M; Morrow, C; Murphy, S; Pearce, B | 1 |
Lin, CC; Moawad, AH; River, LP | 1 |
Delavier-Klutchko, C; Durieu-Trautmann, O; Hoebeke, J; Strosberg, AD | 1 |
Bylund, DB; Chao, WT; Gibbs, SR; Walkenbach, RJ | 1 |
Abbracchio, MP; Berti, F; Cattabeni, F; Daffonchio, L; Hernandez, A; Omini, C | 1 |
Crews, FT; Scott, JA | 1 |
Platt, JE; Slucky, AV; Stone, EA; Trullas, R | 1 |
Altszuler, N; Cherksey, BD; Mendelsohn, SA; Zadunaisky, JA | 1 |
Fialkovskaia, LA; Kuzin, AM; Slozhenikina, LV; Ushakova, TE | 1 |
Aué, GH; Bultsma, T; Dorlas, R; Ijzerman, AP; Timmerman, H | 1 |
Arinze, IJ; Graham, SM; Kawai, Y; Whitsel, C | 1 |
Lang, PH; Lemmer, B | 2 |
Pappano, AJ; Smith, CJ | 1 |
Kazarov, AR; Malatsidze, MA; Sobolev, AS | 1 |
Banerjee, SP; Fan, TH | 1 |
Berlan, M; Carpene, C; Lafontan, M | 1 |
Baker, SP; Liptak, A; Pitha, J | 1 |
Abbracchio, MP; Cattabeni, F; Daffonchio, L; Giani, E; Hernandez, A; Omini, C | 1 |
Banerjee, S; DiStefano, V; Harnish, PP; Northington, FK | 1 |
Abrass, IB; O'Connor, SW; Scarpace, PJ | 1 |
Ratge, D; Wisser, H | 1 |
Abbracchio, MP; Cattabeni, F; Daffonchio, L; Fano, M; Hernandez, A; Omini, C | 1 |
Nagai, S; Ozawa, T; Sugiyama, S; Takamura, T | 1 |
Rodan, GA; Rodan, SB | 1 |
Kanarek, L; Severne, Y; Vauquelin, G | 1 |
Algeri, S; Costantini, C; Cotecchia, S; De Blasi, A; Fratelli, M; Lipartiti, M; Sacchetti, G | 1 |
Aakesson, I; Jacobsen, S; Sager, G; Sandnes, D | 1 |
Kunovská, V; Prásek, J; Prikryl, P; Rysánek, K; Vondrácek, V | 1 |
Jones, SB; Romano, FD | 1 |
Bast, A; Kramer, K; Leurs, R; Rademaker, B; Timmerman, H | 1 |
Jurss, R; Severne, Y; Vauquelin, G | 1 |
Arinze, IJ; Graham, SM; Kawai, Y; Yoshioka, H | 1 |
De Blasi, A; Fratelli, M; Lipartiti, M; Wielosz, M | 1 |
Agrawal, DK; Townley, RG | 1 |
Nelson, KM; Shepherd, RE; Spitzer, JA | 1 |
Humphreys-Beher, MG | 1 |
Khabarov, SV | 1 |
Cheung, WT; Lee, CM; Wong, CC | 1 |
Alnor, J; Auch-Schwelk, W; Gastmann, U; Hirsch, FW; Keul, J; Lehmann, M; Ochs, A | 1 |
Akino, T; Miyamoto, A; Ohshika, H | 1 |
Nagao, T; Naito, K; Yabana, H | 1 |
Honbo, N; Karliner, JS; Simpson, PC; Taylor, JE; Woloszyn, W | 1 |
Conner, MW; Reid, LM | 1 |
Houssay, AB; Levi de Stein, M; Medina, JH; Tumilasci, O; Wolfman, C | 1 |
Cornett, LE; Hiller, C; Hough, A; Norris, JS; Popovich, KJ | 1 |
Gillespie, DD; Manier, DH; Steranka, LR; Sulser, F | 1 |
Kilpatrick, BF; Lefkowitz, RJ; Stiles, GL; Strasser, RH; Taylor, SR | 1 |
Blashkin, IuV; Chirkov, IuIu; Kazarov, AR; Malatsidze, MA; Sobolev, AS | 1 |
Bultsma, T; IJzerman, AP; Timmerman, H; Zaagsma, J | 1 |
Hausen, M; Jacobs, KH; Kutter, A; Mann, JF; Nagel, W; Rascher, W; Ritz, E; Schick, M; Sudhoff, R | 1 |
Hertel, C; Müller, P; Portenier, M; Staehelin, M | 2 |
Montandon, JB; Porzig, H | 1 |
Koshiura, R; Matsunaga, T; Miyamoto, K; Takemoto, N | 1 |
Enna, SJ; Maggi, A; U'Prichard, DC | 1 |
Allred, S; Duriseti, L; Galant, SP; Insel, PA; Underwood, S | 1 |
Cryer, PE; Tohmeh, JF | 1 |
Malbon, CC | 1 |
Briley, M; Cavero, I; Langer, SZ; Roach, AG | 1 |
Delavier-Klutchko, C; Durieu-Trautmann, O; Strosberg, AD; Vauquelin, G | 1 |
Chuang, DM | 1 |
André, C; De Backer, JP; Strosberg, AD; Vauquelin, G | 1 |
Do-Khac, L; Harbon, S; Tanfin-Tougui, Z | 1 |
Baer, M; Chanton, C; Porzig, H | 1 |
Dietz, J; Kaiser, G; Palm, D; Reinhardt, M; Wellstein, A; Wiemer, G | 1 |
Besch, HR; Jones, LR; Manalan, AS; Watanabe, AM | 1 |
Palm, D; Wellstein, A; Wiemer, G | 1 |
Broadley, KJ; Rankin, A | 1 |
Bockaert, J; Homburger, V; Lucas, M | 1 |
Marquardt, DL; Wasserman, SI | 1 |
Abrass, IB; Scarpace, PJ | 3 |
Brockmeier, D; Palm, D; von Hattingberg, HM; Wellstein, A; Wiemer, G | 1 |
Barnes, PJ; Nadel, JA; Roberts, JM; Skoogh, BE | 1 |
Dickinson, KE; Nahorski, SR | 1 |
Chang, RS; Lotti, VJ | 1 |
Baker, SP; Posner, P | 1 |
Hayashi, E; Hayashi, M; Ishima, T; Okada, T; Tomita, T; Yamada, S | 1 |
Kusiak, JW; Pitha, J | 1 |
Gross, DM; Schmitt, CJ; Share, NN | 1 |
Delavier-Klutchko, C; Hoebeke, J; Strosberg, AD | 1 |
Meier, KE; Ruoho, AE | 1 |
Christoffersen, T; Jacobsen, S; Refsnes, M; Sager, G; Sand, TE; Sandnes, D; Westergren, T | 1 |
Koschel, K | 1 |
Baum, BJ; Ito, H; Roth, GS | 1 |
Baum, BJ; Hand, AR; Kousvelari, EE; Kusiak, JW; Pitha, J | 1 |
Hata, F; Ishida, H; Kagawa, K; Kondo, E; Kondo, S; Noguchi, Y | 1 |
Cavey, D; Cavey, MT; Gazith, J; Reichert, U; Shroot, B | 1 |
Flawiá, MM; Kornblihtt, AR; Reig, JA; Torres, HN; Torruella, M | 1 |
Beamish, RE; Corder, DW; Dhalla, NS; Heyliger, CE | 1 |
Feng, YP; Zeng, GY; Zhang, LY | 1 |
Bishopric, NH; Cohen, HJ; Lefkowitz, RJ | 1 |
Chen, TC; Cote, TE; Kebabian, JW | 1 |
Crutcher, KA; Davis, JN | 1 |
Dulis, BH; Wilson, IB | 1 |
DeLean, A; Lefkowitz, RJ; Stadel, JM | 1 |
Kuo, JF; Tse, J; Wrenn, RW | 1 |
Lefkowitz, RJ; Voeikov, VL | 1 |
Korenman, SG; Krall, JF; Levin, LC | 1 |
De Lean, A; Lefkowitz, RJ; Stadel, JM | 1 |
Davis, JN; Kistler, K | 1 |
Barnes, PJ; Dollery, CT; MacDermot, J | 1 |
Briggs, MM; Lefkowitz, RJ | 1 |
Alexander, RW; Barry, WH; Marsh, JD; Neer, EJ; Smith, TW | 1 |
Ben-David, E; Eliahou, H; Gavendo, S; Iaina, A; Kapuler, S; Serban, I | 1 |
Allred, S; Galant, SP; Griffiths, R | 1 |
Davies, JN; Wagner, HR | 1 |
Janowsky, A; Mishra, R; Sulser, F | 1 |
Barabe, J; Bockaert, J; Cantau, B; Homburger, V; Lucas, M; Penit, J | 1 |
Bhalla, RC; Ramanathan, S; Sharma, RV | 1 |
Kajiyama, H; Nomura, Y; Segawa, T | 2 |
Davies, AO; De Lean, A; Lefkowitz, RJ | 1 |
Itoh, T; Watanabe, Y; Yoshida, H | 1 |
Clark, GF; Smith, PB | 1 |
Bégin-Heick, N | 1 |
Chuang, DM; Costa, E; Farber, L; Kinnier, WJ | 1 |
Adams, K; Darovec-Beckerman, C; Manton, MA; Whitsett, JA | 1 |
Bernstein, KJ; Gangat, Y; Triner, L; Verosky, M; Vulliemoz, Y | 1 |
Ray, PD; Rufo, GA; Yorek, MA | 1 |
Barrett, JD; Korenman, SG; Krall, JF | 1 |
De Lean, A; Lefkowitz, RJ; Mullikin-Kilpatrick, D; Sawyer, DD; Stadel, JM | 1 |
Darfler, FJ; Hughes, RJ; Insel, PA | 1 |
Darfler, FJ; Insel, PA; Kennedy, MS | 1 |
Banks, P; Waddington, G | 1 |
Borst, S; Conolly, ME; Hui, KK; Kittrelle, J; Wolfe, RN | 1 |
Caron, MG; Heald, SL; Jeffs, PW; Lefkowitz, RJ; Pitha, J; Shorr, RG; Zjawiony, J | 1 |
De Lean, A; Hoffman, BB; Kent, R; Lefkowitz, RJ; Limbird, L; Michel, T; Stadel, JM | 1 |
Fujita, T; Hirata, Y; Matsukura, S; Sueoka, S; Uchihashi, M | 1 |
Tkachuk, VA; Wollemann, M | 1 |
Cardinali, DP; Luchelli de Fortis, A; Stefano, FJ; Vacas, MI | 1 |
Eden, RS; Lester, RM; Moll, ME; Wallace, AG; Williams, RS | 1 |
Fishman, PH; Mallorga, P; Tallman, JF | 2 |
De Lean, A; Lefkowitz, RJ; Stadel, JM; Stiles, GL | 1 |
Bannister, R; Boylston, AW; Davies, IB; Mathias, CJ; Sever, PS; Sudera, D | 1 |
Baker, SP; Potter, LT | 1 |
Prozialeck, WC; Pylypiw, A; Ross, L | 1 |
Abrass, IB; Davis, JL; Scarpace, PJ | 1 |
Sager, G | 2 |
Higashida, H; Kano-Tanaka, K; Kato, K; Miki, N; Nagatsu, T; Nakano, T; Tanaka, T | 1 |
Hoffman, BB; Lefkowitz, RJ | 1 |
Buja, LM; Bush, LR; Duke, RJ; Hagler, H; McCoy, KE; Mukherjee, A; Willerson, JT | 1 |
Burns, TW; Bylund, DB; Langley, PE; Terry, BE | 1 |
Hayashi, A; Nakahata, N; Suzuki, T | 1 |
Andersson, RG; Johansson, SR | 1 |
Blecher, M; Reilly, TM | 1 |
Moore, JJ; Whitsett, JA; Workman, L | 1 |
Chen, FC; Roeske, WR; Yamamura, HI | 1 |
Billingham, ME; Bristow, MR; Cubicciotti, RS; Ginsburg, R; Harrison, DC; Lurie, K; Minobe, W; Sageman, WS; Stinson, EB | 1 |
Grynne, BH; Toft, IL | 1 |
de Mazancourt, P; Giudicelli, Y; Thotakura, NR | 1 |
Galant, SP; Roan, Y | 1 |
Comai, K; Levin, BE; O'Brien, RA; Sullivan, AC | 1 |
de Vries, K; Kauffman, HF; Koëter, GH; Meurs, H | 2 |
Dax, EM; Partilla, JS | 1 |
Alexander, RW; Galper, JB; Neer, EJ; Smith, TW | 1 |
Broadley, KJ; Hawthorn, MH | 1 |
Andersson, RG; Kuo, JF; Nilsson, OR | 1 |
Kajiyama, H; Nomura, Y; Oki, K | 1 |
Nahorski, SR | 1 |
Hirai, M; Komoriyama, K; Kouyama, H; Shima, S | 2 |
Hasegawa, M; Townley, RG | 1 |
Janowsky, AJ; Manier, DH; Okada, F; Steranka, LR; Sulser, F | 1 |
Axelrod, J; Heisler, S; Reisine, T | 1 |
Caron, MG; Hoffman, BB; Hubbard, M; Lefkowitz, RJ; Stiles, GL | 1 |
Astaldi, A; Roos, D; van de Griend, RJ; van Doorn, R; Wijermans, P | 1 |
Axelrod, J; Heisler, S; Hook, VY; Reisine, TD | 1 |
Falkay, G; Kovacs, L | 1 |
Bühler, FR; Bürgisser, E; Landmann, R | 1 |
Kerry, R; Scrutton, MC | 1 |
Giudicelli, Y; Leneveu, MC; Pecquery, R | 2 |
Abbracchio, MP; Cattabeni, F; Coen, E; Omini, C; Torres-Hernandez, Y | 1 |
Boat, TF; Davis, PB; Dieckman, L; Doershuk, CF; Stern, RC | 1 |
Atkins, FL; Carney, R; Love, S | 1 |
Altszuler, N; Cherksey, B; Mendelsohn, S; Zadunaisky, J | 1 |
Kuriyama, K; Muramatsu, M; Ohkuma, S; Tamura, J | 1 |
Mineo, S; Mishima, T; Mita, H; Tomita, Y; Yamada, S; Yasueda, H | 1 |
Clutter, WE; Cryer, PE; Rosen, SG; Sérusclat, P; Shah, SD; Smith, EB | 1 |
Krzanowski, JJ; Szentivanyi, A | 1 |
Mita, H; Shida, T; Yui, Y | 1 |
Bigl, V; Rothe, T; Schliebs, R | 1 |
Carswell, H; Nahorski, SR | 1 |
Brusovanik, VI; Gorbunov, NV; Kreps, EM; Prilipko, LL; Tiurin, VA | 1 |
Hesch, RD; Meyer, T | 1 |
Britt, S; Galant, SP | 1 |
Haraguchi, K; Hashizume, K; Ichikawa, K; Kobayashi, M; Yamauchi, K | 1 |
Butcher, BT; O'Neil, CE; Reed, MA; Salvaggio, JE | 1 |
Fujiwara, M; Kornblith, PL; McKeever, PE; Nakamura, H; Reisine, TD; Shitara, N; Smith, BH | 1 |
Agli, B; Giudicelli, Y; Lacasa, D; Leneveu, A | 1 |
Levin, BE; Stoddard-Apter, S; Sullivan, AC | 1 |
Smith, PB | 1 |
Drahota, Z; Skobisová, E; Svoboda, P | 1 |
Kawai, M; Nomura, Y; Segawa, T | 1 |
Gillespie, DD; Manier, DH; Mishra, R; Sulser, F | 1 |
Arner, P; Engfeldt, P; Kimura, H; Ostman, J; Wahrenberg, H | 1 |
Kazarov, AR; Rosenkranz, AA; Sobolev, AS | 1 |
Kawai, M; Motomori-Suzaki, E; Nomura, Y; Segawa, T; Yotsumoto, I | 1 |
Gordon, MA; Johnson, DL | 1 |
Limbird, LE; MacMillan, ST | 1 |
Hudson, TH; Johnson, GL | 1 |
Asakura, M; Itirai, M; Shima, S | 1 |
Asakura, M; Hirai, M; Kawashima, Y; Shima, S | 1 |
Gether, U; Kobilka, BK; Lin, S | 1 |
McCulloch, AI; Randall, MD | 1 |
Ganguly, PK; Woo, ND | 1 |
De Montis, MG; Gambarana, C; Meloni, D | 1 |
Inagaki, C; Kitagawa, K; Morita, M; Omori, K; Uriu, T; Yasukura, T | 1 |
Austin, C; Chess-Williams, R | 1 |
Butterfield, MC; Chess-Williams, R | 1 |
Hayashi, H; Hong, RB; Ikegaya, T; Kaneko, M; Kobayashi, A; Masuda, H; Yamazaki, N | 1 |
Gavett, SH; Wills-Karp, M | 1 |
Kotwica, J; Kucharski, J; Muszynska, A; Pesta, M; Superata, J | 1 |
Iams, SG; McConnaughey, MM | 1 |
Chen, XY; Hsu, HK; Liu, MS; Tang, C | 1 |
Hsu, CH; Ma, L; Patterson, E; Robinson, CP; Thadani, U | 1 |
Gesek, FA; White, KE | 1 |
Ballesteros, JA; Gether, U; Ghanouni, P; Kobilka, BK; Lin, S; Weinstein, H | 1 |
Kobilka, BK; Lam, VT; Lee, TW; Seifert, R | 1 |
Schramm, CM | 1 |
Ito, M; Nakagawa, M; Saikawa, T; Takahashi, N; Teshima, Y; Yasunaga, S; Yonemochi, H | 1 |
McLean, AJ; Milligan, G | 1 |
Mills, S | 1 |
Chess-Williams, R; Sellers, DJ | 1 |
Liu, HY; Seifert, R; Wenzel-Seifert, K | 1 |
Chiarenza, AP; Elverdin, JC; Luchelli, MA; Vacas, MI | 1 |
Espinoza, J; Fuhrer, J; Lara, HE; Luza, SM; Miranda, C; Porcile, A; Roblero, L; Romero, C | 1 |
Bordallo, C; Cantabrana, B; Hidalgo, A; Rubín, JM; Sánchez, M; Velasco, L | 1 |
Akahane, M; Inoue, Y; Kawarabayashi, T; Kitamura, K; Kobayashi, M; Kojima, M; Sakakibara, T; Tsukamoto, T; Uzue, S | 1 |
Derkach, KV; Kuznetsova, LA; Pertseva, MN; Plesneva, SA; Shpakov, AO; Shpakova, EA; Uspenskaia, ZI | 1 |
Arias-Montaño, JA; Camacho, J; López-Colombo, A; Ramos-Jiménez, J; Reyes-Esparza, JA; Soria-Jasso, LE | 1 |
Bidasee, KR; Parbhu, SK; Patel, KP; Rozanski, GJ; Shao, CH; Zheng, H | 1 |
Bordallo, C; Bordallo, J; Cantabrana, B; Meana, C; Méndez, M; Sánchez, M; Secades, L; Velasco, L | 1 |
Aránguiz-Urroz, P; Canales, J; Carrillo, C; Copaja, M; Díaz-Araya, G; Lara, H; Lavandero, S; Troncoso, R; Vicencio, JM | 1 |
Arakawa, M; Chakraborty, R; Chelikani, P; Eilers, M; Reeves, PJ; Smith, SO; Upadhyaya, J | 1 |
7 review(s) available for dihydroalprenolol and isoproterenol
Article | Year |
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Biochemical characterization of the beta-adrenergic receptor of the frog erythrocyte.
Topics: Adenylyl Cyclases; Animals; Anura; Binding, Competitive; Dihydroalprenolol; Erythrocyte Membrane; Erythrocytes; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1979 |
Beta-adrenoceptor desensitization in the lung. A phenomenon related to prostanoids.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Dihydroalprenolol; Dinoprostone; Dose-Response Relationship, Drug; Fatty Acids; Gas Chromatography-Mass Spectrometry; Indomethacin; Isoproterenol; Lung; Prostaglandins E; Prostanoic Acids; Receptors, Adrenergic, beta; Trachea | 1985 |
Fat cell adrenoceptors: inter- and intraspecific differences and hormone regulation.
Topics: Adipose Tissue; Albuterol; Animals; Catecholamines; Clonidine; Cyclic AMP; Dihydroalprenolol; Epinephrine; Isoproterenol; Lipolysis; Methoxamine; Phenylephrine; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Species Specificity | 1985 |
Cardiac autonomic receptors. Recent concepts from radiolabeled ligand-binding studies.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Autonomic Nervous System; Columbidae; Dihydroalprenolol; Dogs; Epinephrine; Guanine Nucleotides; Guinea Pigs; Heart Conduction System; Isoproterenol; Myocardium; Pindolol; Propranolol; Rabbits; Radioligand Assay; Ranidae; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Muscarinic; Sensory Receptor Cells | 1982 |
Adrenergic receptors in the heart.
Topics: Animals; Catecholamines; Dihydroalprenolol; Humans; Hypertension; Isoproterenol; Myocardium; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1982 |
Reflections on some aspects of current research in asthma.
Topics: Animals; Asthma; Autoimmune Diseases; Dihydroalprenolol; Guinea Pigs; Humans; Hypersensitivity, Immediate; Isoproterenol; Lymphocytes; Magnetic Resonance Spectroscopy; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Drug; Tomography, Emission-Computed | 1983 |
Desensitization by antidepressants of central norepinephrine receptor systems coupled to adenylate cyclase.
Topics: Adenylyl Cyclases; Adrenal Cortex Hormones; Adrenalectomy; Animals; Antidepressive Agents; Binding, Competitive; Brain; Cyclic AMP; Desipramine; Dihydroalprenolol; Drug Tolerance; Gonadal Steroid Hormones; Hypophysectomy; Isoproterenol; Norepinephrine; Receptors, Adrenergic; Receptors, Adrenergic, beta; Serotonin; Synapses | 1984 |
1 trial(s) available for dihydroalprenolol and isoproterenol
Article | Year |
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Changes in lymphocyte beta-adrenergic receptors in depression and mania.
Topics: Adult; Bipolar Disorder; Clinical Trials as Topic; Cyclic AMP; Depressive Disorder; Desipramine; Dihydroalprenolol; Humans; In Vitro Techniques; Isoproterenol; Lithium; Lymphocytes; Middle Aged; Prostaglandins E; Receptors, Adrenergic; Receptors, Adrenergic, beta; Stimulation, Chemical | 1979 |
335 other study(ies) available for dihydroalprenolol and isoproterenol
Article | Year |
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Quantitative evaluation of the beta 2-adrenoceptor affinity of phenoxypropanolamines and phenylethanolamines.
Topics: Animals; Cattle; Chemical Phenomena; Chemistry; Dihydroalprenolol; Ethanolamines; Guanylyl Imidodiphosphate; Hydrogen-Ion Concentration; Muscles; Propanolamines; Receptors, Adrenergic, beta; Structure-Activity Relationship | 1985 |
Selective alteration in high affinity agonist binding: a mechanism of beta-adrenergic receptor desensitization.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Anura; Binding, Competitive; Dihydroalprenolol; Erythrocyte Membrane; Guanine Nucleotides; In Vitro Techniques; Indicators and Reagents; Isoproterenol; Rana pipiens; Receptors, Adrenergic; Receptors, Adrenergic, beta; Time Factors | 1979 |
The resolution of dopamine and beta 1- and beta 2-adrenergic-sensitive adenylate cyclase activities in homogenates of cat cerebellum, hippocampus and cerebral cortex.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Cats; Cerebellum; Cerebral Cortex; Dihydroalprenolol; Dopamine; Epinephrine; Fluphenazine; Hippocampus; Isoproterenol; Lung; Male; Myocardium; Receptors, Adrenergic, beta | 1979 |
In vitro modulation of CNS beta-receptor number by antidepressants and beta-agonists.
Topics: Adrenergic beta-Agonists; Animals; Antidepressive Agents; Brain; Dihydroalprenolol; In Vitro Techniques; Isoproterenol; Kinetics; Male; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Time Factors | 1979 |
Lisuride hydrogen maleate: an ergoline with beta-adrenergic antagonist activity.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Binding Sites; Cerebellum; Dihydroalprenolol; Ergolines; Isoproterenol; Lisuride; Rabbits; Spiperone | 1979 |
Differential effects of GTP on the coupling of beta-adrenergic receptors to adenylate cyclase from frog and turkey erythrocytes. Application of new methods for the analysis of receptor-effector coupling.
Topics: Adenylyl Cyclases; Animals; Anura; Dihydroalprenolol; Enzyme Activation; Erythrocyte Membrane; Erythrocytes; Guanosine Triphosphate; Isoproterenol; Kinetics; Receptors, Adrenergic; Receptors, Adrenergic, beta; Turkeys | 1979 |
Rat adipocyte beta-adrenergic receptors: evidence in favour of the heterogeneity of agonist-binding sites and against negatively cooperation interactions.
Topics: Adipose Tissue; Animals; Binding, Competitive; Cell Membrane; Dihydroalprenolol; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Male; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1979 |
Characterization of (-)-[3H]dihdroalprenolol binding sites on isolated rat fat cells.
Topics: Adipose Tissue; Alprenolol; Animals; Binding, Competitive; Cyclic AMP; Dihydroalprenolol; Female; Isoproterenol; Kinetics; Phentolamine; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1979 |
Increased number of beta-adrenergic receptors in the hypertrophied myocardium.
Topics: Alprenolol; Animals; Binding, Competitive; Cardiomegaly; Dihydroalprenolol; Isoproterenol; Male; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1979 |
Electroconvulsive treatment: rapid subsensitivity of the norepinephrine receptor coupled adenylate cyclase system in brain linked to down regulation of beta-adrenergic receptors.
Topics: Adenylyl Cyclases; Animals; Brain; Cyclic AMP; Dihydroalprenolol; Electroconvulsive Therapy; Frontal Lobe; Isoproterenol; Limbic System; Male; Norepinephrine; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1979 |
Evidence for a second desensitized state of beta-adrenergic receptor with low affinity for beta-antagonists and normal reactivity towards beta-agonists in adipocyte membranes previously exposed to beta-antagonists.
Topics: Adenylyl Cyclases; Adipose Tissue; Animals; Catecholamines; Cell Membrane; Dihydroalprenolol; Guanylyl Imidodiphosphate; Isoproterenol; Propranolol; Protein Conformation; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1979 |
The effects of common bile duct ligation upon the rat liver beta-adrenergic receptor-adenylate cylase system.
Topics: Adenylyl Cyclases; Animals; Bile Ducts; Cell Membrane; Cholestasis; Dihydroalprenolol; Disease Models, Animal; Enzyme Activation; Female; Glucagon; Isoproterenol; Kinetics; Liver; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1979 |
Denervation-induced changes in alpha and beta adrenergic receptors of the rat submandibular gland.
Topics: Animals; Binding, Competitive; Cell Membrane; Cyclic AMP; Denervation; Dihydroalprenolol; Dihydroergotoxine; Isoproterenol; Kinetics; Male; Potassium; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Submandibular Gland | 1979 |
Opposite effects of acute and repeated administration of desmethylimipramine on adrenergic responsiveness in rat pineal gland.
Topics: Animals; Ascorbic Acid; Catecholamines; Cyclic AMP; Desipramine; Dihydroalprenolol; In Vitro Techniques; Isoproterenol; Male; Norepinephrine; Pineal Gland; Rats; Sympathetic Nervous System; Time Factors | 1979 |
Ontogeny of mammalian myocardial beta-adrenergic receptors.
Topics: Animals; Dihydroalprenolol; Female; Heart; Heart Rate; In Vitro Techniques; Isoproterenol; Kinetics; Mice; Muscle Proteins; Myocardium; Pregnancy; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1979 |
Loss of beta-adrenoceptor binding sites in rat striatum following kainic acid lesions.
Topics: Animals; Axons; Corpus Striatum; Dihydroalprenolol; Isoproterenol; Kainic Acid; Male; Pyrrolidines; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1979 |
Multiple reactive sulfhydryl groups modulate the function of adenylate cyclase coupled beta-adrenergic receptors.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Anura; Dihydroalprenolol; Ethylmaleimide; In Vitro Techniques; Isoproterenol; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta; Sulfhydryl Compounds | 1979 |
A possible role of decreased relaxation mediated by beta-adrenoceptors in bladder outlet obstruction by benign prostatic hyperplasia.
Topics: Adult; Aged; Aged, 80 and over; Colforsin; Dihydroalprenolol; Humans; In Vitro Techniques; Isometric Contraction; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Muscle Relaxation; Potassium Chloride; Prazosin; Propranolol; Prostatic Hyperplasia; Radioligand Assay; Receptors, Adrenergic, beta; Urinary Bladder Neck Obstruction | 1992 |
Relationship between potency of L-isoprenaline and beta-adrenoceptor density estimated in single cells from tracheal smooth muscles of guinea pigs of different ages.
Topics: Aging; Animals; Binding, Competitive; Dihydroalprenolol; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Receptors, Adrenergic, beta; Trachea | 1992 |
Transient elevation of cardiac beta-adrenoceptor responsiveness and receptor number in the streptozotocin-diabetic rat.
Topics: Animals; Binding Sites; Blood Glucose; Calcium; Diabetes Mellitus, Experimental; Dihydroalprenolol; Female; Heart Atria; Insulin; Isoproterenol; Myocardial Contraction; Myocardium; Papillary Muscles; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1992 |
Beta-agonist-induced inhibitory-guanine-nucleotide-binding regulatory protein coupling to adenylate cyclase in mollusc Anodonta cygnea foot muscle sarcolemma.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Amino Acid Sequence; Animals; Binding Sites; Blotting, Western; Cyclic AMP; Dihydroalprenolol; Electrophoresis, Polyacrylamide Gel; GTP-Binding Proteins; Isoproterenol; Molecular Sequence Data; Mollusca; Muscles; Receptors, Adrenergic, beta; Sarcolemma | 1992 |
Effects of foetal treatment with methylazoxymethanol on noradrenergic synapses in rat cerebral cortex.
Topics: Alkylating Agents; Animals; Binding, Competitive; Cerebral Cortex; Dihydroalprenolol; Female; Fetus; Isoproterenol; Ligands; Methylazoxymethanol Acetate; Mitosis; Norepinephrine; Pregnancy; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Synapses | 1992 |
Defective response to cAMP-dependent protein kinase in non-insulin-dependent diabetic heart.
Topics: Adenylyl Cyclases; Animals; Animals, Newborn; Calcium; Cells, Cultured; Cyclic AMP; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 2; Dihydroalprenolol; Electron Transport Complex IV; Heart; Isoproterenol; Kinetics; Male; Myocardial Contraction; Myocardium; Protein Kinases; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Reference Values; Sarcolemma; Sarcoplasmic Reticulum | 1991 |
Characterization of beta-adrenoreceptors of rainbow trout (Oncorhynchus mykiss) erythrocytes.
Topics: Animals; Binding, Competitive; Cell Compartmentation; Dihydroalprenolol; Erythrocytes; Female; Hydrogen-Ion Concentration; Isoproterenol; Male; Propanolamines; Receptors, Adrenergic, beta; Trout | 1991 |
Cocaine and tracheal epithelial function: effects on short circuit current and neurotransmitter receptors.
Topics: Acetylcholine; Animals; Atropine Derivatives; Cocaine; Dihydroalprenolol; Epithelium; Isoproterenol; Ligands; Male; Parasympatholytics; Receptors, Adrenergic, beta; Receptors, Muscarinic; Sodium Channels; Swine; Trachea; Tritium | 1991 |
Differential regulation of bladder beta-adrenergic and muscarinic cholinergic receptors in experimental diabetes.
Topics: Animals; Carbachol; Diabetes Mellitus, Experimental; Dihydroalprenolol; Diuresis; In Vitro Techniques; Isoproterenol; Kinetics; Male; Pindolol; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Muscarinic; Reference Values; Sucrose; Urinary Bladder | 1991 |
Ontogeny of beta-adrenergic receptor-mediated cyclic AMP generating system in primary cultured neurons.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Aging; Animals; Brain; Cell Division; Cells, Cultured; Colforsin; Cyclic AMP; Dihydroalprenolol; Fetus; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Mice; Mice, Inbred Strains; Neurons; Pertussis Toxin; Receptors, Adrenergic, beta; Sodium Fluoride; Virulence Factors, Bordetella | 1991 |
Beta adrenergic receptor alterations in diabetic rat prostate: effects of insulin and dietary myoinositol.
Topics: Adrenergic beta-Antagonists; Animals; Blood Glucose; Body Weight; Diabetes Mellitus, Experimental; Dihydroalprenolol; Dose-Response Relationship, Drug; Drinking; Inositol; Insulin; Isoproterenol; Male; Organ Size; Propanolamines; Propranolol; Prostate; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Streptozocin; Urination | 1991 |
Adrenalectomy-induced alterations in glucagon binding and lipolysis in isolated rat adipocytes.
Topics: 1-Methyl-3-isobutylxanthine; Adenosine Deaminase; Adipose Tissue; Adrenalectomy; Animals; Bucladesine; Cyclic AMP; Dihydroalprenolol; Glucagon; Isoproterenol; Lipolysis; Male; Rats; Rats, Inbred Strains; Receptors, Gastrointestinal Hormone; Receptors, Glucagon | 1990 |
Inverse regulation of calcium channels and beta-adrenergic receptors in virus-transformed human embryonal cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Ca(2+) Mg(2+)-ATPase; Calcium Channels; Cell Line, Transformed; Cell Transformation, Viral; Cyclic AMP; Dihydroalprenolol; Embryo, Mammalian; Humans; Isoproterenol; Muscle, Smooth; Phenylephrine; Radioimmunoassay; Receptors, Adrenergic, beta; Simplexvirus; Trifluoperazine | 1991 |
Reconstitutively active G protein-coupled receptors purified from baculovirus-infected insect cells.
Topics: Adenylyl Cyclases; Animals; Base Sequence; Cell Line; Cell Membrane; Dihydroalprenolol; Epinephrine; Genetic Vectors; GTP-Binding Proteins; Humans; Insect Viruses; Insecta; Iodocyanopindolol; Isoproterenol; Kinetics; Ligands; Molecular Sequence Data; Molecular Weight; Norepinephrine; Pindolol; Receptors, Adrenergic, beta; Receptors, Muscarinic; Turkeys | 1991 |
Serotonergic neurons do not influence the regulation of beta adrenoceptors induced by either desipramine or isoproterenol.
Topics: 5,7-Dihydroxytryptamine; Animals; Desipramine; Dihydroalprenolol; Isoproterenol; Male; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin | 1991 |
Diabetes-induced changes in cardiac beta-adrenoceptor responsiveness: effects of aldose reductase inhibition with ponalrestat.
Topics: Aldehyde Reductase; Animals; Calcium; Colforsin; Diabetes Mellitus, Experimental; Dihydroalprenolol; Female; Heart; In Vitro Techniques; Isoproterenol; Myocardium; Phthalazines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1991 |
Interaction between alpha 2- and beta-adrenergic receptors in rat cerebral cortical membranes: clonidine-induced reduction in agonist and antagonist affinity for beta-adrenergic receptors.
Topics: Animals; Binding, Competitive; Cerebral Cortex; Clonidine; Dihydroalprenolol; Guanosine Triphosphate; Isoproterenol; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Sympathomimetics; Yohimbine | 1991 |
Platelet-activating factor induces nonspecific desensitization to bronchodilators in guinea pigs.
Topics: Airway Resistance; Animals; Desensitization, Immunologic; Dihydroalprenolol; Dinoprostone; Drug Interactions; Guinea Pigs; Isoproterenol; Lung; Male; Methacholine Chloride; Platelet Activating Factor; Tritium | 1991 |
Antagonist characterization of atypical beta adrenoceptors in guinea pig ileum: blockade by alprenolol and dihydroalprenolol.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Dihydroalprenolol; Drug Interactions; Guinea Pigs; Ileum; In Vitro Techniques; Isoproterenol; Male; Muscle, Smooth; Propranolol; Receptors, Adrenergic, beta | 1990 |
Pretreatment with N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline accelerates the electroshock-induced decrease in density of beta-adrenoceptors but not functional downregulation.
Topics: Adrenergic alpha-Antagonists; Animals; Catecholamines; Cerebral Cortex; Cyclic AMP; Dihydroalprenolol; Down-Regulation; Electroshock; Isoproterenol; Male; Quinolines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1990 |
Reovirus type 3 binds to antagonist domains of the beta-adrenergic receptor.
Topics: Adrenal Gland Neoplasms; Animals; Binding, Competitive; Dihydroalprenolol; Glioma; Isoproterenol; Kinetics; L Cells; Mammalian orthoreovirus 3; Mice; Receptors, Adrenergic, beta; Reoviridae; Spiperone | 1990 |
Deficiency of beta-adrenoceptor-mediated relaxation in suncus trachea.
Topics: Animals; Colforsin; Dihydroalprenolol; Eulipotyphla; Guinea Pigs; In Vitro Techniques; Isoproterenol; Kinetics; Male; Membranes; Muscle Relaxation; Muscle, Smooth; Rats; Receptors, Adrenergic, beta; Species Specificity; Trachea | 1990 |
Chronic isoproterenol administration causes altered beta adrenoceptor-Gs-coupling in guinea pig lung.
Topics: Animals; Binding, Competitive; Dihydroalprenolol; Guanosine Triphosphate; Guinea Pigs; Isoproterenol; Lung; Male; Muscle Relaxation; Receptors, Adrenergic, beta | 1990 |
Functional beta-adrenergic receptors in breast cancer cells.
Topics: Breast Neoplasms; Cyclic AMP; Dihydroalprenolol; Female; Humans; Isoproterenol; Receptors, Adrenergic, beta; Tumor Cells, Cultured | 1990 |
Role of beta-adrenoceptor-adenylate cyclase system in the developmental decrease in sensitivity to isoprenaline in foetal and neonatal rat heart.
Topics: Adenylyl Cyclases; Aging; Animals; Animals, Newborn; Colforsin; Dihydroalprenolol; Enzyme Activation; Female; Fetus; Heart; Heart Rate; Isoproterenol; Kinetics; Myocardial Contraction; Myocardium; Pregnancy; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1990 |
Effect of aging on the response of guinea pig trachea to isoprenaline.
Topics: Aging; Animals; Corticosterone; Dihydroalprenolol; Guinea Pigs; In Vitro Techniques; Isoproterenol; Kinetics; Male; Microsomes; Muscle Contraction; Propranolol; Receptors, Adrenergic, beta; Trachea | 1990 |
Increased number of beta-adrenergic receptors on cells of the rat adenohypophysis after thyroid hormone administration.
Topics: Animals; Cyclic AMP; Dihydroalprenolol; Isoproterenol; Male; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Thyroxine; Triiodothyronine | 1990 |
Modulation of cardiac beta-adrenergic receptors by dopamine beta-hydroxylase.
Topics: Animals; Dihydroalprenolol; Dopamine beta-Hydroxylase; Heart Ventricles; In Vitro Techniques; Isoproterenol; Kinetics; Myocardial Contraction; Myocardium; Organ Specificity; Rats; Receptors, Adrenergic, beta; Sarcolemma | 1990 |
Identification and characterization of the beta-adrenergic receptor on neuroblastoma x glioma hybrid NG108-15 cells.
Topics: Alprenolol; Bucladesine; Catecholamines; Cell Differentiation; Dihydroalprenolol; Glioma; Hybrid Cells; Isoproterenol; Kinetics; Neuroblastoma; Receptors, Adrenergic, beta; Stereoisomerism; Tumor Cells, Cultured | 1990 |
Increased number of beta-adrenoceptors in cultured heart cells after propranolol withdrawal.
Topics: Animals; Binding Sites; Cyclic AMP; Dihydroalprenolol; Isoproterenol; Myocardial Contraction; Myocardium; Propranolol; Receptors, Adrenergic, beta | 1990 |
Altered plasma catecholamines and numbers of alpha- and beta-adrenergic receptors in platelets and leucocytes in hyperthyroid patients normalized under antithyroid treatment.
Topics: Adenylyl Cyclases; Adult; Aged; Antithyroid Agents; Blood Platelets; Cell Membrane; Cyclic AMP; Dihydroalprenolol; Epinephrine; Female; Humans; Hyperthyroidism; Isoproterenol; Male; Middle Aged; Monocytes; Norepinephrine; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine | 1985 |
Increased beta-adrenoceptor binding capacity is associated with blunted beta-adrenoceptor-mediated cardiovascular responses in essential hypertension.
Topics: Adult; Catecholamines; Dihydroalprenolol; Humans; Hypertension; Isoproterenol; Leukocytes; Middle Aged; Receptors, Adrenergic, beta; Renin | 1985 |
Characterization of purified dog mastocytoma cells. Autonomic membrane receptors and pharmacologic modulation of histamine release.
Topics: Acetylcholine; Animals; Cyclic AMP; Dihydroalprenolol; Dogs; Histamine Release; In Vitro Techniques; Isoproterenol; Mast-Cell Sarcoma; Phenylephrine; Prazosin; Propranolol; Quinuclidinyl Benzilate; Radioligand Assay; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Cholinergic; Terbutaline | 1985 |
Stimulation of beta-adrenoceptors inhibits calcium-dependent potassium-channels in mouse macrophages.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Calcimycin; Calcium; Cyclic AMP; Dihydroalprenolol; Ethers; Female; Ion Channels; Ionomycin; Isoproterenol; Kinetics; Macrophages; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Potassium; Propranolol; Receptors, Adrenergic, beta | 1986 |
Beta-adrenoceptor blocking activity of diprafenone in anesthetized dogs: comparison with propafenone and propranolol.
Topics: Adrenergic beta-Antagonists; Anesthesia; Animals; Anti-Arrhythmia Agents; Dihydroalprenolol; Dogs; Female; Heart; Isoproterenol; Male; Membranes; Myocardium; Propafenone; Propranolol; Receptors, Adrenergic, beta | 1989 |
Cytosolic factor(s) determines the impaired desensitization of beta-adrenoceptors in the myocardium of spontaneously hypertensive rats.
Topics: Animals; Cell Membrane; Cytosol; Dihydroalprenolol; Isoproterenol; Kinetics; Male; Myocardium; Protease Inhibitors; Protein Kinase Inhibitors; Protein Kinases; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta | 1989 |
Electrophysiological responsiveness to isoproterenol in rat hippocampal slices correlates with changes in beta-adrenergic receptor density induced by chronic morphine treatment.
Topics: Action Potentials; Animals; Dihydroalprenolol; Hippocampus; In Vitro Techniques; Isoproterenol; Male; Morphine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Time Factors | 1989 |
Comparison of two putatively selective radioligands for labeling central nervous system beta-adrenergic receptors: inadequacy of [3H]dihydroalprenolol.
Topics: Alprenolol; Animals; Brain Chemistry; Dihydroalprenolol; Guanosine Triphosphate; Isoproterenol; Kinetics; Male; Propanolamines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin | 1989 |
Chronotropic responses in rats implanted with an acrylic orthopaedic cement.
Topics: Acrylates; Animals; Bone Cements; Bucladesine; Calcium Chloride; Dihydroalprenolol; Female; Glucagon; Heart Rate; Isoproterenol; Papillary Muscles; Rats; Rats, Inbred Strains | 1989 |
Role of thromboxanes in alterations of the diabetic beta-adrenergic system.
Topics: Animals; Biphenyl Compounds; Diabetes Mellitus, Experimental; Dihydroalprenolol; Isoproterenol; Male; Myocardial Contraction; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Sodium-Potassium-Exchanging ATPase; Thromboxane B2 | 1989 |
In vitro pharmacological properties of a series of isoprenaline derivatives.
Topics: Animals; Aorta, Thoracic; Binding, Competitive; Catecholamines; Dihydroalprenolol; Dobutamine; Dogs; Electrophysiology; Female; Guinea Pigs; In Vitro Techniques; Isomerism; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Myocardial Contraction; Papillary Muscles; Potassium; Propanolamines; Rabbits; Receptors, Adrenergic, beta; Xamoterol | 1989 |
Decreased glucagon binding and glucagon-stimulated lipolysis in adipocytes from streptozotocin-diabetic rats.
Topics: Adipose Tissue; Animals; Diabetes Mellitus, Experimental; Dihydroalprenolol; Glucagon; Isoproterenol; Lipolysis; Male; Rats; Rats, Inbred Strains; Receptors, Gastrointestinal Hormone; Receptors, Glucagon | 1989 |
Differential interaction of guanabenz with receptor binding sites in rat brain and kidney.
Topics: Animals; Binding, Competitive; Brain; Clonidine; Dihydroalprenolol; Guanabenz; Guanidines; Guanine Nucleotides; In Vitro Techniques; Isoproterenol; Kidney; Kinetics; Male; Membranes; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Temperature | 1989 |
Distribution and subtype determination of beta-receptors in the spinal cord of the adult rat.
Topics: Adenylyl Cyclases; Animals; Atenolol; Binding, Competitive; Dihydroalprenolol; Isoproterenol; Male; Practolol; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Spinal Cord | 1989 |
Neuropeptides modulate beta-adrenergic agonist binding and receptor downregulation in slices of rat brain.
Topics: Adrenergic beta-Agonists; Adrenocorticotropic Hormone; Animals; Binding, Competitive; Brain; Dihydroalprenolol; Egtazic Acid; In Vitro Techniques; Isoproterenol; Male; Neuropeptides; Rats; Receptors, Adrenergic, beta | 1989 |
An in vivo procedure for the selective inactivation of rat brain cerebral cortical alpha-adrenoceptors using N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ).
Topics: Adrenergic alpha-Antagonists; Animals; Cell Membrane; Cerebral Cortex; Clonidine; Cyclic AMP; Dihydroalprenolol; Inositol Phosphates; Isoproterenol; Male; Norepinephrine; Prazosin; Quinolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine | 1989 |
Effects of calcium channel blockers and ketotifen on beta 2 adrenergic receptor regulation in intact human lymphocytes.
Topics: Adrenergic beta-Antagonists; Calcium Channel Blockers; Cyclic AMP; Dihydroalprenolol; Humans; In Vitro Techniques; Isoproterenol; Ketotifen; Lymphocytes; Propanolamines; Radioimmunoassay; Receptors, Adrenergic, beta | 1989 |
Beta-adrenoceptors in human brain labelled with [3H]dihydroalprenolol and [3H]CGP 12177.
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Brain Chemistry; Dihydroalprenolol; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Practolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 1989 |
Characterization of the inducible serotonin-sensitive dihydroalprenolol binding sites with low affinity for isoproterenol.
Topics: 5,7-Dihydroxytryptamine; Alprenolol; Animals; Binding, Competitive; Brain; Cerebral Ventricles; Dihydroalprenolol; Dihydroxytryptamines; Injections, Intraventricular; Isoproterenol; Kinetics; Male; Rats; Rats, Inbred Strains; Reference Values; Regression Analysis; Serotonin | 1989 |
Characterization of dog fat cell adrenoceptors: variations in alpha-2 and beta adrenergic receptors distribution according to the extent of the fat deposits and the anatomical location.
Topics: Adipose Tissue; Animals; Binding, Competitive; Brimonidine Tartrate; Clonidine; Cyclic AMP; Dihydroalprenolol; Dogs; Epinephrine; Humans; Isoproterenol; Lipolysis; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine | 1987 |
Cardiac post-junctional alpha 1- and beta-adrenoceptors: effects of chronic chemical sympathectomy with 6-hydroxydopamine.
Topics: Animals; Dihydroalprenolol; Guinea Pigs; Heart; Hydroxydopamines; Isoproterenol; Male; Methoxamine; Myocardial Contraction; Oxidopamine; Prazosin; Propranolol; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Sympathectomy, Chemical; Sympathetic Nervous System | 1987 |
Alterations in cardiac beta-adrenoceptor responsiveness and adenylate cyclase system by congestive heart failure in dogs.
Topics: 5'-Nucleotidase; Adenylyl Cyclases; Animals; Chlorides; Colforsin; Dihydroalprenolol; Dobutamine; Dogs; Guanylyl Imidodiphosphate; Heart Failure; Hemodynamics; In Vitro Techniques; Isoproterenol; Kinetics; Manganese; Manganese Compounds; Myocardium; Norepinephrine; Nucleotidases; Receptors, Adrenergic, beta | 1987 |
Haemophilus influenzae-induced decreases in lung beta-adrenoceptor function and number coincide with decreases in spleen noradrenaline.
Topics: Airway Resistance; Animals; Carbachol; Dihydroalprenolol; Guinea Pigs; Haemophilus influenzae; Isoproterenol; Lung; Male; Norepinephrine; Receptors, Adrenergic, beta; Respiratory Hypersensitivity; Spleen | 1987 |
Protein kinases induce isoproterenol desensitization of beta-adrenoceptor-coupled adenylate cyclase system: significance of receptor occupancy.
Topics: Adenylyl Cyclase Inhibitors; Alprostadil; Animals; Bucladesine; Colforsin; Cyclic AMP; Dihydroalprenolol; Guanylyl Imidodiphosphate; In Vitro Techniques; Isoproterenol; Male; Protein Kinase Inhibitors; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Reticulocytes; Theophylline | 1987 |
Time course of resensitization of rat uterine beta-adrenoceptor system.
Topics: Animals; Cyclic AMP; Dihydroalprenolol; Female; Isoproterenol; Kinetics; Myometrium; Phosphoric Diester Hydrolases; Rats; Receptors, Adrenergic, beta | 1988 |
Effects of chronic isoproterenol administration on beta 1-adrenoceptors and growth of pancreas of young and adult rats.
Topics: Aging; Animals; Atenolol; Butoxamine; Cell Differentiation; Cell Membrane; Dihydroalprenolol; DNA; Isoproterenol; Pancreas; Parotid Gland; Quinuclidinyl Benzilate; Rats; Receptors, Adrenergic, beta | 1988 |
Molecular and biological interaction between major histocompatibility complex class I antigens and luteinizing hormone receptors or beta-adrenergic receptors triggers cellular response in mice.
Topics: Animals; Antibodies, Monoclonal; Atrial Function; Cell Membrane; Chorionic Gonadotropin; Dihydroalprenolol; Heart Rate; Histocompatibility Antigens; Immune Sera; Immunization; Immunoglobulin Allotypes; Immunoglobulin G; Immunosorbent Techniques; Isoproterenol; Leydig Cells; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C3H; Myocardial Contraction; Propranolol; Receptors, Adrenergic, beta; Receptors, LH; Testosterone | 1988 |
Beta-adrenergic receptor binding characteristics and responsiveness in cultured Wistar-Kyoto rat arterial smooth muscle cells.
Topics: Animals; Binding, Competitive; Cells, Cultured; Cyclic AMP; Dihydroalprenolol; Isoproterenol; Kinetics; Male; Muscle, Smooth, Vascular; Rats; Rats, Inbred WKY; Receptors, Adrenergic, beta | 1988 |
Glucocorticoid modulation of beta-adrenergic receptors of cultured rat arterial smooth muscle cells.
Topics: Animals; Arteries; Cells, Cultured; Cyclic AMP; Dihydroalprenolol; Glucocorticoids; Isoproterenol; Muscle, Smooth, Vascular; Rats; Rats, Inbred WKY; Receptors, Adrenergic, beta | 1988 |
Differential effects of fluoride on adenylate cyclase activity and guanine nucleotide regulation of agonist high-affinity receptor binding.
Topics: Adenylyl Cyclases; Alprostadil; Animals; Anura; Cell Membrane; Cells, Cultured; Colforsin; Dihydroalprenolol; Epinephrine; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Iodocyanopindolol; Isoproterenol; Pindolol; Receptors, Adrenergic, beta; Sodium Fluoride; Yohimbine | 1988 |
Effects of ketotifen on the responsiveness of peripheral blood lymphocyte beta-adrenergic receptors.
Topics: Adolescent; Adult; Aged; Asthma; Cyclic AMP; Dihydroalprenolol; Female; Humans; In Vitro Techniques; Isoproterenol; Ketotifen; Lymphocytes; Male; Middle Aged; Receptors, Adrenergic, beta | 1988 |
Electroconvulsive shock decreases beta-adrenoceptors despite serotonin lesions.
Topics: 5,7-Dihydroxytryptamine; Animals; Dihydroalprenolol; Electroshock; Isoproterenol; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin | 1988 |
Characterization of beta-adrenoceptors in myometrium of preparturient rats.
Topics: Animals; Binding Sites; Binding, Competitive; Dihydroalprenolol; Female; In Vitro Techniques; Isoproterenol; Kinetics; Labor, Obstetric; Myometrium; Pregnancy; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Uterine Contraction | 1988 |
Irreversible blockade of beta-adrenergic receptors with a bromoacetyl derivative of pindolol.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Dihydroalprenolol; Erythrocytes; Glioma; In Vitro Techniques; Isoproterenol; Pindolol; Rats; Receptors, Adrenergic, beta | 1985 |
A possible mechanism in interaction of a partial agonist with beta-adrenoceptor in guinea-pig taenia caecum: effects of Gpp(NH)p on its two different binding sites.
Topics: Adrenergic beta-Agonists; Animals; Binding Sites; Dihydroalprenolol; Dose-Response Relationship, Drug; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Guinea Pigs; In Vitro Techniques; Intestines; Isoproterenol; Kinetics; Male; Propanolamines; Receptors, Adrenergic, beta | 1985 |
Acute change in the cyclic AMP content of rat mammary acini in vitro. Influence of physiological and pharmacological agents.
Topics: Adrenergic Agonists; Animals; Colforsin; Cyclic AMP; Dihydroalprenolol; Female; Humans; Imidazoles; Isoproterenol; Ligands; Mammary Glands, Animal; Rats; Rats, Inbred Strains; Receptors, Adrenergic | 1985 |
Agonist-induced redistribution of beta-adrenergic receptors on intact human mononuclear leukocytes: redistributed receptors are nonfunctional.
Topics: Adrenergic beta-Antagonists; Adult; Cyclic AMP; Dihydroalprenolol; Humans; In Vitro Techniques; Isoproterenol; Kinetics; Leukocytes; Ligands; Male; Propanolamines; Receptors, Adrenergic, beta | 1985 |
[Effect of pH changes on the binding of agonists and antagonists to the adrenergic beta receptor].
Topics: Acid-Base Equilibrium; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding Sites; Dihydroalprenolol; Dogs; Hydrogen-Ion Concentration; Isoproterenol; Myocardium; Norepinephrine; Receptors, Adrenergic, beta | 1985 |
MY336-a, a novel beta-adrenergic receptor antagonist produced by Streptomyces gabonae.
Topics: Adrenergic beta-Antagonists; Animals; Brain; Cells, Cultured; Dihydroalprenolol; Dogs; Drug Interactions; Guinea Pigs; Isoproterenol; Isoquinolines; Kinetics; Lung; Male; Muscle, Smooth; Myocardial Contraction; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Tetrahydroisoquinolines; Tritium | 1986 |
Differential recovery of beta adrenoreceptor antagonist and agonist high affinity binding sites in the guinea-pig lung after irreversible blockade.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Binding Sites; Dihydroalprenolol; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Lung; Receptors, Adrenergic, beta; Tritium | 1986 |
The significance of beta-adrenoceptor down regulation in the desipramine action in the forced swimming test.
Topics: Adrenergic beta-Antagonists; Animals; Cerebral Cortex; Desipramine; Dihydroalprenolol; Drug Administration Schedule; Isoproterenol; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Swimming | 1986 |
Effects of phospholipases C on the beta-receptor-adenylate cyclase system of chick erythrocyte membranes.
Topics: Adenylyl Cyclases; Animals; Bacillus cereus; Bacillus thuringiensis; Binding, Competitive; Chickens; Clostridium perfringens; Dihydroalprenolol; Dose-Response Relationship, Drug; Epinephrine; Erythrocyte Membrane; Isoproterenol; Norepinephrine; Propranolol; Receptors, Adrenergic, beta; Sphingomyelin Phosphodiesterase; Type C Phospholipases | 1986 |
Shallow agonist competition binding curves for beta-adrenergic receptors: the role of tight agonist binding.
Topics: Adrenergic beta-Agonists; Animals; Binding, Competitive; Cattle; Dihydroalprenolol; GTP-Binding Proteins; Guanosine Triphosphate; In Vitro Techniques; Isoproterenol; Muscles; Receptors, Adrenergic, beta; Time Factors | 1987 |
Calculated and actual changes in beta-adrenoceptor number associated with increases in rat and guinea-pig cardiac sensitivity.
Topics: Animals; Dihydroalprenolol; Guinea Pigs; Heart; Hydroxydopamines; In Vitro Techniques; Isoproterenol; Kinetics; Male; Myocardial Contraction; Oxidopamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Reserpine | 1986 |
Structure-activity relationships of beta-adrenergic receptor-coupled adenylate cyclase: implications of a redox mechanism for the action of agonists at beta-adrenergic receptors.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adrenochrome; Animals; Anura; Benzoquinones; Catecholamines; Chromatography, Liquid; Dihydroalprenolol; Electrochemistry; Erythrocyte Membrane; Isoproterenol; Kinetics; Oxidation-Reduction; Quinones; Receptors, Adrenergic, beta; Structure-Activity Relationship | 1987 |
Comparative studies with the enantiomers of the glycol metabolite of propranolol and their effects on the cardiac beta-adrenoceptor.
Topics: Animals; Dihydroalprenolol; Heart; In Vitro Techniques; Isoproterenol; Kinetics; Male; Myocardial Contraction; Myocardium; Propranolol; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Stereoisomerism | 1987 |
External transport of beta-adrenergic binding sites in ischemic myocardium.
Topics: Adrenergic beta-Antagonists; Animals; Biological Transport, Active; Dihydroalprenolol; Dogs; Isoproterenol; Myocardium; Propranolol; Receptors, Adrenergic, beta | 1987 |
Effects of neurotransmitters on astrocyte glycogen stores in vitro.
Topics: Animals; Animals, Newborn; Astrocytes; Bucladesine; Carbachol; Cells, Cultured; Cerebral Cortex; Colforsin; Dihydroalprenolol; Glycogen; Isoproterenol; Neurotransmitter Agents; Norepinephrine; Phenylephrine; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Receptors, Adrenergic; Receptors, Muscarinic; Receptors, Serotonin; Reserpine; Serotonin | 1988 |
Estrogen increases beta-adrenergic binding in the preterm fetal rabbit lung.
Topics: Amnion; Animals; Binding, Competitive; Dihydroalprenolol; Epinephrine; Estrogens; Female; Fetus; Isoproterenol; Lung; Models, Biological; Norepinephrine; Pregnancy; Rabbits; Receptors, Adrenergic, beta | 1985 |
Altered binding properties of beta-adrenergic receptors and lack of coupling to adenylate cyclase in P815 mastocytoma cells.
Topics: Adenylyl Cyclases; Animals; Cell Line; Cell Membrane; Colforsin; Cyclic AMP; Dihydroalprenolol; Diterpenes; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Mast-Cell Sarcoma; Mice; Mice, Inbred DBA; Neoplasm Proteins; Receptors, Adrenergic, beta; Sarcoma, Experimental; Sodium Fluoride | 1985 |
Characterization of beta-adrenergic receptors in fresh and primary cultured bovine corneal endothelium.
Topics: Animals; Cattle; Cells, Cultured; Cornea; Cyclic AMP; Dihydroalprenolol; Endothelium; Epinephrine; Isoproterenol; Norepinephrine; Propranolol; Receptors, Adrenergic, beta; Time Factors | 1985 |
Increase in serotonin2 receptor density in rat cerebral cortex slices by stimulation of beta-adrenergic receptors.
Topics: Animals; Cerebral Cortex; Dihydroalprenolol; Electroshock; Hydrogen-Ion Concentration; In Vitro Techniques; Isoproterenol; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin; Spiperone | 1985 |
Reduction of the cyclic adenosine 3',5'-monophosphate response to catecholamines in rat brain slices after repeated restraint stress.
Topics: Adrenocorticotropic Hormone; Animals; Brain; Cerebral Cortex; Cyclic AMP; Dihydroalprenolol; Humans; Hypothalamus; Indomethacin; Isoproterenol; Male; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Restraint, Physical; Stress, Psychological | 1985 |
Direct insertion and fluorescence studies of rhodamine-labeled beta-adrenergic receptors in cell membranes.
Topics: Animals; Cell Membrane; Cyclic AMP; Dihydroalprenolol; Erythrocyte Membrane; Islets of Langerhans; Isoproterenol; Kinetics; Male; Rana catesbeiana; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Rhodamines; Tritium | 1985 |
[Mechanisms of the disorder of the hormonal regulation of plasma membrane adenylate cyclase in the rat liver during early ontogeny under in vitro irradiation].
Topics: Adenylyl Cyclases; Animals; Cell Membrane; Dihydroalprenolol; Dose-Response Relationship, Radiation; Enzyme Activation; Fetus; Gamma Rays; Isoproterenol; Liver; Protein Binding; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1985 |
Factors controlling beta 1-adrenoceptor affinity and selectivity.
Topics: Animals; Cattle; Dihydroalprenolol; Guanylyl Imidodiphosphate; Hydrogen-Ion Concentration; In Vitro Techniques; Isoproterenol; Kinetics; Myocardium; Receptors, Adrenergic, beta; Structure-Activity Relationship; Tritium | 1985 |
Hepatic adenylate cyclase. Development-dependent coupling to the beta-adrenergic receptor in the neonate.
Topics: Adenylyl Cyclases; Aging; Animals; Animals, Newborn; Cell Membrane; Cholera Toxin; Dihydroalprenolol; Fetus; Guanosine Triphosphate; Isoproterenol; Kinetics; Liver; Male; Rabbits; Receptors, Adrenergic, beta | 1985 |
Evidence for two specific affinity states of 3H-antagonist binding to cardiac beta-adrenergic receptors and influence of Gpp(NH)p.
Topics: Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Male; Myocardium; Propanolamines; Rats; Receptors, Adrenergic, beta | 1985 |
A role for adenylate cyclase in the subsensitivity to isoproterenol during ontogenesis of the embryonic chick ventricle.
Topics: Adenylyl Cyclases; Animals; Chick Embryo; Chickens; Chlorides; Colforsin; Cyclic AMP; Dihydroalprenolol; Dose-Response Relationship, Drug; Drug Interactions; Guanylyl Imidodiphosphate; Heart; Isoproterenol; Kinetics; Magnesium; Manganese; Manganese Compounds; Muscle Contraction; Myocardium; Receptors, Adrenergic, beta; Sodium Fluoride | 1985 |
Selective protection of cells against X-irradiation. Isoproterenol protects only those cells that possess beta-adrenoreceptors.
Topics: Adenylyl Cyclases; Alprostadil; Animals; Cell Line; Cricetinae; Cyclic AMP; Dihydroalprenolol; Fibroblasts; Isoproterenol; Mice; Propranolol; Receptors, Adrenergic, beta | 1985 |
Age-related reduction of beta-adrenoceptor sensitivity in rat heart occurs by multiple mechanisms.
Topics: Adenylyl Cyclases; Aging; Animals; Cyclic AMP; Dihydroalprenolol; Heart; Isoproterenol; Kinetics; Male; Myocardium; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta | 1985 |
Irreversible inactivation of the beta-adrenoreceptor by a partial agonist. Evidence for selective loss of the agonist high affinity binding sites.
Topics: Adenylyl Cyclases; Animals; Dihydroalprenolol; Guanylyl Imidodiphosphate; Hot Temperature; Isoproterenol; Kinetics; Lung; Norepinephrine; Propranolol; Rats; Receptors, Adrenergic, beta | 1985 |
Arachidonic acid metabolites induce beta-adrenoceptor desensitization in rat lung in vitro.
Topics: Adenylyl Cyclases; Animals; Arachidonic Acid; Arachidonic Acids; Dihydroalprenolol; Dose-Response Relationship, Drug; In Vitro Techniques; Indomethacin; Isoproterenol; Lung; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1985 |
Mechanisms of decreased cerebrospinal fluid production by radiographic contrast media: role of adenylate cyclase activation.
Topics: Adenylyl Cyclases; Animals; Cerebrospinal Fluid; Contrast Media; Diatrizoate; Dihydroalprenolol; Dogs; Dose-Response Relationship, Drug; Enzyme Activation; In Vitro Techniques; Isoproterenol; Male; Receptors, Adrenergic, beta; Tritium | 1986 |
Temperature and isoproterenol modulation of beta-adrenergic receptor characteristics.
Topics: Animals; Binding, Competitive; Cell Membrane; Cold Temperature; Dihydroalprenolol; Isoproterenol; Lung; Nadolol; Propanolamines; Rats; Receptors, Adrenergic, beta | 1986 |
Alpha- and beta-adrenergic receptor activity in circulating blood cells of patients with phaeochromocytoma: effects of adrenalectomy.
Topics: Adrenal Gland Neoplasms; Adrenalectomy; Adult; Blood Platelets; Cyclic AMP; Dihydroalprenolol; Epinephrine; Female; Humans; Hydrocortisone; Isoproterenol; Male; Middle Aged; Monocytes; Norepinephrine; Pheochromocytoma; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine | 1986 |
Functional and biochemical modifications of lung beta-adrenoreceptors after in vivo desensitization: prevention by indomethacin.
Topics: Adenylyl Cyclases; Animals; Cyclic AMP; Dihydroalprenolol; Indomethacin; Injections, Intraperitoneal; Isoproterenol; Lung; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Tritium | 1986 |
Mechanism responsible for "down regulation" during successive beta-agonist administration in rat hearts.
Topics: Adenosine Triphosphate; Animals; Cell Membrane; Dihydroalprenolol; Fatty Acids; Isoproterenol; Male; Myocardium; Phospholipases; Phospholipases A; Phospholipids; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1985 |
Dexamethasone effects on beta-adrenergic receptors and adenylate cyclase regulatory proteins Gs and Gi in ROS 17/2.8 cells.
Topics: Adenosine Diphosphate Ribose; Adenylyl Cyclases; Animals; Cell Line; Cholera Toxin; Cyclic AMP; Cycloheximide; Dexamethasone; Dihydroalprenolol; Enzyme Activation; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Molecular Weight; NAD; Osteosarcoma; Rats; Receptors, Adrenergic, beta | 1986 |
Agonist-mediated conformational changes of beta-adrenoceptors could occur independent of functional coupling to Ns.
Topics: Adenylyl Cyclases; Animals; Dihydroalprenolol; Erythrocyte Membrane; Ethylmaleimide; GTP-Binding Proteins; In Vitro Techniques; Isoproterenol; Kinetics; Protein Conformation; Receptors, Adrenergic, beta; Thermodynamics; Turkeys | 1986 |
Stress induced desensitization of lymphocyte beta-adrenoceptors in young and aged rats.
Topics: Age Factors; Animals; Corticosterone; Dihydroalprenolol; Isoproterenol; Lymphocytes; Male; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Restraint, Physical; Stress, Physiological | 1986 |
Effect of serum, alpha-1 acid glycoprotein, lipoproteins and albumin on human mononuclear leucocyte beta-adrenoceptors.
Topics: Alprenolol; Blood; Blood Proteins; Cyclic AMP; Dihydroalprenolol; Humans; Isoproterenol; Leukocytes; Lipoproteins; Orosomucoid; Propranolol; Receptors, Adrenergic, beta; Serum Albumin; Theophylline | 1986 |
[Interindividual changes in the specific binding of 3H-dihydroalprenolol by beta 2-adrenergic lymphocytic receptors in essential hypertension].
Topics: Adult; Alprenolol; Dihydroalprenolol; Humans; Hypertension; Isoproterenol; Lymphocytes; Male; Receptors, Adrenergic, beta | 1986 |
Characteristics of myocardial beta-adrenergic receptors during endotoxicosis in the rat.
Topics: Animals; Binding, Competitive; Dihydroalprenolol; Endotoxins; Isoproterenol; Male; Myocardium; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Salmonella enteritidis | 1986 |
The effects of 4-hydroxy-2,3-trans-nonenal on beta-adrenoceptors of rat lung membranes.
Topics: Aldehydes; Alkylation; Animals; Dihydroalprenolol; In Vitro Techniques; Isoproterenol; Lipid Peroxides; Lung; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1986 |
Deglycosylated mammalian beta 2-adrenergic receptors are still able to undergo functional coupling to Ns.
Topics: Adenylyl Cyclases; Affinity Labels; Animals; Cell Membrane; Chromatography, Affinity; Cricetinae; Dihydroalprenolol; Ethylmaleimide; Glycoside Hydrolases; Glycosylation; Iodocyanopindolol; Isoproterenol; Lung; Mannosyl-Glycoprotein Endo-beta-N-Acetylglucosaminidase; Neuraminidase; Photochemistry; Pindolol; Receptors, Adrenergic, beta | 1986 |
Beta-adrenergic receptors in guinea-pig liver plasma membranes and thermal lability of [3H]dihydroalprenolol binding sites.
Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Alprenolol; Animals; Binding, Competitive; Cell Membrane; Cholera Toxin; Dihydroalprenolol; Guanylyl Imidodiphosphate; Guinea Pigs; Hot Temperature; Iodocyanopindolol; Isoproterenol; Liver; Male; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Virulence Factors, Bordetella | 1986 |
Regulation of beta adrenergic receptors on rat mononuclear leukocytes by stress: receptor redistribution and down-regulation are altered with aging.
Topics: Aging; Animals; Cyclic AMP; Dihydroalprenolol; Isoproterenol; Male; Monocytes; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Restraint, Physical; Stress, Physiological; Time Factors | 1987 |
Effect of platelet-activating factor on beta-adrenoceptors in human lung.
Topics: Cell Membrane; Dihydroalprenolol; Histamine; Humans; In Vitro Techniques; Isoproterenol; Kinetics; Lung; Methacholine Chloride; Methacholine Compounds; Platelet Activating Factor; Receptors, Adrenergic, beta; Trachea | 1987 |
Lipolysis and beta-adrenergic receptor binding on adipocytes of spontaneously hypertensive rats.
Topics: Adipose Tissue; Animals; Cyclic AMP; Dihydroalprenolol; Hypertension; Isoproterenol; Lipolysis; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Rats, Inbred WKY; Receptors, Adrenergic, beta; Sodium Fluoride | 1987 |
Elimination of isoproterenol-induced proline-rich protein biosynthesis in rat salivary glands after adult thyroidectomy.
Topics: Animals; Cyclic AMP; Dihydroalprenolol; Electrophoresis, Polyacrylamide Gel; Isoproterenol; Male; Peptide Biosynthesis; Peptides; Proline-Rich Protein Domains; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Salivary Glands; Thyroidectomy | 1987 |
[Characteristics of beta-adrenoreceptors of L-1210 leukemia and its sarcolysine-resistant variant].
Topics: Adenylyl Cyclases; Animals; Cyclic AMP; Dihydroalprenolol; Drug Resistance; Enzyme Activation; Isoproterenol; Leukemia L1210; Melphalan; Mice; Mice, Inbred Strains; Neoplasm Transplantation; Receptors, Adrenergic, beta | 1987 |
Neonatal monosodium-L-glutamate treatment reduced lipolytic response of rat epididymal adipose tissue.
Topics: Adenosine Deaminase; Adipose Tissue; Animals; Animals, Newborn; Cerebral Cortex; Dihydroalprenolol; Dose-Response Relationship, Drug; Glutamates; Isoproterenol; Lipolysis; Male; Rats; Sodium Glutamate | 1988 |
[Primary orthostatic hypotension].
Topics: Adult; Blood Platelets; Blood Pressure; Catecholamines; Chronic Disease; Dihydroalprenolol; Humans; Hypotension, Orthostatic; Isoproterenol; Male; Norepinephrine; Physical Exertion; Posture; Receptors, Adrenergic; Yohimbine | 1986 |
Effects of isoproterenol pretreatment on phosphatidylinositol turnover in rat parotid gland.
Topics: Animals; Dihydroalprenolol; Epinephrine; In Vitro Techniques; Isoproterenol; Lipid Metabolism; Male; Parotid Gland; Phosphatidylinositols; Prazosin; Rats; Rats, Inbred Strains | 1986 |
Effect of chronic administration of denopamine (TA-064), a new positive inotropic agent, on cardiac response of rats to denopamine.
Topics: Anesthesia; Animals; Dihydroalprenolol; Drug Tolerance; Ethanolamines; Heart Rate; Isoproterenol; Male; Myocardial Contraction; Organ Size; Rats; Rats, Inbred Strains; Stimulation, Chemical | 1986 |
Adrenergic receptor characteristics of cardiac myocytes cultured in serum-free medium: comparison with serum-supplemented medium.
Topics: Animals; Blood; Culture Media; Dihydroalprenolol; Isoproterenol; Myocardium; Propranolol; Rats; Receptors, Adrenergic; Stereoisomerism | 1985 |
Mapping of beta-adrenergic receptors in rat lung: effect of isoproterenol.
Topics: Animals; Autoradiography; Bronchi; Dihydroalprenolol; Epithelium; Isoproterenol; Lung; Male; Muscle, Smooth; Pulmonary Alveoli; Pulmonary Artery; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1984 |
Rapid recovery of cardiac beta-adrenergic receptors after isoproterenol-induced "down"-regulation.
Topics: Adenosine Triphosphate; Animals; Colchicine; Cyclic AMP; Cytoplasm; Dihydroalprenolol; Drug Tolerance; Isoproterenol; Male; Monensin; Myocardium; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1984 |
Thyroid hormone regulation of adrenergic receptors and beta-adrenergic responsiveness in the rat submandibular gland.
Topics: Animals; Dihydroalprenolol; Hyperthyroidism; Hypothyroidism; Isoproterenol; Kinetics; Male; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Saliva; Submandibular Gland; Thyroidectomy; Thyroxine; Triiodothyronine | 1984 |
"Spare" beta-adrenergic receptors of rat white adipocyte membranes.
Topics: Adenylyl Cyclases; Adipose Tissue; Alprenolol; Animals; Cell Membrane; Cyclic AMP; Dihydroalprenolol; Guanine Nucleotides; Guanylyl Imidodiphosphate; In Vitro Techniques; Isoproterenol; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1984 |
Characterization of a beta-adrenergic receptor in porcine trachealis muscle.
Topics: Adenylyl Cyclases; Animals; Cell Membrane; Cyclic AMP; Dihydroalprenolol; GTP-Binding Proteins; Guanosine Monophosphate; Guanosine Triphosphate; Isoproterenol; Microscopy, Electron; Muscle Contraction; Muscle, Smooth; Receptors, Adrenergic, beta; Stimulation, Chemical; Swine; Trachea | 1984 |
A pivotal role for serotonin (5HT) in the regulation of beta adrenoceptors by antidepressants: reversibility of the action parachlorophenylalanine by 5-hydroxytroptophan.
Topics: 5-Hydroxytryptophan; Adenylyl Cyclases; Animals; Binding, Competitive; Cerebral Cortex; Desipramine; Dihydroalprenolol; Fenclonine; Isoproterenol; Male; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Serotonin; Synapses; Tryptophan Hydroxylase | 1984 |
Endogenous proteinases modulate the function of the beta-adrenergic receptor-adenylate cyclase system.
Topics: Adenylyl Cyclases; Affinity Labels; Animals; Azides; Binding, Competitive; Dihydroalprenolol; Electrophoresis, Polyacrylamide Gel; Endopeptidases; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Lung; Male; Membrane Proteins; Molecular Weight; Propanolamines; Protease Inhibitors; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1984 |
[Desensitization of beta-adrenoreceptors and its influence on manifestations of the antiradiation effect of isoproterenol].
Topics: Adenylyl Cyclases; Animals; Cell Survival; Cells, Cultured; Cricetinae; Cricetulus; Cyclic AMP; Dihydroalprenolol; Drug Tolerance; Isoproterenol; Radiation Tolerance; Radiation-Protective Agents; Receptors, Adrenergic, beta; Time Factors | 1984 |
The relation between ionization and affinity of beta-adrenoceptor ligands.
Topics: Animals; Cattle; Chemical Phenomena; Chemistry, Physical; Cyclic AMP; Dihydroalprenolol; Epinephrine; Guanylyl Imidodiphosphate; In Vitro Techniques; Isoproterenol; Kinetics; Ligands; Membranes; Muscle Proteins; Muscles; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism | 1984 |
Adrenergic responsiveness in experimental uremia.
Topics: Adenylyl Cyclases; Animals; Colforsin; Dihydroalprenolol; Diterpenes; Isoproterenol; Norepinephrine; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Uremia | 1984 |
Some unique properties of CGP-12177.
Topics: Adenylyl Cyclases; Animals; Cell Line; Cyclic AMP; Digitonin; Dihydroalprenolol; Glioma; Isoproterenol; Propanolamines; Rats; Receptors, Adrenergic, beta; Stereoisomerism | 1984 |
Changes in beta-adrenoceptor binding properties and receptor-cyclase coupling during in vitro maturation of rat reticulocytes.
Topics: Adenosine Triphosphate; Adenylyl Cyclases; Animals; Cells, Cultured; Cyclic AMP; Dihydroalprenolol; Isoproterenol; Propanolamines; Rats; Receptors, Adrenergic, beta; Reticulocytes | 1984 |
Studies on responsiveness of hepatoma cells to catecholamines. I. Lack of beta-adrenergic responsiveness in rat ascites hepatoma AH13 cells.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclases; Animals; Binding Sites; Catecholamines; Cell Line; Dihydroalprenolol; Female; Isoproterenol; Kinetics; Liver; Liver Neoplasms, Experimental; Propranolol; Rats; Receptors, Adrenergic, beta | 1984 |
Circadian-phase-dependency in [3H]-dihydroalprenolol binding to rat heart ventricular membranes.
Topics: Alprenolol; Animals; Circadian Rhythm; Dihydroalprenolol; Guanine Nucleotides; Heart Ventricles; Isoproterenol; Male; Myocardium; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Reserpine; Sarcolemma | 1984 |
beta-Adrenergic regulation of alpha 2-adrenergic receptors in the central nervous system.
Topics: Adrenergic alpha-Agonists; Animals; Brain; Clonidine; Dihydroalprenolol; In Vitro Techniques; Isoproterenol; Male; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Sotalol | 1980 |
Beta adrenergic receptors of polymorphonuclear particulates in bronchial asthma.
Topics: Adenylyl Cyclases; Adolescent; Adrenergic beta-Agonists; Adult; Aged; Asthma; Dihydroalprenolol; Female; Humans; Isoproterenol; Male; Middle Aged; Neutrophils; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Biphasic adrenergic modulation of beta-adrenergic receptors in man. Agonist-induced early increment and late decrement in beta-adrenergic receptor number.
Topics: Adrenergic beta-Agonists; Dihydroalprenolol; Epinephrine; Humans; Isoproterenol; Leukocyte Count; Lymphocytes; Male; Monocytes; Neutrophils; Receptors, Adrenergic; Receptors, Adrenergic, beta; Time Factors | 1980 |
The effects of thyroid status on the modulation of fat cell beta-adrenergic receptor agonist affinity by guanine nucleotides.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Animals; Dihydroalprenolol; Female; Guanine Nucleotides; Isoproterenol; Propranolol; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Thyroid Gland | 1980 |
Evidence against beta-adrenoceptor blocking activity of diltiazem, a drug with calcium antagonist properties.
Topics: Adrenergic beta-Antagonists; Animals; Benzazepines; Calcium; Dihydroalprenolol; Diltiazem; Dose-Response Relationship, Drug; Heart Atria; Heart Rate; Isoproterenol; Male; Propranolol; Rats | 1980 |
Visualization of the turkey erythrocyte beta-adrenergic receptor.
Topics: Adenylyl Cyclases; Animals; Chromatography, Affinity; Dihydroalprenolol; Erythrocyte Membrane; Erythrocytes; GTP Phosphohydrolases; Isoproterenol; Molecular Weight; Receptors, Adrenergic; Receptors, Adrenergic, beta; Turkeys | 1980 |
Inhibitors of transglutaminase prevent agonist-mediated internalization of beta-adrenergic receptors.
Topics: Adrenergic beta-Agonists; Animals; Cytosol; Dihydroalprenolol; Erythrocyte Membrane; Erythrocytes; gamma-Glutamyltransferase; Isoproterenol; Kinetics; Methylamines; Rana catesbeiana; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Identification and chemical characterisation of beta-adrenergic receptors in intact turkey erythrocytes.
Topics: Adrenergic beta-Agonists; Animals; Dihydroalprenolol; Dithiothreitol; Erythrocytes; Ethylmaleimide; Isoproterenol; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta; Turkeys | 1981 |
Agonist-induced desensitization of beta-adrenergic receptors in rat myometrium.
Topics: Adrenergic beta-Agonists; Animals; Cell Membrane; Cyclic AMP; Dihydroalprenolol; Estrogens; Female; Isoproterenol; Kinetics; Male; Myometrium; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Uterus | 1981 |
Properties of beta-adrenoceptor sites in metabolizing and nonmetabolizing rat reticulocytes and in resealed reticulocyte ghosts.
Topics: Adrenergic beta-Antagonists; Animals; Cell Membrane; Cold Temperature; Cytosol; Dihydroalprenolol; Energy Metabolism; Female; Isoproterenol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Reticulocytes; Timolol | 1981 |
Desensitization of the beta-adrenoceptor-adenylate cyclase system of immature erythrocytes by in-vivo treatment of rats with isoprenaline.
Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Cyclic AMP; Dihydroalprenolol; Dose-Response Relationship, Drug; Erythrocytes; Isoproterenol; Male; Papaverine; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Beta-adrenoceptor sites in maturing red blood cells of the rat: differing development of agonist and antagonist binding.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dihydroalprenolol; Erythrocytes; Isoproterenol; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Reticulocytes; Time Factors | 1982 |
Characteristics of beta-adrenergic-agonist binding to rat adipocyte membranes. Evidence that (+/-)-[3H]hydroxybenzylisoproterenol interacts selectively with the adipocyte beta-adrenergic receptors.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Animals; Binding, Competitive; Cell Membrane; Dihydroalprenolol; Isoproterenol; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1982 |
Comparison of the apparent irreversible beta-adrenoceptor antagonist Ro 03-7894 with propranolol in cardiac ventricular muscle by pharmacological and radioligand binding techniques.
Topics: Adrenergic beta-Antagonists; Animals; Benzofurans; Binding, Competitive; Cell Membrane; Dihydroalprenolol; Female; Guinea Pigs; Heart; Heart Ventricles; Isoproterenol; Male; Myocardial Contraction; Propranolol; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1982 |
Turn on and turn off reactions of beta-adrenergic-sensitive adenylate cyclase in control and desensitized C6 glioma cells.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Cell Line; Dihydroalprenolol; Enzyme Activation; Epinephrine; Glioma; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Propranolol; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1982 |
Characterization of the rat mast cell beta-adrenergic receptor in resting and stimulated cells by radioligand binding.
Topics: Adrenergic beta-Agonists; Animals; Binding, Competitive; Cattle; Cyclic AMP; Dihydroalprenolol; Dinitrobenzenes; Immunoglobulin E; Isoproterenol; Mast Cells; Propranolol; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Serum Albumin, Bovine; Stereoisomerism | 1982 |
Desensitization of adenylate cyclase and down regulation of beta adrenergic receptors after in vivo administration of beta agonist.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Binding, Competitive; Dihydroalprenolol; Female; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Lung; Metaproterenol; Rats; Rats, Inbred F344; Receptors, Adrenergic; Receptors, Adrenergic, beta; Sodium Fluoride | 1982 |
Properties of agonist binding at the beta-adrenoceptor of the rat reticulocyte.
Topics: Adrenergic beta-Agonists; Animals; Binding, Competitive; Dihydroalprenolol; Erythrocyte Membrane; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Reticulocytes; Stereoisomerism; Temperature | 1982 |
Characterization of beta adrenoceptor subtypes in canine airway smooth muscle by radioligand binding and physiological responses.
Topics: Adrenergic beta-Agonists; Animals; Binding, Competitive; Cell Membrane; Dihydroalprenolol; Dogs; Electric Stimulation; Epinephrine; Isoproterenol; Kinetics; Muscle Contraction; Muscle, Smooth; Propranolol; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, beta; Trachea | 1983 |
Agonist binding to mammalian beta 1 and beta 2 adrenoceptors: modulation by guanine nucleotides and magnesium.
Topics: Adrenergic beta-Agonists; Albuterol; Animals; Cell Membrane; Dihydroalprenolol; Guanine Nucleotides; In Vitro Techniques; Isoproterenol; Lung; Magnesium; Male; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1983 |
Characterization of beta-adrenergic receptors in the rat vas deferens using [3H]-dihydroalprenolol binding.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; Isoproterenol; Male; Muscle Contraction; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Vas Deferens | 1983 |
The effect of the beta-adrenoreceptor antagonist Ro03-7894 on rat atrial tension development and (-)-[3H]dihydroalprenolol binding to cardiac and lung membranes.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Benzofurans; Cell Membrane; Dihydroalprenolol; Isoproterenol; Kinetics; Lung; Male; Myocardial Contraction; Myocardium; Rats | 1983 |
Alterations in cardiac alpha and beta adrenoceptors during the development of spontaneous hypertension.
Topics: Adrenergic alpha-Antagonists; Aging; Animals; Dihydroalprenolol; Dioxanes; Heart Ventricles; Hypertension; Isoproterenol; Male; Myocardium; Papillary Muscles; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Tritium | 1984 |
Determination of the desensitization of beta-adrenergic receptors by [3H]CGP-12177.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Binding Sites; Binding, Competitive; Cell Line; Cell Membrane; Centrifugation, Density Gradient; Dihydroalprenolol; Glioma; Humans; Isoproterenol; Propanolamines; Receptors, Adrenergic, beta | 1983 |
Interaction of a beta-adrenergic partial agonist with its receptor in guinea-pig taenia caecum.
Topics: Adrenergic beta-Agonists; Animals; Carteolol; Cecum; Dihydroalprenolol; Ethanolamines; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Microsomes; Muscle, Smooth; Radioligand Assay; Receptors, Adrenergic, beta | 1984 |
Inhibition of cardiac adenylate cyclase by an irreversible beta-adrenergic blocker.
Topics: Adenylyl Cyclase Inhibitors; Adrenergic beta-Antagonists; Animals; Dihydroalprenolol; In Vitro Techniques; Isoproterenol; Male; Myocardium; Rats | 1984 |
Beta-adrenergic receptor subtypes in iris-ciliary body of rabbits.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Binding, Competitive; Ciliary Body; Dihydroalprenolol; Female; Guinea Pigs; Heart Atria; Iris; Isoproterenol; Kinetics; Rabbits; Radioligand Assay; Receptors, Adrenergic, beta; Trachea | 1984 |
The human carcinoma cell line A431 possesses large numbers of functional beta-adrenergic receptors.
Topics: Adrenergic beta-Antagonists; Binding, Competitive; Carcinoma, Squamous Cell; Cell Line; Dihydroalprenolol; Humans; Isoproterenol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism | 1984 |
Uptake of L-[propyl-2,3-3H]dihydroalprenolol by intact HeLa cells.
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Biological Transport; Cell Membrane; Chloroquine; Cold Temperature; Diffusion; Dihydroalprenolol; HeLa Cells; Humans; Hydrogen-Ion Concentration; Isoproterenol; Phentolamine; Pindolol; Receptors, Adrenergic, beta; Valinomycin | 1984 |
A comparison of the binding characteristics of the beta-adrenoceptor antagonists 3H-dihydroalprenolol and 125I-iodocyanopindolol in rat liver.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Kinetics; Liver; Liver Regeneration; Male; Membranes; Pindolol; Prazosin; Rats; Rats, Inbred Strains | 1984 |
A hormone-independent rise of adenosine 3',5'-monophosphate desensitizes coupling of beta-adrenergic receptors to adenylate cyclase in rat glioma C6-cells.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Carrier Proteins; Cholera Toxin; Cyclic AMP; Dihydroalprenolol; Fluorides; Glioma; Guanosine Triphosphate; Isoproterenol; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Beta-adrenergic regulation of rat parotid gland exocrine protein secretion during aging.
Topics: Aging; Amylases; Animals; Dihydroalprenolol; Dose-Response Relationship, Drug; In Vitro Techniques; Isoproterenol; Kinetics; Male; Parotid Gland; Propranolol; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Bromoacetylalprenololmenthane: a potent irreversible antagonist of beta adrenergic elicited protein exocytosis in rat parotid cells.
Topics: Adrenergic beta-Antagonists; Alprenolol; Amylases; Animals; Cyclohexane Monoterpenes; Depression, Chemical; Dihydroalprenolol; Exocytosis; Isoproterenol; Male; Microscopy, Electron; Parotid Gland; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1983 |
beta-Adrenoceptor alterations coupled with secretory response in rat parotid tissue.
Topics: Acetylcholine; Amylases; Animals; Cyclic AMP; Dihydroalprenolol; Dioxanes; Isoproterenol; Male; Parotid Gland; Phenylephrine; Propranolol; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Time Factors | 1983 |
Characterization of the beta-adrenergic receptors of cultured human epidermal keratinocytes.
Topics: Binding, Competitive; Cell Membrane; Cells, Cultured; Dihydroalprenolol; Epidermis; Humans; Infant; Isoproterenol; Keratins; Kinetics; Male; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism | 1983 |
Reconstitution of a hormone-sensitive adenylate cyclase with membrane extracts from Neurospora and avian erythrocytes.
Topics: Adenylyl Cyclases; Animals; Cell Membrane; Cholera Toxin; Dihydroalprenolol; Erythrocyte Membrane; Erythrocytes; Isoproterenol; Kinetics; Male; Neurospora; Neurospora crassa; Species Specificity; Testis; Turkeys | 1983 |
Defect in the adrenergic receptor-adenylate cyclase system during development of catecholamine-induced cardiomyopathy.
Topics: Adenylyl Cyclases; Animals; Cardiomegaly; Dihydroalprenolol; Dihydroergotoxine; Epinephrine; Isoproterenol; Male; Myocardium; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Sodium Fluoride | 1984 |
[Effect of puerarin and analogues of daidzein on adrenoceptors].
Topics: Adenylyl Cyclases; Animals; Dihydroalprenolol; Dose-Response Relationship, Drug; Flavonoids; In Vitro Techniques; Isoflavones; Isoproterenol; Myocardial Contraction; Rabbits; Rats; Receptors, Adrenergic | 1984 |
Beta adrenergic receptors in lymphocyte subpopulations.
Topics: B-Lymphocytes; Binding Sites; Binding, Competitive; Cyclic AMP; Dihydroalprenolol; Female; Humans; Isoproterenol; Lymphocytes; Male; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta; T-Lymphocytes | 1980 |
Guanosine triphosphate: an endogenous compound in the rabbit cerebellar cortex which couples the beta-adrenergic receptor to adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Cerebellar Cortex; Culture Techniques; Dihydroalprenolol; Enzyme Activation; Guanosine Diphosphate; Guanosine Triphosphate; Isoproterenol; Rabbits; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Hippocampal alpha- and beta-adrenergic receptors: comparison of [3H]dihydroalprenolol and [3H]WB 4101 binding with noradrenergic innervation in the rat.
Topics: Alprenolol; Animals; Binding Sites; Binding, Competitive; Dihydroalprenolol; Epinephrine; Hippocampus; Isoproterenol; Microscopy, Fluorescence; Norepinephrine; Radioligand Assay; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Synaptosomes | 1980 |
The beta-adrenergic receptor of live human polymorphonuclear leukocytes.
Topics: Binding, Competitive; Colchicine; Cyclic AMP; Dihydroalprenolol; Humans; Isoproterenol; Kinetics; Lysosomes; Neutrophils; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
A high affinity agonist . beta-adrenergic receptor complex is an intermediate for catecholamine stimulation of adenylate cyclase in turkey and frog erythrocyte membranes.
Topics: Adenylyl Cyclases; Animals; Anura; Catecholamines; Computers; Dihydroalprenolol; Enzyme Activation; Erythrocyte Membrane; Erythrocytes; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta; Turkeys | 1980 |
Thyroxine-induced changes in characteristics and activities of beta-adrenergic receptors and adenosine 3',5'-monophosphate and guanosine 3',5'-monophosphate systems in the heart may be related to reputed catecholamine supersensitivity in hyperthyroidism.
Topics: Adenylyl Cyclases; Animals; Cardiomegaly; Cyclic AMP; Cyclic GMP; Dihydroalprenolol; Fluorides; Heart; Hyperthyroidism; Isoproterenol; Kinetics; Male; Myocardium; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Thyroxine | 1980 |
Effects of local anesthetics on guanyl nucleotide modulation of the catecholamine-sensitive adenylate cyclase system and on beta-adrenergic receptors.
Topics: Adenylyl Cyclases; Anesthetics, Local; Animals; Anura; Catecholamines; Dihydroalprenolol; Erythrocyte Membrane; Guanine Nucleotides; In Vitro Techniques; Isoproterenol; Receptors, Adrenergic; Receptors, Adrenergic, beta; Tetracaine | 1980 |
Agonist-dependent desensitization of myometrial beta-adrenergic catecholamine-sensitive adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Dihydroalprenolol; Female; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Myometrium; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Uterus | 1980 |
A ternary complex model explains the agonist-specific binding properties of the adenylate cyclase-coupled beta-adrenergic receptor.
Topics: Adenylyl Cyclases; Alprenolol; Animals; Anura; Binding Sites; Binding, Competitive; Dihydroalprenolol; Erythrocyte Membrane; Erythrocytes; Isoproterenol; Kinetics; Mathematics; Protein Binding; Receptors, Adrenergic; Receptors, Adrenergic, beta; Turkeys | 1980 |
beta-adrenergic supersensitivity in rat brainstem during clonidine withdrawal.
Topics: Animals; Brain Stem; Clonidine; Cyclic AMP; Dihydroalprenolol; Humans; Isoproterenol; Male; Propranolol; Protein Binding; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Substance Withdrawal Syndrome; Time Factors | 1980 |
Increased pulmonary alpha-adrenergic and reduced beta-adrenergic receptors in experimental asthma.
Topics: Adenylyl Cyclases; Animals; Asthma; Dihydroalprenolol; Disease Models, Animal; Enzyme Activation; Guinea Pigs; Isoproterenol; Lung; Ovalbumin; Prazosin; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1980 |
Parallel modulation of catecholamine activation of adenylate cyclase and formation of the high-affinity agonist.receptor complex in turkey erythrocyte membranes by temperature and cis-vaccenic acid.
Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Dihydroalprenolol; Enzyme Activation; Erythrocyte Membrane; Erythrocytes; Isoproterenol; Kinetics; Receptors, Adrenergic; Receptors, Adrenergic, beta; Temperature; Turkeys | 1980 |
Evidence for uncoupling of the beta receptor-adenylate cyclase complex.
Topics: Adenylyl Cyclases; Animals; Chick Embryo; Dihydroalprenolol; Heart Ventricles; Isoproterenol; Myocardial Contraction; Receptors, Adrenergic; Receptors, Adrenergic, beta; Ventricular Function | 1980 |
beta 1-Adrenergic receptors in kidney tubular cell membrane in the rat.
Topics: Alprenolol; Animals; Cell Membrane; Depression, Chemical; Dihydroalprenolol; Epinephrine; Isoproterenol; Kidney Tubules; Kinetics; Norepinephrine; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Characterization of adenylate cyclase activity in asthmatic neutrophil sonicates.
Topics: Adenylyl Cyclases; Adult; Aged; Asthma; Cyclic AMP; Dihydroalprenolol; Female; Histamine; Humans; Isoproterenol; Male; Middle Aged; Neutrophils; Prostaglandins E; Receptors, Adrenergic; Receptors, Adrenergic, beta; Sodium Fluoride; Sonication | 1980 |
Decreased beta-adrenergic responses in the female rat brain are eliminated by ovariectomy: correlation of [3H]dihydroalprenolol binding and catecholamine stimulated cyclic AMP levels.
Topics: Alprenolol; Animals; Binding Sites; Castration; Cerebral Cortex; Cyclic AMP; Dihydroalprenolol; Estrogens; Estrus; Female; Isoproterenol; Male; Pregnancy; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Action of mianserin and zimelidine on the norepinephrine receptor coupled adenylate cyclase system in brain: subsensitivity without reduction in beta-adrenergic receptor binding.
Topics: Adenylyl Cyclases; Animals; Brain; Brompheniramine; Dibenzazepines; Dihydroalprenolol; Isoproterenol; Kinetics; Male; Mianserin; Pyridines; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Zimeldine | 1980 |
Further evidence that desensitization of beta-adrenergic-sensitive adenylate cyclase proceeds in two steps. Modification of the coupling and loss of beta-adrenergic receptors.
Topics: Adenylyl Cyclases; Animals; Cell Line; Cycloheximide; Dihydroalprenolol; Enzyme Activation; Glioma; Isoproterenol; Kinetics; Mathematics; Mice; Prostaglandins E; Puromycin; Receptors, Adrenergic; Receptors, Adrenergic, beta; Temperature | 1980 |
Ontogenetic development of isoproterenol subsensitivity of myocardial adenylate cyclase and beta-adrenergic receptors in spontaneously hypertensive rats.
Topics: Adenylyl Cyclases; Aging; Animals; Body Weight; Cell Membrane; Dihydroalprenolol; Heart; Hypertension; Isoproterenol; Kinetics; Myocardium; Organ Size; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Hypersensitivity of cardiac beta-adrenergic receptors after neonatal treatment of rats with 6-hydroxydopa.
Topics: Animals; Animals, Newborn; Binding Sites; Dihydroalprenolol; Dihydroxyphenylalanine; Female; Heart; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Myocardium; Norepinephrine; Ornithine Decarboxylase; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Myocardial beta-adrenergic receptors from adrenalectomized rats: impaired formation of high-affinity agonist-receptor complexes.
Topics: Adenylyl Cyclases; Adrenal Glands; Adrenalectomy; Alprenolol; Animals; Computers; Dihydroalprenolol; In Vitro Techniques; Isoproterenol; Male; Myocardium; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Developmental change of beta-adrenergic receptors in rat brain.
Topics: Age Factors; Animals; Binding Sites; Brain Chemistry; Dihydroalprenolol; In Vitro Techniques; Isoproterenol; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Synaptic Membranes | 1980 |
Beta-adrenergic receptor-adenylate cyclase alterations during the postnatal development of skeletal muscle.
Topics: Adenylyl Cyclases; Animals; Catecholamines; Cell Membrane; Dihydroalprenolol; Epinephrine; Female; Guanosine Triphosphate; Isoproterenol; Muscle Development; Norepinephrine; Phospholipids; Rabbits; Receptors, Adrenergic; Receptors, Adrenergic, beta; Sarcolemma; Sodium Fluoride; Sodium-Potassium-Exchanging ATPase | 1980 |
Adenylate cyclase in lean and obese (ob/ob) mouse epididymal white adipocytes.
Topics: Adenylyl Cyclases; Adipose Tissue; Animals; Cell Membrane; Dihydroalprenolol; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Male; Mice; Mice, Inbred C57BL; Mice, Obese; Receptors, Adrenergic, beta; Sodium Fluoride; Species Specificity | 1980 |
A biochemical study of receptor internalization during beta-adrenergic receptor desensitization in frog erythrocytes.
Topics: Adenylyl Cyclases; Animals; Blood Proteins; Cytosol; Dihydroalprenolol; Erythrocyte Membrane; Erythrocytes; In Vitro Techniques; Isoproterenol; Rana catesbeiana; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
II. Beta-adrenergic receptors and catecholamine sensitive adenylate cyclase in the developing rat lung.
Topics: Adenylyl Cyclases; Animals; Benzyl Alcohols; Catecholamines; Cell Membrane; Dihydroalprenolol; Enzyme Activation; Epinephrine; Female; Isoproterenol; Lung; Male; Norepinephrine; Pindolol; Pregnancy; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Human lymphocyte beta-adrenergic receptors are unaltered with age.
Topics: Adolescent; Adult; Aged; Aging; Dihydroalprenolol; Epinephrine; Female; Humans; Isoproterenol; Lymphocytes; Male; Middle Aged; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Halothane effect on beta-adrenergic receptors in canine myocardium.
Topics: Adenylyl Cyclases; Animals; Cell Membrane; Cyclic AMP; Dihydroalprenolol; Dogs; Female; Guanosine Triphosphate; Halothane; Heart; Isoproterenol; Male; Myocardium; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
The influences of glucagon, epinephrine and alpha- and beta-adrenergic agents on glycogenolysis in isolated rabbit hepatocytes and perfused livers.
Topics: Alprenolol; Animals; Bucladesine; Cyclic AMP; Dihydroalprenolol; Epinephrine; Glucagon; In Vitro Techniques; Isoproterenol; Liver; Liver Glycogen; Male; Phentolamine; Phenylephrine; Rabbits | 1981 |
Coupling of beta-adrenoreceptors in rat uterine smooth muscle.
Topics: Adenylyl Cyclases; Animals; Cyclic AMP; Dihydroalprenolol; Female; Guanylyl Imidodiphosphate; Isoproterenol; Muscle Relaxation; Myometrium; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Uterine Contraction; Uterus | 1981 |
Catecholamine-induced desensitization in turkey erythrocytes: cAMP mediated impairment of high affinity agonist binding without alteration in receptor number.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Binding, Competitive; Cyclic AMP; Dihydroalprenolol; Drug Tolerance; Erythrocytes; Isoproterenol; Receptors, Adrenergic; Receptors, Adrenergic, beta; Turkeys | 1981 |
Characterization of serum-induced alterations in the cyclic AMP pathway in S49 lymphoma cells.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclases; Animals; Blood; Cell Line; Cholera Toxin; Culture Media; Cyclic AMP; Dihydroalprenolol; Isoproterenol; Kinetics; Lymphoma; Mice; Receptors, Adrenergic, alpha | 1981 |
Cholera toxin can recouple hormone receptors that are uncoupled from adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Cell Line; Cholera Toxin; Cyclic AMP; Dihydroalprenolol; Isoproterenol; Prostaglandins E; Receptors, Adrenergic, beta; Receptors, Cell Surface | 1981 |
The development of pre- and postsynaptic components of the noradrenergic system in the rat cerebellum.
Topics: Adenylyl Cyclases; Aging; Animals; Brain; Cerebellum; Dihydroalprenolol; Female; Isoproterenol; Kinetics; Male; Norepinephrine; Rats; Receptors, Adrenergic, beta; Synapses | 1981 |
Extracellular magnesium is not required for beta adrenergic drug-receptor interactions in intact human lymphocytes.
Topics: Adenylyl Cyclases; Cyclic AMP; Dihydroalprenolol; Extracellular Space; Humans; In Vitro Techniques; Isoproterenol; Lymphocytes; Magnesium; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Isolation and characterization of the beta-adrenergic receptor of frog erythrocytes and development of potential affinity ligands.
Topics: Affinity Labels; Animals; Binding, Competitive; Dihydroalprenolol; Erythrocyte Membrane; Erythrocytes; Isoproterenol; Kinetics; Ligands; Molecular Weight; Ranidae; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Molecular pharmacology of adenylate cyclase-coupled alpha- and beta-adrenergic receptors.
Topics: Adenylyl Cyclases; Alprenolol; Animals; Blood Platelets; Cell Membrane; Dihydroalprenolol; Epinephrine; Erythrocyte Membrane; Erythrocytes; Guanosine Triphosphate; Isoproterenol; Kinetics; Ranidae; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1981 |
Presence of ectopic beta-adrenergic receptors on human adrenocortical cortisol-producing adenomas.
Topics: Adenoma; Adrenal Cortex; Adrenal Gland Neoplasms; Adrenocorticotropic Hormone; Adult; Cell Membrane; Cushing Syndrome; Dihydroalprenolol; Epinephrine; Female; Humans; Hydrocortisone; Isoproterenol; Middle Aged; Phentolamine; Propranolol; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
The effect of alprenolol on the beta-receptor and adenylate cyclase activity in rabbit heart membranes.
Topics: Adenylyl Cyclases; Alprenolol; Animals; Cell Membrane; Dihydroalprenolol; Guanine Nucleotides; Heart; In Vitro Techniques; Isoproterenol; Myocardium; Rabbits; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Superior cervical ganglionectomy depresses norepinephrine uptake, increases the density of alpha-adrenoceptor sites, and induces supersensitivity to adrenergic drugs in rat medial basal hypothalamus.
Topics: Animals; Dihydroalprenolol; Ganglia, Sympathetic; Hypothalamus; Isoproterenol; Kinetics; Levodopa; Male; Norepinephrine; Phentolamine; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Tubulin | 1981 |
Autonomic mechanisms of training bradycardia: beta-adrenergic receptors in humans.
Topics: Adult; Dihydroalprenolol; Female; Heart Rate; Humans; Isoproterenol; Lymphocytes; Male; Physical Education and Training; Receptors, Adrenergic; Receptors, Adrenergic, beta; Running | 1981 |
Catecholamine-induced desensitization of adenylate cyclase in rat glioma C6 cells. Evidence for a specific uncoupling of beta-adrenergic receptors from a functional regulatory component of adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Catecholamines; Cells, Cultured; Cholera Toxin; Dihydroalprenolol; Glioma; Isoproterenol; Neoplasms, Experimental; Quinacrine; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Differences in the beta-adrenergic responsiveness between high and low passage rat glioma C6 cells.
Topics: Adenylyl Cyclases; Animals; Cell Line; Cell Membrane; Cholera Toxin; Cyclic AMP; Dihydroalprenolol; G(M1) Ganglioside; Glioma; Isoproterenol; Kinetics; Neoplasms, Experimental; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Hypothyroidism modulates beta adrenergic receptor adenylate cyclase interactions in rat reticulocytes.
Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Dihydroalprenolol; GTP-Binding Proteins; Hypothyroidism; Isoproterenol; Models, Biological; Protein Binding; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Receptors, Cell Surface; Reticulocytes; Thyroidectomy | 1981 |
beta-Receptor numbers and thermodynamics in denervation supersensitivity.
Topics: Adult; Aged; Autonomic Nervous System Diseases; Dihydroalprenolol; Dose-Response Relationship, Drug; Female; Heart Rate; Humans; Isoproterenol; Lymphocytes; Male; Nerve Degeneration; Receptors, Adrenergic; Receptors, Adrenergic, beta; Shy-Drager Syndrome; Temperature; Thermodynamics | 1981 |
Altered states of cardiac beta-adrenoreceptors.
Topics: Alprenolol; Animals; Ascorbic Acid; Chymotrypsin; Dihydroalprenolol; Dogs; Female; Hot Temperature; Isoproterenol; Male; Myocardium; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Development of beta-adrenergic receptors and the in vitro accumulation of cyclic AMP in the chick spinal cord.
Topics: Adenylyl Cyclases; Animals; Cell Differentiation; Chick Embryo; Chickens; Cyclic AMP; Dihydroalprenolol; Epinephrine; Isoproterenol; Norepinephrine; Phosphoric Diester Hydrolases; Receptors, Adrenergic; Receptors, Adrenergic, beta; Spinal Cord | 1982 |
Isoproterenol responsiveness and myocardial beta-adrenergic receptors in young and old rats.
Topics: Aging; Animals; Dihydroalprenolol; Female; Heart Rate; Isoproterenol; Lung; Lymphocytes; Myocardium; Rats; Rats, Inbred F344; Receptors, Adrenergic; Receptors, Adrenergic, alpha | 1982 |
Receptor binding sites for beta-adrenergic ligands on human erythrocytes.
Topics: Adult; Alprenolol; Binding, Competitive; Cyclic AMP; Dihydroalprenolol; Erythrocyte Membrane; Erythrocytes; Humans; Isoproterenol; Kinetics; Propranolol; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1982 |
Receptor-associated changes of the catecholamine-sensitive adenylate cyclase in glioma cells doubly transformed with Moloney sarcoma virus.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenosine Triphosphate; Adenylyl Cyclases; Animals; Cell Transformation, Neoplastic; Cell Transformation, Viral; Cells, Cultured; Chromosome Aberrations; Dihydroalprenolol; Glioma; Isoproterenol; Kinetics; Male; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Sarcoma Viruses, Murine | 1982 |
Relationship between beta-adrenergic receptor numbers and physiological responses during experimental canine myocardial ischemia.
Topics: Animals; Coronary Circulation; Coronary Disease; Cyclic AMP; Dihydroalprenolol; Dogs; Female; Heart Ventricles; Isoproterenol; Male; Phosphorylase b; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1982 |
Studies on desensitization of adrenergic receptors of human adipocytes.
Topics: Adipose Tissue; Clonidine; Cyclic AMP; Dihydroalprenolol; Epinephrine; Humans; Isoproterenol; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine | 1982 |
Temperature dependence if beta-receptor mediated relaxation in rabbit intestine.
Topics: Animals; Cyclic AMP; Dihydroalprenolol; Female; In Vitro Techniques; Intestines; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Phentolamine; Propranolol; Rabbits; Receptors, Adrenergic; Receptors, Adrenergic, beta; Temperature | 1982 |
Mechanisms of beta-adrenergic desensitization in rat myometrium.
Topics: Adenylyl Cyclases; Animals; Cyclic AMP; Dihydroalprenolol; Drug Tolerance; Female; Isoproterenol; Myometrium; Phosphoric Diester Hydrolases; Protein Kinases; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Uterine Contraction | 1981 |
On the mechanism of isoproterenol-induced desensitization of adenylate cyclase in cultured differentiated hepatocytes.
Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Cell Line; Clone Cells; Cyclic AMP; Dihydroalprenolol; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Liver; Rats; Sodium Fluoride | 1982 |
Trophoblastic cells of the hydatidiform mole contain a beta 1-subtype adrenergic receptor.
Topics: Adenylyl Cyclases; Adolescent; Adult; Dihydroalprenolol; Epinephrine; Female; Guanylyl Imidodiphosphate; Humans; Hydatidiform Mole; Isoproterenol; Norepinephrine; Pregnancy; Receptors, Adrenergic; Receptors, Adrenergic, beta; Trophoblasts; Uterine Neoplasms | 1982 |
Adenylate cyclase and beta adrenergic receptor development in the mouse heart.
Topics: Adenylyl Cyclases; Aging; Animals; Animals, Newborn; Dihydroalprenolol; Female; Fetal Heart; Heart; In Vitro Techniques; Isoproterenol; Mice; Myocardium; Pregnancy; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1982 |
Decreased catecholamine sensitivity and beta-adrenergic-receptor density in failing human hearts.
Topics: Adenylyl Cyclases; Adolescent; Adult; Catecholamines; Contractile Proteins; Creatine Kinase; Dihydroalprenolol; Female; Fluorides; Heart Failure; Histamine; Humans; Hydroxyproline; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Myocardial Contraction; Myocardium; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, beta; Tritium | 1982 |
The action of six lipid perturbing substances on hormone receptor adenylate cyclase complex in turkey erythrocytes and intestinal mucosa cells.
Topics: Adenylyl Cyclases; Animals; Cyclic AMP; Detergents; Dihydroalprenolol; Erythrocyte Membrane; Erythrocytes; In Vitro Techniques; Intestinal Mucosa; Isoproterenol; Male; Proteins; Rats; Receptors, Cell Surface; Surface-Active Agents; Turkeys | 1982 |
Evidence for a defect in the number of beta-adrenergic receptors and in the adenylate cyclase responsiveness to guanine nucleotides in fat cells after adrenalectomy.
Topics: Adenosine Deaminase; Adenylyl Cyclases; Adipose Tissue; Adrenalectomy; Animals; Cell Membrane; Dihydroalprenolol; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1982 |
Decreased neutrophil beta adrenergic receptors in the neonate.
Topics: Cyclic AMP; Dihydroalprenolol; Fetal Blood; Humans; Infant, Newborn; Isoproterenol; Neutrophils; Receptors, Adrenergic; Receptors, Adrenergic, beta; Tritium | 1982 |
Abnormal brown adipose composition and beta-adrenoceptor binding in obese Zucker rats.
Topics: Adipose Tissue, Brown; Animals; Body Weight; Dihydroalprenolol; Epinephrine; Isoproterenol; Lipolysis; Male; Norepinephrine; Obesity; Rats; Rats, Zucker; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1982 |
The beta-adrenergic system and allergic bronchial asthma: changes in lymphocyte beta-adrenergic receptor number and adenylate cyclase activity after an allergen-induced asthmatic attack.
Topics: Adenylyl Cyclases; Adolescent; Adult; Allergens; Asthma; Bronchial Provocation Tests; Dihydroalprenolol; Forced Expiratory Volume; Guanylyl Imidodiphosphate; Humans; Isoproterenol; Lymphocytes; Male; Mites; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1982 |
Adrenergic ligand liposolubility in membranes. Direct assessment in a beta-adrenergic binding system.
Topics: Adipose Tissue; Animals; Binding, Competitive; Dihydroalprenolol; Isoproterenol; Ligands; Membrane Lipids; Membranes; Receptors, Adrenergic; Receptors, Adrenergic, beta; Solubility; Sympathomimetics | 1982 |
Non-co-ordinate development of beta-adrenergic receptors and adenylate cyclase in chick heart.
Topics: Adenylyl Cyclases; Animals; Chick Embryo; Dihydroalprenolol; Guanylyl Imidodiphosphate; Heart; In Vitro Techniques; Isoproterenol; Kinetics; Myocardium; Receptors, Adrenergic; Receptors, Adrenergic, beta; Time Factors | 1982 |
beta-Adrenoceptor ligand binding and supersensitivity to isoprenaline of ventricular muscle after chronic reserpine pretreatment.
Topics: Animals; Calcium; Dihydroalprenolol; Female; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Ligands; Male; Membranes; Myocardial Contraction; Myocardium; Papillary Muscles; Receptors, Adrenergic; Receptors, Adrenergic, beta; Reserpine | 1982 |
beta-Adrenoceptor-adenosine 3',5-monophosphate system in human leucocytes before and after treatment for hyperthyroidism.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclases; Binding, Competitive; Cyclic AMP; Dihydroalprenolol; Enzyme Activation; Female; Humans; Hyperthyroidism; Isoproterenol; Leukocytes; Male; Middle Aged; Protein Kinases; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1983 |
Influence of repeated administration of desmethylimipramine on beta adrenergic and muscarinic cholinergic receptors and 45Ca++ binding to sarcoplasmic reticulum in the rat heart.
Topics: Acetylcholine; Animals; Calcium; Desipramine; Dihydroalprenolol; Heart; Isoproterenol; Male; Myocardial Contraction; Myocardium; Norepinephrine; Ornithine Decarboxylase; Propranolol; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Receptors, Cholinergic; Receptors, Muscarinic; Sarcoplasmic Reticulum | 1982 |
alpha and beta-adrenoceptor coupling to adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Dihydroalprenolol; Guanosine Triphosphate; Isoproterenol; Lung; Microsomes; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1982 |
Blockade of heterologous desensitization of prostate adenylate cyclase without blockade of homologous down regulation of receptors or loss of GTP regulation of agonist binding.
Topics: Acetylcholine; Adenylyl Cyclases; Animals; Calcimycin; Dihydroalprenolol; Guanosine Triphosphate; Isoproterenol; Male; Potassium; Prostate; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1983 |
Difference between lung and spleen susceptibility of beta-adrenergic receptors to desensitization by terbutaline.
Topics: Animals; Cells, Cultured; Dihydroalprenolol; Humans; Isoproterenol; Lung; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Spleen; Terbutaline | 1983 |
Serotonergic denervation changes binding characteristics of beta-adrenoceptors in rat cortex.
Topics: Animals; Cerebral Cortex; Denervation; Dihydroalprenolol; Isoproterenol; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Serotonin | 1982 |
Decreased beta-adrenergic agonist affinity and adenylate cyclase activity in senescent rat lung.
Topics: Adenylyl Cyclases; Aging; Animals; Binding, Competitive; Colforsin; Dihydroalprenolol; Diterpenes; Female; Guanylyl Imidodiphosphate; Isoproterenol; Lung; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Temperature | 1983 |
Desensitization of beta 2-adrenergic receptors and adrenocorticotropin release.
Topics: Adrenocorticotropic Hormone; Animals; Cell Line; Colforsin; Cyclic AMP; Dihydroalprenolol; Diterpenes; Isoproterenol; Mice; Pituitary Gland, Anterior; Pituitary Neoplasms; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1983 |
Guanine nucleotides and alpha 1 adrenergic receptors in the heart.
Topics: Animals; Binding, Competitive; Dihydroalprenolol; Epinephrine; Guanine Nucleotides; Guanylyl Imidodiphosphate; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Myocardium; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha | 1983 |
Low beta-adrenergic receptor concentration on human thymocytes.
Topics: Adenosine; Alprostadil; Animals; Cyclic AMP; Dihydroalprenolol; Humans; Isoproterenol; Mice; Mice, Inbred Strains; Phosphodiesterase Inhibitors; Prostaglandins E; Receptors, Adrenergic; Receptors, Adrenergic, beta; T-Lymphocytes | 1983 |
Activation of beta 2-adrenergic receptors on mouse anterior pituitary tumor cells increases cyclic adenosine 3':5'-monophosphate synthesis and adrenocorticotropin release.
Topics: Adrenocorticotropic Hormone; Animals; Cell Line; Cell Membrane; Cyclic AMP; Dihydroalprenolol; Epinephrine; Isoproterenol; Kinetics; Mice; Neoplasms, Experimental; Norepinephrine; Pituitary Gland, Anterior; Pituitary Neoplasms; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1983 |
Beta-adrenergic receptors in early human placenta characterization of [3H]-dihydroalprenolol binding.
Topics: Alprenolol; Binding, Competitive; Dihydroalprenolol; Epinephrine; Female; Humans; Isoproterenol; Kinetics; Membranes; Norepinephrine; Placenta; Pregnancy; Pregnancy Trimester, First; Receptors, Adrenergic; Receptors, Adrenergic, beta; Substrate Specificity | 1983 |
A possible mechanism of action of a beta-adrenergic partial agonist (carteolol) in guinea pig taenia caecum.
Topics: Animals; Carteolol; Cecum; Cyclic AMP; Dihydroalprenolol; Guinea Pigs; In Vitro Techniques; Isoproterenol; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Propanolamines; Proteins | 1983 |
Human lymphocytes as a model for beta-adrenergic receptors in clinical investigation.
Topics: Adolescent; Adult; Aged; Dihydroalprenolol; Female; Guanylyl Imidodiphosphate; Humans; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Kinetics; Lymphocytes; Male; Middle Aged; Models, Biological; Pindolol; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1983 |
Binding of [3H]-dihydroalprenolol and [3H]-acetobutolol to human blood platelets is not related to occupancy of beta-adrenoceptors.
Topics: Acebutolol; Alprenolol; Blood Platelets; Butoxamine; Dihydroalprenolol; Humans; Isoproterenol; Kinetics; Practolol; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1983 |
Possible influence of noradrenaline on beta-adrenergic and muscarinic cholinergic receptors in rat heart: effects of 6-hydroxydopa, isoproterenol, and desmethylimipramine.
Topics: Animals; Desipramine; Dihydroalprenolol; Dihydroxyphenylalanine; Female; Heart; Isoproterenol; Male; Myocardium; Norepinephrine; Ornithine Decarboxylase; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Receptors, Cholinergic; Receptors, Muscarinic | 1983 |
Characterization of the beta-adrenergic receptors of hamster white fat cells. Evidence against an important role for the alpha 2-receptor subtype in the adrenergic control of lipolysis.
Topics: Adipose Tissue; Animals; Binding, Competitive; Cricetinae; Dihydroalprenolol; Isoproterenol; Kinetics; Lipolysis; Male; Mesocricetus; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1983 |
Beta-adrenoceptor desensitization in rat lung: functional and biochemical aspects.
Topics: Adenylyl Cyclases; Animals; Carbachol; Dihydroalprenolol; In Vitro Techniques; Isoproterenol; Lung; Male; Membranes; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1983 |
Beta adrenergic receptors in lymphocytes and granulocytes from patients with cystic fibrosis.
Topics: Adolescent; Adult; Cyclic AMP; Cystic Fibrosis; Dihydroalprenolol; Granulocytes; Heterozygote; Humans; Isoproterenol; Kinetics; Lymphocytes; Middle Aged; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1983 |
Regression of thyroid hormone induced cardiac hypertrophy: effect on cardiac beta receptors and adenyl cyclase activity.
Topics: Adenylyl Cyclases; Animals; Cardiomegaly; Cell Membrane; Dihydroalprenolol; Isoproterenol; Kinetics; Male; Myocardium; Organ Size; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Thyroxine; Triiodothyronine | 1983 |
beta-2 adrenergic receptors on intact human erythrocytes.
Topics: Alprenolol; Binding, Competitive; Cyclic AMP; Dihydroalprenolol; Erythrocytes; Humans; In Vitro Techniques; Isoproterenol; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1983 |
Displacement of alpha- and beta-radioligands by specific adrenergic agonists in rat pancreatic islets.
Topics: Animals; Binding, Competitive; Clonidine; Dihydroalprenolol; Dihydroergotoxine; Epinephrine; In Vitro Techniques; Islets of Langerhans; Isoproterenol; Ligands; Male; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1983 |
Alteration in the effect of GTP on cerebral beta-adrenergic receptor binding during morphine withdrawal.
Topics: Animals; Dihydroalprenolol; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Humans; Isoproterenol; Kinetics; Male; Morphine Dependence; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Subcellular Fractions; Substance Withdrawal Syndrome | 1983 |
[Effect of neuraminidase on the beta-adrenergic receptor].
Topics: Animals; Asthma; Cyclic AMP; Dihydroalprenolol; Guinea Pigs; Humans; Isoproterenol; Lymphocytes; Male; Neuraminidase; Propranolol; Receptors, Adrenergic, beta | 1983 |
Involvement of microtubules in the isoproterenol-induced 'down'-regulation of myocardial beta-adrenergic receptors.
Topics: Animals; Binding, Competitive; Cell Membrane; Colchicine; Dihydroalprenolol; Isoproterenol; Kinetics; Male; Microtubules; Myocardium; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1983 |
Mononuclear leukocyte beta 2-adrenergic receptors and adenylate cyclase sensitivity in insulin-dependent diabetes mellitus.
Topics: Adenylyl Cyclases; Adult; Autonomic Nervous System; Blood Pressure; Cell Membrane; Diabetes Mellitus, Type 1; Dihydroalprenolol; Female; Heart Rate; Humans; Isoproterenol; Leukocytes; Male; Receptors, Adrenergic, beta | 1983 |
Changes of beta-adrenergic receptor number and catecholamine-sensitive adenylate cyclase in guinea pig lung after inhalation of histamine aerosol.
Topics: Adenylyl Cyclases; Aerosols; Animals; Dihydroalprenolol; Guinea Pigs; Histamine; Isoproterenol; Lung; Prazosin; Quinuclidinyl Benzilate; Receptors, Adrenergic, beta; Sodium Fluoride; Tritium | 1983 |
[Measurement of radioligand binding to beta-adrenergic and benzodiazepine receptors in the cerebral cortex of the rat. Comparison of filtration and centrifugation technics].
Topics: Animals; Cerebral Cortex; Dihydroalprenolol; Filtration; Flunitrazepam; Isoproterenol; Proteins; Radioligand Assay; Rats; Receptors, Adrenergic, beta; Receptors, Cell Surface; Receptors, GABA-A; Ultracentrifugation | 1983 |
Beta-adrenoceptor heterogeneity in guinea-pig airways: comparison of functional and receptor labelling studies.
Topics: Animals; Binding, Competitive; Bronchi; Dihydroalprenolol; Guinea Pigs; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Lung; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Respiratory System; Trachea | 1983 |
[Monoacylglycerophosphatide formation during ligand-receptor interaction in the plasma membranes of brain synaptosomes. A possible mechanism of receptor desensitization].
Topics: Animals; Brain; Dihydroalprenolol; Drug Interactions; Fatty Acids; Hydrolysis; Isoproterenol; Ligands; Phosphatidic Acids; Phospholipases A; Phospholipids; Protein Binding; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Neurotransmitter; Synaptosomes | 1983 |
Studies on cyclic nucleotides in the adrenal gland. XI. Adrenergic regulation of adenylate cyclase activity in the adrenal cortex.
Topics: Adenylyl Cyclases; Adrenal Cortex; Adrenocorticotropic Hormone; Albuterol; Animals; Cell Membrane; Dihydroalprenolol; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Male; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1984 |
Triiodothyronamine--a beta-adrenergic metabolite of triiodothyronine?
Topics: Animals; Decarboxylation; Dihydroalprenolol; Diiodothyronines; Dopamine; Epinephrine; Erythrocytes; In Vitro Techniques; Isoproterenol; Norepinephrine; Receptors, Adrenergic, beta; Thyroxine; Triiodothyronine; Triiodothyronine, Reverse; Turkeys | 1983 |
Uncoupling of the beta-adrenergic receptor as a mechanism of in vitro neutrophil desensitization.
Topics: Blood Proteins; Cyclic AMP; Cycloheximide; Dihydroalprenolol; Drug Resistance; Epinephrine; Histamine; Humans; Isoproterenol; Kinetics; Membranes; Neutrophils; Norepinephrine; Prostaglandins E; Receptors, Adrenergic, beta; Uncoupling Agents | 1984 |
[Effect of thyroid hormones on the beta-adrenergic receptor internalization in isolated rat hepatocytes].
Topics: Alprenolol; Animals; Cadaverine; Dihydroalprenolol; In Vitro Techniques; Isoproterenol; Liver; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Thyroidectomy; Thyroxine | 1983 |
In vitro effects of aqueous cotton dust extract on leucocyte cyclic adenosine monophosphate levels.
Topics: Adult; Cell Survival; Cyclic AMP; Dihydroalprenolol; Dust; Female; Gossypium; Humans; Isoproterenol; Kinetics; Lymphocytes; Male; Monocytes; Receptors, Adrenergic, beta; Tritium | 1984 |
The beta-adrenergic receptor system in human glioma-derived cell lines: the mode of phosphodiesterase induction and the macromolecules phosphorylated by cyclic AMP-dependent protein kinase.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclases; Animals; Cell Line; Cyclic AMP; Cytosol; Dihydroalprenolol; Enzyme Induction; Glioma; Humans; Isoproterenol; Kinetics; Phosphoproteins; Phosphorylation; Protein Kinases; Rats; Receptors, Adrenergic, beta | 1984 |
In vivo desensitization of the beta, but not the alpha 2-adrenoreceptor-coupled-adenylate cyclase system in hamster white adipocytes after administration of epinephrine.
Topics: Adenylyl Cyclases; Adipose Tissue; Adrenocorticotropic Hormone; Animals; Cricetinae; Cyclic AMP; Dihydroalprenolol; Epinephrine; Glycerol; Isoproterenol; Kinetics; Male; Mesocricetus; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1984 |
Comparison of changes in the characteristics of beta-adrenoceptors and responsiveness of human circulating lymphocytes during and after chronic administration of pindolol and propranolol.
Topics: Adult; Cell Membrane; Cyclic AMP; Dihydroalprenolol; Humans; Isoproterenol; Lymphocytes; Male; Pindolol; Propranolol; Receptors, Adrenergic, beta; Substance Withdrawal Syndrome | 1984 |
Central activation and peripheral function of sympatho-adrenal and cardiovascular systems in the Zucker rat.
Topics: Adrenal Glands; Animals; Blood Pressure; Cardiovascular System; Dihydroalprenolol; Electric Stimulation; Epinephrine; Heart Rate; Isoproterenol; Male; Norepinephrine; Obesity; Rats; Rats, Mutant Strains; Rats, Zucker; Receptors, Adrenergic, beta; Sympathetic Nervous System; Ventromedial Hypothalamic Nucleus | 1984 |
Developmental alterations in guanine nucleotide regulation of the beta-adrenergic receptor-adenylate cyclase system of skeletal muscle.
Topics: Adenylyl Cyclases; Animals; Cholera Toxin; Cyclic AMP; Dihydroalprenolol; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Muscle Development; Muscles; Rabbits; Receptors, Adrenergic, beta; Sodium Fluoride | 1984 |
Postnatal development of the beta-adrenergic receptor complex in brown adipose tissue of the rat.
Topics: Adenylyl Cyclases; Adipose Tissue, Brown; Alprenolol; Animals; Animals, Newborn; Binding Sites; Dihydroalprenolol; Enzyme Activation; Female; Isoproterenol; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Sodium Fluoride | 1984 |
The interaction between beta- and alpha 2-adrenoceptors in cerebral cortical membranes: isoproterenol-induced increase in [3H]clonidine binding in rats.
Topics: Animals; Ascorbic Acid; Cell Membrane; Cerebral Cortex; Clonidine; Dihydroalprenolol; Isoproterenol; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Temperature | 1984 |
Dynamics of the lymphocyte beta-adrenoceptor system in patients with allergic bronchial asthma.
Topics: Adenylyl Cyclases; Adolescent; Adult; Asthma; Bronchial Provocation Tests; Cell Membrane; Dihydroalprenolol; Female; Guanosine Diphosphate; Guanosine Triphosphate; Humans; Isoproterenol; Lymphocytes; Male; Propranolol; Receptors, Adrenergic, beta; Respiratory Hypersensitivity | 1984 |
Influence of fasting on lipolytic response to adrenergic agonists and on adrenergic receptors in subcutaneous adipocytes.
Topics: Adipose Tissue; Adult; Clonidine; Dihydroalprenolol; Fasting; Female; Glycerol; Humans; In Vitro Techniques; Isoproterenol; Lipolysis; Middle Aged; Receptors, Adrenergic; Sympathomimetics; Theophylline | 1984 |
A study of mechanisms of post-irradiation changes in adenylate-cyclase activity.
Topics: Adenylyl Cyclases; Animals; Dihydroalprenolol; Dose-Response Relationship, Radiation; Erythrocyte Membrane; Erythrocytes; In Vitro Techniques; Isoproterenol; Lipid Peroxides; Membrane Lipids; Rana temporaria; Sodium Fluoride; Stimulation, Chemical | 1983 |
Influences of isoproterenol pretreatment on cerebral cortical bindings of [3H]clonidine and [3H]dihydroalprenolol in infant and adult rats.
Topics: Alprenolol; Animals; Cerebral Cortex; Clonidine; Dihydroalprenolol; Female; Isoproterenol; Male; Rats; Rats, Inbred Strains; Tritium | 1983 |
Characteristics of adrenergic binding sites associated with murine lymphocytes isolated from spleen.
Topics: Animals; Binding Sites; Binding, Competitive; Cell Membrane; Dihydroalprenolol; In Vitro Techniques; Isoproterenol; Kinetics; Lymphocytes; Mice; Receptors, Adrenergic; Spleen; Sympathomimetics | 1980 |
Mn2+-uncoupling of the catecholamine-sensitive adenylate cyclase system of rat reticulocytes. Parallel effects on cholera toxin-catalyzed ADP-ribosylation of the system.
Topics: Adenosine Diphosphate Ribose; Adenylyl Cyclases; Animals; Catecholamines; Cholera Toxin; Dihydroalprenolol; Guanylyl Imidodiphosphate; Isoproterenol; Magnesium; Manganese; Molecular Weight; Nucleoside Diphosphate Sugars; Rats; Reticulocytes | 1981 |
Functional alterations in components of pigeon erythrocyte adenylate cyclase following desensitization to isoproterenol.
Topics: Adenylyl Cyclases; Animals; Cells, Cultured; Cholera Toxin; Columbidae; Dihydroalprenolol; Drug Tolerance; Erythrocyte Membrane; Erythrocytes; Isoproterenol | 1981 |
Regulation of the adenylate cyclase system by catecholamines in the rat prostate.
Topics: Adenylyl Cyclases; Animals; Catecholamines; Dihydroalprenolol; Dopamine; Haloperidol; In Vitro Techniques; Isoproterenol; Male; Membranes; Propranolol; Prostate; Rats | 1980 |
Effects of androgens on isoproterenol-sensitive adenylate cyclase system of the rat prostate.
Topics: Adenylyl Cyclases; Androgens; Animals; Dihydroalprenolol; Fluorides; Guanylyl Imidodiphosphate; In Vitro Techniques; Isoproterenol; Male; Membranes; Prostate; Rats | 1980 |
Fluorescent labeling of purified beta 2 adrenergic receptor. Evidence for ligand-specific conformational changes.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Line; Cysteine; Dihydroalprenolol; Fluorescent Dyes; Histidine; Humans; Isoproterenol; Kinetics; Ligands; Models, Structural; Oxadiazoles; Protein Conformation; Receptors, Adrenergic, beta-2; Recombinant Proteins; Sensitivity and Specificity; Sequence Tagged Sites; Spectrometry, Fluorescence; Spodoptera; Time Factors; Transfection | 1995 |
The involvement of ATP-sensitive potassium channels in beta-adrenoceptor-mediated vasorelaxation in the rat isolated mesenteric arterial bed.
Topics: Adenosine Triphosphate; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Binding, Competitive; Bucladesine; Dihydroalprenolol; Dobutamine; Glyburide; In Vitro Techniques; Isoproterenol; Male; Mesenteric Arteries; Muscle Relaxation; Muscle, Smooth, Vascular; Potassium Channel Blockers; Potassium Channels; Radioligand Assay; Rats; Rats, Wistar; Terbutaline; Vasodilation; Vasodilator Agents; Verapamil | 1995 |
Neuropeptide Y prevents agonist-stimulated increases in contractility.
Topics: Animals; Dihydroalprenolol; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Neuropeptide Y; Phenylephrine; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1995 |
Alpha-methyl-para-tyrosine antagonizes the effect of chronic imipramine on learned helplessness in rats.
Topics: Adenylyl Cyclases; alpha-Methyltyrosine; Animals; Cerebral Cortex; Dihydroalprenolol; Down-Regulation; Helplessness, Learned; Imipramine; Isoproterenol; Male; Membranes; Methyltyrosines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Tyrosine 3-Monooxygenase | 1993 |
A cytosolic peptide potentiates the GTP effect on beta-adrenergic response of adenylate cyclase.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Binding, Competitive; Cytosol; Dihydroalprenolol; Electrophoresis, Polyacrylamide Gel; Enzyme Activation; Female; Guanosine Triphosphate; Isoproterenol; Peptides; Rats; Rats, Wistar | 1994 |
The in-vitro effects of insulin and the effects of acute fasting on cardiac beta-adrenoceptor responses in the short-term streptozotocin-diabetic rat.
Topics: Analysis of Variance; Animals; Blood Glucose; Colforsin; Diabetes Mellitus, Experimental; Dihydroalprenolol; Fasting; Female; Heart; In Vitro Techniques; Insulin; Isoproterenol; Myocardium; Papillary Muscles; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Streptozocin | 1994 |
Potentiation of alpha-adrenoceptor-mediated responses following chronic beta-adrenoceptor stimulation in the rat heart.
Topics: Adrenergic beta-Agonists; Animals; Cardiac Pacing, Artificial; Dihydroalprenolol; Drug Implants; Drug Synergism; Heart; Heart Atria; In Vitro Techniques; Isoproterenol; Kinetics; Male; Myocardial Contraction; Norepinephrine; Papillary Muscles; Phenylephrine; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha | 1993 |
Effects of hydrogen peroxide on stimulatory guanine nucleotide-binding protein in rat heart.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Binding Sites; Colforsin; Cyclic AMP; Dihydroalprenolol; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Heart; Hydrogen Peroxide; In Vitro Techniques; Isoproterenol; Lymphoma; Male; Myocardium; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Tumor Cells, Cultured | 1993 |
Elevated lung G protein levels and muscarinic receptor affinity in a mouse model of airway hyperreactivity.
Topics: Animals; Binding, Competitive; Bronchial Hyperreactivity; Cell Membrane; Dihydroalprenolol; Disease Models, Animal; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Lung; Male; Mice; Mice, Inbred A; Mice, Inbred C3H; Molecular Weight; Quinuclidinyl Benzilate; Receptors, Adrenergic, beta-2; Receptors, Muscarinic; Species Specificity | 1993 |
Beta-adrenergic receptors in corpora lutea from different stages of the estrous cycle in conscious and slaughtered cattle.
Topics: Animals; Cattle; Cell Membrane; Corpus Luteum; Dihydroalprenolol; Epinephrine; Estrus; Female; Isoproterenol; Norepinephrine; Progesterone; Receptors, Adrenergic, beta; Tritium | 1994 |
Sex hormones change adrenoceptors in blood vessels of the spontaneously hypertensive rat.
Topics: Animals; Arteries; Blood Pressure; Dihydroalprenolol; Hypertension; Isoproterenol; Kinetics; Male; Norepinephrine; Orchiectomy; Prazosin; Rats; Rats, Inbred SHR; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Testis; Testosterone | 1993 |
Externalization and internalization of (Na+ + K+)-ATPase in rat heart during different phases of sepsis.
Topics: Adenosine Triphosphate; Affinity Labels; Animals; Azides; Binding, Competitive; Dihydroalprenolol; Guanylyl Imidodiphosphate; Isoproterenol; Male; Myocardium; Ouabain; Photochemistry; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Sarcolemma; Sepsis | 1993 |
Ricin depresses cardiac function in the rabbit heart.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dihydroalprenolol; Electrocardiography; Heart; In Vitro Techniques; Isoproterenol; Myocardial Contraction; Myocardium; Oxygen Consumption; Propranolol; Rabbits; Receptors, Adrenergic, beta; Ricin; Ventricular Function, Left | 1996 |
Molecular and functional identification of beta-adrenergic receptors in distal convoluted tubule cells.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Calcium; Cells, Cultured; Cyclic AMP; Dihydroalprenolol; Isoproterenol; Kidney Tubules, Distal; Mice; Propranolol; Receptors, Adrenergic, beta; RNA, Messenger; Sodium | 1997 |
Agonists induce conformational changes in transmembrane domains III and VI of the beta2 adrenoceptor.
Topics: Adrenergic beta-Agonists; Amino Acid Sequence; Computer Simulation; Cysteine; Dihydroalprenolol; Fluorescent Dyes; Isoproterenol; Models, Molecular; Molecular Sequence Data; Mutation; Protein Conformation; Receptors, Adrenergic, beta-2; Spectrometry, Fluorescence | 1997 |
Reconstitution of beta2-adrenoceptor-GTP-binding-protein interaction in Sf9 cells--high coupling efficiency in a beta2-adrenoceptor-G(s alpha) fusion protein.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; beta-Adrenergic Receptor Kinases; Binding, Competitive; Cell Line; Cell Membrane; Cyclic AMP-Dependent Protein Kinases; Dihydroalprenolol; GTP Phosphohydrolases; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanosine Triphosphate; Isoproterenol; Kinetics; Polymerase Chain Reaction; Propanolamines; Rats; Receptors, Adrenergic, beta; Recombinant Fusion Proteins; Spodoptera; Transfection | 1998 |
beta-adrenergic relaxation of rabbit tracheal smooth muscle: a receptor deficit that improves with corticosteroid administration.
Topics: Acetylcholine; Adrenal Cortex Hormones; Adrenergic beta-Agonists; Animals; Anti-Inflammatory Agents; Cyclic AMP; Dexamethasone; Dihydroalprenolol; Dose-Response Relationship, Drug; Drug Interactions; GTP-Binding Protein alpha Subunits, Gi-Go; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Protein Binding; Rabbits; Radioligand Assay; Receptors, Adrenergic, beta; Trachea; Vasodilator Agents | 2000 |
Rapid electrical stimulation of contraction reduces the density of beta-adrenergic receptors and responsiveness of cultured neonatal rat cardiomyocytes. Possible involvement of microtubule disassembly secondary to mechanical stress.
Topics: Acetylcholine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Antineoplastic Agents, Phytogenic; Cells, Cultured; Colforsin; Diacetyl; Dihydroalprenolol; Down-Regulation; Electric Stimulation; Enzyme Inhibitors; Heart Failure; Isoproterenol; Microtubules; Muscle Fibers, Skeletal; Myocardial Contraction; Myocardium; Pacemaker, Artificial; Paclitaxel; Propanolamines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Stress, Mechanical; Tritium; Vasodilator Agents | 2000 |
Ligand regulation of green fluorescent protein-tagged forms of the human beta(1)- and beta(2)-adrenoceptors; comparisons with the unmodified receptors.
Topics: Betaxolol; Binding, Competitive; Cell Line; Dihydroalprenolol; Endocytosis; Green Fluorescent Proteins; Humans; Isoproterenol; Kinetics; Ligands; Luminescent Proteins; Microscopy, Confocal; Oligopeptides; Peptides; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Fusion Proteins; Tritium | 2000 |
Beta-adrenergic receptor subtypes mediating lipolysis in porcine adipocytes. Studies with BRL-37344, a putative beta3-adrenergic agonist.
Topics: Adenylyl Cyclases; Adipocytes; Adrenergic beta-Agonists; Animals; Cell Fractionation; Dihydroalprenolol; Ethanolamines; Intracellular Membranes; Isoproterenol; Lipolysis; Muscle, Skeletal; Receptors, Adrenergic, beta; Swine | 2000 |
The effect of streptozotocin-induced diabetes on cardiac beta-adrenoceptor subtypes in the rat.
Topics: Adrenergic beta-Agonists; Animals; Binding Sites; Blood Glucose; Blood Pressure; Body Weight; Diabetes Mellitus, Experimental; Dihydroalprenolol; Heart Rate; Imidazoles; Isoproterenol; Male; Myocardium; Perfusion; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Stimulation, Chemical; Streptozocin | 2001 |
The olfactory G protein G(alphaolf) possesses a lower GDP-affinity and deactivates more rapidly than G(salphashort): consequences for receptor-coupling and adenylyl cyclase activation.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Alternative Splicing; Animals; Cell Line; Cell Membrane; Dihydroalprenolol; Dobutamine; Ephedrine; Genetic Variation; GTP-Binding Protein alpha Subunits; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanosine Triphosphate; Heterotrimeric GTP-Binding Proteins; Isoproterenol; Kinetics; Rats; Receptors, Adrenergic, beta-2; Recombinant Fusion Proteins; Recombinant Proteins; Spodoptera; Transfection | 2001 |
Daily changes in beta-adrenergic sensitivity of rat submandibular gland. Correlation with beta-adrenoceptor rhythm.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Circadian Rhythm; Dihydroalprenolol; Feeding Behavior; Female; Isoproterenol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Saliva; Submandibular Gland; Superior Cervical Ganglion; Tritium | 2001 |
Release of norepinephrine from human ovary: coupling to steroidogenic response.
Topics: Adrenergic beta-Agonists; Adult; Binding Sites; Calcium; Cell Membrane; Cells, Cultured; Dihydroalprenolol; Dopamine; Electric Stimulation; Epinephrine; Ethanolamines; Female; Granulosa Cells; Humans; Isoproterenol; Middle Aged; Norepinephrine; Ovary; Progesterone; Receptors, Adrenergic, beta; Tritium | 2001 |
Intracellular cAMP increases during the positive inotropism induced by androgens in isolated left atrium of rat.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Androgens; Animals; Atenolol; Atrial Function; Binding, Competitive; Cattle; Cyclic AMP; Dihydroalprenolol; Dihydrotestosterone; Dose-Response Relationship, Drug; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Membranes; Myocardial Contraction; Phosphodiesterase Inhibitors; Rats; Rats, Wistar; Reserpine; Serum Albumin, Bovine; Tritium | 2002 |
Diversity of inhibitory responses to beta2-stimulants shown by term-pregnant human myometria in vitro is partly due to differences in receptor density.
Topics: Acetamides; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Binding Sites; Binding, Competitive; Delivery, Obstetric; Dihydroalprenolol; Female; Humans; In Vitro Techniques; Isoproterenol; Membrane Potentials; Myometrium; Naphthalenes; Osmolar Concentration; Pregnancy; Receptors, Adrenergic, beta; Tocolytic Agents; Uterine Contraction | 2002 |
[Molecular mechanisms of regulatory action of adrenergic receptor agonists on functional activity of adenylyl cyclase signaling system of the ciliates Dileptus anser and Tetrahymena pyriformis].
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cell Membrane; Ciliophora; Dihydroalprenolol; Enzyme Activation; Epinephrine; Guanosine Triphosphate; Isoproterenol; Signal Transduction; Tetrahymena pyriformis | 2004 |
Histamine augments beta2-adrenoceptor-induced cyclic AMP accumulation in human prostate cancer cells DU-145 independently of known histamine receptors.
Topics: Cell Line, Tumor; Cyclic AMP; Dihydroalprenolol; Histamine; Humans; Isoproterenol; Male; Prostatic Neoplasms; Receptors, Adrenergic, beta-2; Receptors, Histamine; Zinc | 2007 |
Exercise training initiated after the onset of diabetes preserves myocardial function: effects on expression of beta-adrenoceptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blotting, Western; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 1; Dihydroalprenolol; Echocardiography; Exercise Therapy; Heart Rate; Hemodynamics; Isoproterenol; Male; Myocardial Contraction; Myocardium; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Stroke Volume; Time Factors; Ventricular Function, Left | 2008 |
Putrescine modulation of acute activation of the beta-adrenergic system in the left atrium of rat.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiotonic Agents; Chromatography, High Pressure Liquid; Cyclic AMP; Dihydroalprenolol; Eflornithine; Enzyme Inhibitors; Heart; Heart Atria; Isoproterenol; Male; Membranes; Myocardium; Putrescine; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Spermidine; Spermine | 2008 |
Beta(2)-adrenergic receptor regulates cardiac fibroblast autophagy and collagen degradation.
Topics: Adenine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Autophagy; Blotting, Western; Cells, Cultured; Collagen; Dihydroalprenolol; Dose-Response Relationship, Drug; Fibroblasts; Isoproterenol; Male; Microscopy, Electron, Transmission; Myocardium; Norepinephrine; Propanolamines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-2; Tritium | 2011 |
Structural and functional roles of small group-conserved amino acids present on helix-H7 in the β(2)-adrenergic receptor.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amino Acid Substitution; Amino Acids; Animals; Binding Sites; Chlorocebus aethiops; COS Cells; Cricetinae; Cyclic AMP; Dihydroalprenolol; Glycine; HEK293 Cells; Humans; Hydrogen Bonding; Isoproterenol; Models, Molecular; Mutation; Protein Binding; Protein Structure, Secondary; Protein Structure, Tertiary; Radioligand Assay; Receptors, Adrenergic, beta-2; Serine; Structure-Activity Relationship | 2011 |