dihydroalprenolol has been researched along with cgp 12177 in 31 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 21 (67.74) | 18.7374 |
1990's | 7 (22.58) | 18.2507 |
2000's | 3 (9.68) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bultsma, T; Donné-Op den Kelder, GM; Rademaker, B; Timmerman, H | 1 |
McNeel, RL; Mersmann, HJ | 1 |
Moon, TW; Perry, SF; Reid, SD | 1 |
Kállay, Z; Marko, V; Smisterová, J; Soltés, L | 1 |
Coury, A; Guyard, A; Rumigny, JF | 1 |
Creese, I; Riva, MA | 2 |
Hui, KK; Yu, JL | 1 |
Cheetham, SC; Crompton, MR; De Paermentier, F; Horton, RW | 1 |
De Blasi, A; Fratelli, M; Insel, PA; Lipartiti, M; Motulsky, HJ | 1 |
Henneberry, RC; Jahangeer, S; Lysko, PG | 1 |
Contreras, ML; Molinoff, PB; Wolfe, BB | 1 |
Limas, C; Limas, CJ | 2 |
Lang, PH; Lemmer, B | 1 |
Algeri, S; Costantini, C; Cotecchia, S; De Blasi, A; Fratelli, M; Lipartiti, M; Sacchetti, G | 1 |
Arinze, IJ; Graham, SM; Kawai, Y; Yoshioka, H | 1 |
De Blasi, A; Fratelli, M; Lipartiti, M; Wielosz, M | 1 |
Marttila, T; Niina, O; Nikinmaa, M | 1 |
Hertel, C; Müller, P; Portenier, M; Staehelin, M | 2 |
Montandon, JB; Porzig, H | 1 |
Baer, M; Chanton, C; Porzig, H | 1 |
Delavier-Klutchko, C; Hoebeke, J; Strosberg, AD | 1 |
Mutschler, E; Palm, D; Schäfer-Korting, M; Wellstein, A; Wiemer, G | 1 |
Kobilka, BK; von Zastrow, M | 1 |
Mersmann, HJ | 1 |
Cloutier, MM; Guernsey, L; Schramm, CM | 1 |
Ito, M; Nakagawa, M; Saikawa, T; Takahashi, N; Teshima, Y; Yasunaga, S; Yonemochi, H | 1 |
McLean, AJ; Milligan, G | 1 |
Alewijnse, AE; Michel, MC; Michel-Reher, MB; Niclauss, N | 1 |
31 other study(ies) available for dihydroalprenolol and cgp 12177
Article | Year |
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Mapping of the beta 2-adrenoceptor on Chang liver cells. Differences between high- and low-affinity receptor states.
Topics: Cell Membrane; Cells, Cultured; Guanylyl Imidodiphosphate; Hydrogen Bonding; Iodocyanopindolol; Liver; Models, Molecular; Pindolol; Protein Conformation; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Dopamine D2; Stereoisomerism; Structure-Activity Relationship | 1988 |
Ligand binding to the porcine adipose tissue beta-adrenergic receptor.
Topics: Adipose Tissue; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Dihydroalprenolol; Guanosine Triphosphate; Kinetics; Ligands; Molecular Conformation; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Swine; Temperature; Time Factors | 1992 |
Characterization of beta-adrenoreceptors of rainbow trout (Oncorhynchus mykiss) erythrocytes.
Topics: Animals; Binding, Competitive; Cell Compartmentation; Dihydroalprenolol; Erythrocytes; Female; Hydrogen-Ion Concentration; Isoproterenol; Male; Propanolamines; Receptors, Adrenergic, beta; Trout | 1991 |
Evaluation of 3H-CGP 12177 and 3H-DHA binding to beta 2-adrenoceptors of rat reticulocytes by means of affinity spectra.
Topics: Animals; Binding Sites; Dihydroalprenolol; Female; In Vitro Techniques; Male; Propanolamines; Radioligand Assay; Rats; Receptors, Adrenergic, beta; Reticulocytes | 1991 |
Characterization of beta-adrenoceptors in synaptoneurosomes from rat brain: [3H]dihydroalprenolol versus [3H]CGP 12177.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Brain Chemistry; Dihydroalprenolol; Propanolamines; Radioligand Assay; Rats; Receptors, Adrenergic, beta; Synaptosomes; Tritium | 1990 |
Comparison of two putatively selective radioligands for labeling central nervous system beta-adrenergic receptors: inadequacy of [3H]dihydroalprenolol.
Topics: Alprenolol; Animals; Brain Chemistry; Dihydroalprenolol; Guanosine Triphosphate; Isoproterenol; Kinetics; Male; Propanolamines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin | 1989 |
Reevaluation of the regulation of beta-adrenergic receptor binding by desipramine treatment.
Topics: Animals; Desipramine; Dihydroalprenolol; Fenclonine; Kinetics; Male; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin | 1989 |
Effects of calcium channel blockers and ketotifen on beta 2 adrenergic receptor regulation in intact human lymphocytes.
Topics: Adrenergic beta-Antagonists; Calcium Channel Blockers; Cyclic AMP; Dihydroalprenolol; Humans; In Vitro Techniques; Isoproterenol; Ketotifen; Lymphocytes; Propanolamines; Radioimmunoassay; Receptors, Adrenergic, beta | 1989 |
Beta-adrenoceptors in human brain labelled with [3H]dihydroalprenolol and [3H]CGP 12177.
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Brain Chemistry; Dihydroalprenolol; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Practolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 1989 |
Agonist-induced redistribution of beta-adrenergic receptors on intact human mononuclear leukocytes: redistributed receptors are nonfunctional.
Topics: Adrenergic beta-Antagonists; Adult; Cyclic AMP; Dihydroalprenolol; Humans; In Vitro Techniques; Isoproterenol; Kinetics; Leukocytes; Ligands; Male; Propanolamines; Receptors, Adrenergic, beta | 1985 |
Transport of beta-adrenergic antagonists in the absence of beta-adrenergic receptors in rat pituitary tumor cells.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Biological Transport; Cell Line; Colforsin; Cyclic AMP; Dihydroalprenolol; Epinephrine; Hydrogen-Ion Concentration; Imipramine; Kinetics; Monensin; Norepinephrine; Nucleotides; Oligomycins; Ouabain; Pituitary Neoplasms; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta; Reserpine; Serotonin; Temperature | 1986 |
Kinetic analysis of the interactions of agonists and antagonists with beta adrenergic receptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Bupranolol; Cell Line; Computers; Dihydroalprenolol; Kinetics; Mathematics; Pindolol; Propanolamines; Time Factors | 1986 |
Altered intracellular adrenoceptor distribution in myocardium of spontaneously hypertensive rats.
Topics: Adrenergic beta-Agonists; Animals; Cardiomegaly; Cell Membrane; Cytosol; Dihydroalprenolol; Hypertension; Myocardial Contraction; Myocardium; Prazosin; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Tissue Distribution | 1987 |
Evidence for two specific affinity states of 3H-antagonist binding to cardiac beta-adrenergic receptors and influence of Gpp(NH)p.
Topics: Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Male; Myocardium; Propanolamines; Rats; Receptors, Adrenergic, beta | 1985 |
Stress induced desensitization of lymphocyte beta-adrenoceptors in young and aged rats.
Topics: Age Factors; Animals; Corticosterone; Dihydroalprenolol; Isoproterenol; Lymphocytes; Male; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Restraint, Physical; Stress, Physiological | 1986 |
Beta-adrenergic receptors in guinea-pig liver plasma membranes and thermal lability of [3H]dihydroalprenolol binding sites.
Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Alprenolol; Animals; Binding, Competitive; Cell Membrane; Cholera Toxin; Dihydroalprenolol; Guanylyl Imidodiphosphate; Guinea Pigs; Hot Temperature; Iodocyanopindolol; Isoproterenol; Liver; Male; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Virulence Factors, Bordetella | 1986 |
Regulation of beta adrenergic receptors on rat mononuclear leukocytes by stress: receptor redistribution and down-regulation are altered with aging.
Topics: Aging; Animals; Cyclic AMP; Dihydroalprenolol; Isoproterenol; Male; Monocytes; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Restraint, Physical; Stress, Physiological; Time Factors | 1987 |
Binding of beta-adrenergic antagonists 3H-DHA and 3H-CGP 12177 to intact rainbow trout (Salmo gairdneri) and carp (Cyprinus carpio) red blood cells.
Topics: Alprenolol; Animals; Carps; Cyprinidae; Dihydroalprenolol; Erythrocytes; Ligands; Membrane Lipids; Propanolamines; Salmonidae; Trout | 1988 |
Rapid recovery of cardiac beta-adrenergic receptors after isoproterenol-induced "down"-regulation.
Topics: Adenosine Triphosphate; Animals; Colchicine; Cyclic AMP; Cytoplasm; Dihydroalprenolol; Drug Tolerance; Isoproterenol; Male; Monensin; Myocardium; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1984 |
Some unique properties of CGP-12177.
Topics: Adenylyl Cyclases; Animals; Cell Line; Cyclic AMP; Digitonin; Dihydroalprenolol; Glioma; Isoproterenol; Propanolamines; Rats; Receptors, Adrenergic, beta; Stereoisomerism | 1984 |
Changes in beta-adrenoceptor binding properties and receptor-cyclase coupling during in vitro maturation of rat reticulocytes.
Topics: Adenosine Triphosphate; Adenylyl Cyclases; Animals; Cells, Cultured; Cyclic AMP; Dihydroalprenolol; Isoproterenol; Propanolamines; Rats; Receptors, Adrenergic, beta; Reticulocytes | 1984 |
Properties of beta-adrenoceptor sites in metabolizing and nonmetabolizing rat reticulocytes and in resealed reticulocyte ghosts.
Topics: Adrenergic beta-Antagonists; Animals; Cell Membrane; Cold Temperature; Cytosol; Dihydroalprenolol; Energy Metabolism; Female; Isoproterenol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Reticulocytes; Timolol | 1981 |
Determination of the desensitization of beta-adrenergic receptors by [3H]CGP-12177.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Binding Sites; Binding, Competitive; Cell Line; Cell Membrane; Centrifugation, Density Gradient; Dihydroalprenolol; Glioma; Humans; Isoproterenol; Propanolamines; Receptors, Adrenergic, beta | 1983 |
The human carcinoma cell line A431 possesses large numbers of functional beta-adrenergic receptors.
Topics: Adrenergic beta-Antagonists; Binding, Competitive; Carcinoma, Squamous Cell; Cell Line; Dihydroalprenolol; Humans; Isoproterenol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism | 1984 |
Simple and reliable radioreceptor assay for beta-adrenoceptor antagonists and active metabolites in native human plasma.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Carteolol; Dihydroalprenolol; Erythrocyte Membrane; Female; Humans; Male; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Time Factors | 1984 |
Antagonist-dependent and -independent steps in the mechanism of adrenergic receptor internalization.
Topics: Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Antibodies, Monoclonal; Azides; Cell Line, Transformed; Cell Membrane; Cold Temperature; Dihydroalprenolol; Endocytosis; Epitopes; Humans; Microscopy, Immunoelectron; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-2; Recombinant Proteins; Sodium Azide; Tritium | 1994 |
Evidence of classic beta 3-adrenergic receptors in porcine adipocytes.
Topics: Adipocytes; Adrenergic beta-Antagonists; Animals; Binding Sites; Binding, Competitive; Cell Membrane; Dihydroalprenolol; Iodocyanopindolol; Magnesium Chloride; Male; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; RNA; Swine; Tritium | 1996 |
Tannin inhibits the cAMP-beta-adrenergic receptor pathway in bovine tracheal epithelium.
Topics: Acetylcysteine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cattle; Chloride Channels; Cyclic AMP; Dihydroalprenolol; Epithelium; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Hydrolyzable Tannins; Propanolamines; Receptors, Adrenergic, beta; Trachea | 1998 |
Rapid electrical stimulation of contraction reduces the density of beta-adrenergic receptors and responsiveness of cultured neonatal rat cardiomyocytes. Possible involvement of microtubule disassembly secondary to mechanical stress.
Topics: Acetylcholine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Antineoplastic Agents, Phytogenic; Cells, Cultured; Colforsin; Diacetyl; Dihydroalprenolol; Down-Regulation; Electric Stimulation; Enzyme Inhibitors; Heart Failure; Isoproterenol; Microtubules; Muscle Fibers, Skeletal; Myocardial Contraction; Myocardium; Pacemaker, Artificial; Paclitaxel; Propanolamines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Stress, Mechanical; Tritium; Vasodilator Agents | 2000 |
Ligand regulation of green fluorescent protein-tagged forms of the human beta(1)- and beta(2)-adrenoceptors; comparisons with the unmodified receptors.
Topics: Betaxolol; Binding, Competitive; Cell Line; Dihydroalprenolol; Endocytosis; Green Fluorescent Proteins; Humans; Isoproterenol; Kinetics; Ligands; Luminescent Proteins; Microscopy, Confocal; Oligopeptides; Peptides; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Fusion Proteins; Tritium | 2000 |
Comparison of three radioligands for the labelling of human beta-adrenoceptor subtypes.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Dihydroalprenolol; Ethanolamines; Humans; Iodine Radioisotopes; Iodocyanopindolol; Isotope Labeling; Kinetics; Propanolamines; Protein Binding; Radioligand Assay; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Tetrahydronaphthalenes; Tritium | 2006 |