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dihydroalprenolol and cgp 12177

dihydroalprenolol has been researched along with cgp 12177 in 31 studies

Research

Studies (31)

TimeframeStudies, this research(%)All Research%
pre-199021 (67.74)18.7374
1990's7 (22.58)18.2507
2000's3 (9.68)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bultsma, T; Donné-Op den Kelder, GM; Rademaker, B; Timmerman, H1
McNeel, RL; Mersmann, HJ1
Moon, TW; Perry, SF; Reid, SD1
Kállay, Z; Marko, V; Smisterová, J; Soltés, L1
Coury, A; Guyard, A; Rumigny, JF1
Creese, I; Riva, MA2
Hui, KK; Yu, JL1
Cheetham, SC; Crompton, MR; De Paermentier, F; Horton, RW1
De Blasi, A; Fratelli, M; Insel, PA; Lipartiti, M; Motulsky, HJ1
Henneberry, RC; Jahangeer, S; Lysko, PG1
Contreras, ML; Molinoff, PB; Wolfe, BB1
Limas, C; Limas, CJ2
Lang, PH; Lemmer, B1
Algeri, S; Costantini, C; Cotecchia, S; De Blasi, A; Fratelli, M; Lipartiti, M; Sacchetti, G1
Arinze, IJ; Graham, SM; Kawai, Y; Yoshioka, H1
De Blasi, A; Fratelli, M; Lipartiti, M; Wielosz, M1
Marttila, T; Niina, O; Nikinmaa, M1
Hertel, C; Müller, P; Portenier, M; Staehelin, M2
Montandon, JB; Porzig, H1
Baer, M; Chanton, C; Porzig, H1
Delavier-Klutchko, C; Hoebeke, J; Strosberg, AD1
Mutschler, E; Palm, D; Schäfer-Korting, M; Wellstein, A; Wiemer, G1
Kobilka, BK; von Zastrow, M1
Mersmann, HJ1
Cloutier, MM; Guernsey, L; Schramm, CM1
Ito, M; Nakagawa, M; Saikawa, T; Takahashi, N; Teshima, Y; Yasunaga, S; Yonemochi, H1
McLean, AJ; Milligan, G1
Alewijnse, AE; Michel, MC; Michel-Reher, MB; Niclauss, N1

Other Studies

31 other study(ies) available for dihydroalprenolol and cgp 12177

ArticleYear
Mapping of the beta 2-adrenoceptor on Chang liver cells. Differences between high- and low-affinity receptor states.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:6

    Topics: Cell Membrane; Cells, Cultured; Guanylyl Imidodiphosphate; Hydrogen Bonding; Iodocyanopindolol; Liver; Models, Molecular; Pindolol; Protein Conformation; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Dopamine D2; Stereoisomerism; Structure-Activity Relationship

1988
Ligand binding to the porcine adipose tissue beta-adrenergic receptor.
    Journal of animal science, 1992, Volume: 70, Issue:3

    Topics: Adipose Tissue; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Dihydroalprenolol; Guanosine Triphosphate; Kinetics; Ligands; Molecular Conformation; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Swine; Temperature; Time Factors

1992
Characterization of beta-adrenoreceptors of rainbow trout (Oncorhynchus mykiss) erythrocytes.
    The Journal of experimental biology, 1991, Volume: 158

    Topics: Animals; Binding, Competitive; Cell Compartmentation; Dihydroalprenolol; Erythrocytes; Female; Hydrogen-Ion Concentration; Isoproterenol; Male; Propanolamines; Receptors, Adrenergic, beta; Trout

1991
Evaluation of 3H-CGP 12177 and 3H-DHA binding to beta 2-adrenoceptors of rat reticulocytes by means of affinity spectra.
    Journal of receptor research, 1991, Volume: 11, Issue:6

    Topics: Animals; Binding Sites; Dihydroalprenolol; Female; In Vitro Techniques; Male; Propanolamines; Radioligand Assay; Rats; Receptors, Adrenergic, beta; Reticulocytes

1991
Characterization of beta-adrenoceptors in synaptoneurosomes from rat brain: [3H]dihydroalprenolol versus [3H]CGP 12177.
    Biochemical Society transactions, 1990, Volume: 18, Issue:3

    Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Brain Chemistry; Dihydroalprenolol; Propanolamines; Radioligand Assay; Rats; Receptors, Adrenergic, beta; Synaptosomes; Tritium

1990
Comparison of two putatively selective radioligands for labeling central nervous system beta-adrenergic receptors: inadequacy of [3H]dihydroalprenolol.
    Molecular pharmacology, 1989, Volume: 36, Issue:1

    Topics: Alprenolol; Animals; Brain Chemistry; Dihydroalprenolol; Guanosine Triphosphate; Isoproterenol; Kinetics; Male; Propanolamines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin

1989
Reevaluation of the regulation of beta-adrenergic receptor binding by desipramine treatment.
    Molecular pharmacology, 1989, Volume: 36, Issue:1

    Topics: Animals; Desipramine; Dihydroalprenolol; Fenclonine; Kinetics; Male; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin

1989
Effects of calcium channel blockers and ketotifen on beta 2 adrenergic receptor regulation in intact human lymphocytes.
    Research communications in chemical pathology and pharmacology, 1989, Volume: 65, Issue:1

    Topics: Adrenergic beta-Antagonists; Calcium Channel Blockers; Cyclic AMP; Dihydroalprenolol; Humans; In Vitro Techniques; Isoproterenol; Ketotifen; Lymphocytes; Propanolamines; Radioimmunoassay; Receptors, Adrenergic, beta

1989
Beta-adrenoceptors in human brain labelled with [3H]dihydroalprenolol and [3H]CGP 12177.
    European journal of pharmacology, 1989, Aug-29, Volume: 167, Issue:3

    Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Brain Chemistry; Dihydroalprenolol; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Practolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta

1989
Agonist-induced redistribution of beta-adrenergic receptors on intact human mononuclear leukocytes: redistributed receptors are nonfunctional.
    The Journal of clinical endocrinology and metabolism, 1985, Volume: 61, Issue:6

    Topics: Adrenergic beta-Antagonists; Adult; Cyclic AMP; Dihydroalprenolol; Humans; In Vitro Techniques; Isoproterenol; Kinetics; Leukocytes; Ligands; Male; Propanolamines; Receptors, Adrenergic, beta

1985
Transport of beta-adrenergic antagonists in the absence of beta-adrenergic receptors in rat pituitary tumor cells.
    Biochemical pharmacology, 1986, Aug-15, Volume: 35, Issue:16

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Biological Transport; Cell Line; Colforsin; Cyclic AMP; Dihydroalprenolol; Epinephrine; Hydrogen-Ion Concentration; Imipramine; Kinetics; Monensin; Norepinephrine; Nucleotides; Oligomycins; Ouabain; Pituitary Neoplasms; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta; Reserpine; Serotonin; Temperature

1986
Kinetic analysis of the interactions of agonists and antagonists with beta adrenergic receptors.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Bupranolol; Cell Line; Computers; Dihydroalprenolol; Kinetics; Mathematics; Pindolol; Propanolamines; Time Factors

1986
Altered intracellular adrenoceptor distribution in myocardium of spontaneously hypertensive rats.
    The American journal of physiology, 1987, Volume: 253, Issue:4 Pt 2

    Topics: Adrenergic beta-Agonists; Animals; Cardiomegaly; Cell Membrane; Cytosol; Dihydroalprenolol; Hypertension; Myocardial Contraction; Myocardium; Prazosin; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Tissue Distribution

1987
Evidence for two specific affinity states of 3H-antagonist binding to cardiac beta-adrenergic receptors and influence of Gpp(NH)p.
    Journal of cyclic nucleotide and protein phosphorylation research, 1985, Volume: 10, Issue:4

    Topics: Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Male; Myocardium; Propanolamines; Rats; Receptors, Adrenergic, beta

1985
Stress induced desensitization of lymphocyte beta-adrenoceptors in young and aged rats.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:4

    Topics: Age Factors; Animals; Corticosterone; Dihydroalprenolol; Isoproterenol; Lymphocytes; Male; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Restraint, Physical; Stress, Physiological

1986
Beta-adrenergic receptors in guinea-pig liver plasma membranes and thermal lability of [3H]dihydroalprenolol binding sites.
    Biochemical pharmacology, 1986, Dec-15, Volume: 35, Issue:24

    Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Alprenolol; Animals; Binding, Competitive; Cell Membrane; Cholera Toxin; Dihydroalprenolol; Guanylyl Imidodiphosphate; Guinea Pigs; Hot Temperature; Iodocyanopindolol; Isoproterenol; Liver; Male; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Virulence Factors, Bordetella

1986
Regulation of beta adrenergic receptors on rat mononuclear leukocytes by stress: receptor redistribution and down-regulation are altered with aging.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:1

    Topics: Aging; Animals; Cyclic AMP; Dihydroalprenolol; Isoproterenol; Male; Monocytes; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Restraint, Physical; Stress, Physiological; Time Factors

1987
Binding of beta-adrenergic antagonists 3H-DHA and 3H-CGP 12177 to intact rainbow trout (Salmo gairdneri) and carp (Cyprinus carpio) red blood cells.
    General and comparative endocrinology, 1988, Volume: 70, Issue:3

    Topics: Alprenolol; Animals; Carps; Cyprinidae; Dihydroalprenolol; Erythrocytes; Ligands; Membrane Lipids; Propanolamines; Salmonidae; Trout

1988
Rapid recovery of cardiac beta-adrenergic receptors after isoproterenol-induced "down"-regulation.
    Circulation research, 1984, Volume: 55, Issue:4

    Topics: Adenosine Triphosphate; Animals; Colchicine; Cyclic AMP; Cytoplasm; Dihydroalprenolol; Drug Tolerance; Isoproterenol; Male; Monensin; Myocardium; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1984
Some unique properties of CGP-12177.
    Journal of receptor research, 1984, Volume: 4, Issue:1-6

    Topics: Adenylyl Cyclases; Animals; Cell Line; Cyclic AMP; Digitonin; Dihydroalprenolol; Glioma; Isoproterenol; Propanolamines; Rats; Receptors, Adrenergic, beta; Stereoisomerism

1984
Changes in beta-adrenoceptor binding properties and receptor-cyclase coupling during in vitro maturation of rat reticulocytes.
    Journal of receptor research, 1984, Volume: 4, Issue:1-6

    Topics: Adenosine Triphosphate; Adenylyl Cyclases; Animals; Cells, Cultured; Cyclic AMP; Dihydroalprenolol; Isoproterenol; Propanolamines; Rats; Receptors, Adrenergic, beta; Reticulocytes

1984
Properties of beta-adrenoceptor sites in metabolizing and nonmetabolizing rat reticulocytes and in resealed reticulocyte ghosts.
    Naunyn-Schmiedeberg's archives of pharmacology, 1981, Volume: 317, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Cell Membrane; Cold Temperature; Cytosol; Dihydroalprenolol; Energy Metabolism; Female; Isoproterenol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Reticulocytes; Timolol

1981
Determination of the desensitization of beta-adrenergic receptors by [3H]CGP-12177.
    The Biochemical journal, 1983, Dec-15, Volume: 216, Issue:3

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Binding Sites; Binding, Competitive; Cell Line; Cell Membrane; Centrifugation, Density Gradient; Dihydroalprenolol; Glioma; Humans; Isoproterenol; Propanolamines; Receptors, Adrenergic, beta

1983
The human carcinoma cell line A431 possesses large numbers of functional beta-adrenergic receptors.
    FEBS letters, 1984, Apr-24, Volume: 169, Issue:2

    Topics: Adrenergic beta-Antagonists; Binding, Competitive; Carcinoma, Squamous Cell; Cell Line; Dihydroalprenolol; Humans; Isoproterenol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism

1984
Simple and reliable radioreceptor assay for beta-adrenoceptor antagonists and active metabolites in native human plasma.
    European journal of clinical pharmacology, 1984, Volume: 27, Issue:5

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Carteolol; Dihydroalprenolol; Erythrocyte Membrane; Female; Humans; Male; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Time Factors

1984
Antagonist-dependent and -independent steps in the mechanism of adrenergic receptor internalization.
    The Journal of biological chemistry, 1994, Jul-15, Volume: 269, Issue:28

    Topics: Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Antibodies, Monoclonal; Azides; Cell Line, Transformed; Cell Membrane; Cold Temperature; Dihydroalprenolol; Endocytosis; Epitopes; Humans; Microscopy, Immunoelectron; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-2; Recombinant Proteins; Sodium Azide; Tritium

1994
Evidence of classic beta 3-adrenergic receptors in porcine adipocytes.
    Journal of animal science, 1996, Volume: 74, Issue:5

    Topics: Adipocytes; Adrenergic beta-Antagonists; Animals; Binding Sites; Binding, Competitive; Cell Membrane; Dihydroalprenolol; Iodocyanopindolol; Magnesium Chloride; Male; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; RNA; Swine; Tritium

1996
Tannin inhibits the cAMP-beta-adrenergic receptor pathway in bovine tracheal epithelium.
    The American journal of physiology, 1998, Volume: 274, Issue:2

    Topics: Acetylcysteine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cattle; Chloride Channels; Cyclic AMP; Dihydroalprenolol; Epithelium; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Hydrolyzable Tannins; Propanolamines; Receptors, Adrenergic, beta; Trachea

1998
Rapid electrical stimulation of contraction reduces the density of beta-adrenergic receptors and responsiveness of cultured neonatal rat cardiomyocytes. Possible involvement of microtubule disassembly secondary to mechanical stress.
    Circulation, 2000, Jun-06, Volume: 101, Issue:22

    Topics: Acetylcholine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Antineoplastic Agents, Phytogenic; Cells, Cultured; Colforsin; Diacetyl; Dihydroalprenolol; Down-Regulation; Electric Stimulation; Enzyme Inhibitors; Heart Failure; Isoproterenol; Microtubules; Muscle Fibers, Skeletal; Myocardial Contraction; Myocardium; Pacemaker, Artificial; Paclitaxel; Propanolamines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Stress, Mechanical; Tritium; Vasodilator Agents

2000
Ligand regulation of green fluorescent protein-tagged forms of the human beta(1)- and beta(2)-adrenoceptors; comparisons with the unmodified receptors.
    British journal of pharmacology, 2000, Volume: 130, Issue:8

    Topics: Betaxolol; Binding, Competitive; Cell Line; Dihydroalprenolol; Endocytosis; Green Fluorescent Proteins; Humans; Isoproterenol; Kinetics; Ligands; Luminescent Proteins; Microscopy, Confocal; Oligopeptides; Peptides; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Fusion Proteins; Tritium

2000
Comparison of three radioligands for the labelling of human beta-adrenoceptor subtypes.
    Naunyn-Schmiedeberg's archives of pharmacology, 2006, Volume: 374, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Dihydroalprenolol; Ethanolamines; Humans; Iodine Radioisotopes; Iodocyanopindolol; Isotope Labeling; Kinetics; Propanolamines; Protein Binding; Radioligand Assay; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Tetrahydronaphthalenes; Tritium

2006