dihydroalprenolol and alprenolol
dihydroalprenolol has been researched along with alprenolol in 139 studies
Research
Studies (139)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 132 (94.96) | 18.7374 |
1990's | 7 (5.04) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors
Authors | Studies |
---|---|
Bultsma, T; Donné-Op den Kelder, GM; Rademaker, B; Timmerman, H | 1 |
Bottari, S; Strosberg, AD; Vauquelin, G | 1 |
Cabelli, RJ; Malbon, CC | 1 |
Barnett, DB; Howlett, DR; Nahorski, SR; Rugg, EL | 1 |
Limas, CJ | 1 |
Bhalla, R; Winek, R | 2 |
Cannon, B; Houstĕk, J; Snochowski, M; Svartengren, J; Svoboda, P | 1 |
Nahorski, SR; Richardson, A | 2 |
Adham, N; Blue, DR; Bond, RA; Clarke, DE; Delmendo, R; Eglen, RM; Michel, AD; Whiting, RL | 1 |
Coury, A; Guyard, A; Rumigny, JF | 1 |
Cheng, KW; Ghahary, A | 1 |
Ernsberger, P; Iacovitti, L; Reis, DJ | 1 |
Alexander, E; Friedman, AH | 1 |
Galbani, P; Pompeiano, M; Ronca-Testoni, S | 1 |
Creese, I; Riva, MA | 1 |
Kellar, KJ; Stockmeier, CA | 1 |
Cheetham, SC; Crompton, MR; De Paermentier, F; Horton, RW | 1 |
Gillespie, DD; Manier, DH; Sulser, F | 1 |
Dermon, CR; Kouvelas, ED | 2 |
Nagatomo, T; Tsuchihashi, H | 5 |
Coscia, E; Daw, NW; Parkinson, D | 1 |
Klimek, V; Mogilnicka, E; Nowak, G; Wedzony, K | 1 |
Kusiak, JW; Liptak, A; Pitha, J | 1 |
Hayashi, T; Kunihara, M; Tadokoro, S | 1 |
Baker, SP; Muther, TF; Nelson, CA; Pitha, J | 1 |
Klempner, MS; Styrt, B | 1 |
Amenta, F; Cavallotti, C; De Rossi, M | 1 |
Agid, Y; Cash, R; Lasbennes, F; Sercombe, R; Seylaz, J | 1 |
Lang, PH; Lemmer, B | 2 |
Homcy, CJ; Sawutz, DG; Sylvestre, D | 1 |
Nagatomo, T; Sasaki, M; Tsuchihashi, H | 1 |
Buja, LM; Calianos, TA; Muntz, KH; Vandermolen, DT; Willerson, JT | 1 |
Biegon, A | 1 |
Aakesson, I; Jacobsen, S; Sager, G; Sandnes, D | 1 |
Kunovská, V; Prásek, J; Prikryl, P; Rysánek, K; Vondrácek, V | 1 |
McGonigle, P; Molinoff, PB; Neve, KA | 1 |
Borda, E; Perez Leiros, C | 1 |
Arinze, IJ; Graham, SM; Kawai, Y; Yoshioka, H | 1 |
Aalbers, C; Carstens, ME; Chalton, DO; Engelbrecht, AH; Gagiano, CA; Russell, VA; Taljaard, JJ | 1 |
Alam, BS; Alam, SQ; Ren, YF | 2 |
Marttila, T; Niina, O; Nikinmaa, M | 1 |
Chamat, S; Engelborghs, Y; Hoebeke, J; Strosberg, AD | 1 |
Bunn, SJ; Hanley, MR; Wilkin, GP | 1 |
Brière, R; Diop, L; Grondin, L; Reader, TA | 1 |
Bigl, V; Schliebs, R | 2 |
Bogdany, A; Borsodi, A; Grigorian, G; Halasz, N; Toth, G | 1 |
Leysen, JE; Peeters, G; Roets, E | 1 |
Agli, B; Giudicelli, Y; Lacasa, D | 1 |
Gurevich, VV; Voeĭkov, VL | 1 |
Il'inskiĭ, OB; Krasnikova, TL; Parfenova, EV; Radiukhin, VA; Shkhvatsabaia, IK | 1 |
Eckelman, WC; Francis, B; Gibson, RE; Reba, RC; Rzeszotarski, WJ; Vieras, F | 1 |
Caron, MG; Lefkowitz, RJ; Srinivasan, Y | 1 |
Mauger, JP; Worcel, M | 1 |
Sulakhe, PV; Wei, JW | 1 |
Caron, MG; Lefkowitz, RJ; Nasrin, N; Pitha, J; Zjawiony, J | 1 |
Cheng, JB; Cornett, LE; Goldfien, A; Roberts, JM | 1 |
Burnam, MH; Rose, DM; Sethna, DH; Shell, WE; Stern, CS | 1 |
Stone, EA; U'Prichard, DC | 1 |
Goldfien, A; Hayashida, DN; Leung, R; Roberts, JM | 1 |
Baker, SP; Dax, EM; Hughes, BA; Kusiak, JW; Pitha, J | 1 |
Pong, SF; Tinkham, CL | 1 |
Fujimura, H; Imai, H; Niwa, M; Nozaki, M; Tsurumi, K | 1 |
Chang, RS; Lotti, VJ | 1 |
Bhanot, R; Eskes, G; Moger, WH; Wilkinson, DA; Wilkinson, M | 1 |
Baker, SP; Posner, P | 1 |
Kusiak, JW; Pitha, J | 2 |
Erdö, SL; Laszlovszky, I | 1 |
Matsumoto, G | 1 |
Gross, DM; Schmitt, CJ; Share, NN | 1 |
Crankshaw, DJ; Ruzycky, AL | 1 |
Meier, KE; Ruoho, AE | 2 |
Nakazawa, T; Nomura, S; Sakaida, S; Ukei, N | 1 |
Christoffersen, T; Jacobsen, S; Refsnes, M; Sager, G; Sand, TE; Sandnes, D; Westergren, T | 1 |
Bani-Sacchi, T; Blandina, P; Fantozzi, R; Galli, A; Giotti, A; Mannaioni, PF; Masini, E; Zilletti, L | 1 |
Baum, BJ; Hand, AR; Kousvelari, EE; Kusiak, JW; Pitha, J | 1 |
Crutcher, KA; Davis, JN | 1 |
Baker, SP; Potter, LT | 2 |
Baer, M; Porzig, H | 1 |
De Lean, A; Lefkowitz, RJ; Stadel, JM | 1 |
Boriskina, GM; Postnov, IuV | 1 |
Johnston, CI; Woodcock, EA | 1 |
Ben-David, E; Eliahou, H; Gavendo, S; Iaina, A; Kapuler, S; Serban, I | 1 |
Davies, JN; Wagner, HR | 1 |
Borsodi, A; Thang, NX; Wollemann, M | 1 |
Davies, AO; De Lean, A; Lefkowitz, RJ | 1 |
Chuang, DM; Costa, E; Kinnier, WJ | 1 |
Jordan, AW | 1 |
Sha'afi, RI; Wacholtz, MC | 1 |
Ray, PD; Rufo, GA; Yorek, MA | 1 |
Higuchi, H; Lai, RT; Maeda, H; Watanabe, Y; Yoshida, H | 1 |
Rexroad, CE | 1 |
Culvenor, AJ; Jarrott, B | 1 |
De Lean, A; Hoffman, BB; Kent, R; Lefkowitz, RJ; Limbird, L; Michel, T; Stadel, JM | 1 |
Davis, JN; Giron, LT | 1 |
Tkachuk, VA; Wollemann, M | 1 |
Moustafa, E; Wong, M | 1 |
Sager, G | 2 |
Boriskina, GM | 1 |
Altiere, RJ; Douglas, JS; Gillis, CN | 1 |
Maderspach, K; Nemecz, G; Yigiter, M | 1 |
Dax, EM; Gregerman, RI; Partilla, JS | 1 |
Roeske, WR; Yamada, S; Yamamura, HI | 1 |
Bruynzeel, PL; Kauffman, HF; Meurs, H; van den Bogaard, W | 1 |
Falkay, G; Kovacs, L | 1 |
Kerry, R; Scrutton, MC | 1 |
Noack, E; Schuhmacher, P | 1 |
Imai, S; Nagatomo, T; Sasaki, M; Tsuchihashi, H | 1 |
Bergdolt, E; Keul, J; Lehmann, M; Porzig, H; Schmid, P | 1 |
Haraguchi, K; Hashizume, K; Ichikawa, K; Kobayashi, M; Yamauchi, K | 1 |
Erickson, RP; Markovac, J | 1 |
Altszuler, N; Cherksey, B | 1 |
Drahota, Z; Skobisová, E; Svoboda, P | 1 |
Bruynzeel, PL; de Jong, JG; Hamelink, ML; Kok, PT | 1 |
Kawai, M; Nomura, Y; Sakaue, T; Segawa, T; Watanabe, C | 1 |
Bruinink, A; Lichtensteiger, W | 1 |
Kawai, M; Motomori-Suzaki, E; Nomura, Y; Segawa, T; Yotsumoto, I | 1 |
Heikkila, RE | 1 |
Imai, M; Kusano, E; Nakamura, R | 1 |
Chamat, S; Hoebeke, J; Strosberg, AD | 1 |
Cavanagh, HD; Colley, AM | 1 |
Dulis, BH; Wilson, IB | 1 |
Hendley, ED; Myers, MM; Whittemore, SR | 1 |
Arbilla, S; Depoortere, H; Langer, SZ; Mogilnicka, E | 1 |
Morimoto, C; Okuda, H; Tsujita, T | 1 |
Ogawa, N | 1 |
Reviews
1 review(s) available for dihydroalprenolol and alprenolol
Article | Year |
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[Analysis and characterization of ligand-receptor binding systems].
Topics: Alprenolol; Animals; Atropine; Binding, Competitive; Carbachol; Dihydroalprenolol; Humans; Ligands; Metoprolol; Receptors, Cell Surface; Receptors, Neurotransmitter | 1997 |
Other Studies
138 other study(ies) available for dihydroalprenolol and alprenolol
Article | Year |
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Mapping of the beta 2-adrenoceptor on Chang liver cells. Differences between high- and low-affinity receptor states.
Topics: Cell Membrane; Cells, Cultured; Guanylyl Imidodiphosphate; Hydrogen Bonding; Iodocyanopindolol; Liver; Models, Molecular; Pindolol; Protein Conformation; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Dopamine D2; Stereoisomerism; Structure-Activity Relationship | 1988 |
Agonist- induced transconformation of beta-adrenergic receptors, and adenylate cyclase activation [proceedings].
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; Enzyme Activation; Erythrocytes; Ethylmaleimide; Kinetics; Receptors, Adrenergic; Receptors, Adrenergic, beta; Turkeys | 1979 |
Characterization of (-)-[3H]dihdroalprenolol binding sites on isolated rat fat cells.
Topics: Adipose Tissue; Alprenolol; Animals; Binding, Competitive; Cyclic AMP; Dihydroalprenolol; Female; Isoproterenol; Kinetics; Phentolamine; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1979 |
Pharmacological characteristics of beta-adrenoceptor binding sites in intact and sympathectomized rat spleen.
Topics: Alprenolol; Animals; Binding Sites; Dihydroalprenolol; Hydroxydopamines; Male; Membranes; Norepinephrine; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Spleen; Sympathetic Nervous System | 1979 |
Increased number of beta-adrenergic receptors in the hypertrophied myocardium.
Topics: Alprenolol; Animals; Binding, Competitive; Cardiomegaly; Dihydroalprenolol; Isoproterenol; Male; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1979 |
[3H]Dihydroalprenolol binding sites in rat myocardium: relationship between a single binding site population and the concentration of radioligand.
Topics: Alprenolol; Animals; Cell Membrane; Dihydroalprenolol; Isotope Labeling; Kinetics; Male; Myocardium; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Tritium | 1979 |
High number of high-affinity binding sites for (-)-[3H]dihydroalprenolol on isolated hamster brown-fat cells. A study of the beta-adrenergic receptors.
Topics: Adipose Tissue, Brown; Alprenolol; Animals; Cricetinae; Dihydroalprenolol; Kinetics; Mesocricetus; Oxygen Consumption; Receptors, Adrenergic; Receptors, Adrenergic, beta; Sympatholytics; Sympathomimetics | 1979 |
Pitfalls in the assessment of the specific binding of(-)[3H]-dihydroalprenolol to beta-adrenoceptors [proceedings].
Topics: Alprenolol; Animals; Cattle; Dihydroalprenolol; In Vitro Techniques; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1979 |
Antagonist characterization of atypical beta adrenoceptors in guinea pig ileum: blockade by alprenolol and dihydroalprenolol.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Dihydroalprenolol; Drug Interactions; Guinea Pigs; Ileum; In Vitro Techniques; Isoproterenol; Male; Muscle, Smooth; Propranolol; Receptors, Adrenergic, beta | 1990 |
Characterization of beta-adrenoceptors in synaptoneurosomes from rat brain: [3H]dihydroalprenolol versus [3H]CGP 12177.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Brain Chemistry; Dihydroalprenolol; Propanolamines; Radioligand Assay; Rats; Receptors, Adrenergic, beta; Synaptosomes; Tritium | 1990 |
Identification and characterization of the beta-adrenergic receptor on neuroblastoma x glioma hybrid NG108-15 cells.
Topics: Alprenolol; Bucladesine; Catecholamines; Cell Differentiation; Dihydroalprenolol; Glioma; Hybrid Cells; Isoproterenol; Kinetics; Neuroblastoma; Receptors, Adrenergic, beta; Stereoisomerism; Tumor Cells, Cultured | 1990 |
Astrocytes cultured from specific brain regions differ in their expression of adrenergic binding sites.
Topics: Alprenolol; Animals; Astrocytes; Brain; Cells, Cultured; Clonidine; Dihydroalprenolol; Glial Fibrillary Acidic Protein; Rats; Receptors, Adrenergic | 1990 |
The identification of adrenergic receptors in human pial membranes.
Topics: Alprenolol; Cerebral Veins; Dihydroalprenolol; Humans; Pia Mater; Prazosin; Receptors, Adrenergic; Yohimbine | 1990 |
Distribution of beta-adrenergic receptors in different cortical and nuclear regions of cat cerebellum, as revealed by binding studies.
Topics: Alprenolol; Animals; Binding, Competitive; Cats; Cerebellar Nuclei; Cerebral Cortex; Dihydroalprenolol; Metoprolol; Receptors, Adrenergic, beta | 1989 |
Comparison of two putatively selective radioligands for labeling central nervous system beta-adrenergic receptors: inadequacy of [3H]dihydroalprenolol.
Topics: Alprenolol; Animals; Brain Chemistry; Dihydroalprenolol; Guanosine Triphosphate; Isoproterenol; Kinetics; Male; Propanolamines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin | 1989 |
Serotonin depletion unmasks serotonergic component of [3H]dihydroalprenolol binding in rat brain.
Topics: 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Alprenolol; Animals; Brain; Dihydroalprenolol; Fenclonine; In Vitro Techniques; Iodocyanopindolol; Male; p-Chloroamphetamine; Pindolol; Piperazines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes | 1989 |
Beta-adrenoceptors in human brain labelled with [3H]dihydroalprenolol and [3H]CGP 12177.
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Brain Chemistry; Dihydroalprenolol; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Practolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 1989 |
Characterization of the inducible serotonin-sensitive dihydroalprenolol binding sites with low affinity for isoproterenol.
Topics: 5,7-Dihydroxytryptamine; Alprenolol; Animals; Binding, Competitive; Brain; Cerebral Ventricles; Dihydroalprenolol; Dihydroxytryptamines; Injections, Intraventricular; Isoproterenol; Kinetics; Male; Rats; Rats, Inbred Strains; Reference Values; Regression Analysis; Serotonin | 1989 |
Quantitative analysis of the localization of adrenergic binding sites in chick brain.
Topics: Alprenolol; Animals; Autoradiography; Brain; Chickens; Clonidine; Dihydroalprenolol; Dioxanes; Dioxins; Receptors, Adrenergic | 1989 |
Characterization of 3H-dihydroalprenolol binding to beta-adrenergic receptors of rat brain: two binding sites of racemic propranolol in displacement experiments.
Topics: Alprenolol; Animals; Binding, Competitive; Brain; Dihydroalprenolol; Propranolol; Rats; Receptors, Adrenergic, beta | 1987 |
Effects of choline and inositol on 3H-dihydroalprenolol and 125I-iodocyanopindolol bindings to beta-adrenergic receptors of the guinea pig cerebral cortical membranes.
Topics: Alprenolol; Animals; Cerebral Cortex; Choline; Dihydroalprenolol; Guinea Pigs; In Vitro Techniques; Inositol; Iodocyanopindolol; Male; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1988 |
Identification and localization of adrenergic receptors in cat visual cortex.
Topics: Alprenolol; Animals; Cats; Dihydroalprenolol; Female; Male; Prazosin; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Visual Cortex; Yohimbine | 1988 |
The importance of timing for the action of alpha 1- or beta-agonists: possible relationship with the density of [3H]prazosin and [3H]dihydroalprenolol binding sites.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Alprenolol; Animals; Binding Sites; Dihydroalprenolol; Exploratory Behavior; In Vitro Techniques; Male; Prazosin; Rats; Rats, Inbred Strains; Time Factors; Tritium | 1985 |
Alkylating beta-blockers: activity of isomeric bromoacetyl alprenolol menthanes.
Topics: Adrenergic beta-Antagonists; Affinity Labels; Alprenolol; Animals; Cell Membrane; Dihydroalprenolol; Isomerism; Lung; Magnetic Resonance Spectroscopy; Molecular Conformation; Myocardium; Rats; Receptors, Adrenergic, beta; Structure-Activity Relationship | 1985 |
Changes in 3H-spiperone, 3H-WB 4101 and 3H-dihydroalprenolol bindings to brain membranes produced by postnatal pretreatment with chlorpromazine in adult rats.
Topics: Adrenergic alpha-Antagonists; Alprenolol; Animals; Animals, Newborn; Brain; Butyrophenones; Chlorpromazine; Dihydroalprenolol; Dioxanes; Dioxins; Female; Kinetics; Male; Membranes; Rats; Rats, Inbred Strains; Spiperone | 1985 |
Differential recovery of beta adrenoreceptor antagonist and agonist high affinity binding sites in the guinea-pig lung after irreversible blockade.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Binding Sites; Dihydroalprenolol; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Lung; Receptors, Adrenergic, beta; Tritium | 1986 |
Lysosomotropic behavior of adrenergic antagonists in interactions with human neutrophils.
Topics: Adrenergic beta-Agonists; Affinity Labels; Alprenolol; Azides; Cell Membrane; Dihydroalprenolol; Humans; Kinetics; Lysosomes; Neutrophils; Propanolamines | 1988 |
Histoautoradiographic localization of (-)-3H-dihydroalprenolol in rabbit aorta.
Topics: Alprenolol; Animals; Aorta; Autoradiography; Dihydroalprenolol; Female; In Vitro Techniques; Male; Rabbits; Receptors, Adrenergic, beta; Tritium | 1985 |
Influence of polymeric effectors on binding of 3H-dihydroalprenolol to beta-adrenergic receptor of rat brain.
Topics: Alprenolol; Animals; Brain; Cell Membrane; Dihydroalprenolol; DNA; Gelatin; Heparin; Histones; In Vitro Techniques; Male; Membrane Potentials; Polymers; Polymyxin B; Polysaccharides; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Serum Albumin, Bovine; Surface Properties | 1985 |
Adrenergic receptors on cerebral microvessels in control and parkinsonian subjects.
Topics: Aged; Alprenolol; Capillaries; Cerebrovascular Circulation; Clonidine; Dihydroalprenolol; Humans; Kinetics; Parkinson Disease; Prazosin; Quinazolines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Reference Values | 1985 |
Evidence for two specific affinity states of 3H-antagonist binding to cardiac beta-adrenergic receptors and influence of Gpp(NH)p.
Topics: Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Male; Myocardium; Propanolamines; Rats; Receptors, Adrenergic, beta | 1985 |
Characterization of monoclonal antibodies to the beta-adrenergic antagonist alprenolol as models of the receptor binding site.
Topics: Alprenolol; Animals; Antibodies, Monoclonal; Ascitic Fluid; Binding Sites, Antibody; Binding, Competitive; Dihydroalprenolol; Hybridomas; Iodocyanopindolol; Mice; Models, Biological; Pindolol; Receptors, Adrenergic, beta | 1985 |
Binding characteristics of 3H-dihydroalprenolol to beta-adrenergic receptors of rat brain: influence of lectins.
Topics: Alprenolol; Animals; Brain; Carbohydrate Metabolism; Dihydroalprenolol; In Vitro Techniques; Lectins; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Tritium | 1985 |
Binding characteristics of 3H-dihydroalprenolol to beta-adrenergic receptors of rat brain: influence of exo- and endo-glycosidases and glycopeptidase.
Topics: Alprenolol; Amidohydrolases; Animals; Brain; Carbohydrate Metabolism; Dihydroalprenolol; Glycoside Hydrolases; In Vitro Techniques; Kinetics; Peptide-N4-(N-acetyl-beta-glucosaminyl) Asparagine Amidase; Rats; Receptors, Adrenergic, beta | 1985 |
Binding characteristics of [3H]dihydroalprenolol to beta-adrenergic receptors of rat brain: comparison with those of rat heart treated with neuraminidase.
Topics: Alprenolol; Animals; Brain; Dihydroalprenolol; In Vitro Techniques; Male; Myocardium; Neuraminidase; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1985 |
Differences in affinity of cardiac beta-adrenergic receptors for [3H]dihydroalprenolol.
Topics: Alprenolol; Animals; Arterioles; Autoradiography; Coronary Circulation; Coronary Vessels; Dihydroalprenolol; Dogs; Muscle, Smooth; Myocardium; Nervous System; Receptors, Adrenergic, beta; Tissue Distribution; Tritium | 1986 |
Effect of chronic desipramine treatment on dihydroalprenolol, imipramine, and desipramine binding sites: a quantitative autoradiographic study in the rat brain.
Topics: Alprenolol; Animals; Autoradiography; Binding Sites; Brain; Desipramine; Dihydroalprenolol; Imipramine; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Time Factors; Tissue Distribution | 1986 |
Effect of serum, alpha-1 acid glycoprotein, lipoproteins and albumin on human mononuclear leucocyte beta-adrenoceptors.
Topics: Alprenolol; Blood; Blood Proteins; Cyclic AMP; Dihydroalprenolol; Humans; Isoproterenol; Leukocytes; Lipoproteins; Orosomucoid; Propranolol; Receptors, Adrenergic, beta; Serum Albumin; Theophylline | 1986 |
[Interindividual changes in the specific binding of 3H-dihydroalprenolol by beta 2-adrenergic lymphocytic receptors in essential hypertension].
Topics: Adult; Alprenolol; Dihydroalprenolol; Humans; Hypertension; Isoproterenol; Lymphocytes; Male; Receptors, Adrenergic, beta | 1986 |
Quantitative analysis of the selectivity of radioligands for subtypes of beta adrenergic receptors.
Topics: Alprenolol; Animals; Cell Line; Dihydroalprenolol; Dose-Response Relationship, Drug; Glioma; Heart Atria; Humans; Iodocyanopindolol; Kinetics; Mathematics; Pindolol; Receptors, Adrenergic, beta; Software | 1986 |
Characterization of (-)-(3H)-DHA binding to intact mouse lymphocytes: effect of experimental autoimmune orchitis on beta-adrenoceptor expression.
Topics: Alprenolol; Animals; Autoimmune Diseases; Binding, Competitive; Dihydroalprenolol; Kinetics; Lymphocytes; Male; Mice; Orchitis; Propranolol; Receptors, Adrenergic, beta; Testis | 1986 |
Beta-adrenergic receptors in guinea-pig liver plasma membranes and thermal lability of [3H]dihydroalprenolol binding sites.
Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Alprenolol; Animals; Binding, Competitive; Cell Membrane; Cholera Toxin; Dihydroalprenolol; Guanylyl Imidodiphosphate; Guinea Pigs; Hot Temperature; Iodocyanopindolol; Isoproterenol; Liver; Male; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Virulence Factors, Bordetella | 1986 |
Beta-adrenoceptors on lymphocytes of patients with major depressive disorder.
Topics: Adult; Alprenolol; Cell Membrane; Depressive Disorder; Dexamethasone; Dihydroalprenolol; Female; Humans; Lymphocytes; Male; Middle Aged; Receptors, Adrenergic, beta; Tritium | 1987 |
Effect of cholesterol feeding on membrane fluidity, (Na+ + K+)ATPase, adenylate cyclase, [3H]-ouabain-, and [3H]-dihydroalprenolol-binding in rat submandibular salivary glands.
Topics: Adenylyl Cyclases; Alprenolol; Animals; Cell Membrane; Cholesterol, Dietary; Dihydroalprenolol; Kinetics; Male; Membrane Fluidity; Ouabain; Rats; Rats, Inbred Strains; Sodium-Potassium-Exchanging ATPase; Submandibular Gland | 1987 |
Binding properties, regional ontogeny and localization of adrenergic receptors in chick brain.
Topics: Alprenolol; Animals; Binding, Competitive; Brain; Chick Embryo; Chickens; Clonidine; Dihydroalprenolol; Dioxanes; Dioxins; Kinetics; Receptors, Adrenergic | 1988 |
[3H]forskolin- and [3H]dihydroalprenolol-binding sites and adenylate cyclase activity in heart of rats fed diets containing different oils.
Topics: Adenylyl Cyclases; Alprenolol; Animals; Binding Sites; Cell Membrane; Coconut Oil; Colforsin; Corn Oil; Dietary Fats; Dihydroalprenolol; Fish Oils; Male; Membrane Lipids; Myocardium; Phospholipids; Plant Oils; Rats; Rats, Inbred Strains; Tritium | 1988 |
Binding of beta-adrenergic antagonists 3H-DHA and 3H-CGP 12177 to intact rainbow trout (Salmo gairdneri) and carp (Cyprinus carpio) red blood cells.
Topics: Alprenolol; Animals; Carps; Cyprinidae; Dihydroalprenolol; Erythrocytes; Ligands; Membrane Lipids; Propanolamines; Salmonidae; Trout | 1988 |
The immune response towards beta-adrenergic ligands and their receptors--VII. Equilibrium and kinetic binding studies of l-alprenolol to a monoclonal anti-alprenolol antibody.
Topics: Alprenolol; Animals; Antibodies, Monoclonal; Antigen-Antibody Complex; Antigen-Antibody Reactions; Chemical Phenomena; Chemistry, Physical; Dihydroalprenolol; Haptens; Immunoglobulin G; Kinetics; Mice; Mice, Inbred BALB C; Radioimmunoassay; Thermodynamics | 1987 |
Autoradiographic localization of peripheral benzodiazepine, dihydroalprenolol and arginine vasopressin binding sites in the pituitaries of control, stalk transected and Brattleboro rats.
Topics: Alprenolol; Animals; Arginine Vasopressin; Autoradiography; Benzodiazepines; Benzodiazepinones; Binding Sites; Dihydroalprenolol; gamma-Aminobutyric Acid; Glial Fibrillary Acidic Protein; Intermediate Filament Proteins; Male; Pituitary Gland; Rats; Rats, Brattleboro; Rats, Inbred Strains; Spiperone | 1986 |
Adrenergic receptor and catecholamine distribution in rat cerebral cortex: binding studies with [3H]prazosin, [3H]idazoxan and [3H]dihydroalprenolol.
Topics: Alprenolol; Animals; Catecholamines; Cerebral Cortex; Chromatography, High Pressure Liquid; Dihydroalprenolol; Dioxanes; Dioxins; Electrochemistry; Idazoxan; Male; Prazosin; Rats; Receptors, Adrenergic; Tissue Distribution; Tritium | 1987 |
Kinetics of the interaction of dihydroalprenolol with beta-adrenergic receptors in rat cerebral cortex.
Topics: Alprenolol; Animals; Cerebral Cortex; Dihydroalprenolol; Drug Interactions; Female; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Temperature; Thermodynamics | 1984 |
Purification and characterization of beta-adrenoreceptor rich heart plasma membrane.
Topics: 5'-Nucleotidase; Adenylyl Cyclases; Alprenolol; Animals; Cell Membrane; Dihydroalprenolol; In Vitro Techniques; Muscle Proteins; Myocardium; Nucleotidases; Rabbits; Receptors, Adrenergic, beta; Sarcolemma; Sodium-Potassium-Exchanging ATPase | 1983 |
A simple non-parametric procedure for rapid estimation of Scatchard parameters.
Topics: Alprenolol; Animals; Cerebral Cortex; Dihydroalprenolol; Kinetics; Mathematics; Methods; Models, Biological; Rats; Receptors, Adrenergic, beta | 1984 |
Identification of beta-adrenoceptors in bovine teat muscles by 3H-dihydroalprenolol binding.
Topics: Alprenolol; Animals; Cattle; Dihydroalprenolol; Female; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Mammary Glands, Animal; Muscle, Smooth; Radioligand Assay; Receptors, Adrenergic, beta; Tritium; Tromethamine | 1984 |
"Spare" beta-adrenergic receptors of rat white adipocyte membranes.
Topics: Adenylyl Cyclases; Adipose Tissue; Alprenolol; Animals; Cell Membrane; Cyclic AMP; Dihydroalprenolol; Guanine Nucleotides; Guanylyl Imidodiphosphate; In Vitro Techniques; Isoproterenol; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1984 |
[Separation of [3H]dihydroalprenolol, free or bound to solubilized beta-adrenergic receptors, on a cation-exchange resin].
Topics: Alprenolol; Animals; Cattle; Cerebellum; Chromatography, Ion Exchange; Dihydroalprenolol; In Vitro Techniques; Kinetics; Radioligand Assay; Rats; Receptors, Adrenergic, beta; Reticulocytes | 1983 |
[Changes in the density of human lymphocyte beta-adrenergic receptors in hypertension].
Topics: Adult; Alprenolol; Dihydroalprenolol; Humans; Hypertension; Lymphocytes; Male; Phentolamine; Radioligand Assay; Receptors, Adrenergic, beta | 1984 |
Circadian-phase-dependency in [3H]-dihydroalprenolol binding to rat heart ventricular membranes.
Topics: Alprenolol; Animals; Circadian Rhythm; Dihydroalprenolol; Guanine Nucleotides; Heart Ventricles; Isoproterenol; Male; Myocardium; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Reserpine; Sarcolemma | 1984 |
In vivo receptor binding of iodinated beta-adrenoceptor blockers.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Carbazoles; Dihydroalprenolol; Guinea Pigs; Iodine Radioisotopes; Levobunolol; Lung; Male; Myocardium; Practolol; Proadifen; Propanolamines; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Affinity chromatography of the beta-adrenergic receptor and characterization of antibodies raised against purified receptor preparations.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Antibodies; Anura; Binding, Competitive; Chromatography, Affinity; Dihydroalprenolol; Erythrocyte Membrane; Receptors, Adrenergic; Receptors, Adrenergic, beta; Stereoisomerism | 1980 |
Relationship between the (--)-[3H]-dihydroalprenolol binding to beta-adrenoceptors and transmembrane 86Rb efflux of the BC3H1 nonfusing muscle cell line.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Cell Line; Cell Membrane; Dihydroalprenolol; Membranes; Muscles; Radioisotopes; Receptors, Adrenergic; Receptors, Adrenergic, beta; Rubidium | 1980 |
Identity of [3H]dihydroalprenolol binding sites and beta-2 adrenergic receptors coupled with adenylate cyclase in guinea-pig skeletal muscle sarcolemma: general properties and structure-activity relationships.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Binding Sites; Catecholamines; Dihydroalprenolol; Dose-Response Relationship, Drug; Guanosine Monophosphate; Guinea Pigs; Kinetics; Receptors, Adrenergic; Receptors, Adrenergic, beta; Sarcolemma; Species Specificity; Stereoisomerism; Structure-Activity Relationship; Temperature; Time Factors; Tritium | 1980 |
Potent beta-adrenergic antagonist possessing chemically reactive group.
Topics: Adrenergic beta-Agonists; Alprenolol; Animals; Binding, Competitive; Cyclohexane Monoterpenes; Dihydroalprenolol; Erythrocyte Membrane; Kinetics; Ranidae; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Identification of beta-adrenergic receptors using [3H]dihydroalprenolol in fetal sheep heart: direct evidence of qualitative similarity to the receptors in adult sheep heart.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Aging; Alprenolol; Animals; Dihydroalprenolol; Female; Fetal Heart; In Vitro Techniques; Myocardial Contraction; Pregnancy; Receptors, Adrenergic; Receptors, Adrenergic, beta; Sheep | 1981 |
Differences in beta-adrenoceptor binding in anterior and inferior myocardial wall microsomes of normal canine left ventricle.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Binding Sites; Dihydroalprenolol; Dogs; Heart Ventricles; Kinetics; Male; Microsomes; Myocardium; Receptors, Adrenergic; Receptors, Adrenergic, beta; Stereoisomerism | 1981 |
[3H]dihydroalprenolol binding in the rat brainstem.
Topics: Adrenergic beta-Agonists; Alprenolol; Animals; Brain Stem; Dihydroalprenolol; In Vitro Techniques; Kinetics; Male; Membranes; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Human myometrial adrenergic receptors: identification of the beta-adrenergic receptor by [3H]dihydroalprenolol binding.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Dihydroalprenolol; Ethanolamines; Female; Humans; Myometrium; Postural Balance; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta; Uterus | 1982 |
Regeneration of beta-adrenergic receptors in senescent rats: a study using an irreversible binding antagonist.
Topics: Adrenergic beta-Antagonists; Aging; Alprenolol; Animals; Brain; Cyclohexane Monoterpenes; Dihydroalprenolol; Kinetics; Lung; Myocardium; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1982 |
Displacement of [3H]dihydroalprenolol binding from rat heart and lung by acebutolol, diacetolol and D-diacetolol.
Topics: Acebutolol; Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; In Vitro Techniques; Isomerism; Lung; Myocardium; Rats; Rats, Inbred Strains; Tritium | 1983 |
[Influence of indomethacin and clidanac on the blood pressure lowering effect of beta-blockers].
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Blood Pressure; Dihydroalprenolol; Drug Interactions; Guinea Pigs; Heart Rate; In Vitro Techniques; Indans; Indenes; Indomethacin; Injections, Intravenous; Male; Pindolol; Propranolol; Rabbits; Radioligand Assay; Receptors, Adrenergic, beta | 1983 |
Characterization of beta-adrenergic receptors in the rat vas deferens using [3H]-dihydroalprenolol binding.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; Isoproterenol; Male; Muscle Contraction; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Vas Deferens | 1983 |
Photoperiodic modification of opiate but not beta-adrenergic or benzodiazepine binding sites in hamster brain.
Topics: Alprenolol; Animals; Anti-Anxiety Agents; Binding Sites; Body Weight; Brain; Cricetinae; Dihydroalprenolol; Flunitrazepam; Male; Naloxone; Organ Size; Periodicity; Photic Stimulation; Testis | 1983 |
The effect of the beta-adrenoreceptor antagonist Ro03-7894 on rat atrial tension development and (-)-[3H]dihydroalprenolol binding to cardiac and lung membranes.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Benzofurans; Cell Membrane; Dihydroalprenolol; Isoproterenol; Kinetics; Lung; Male; Myocardial Contraction; Myocardium; Rats | 1983 |
Beta-adrenoreceptor antagonists with multiple pharmacophores: persistent inhibition of rat heart adenylate cyclase.
Topics: Adenylyl Cyclase Inhibitors; Adrenergic beta-Antagonists; Alprenolol; Animals; Dihydroalprenolol; Dose-Response Relationship, Drug; Male; Myocardium; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Structure-Activity Relationship | 1983 |
Characterization of beta-adrenergic receptors in rat ovary.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; Female; In Vitro Techniques; Kinetics; Ovary; Rats; Receptors, Adrenergic, beta; Stereoisomerism; Tritium | 1983 |
[Characteristics of lipolytic activities in the genetically obese Zucker fatty rats--experimental study on (-)-[3H]dihydroalprenolol binding in the intact fat cells].
Topics: Adipose Tissue; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Cells, Cultured; Cyclic AMP; Dihydroalprenolol; Fatty Acids, Nonesterified; Lipolysis; Obesity; Phentolamine; Rats; Rats, Inbred Strains; Rats, Zucker | 1983 |
Beta-adrenergic receptor subtypes in iris-ciliary body of rabbits.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Binding, Competitive; Ciliary Body; Dihydroalprenolol; Female; Guinea Pigs; Heart Atria; Iris; Isoproterenol; Kinetics; Rabbits; Radioligand Assay; Receptors, Adrenergic, beta; Trachea | 1984 |
Characterization of putative beta-adrenoceptors in the myometrium of the pregnant ewe: correlation between the binding of [3H] dihydroalprenolol and the inhibition of myometrial contractility in vitro.
Topics: Adrenergic beta-Agonists; Albuterol; Alprenolol; Animals; Atenolol; Dihydroalprenolol; Dose-Response Relationship, Drug; Female; Myometrium; Pregnancy; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Sheep; Uterine Contraction | 1984 |
Uptake of L-[propyl-2,3-3H]dihydroalprenolol by intact HeLa cells.
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Biological Transport; Cell Membrane; Chloroquine; Cold Temperature; Diffusion; Dihydroalprenolol; HeLa Cells; Humans; Hydrogen-Ion Concentration; Isoproterenol; Phentolamine; Pindolol; Receptors, Adrenergic, beta; Valinomycin | 1984 |
Identification of beta-adrenergic receptors in mouse brain with 3H-dihydroalprenolol.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Cerebral Cortex; Dihydroalprenolol; Male; Mice; Rats; Receptors, Adrenergic, beta; Species Specificity | 1983 |
A comparison of the binding characteristics of the beta-adrenoceptor antagonists 3H-dihydroalprenolol and 125I-iodocyanopindolol in rat liver.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Kinetics; Liver; Liver Regeneration; Male; Membranes; Pindolol; Prazosin; Rats; Rats, Inbred Strains | 1984 |
Mapping of mammalian beta-adrenoreceptors by use of macromolecular alprenolol derivatives. A comparison with amphibian erythrocyte receptors.
Topics: Alprenolol; Animals; Anura; Chemical Phenomena; Chemistry; Dextrans; Dihydroalprenolol; Erythrocytes; In Vitro Techniques; Kinetics; Lung; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1982 |
Presence of functionally active beta-adrenoceptors in rat mast cells. Correlation between (--)[3H]-dihydroalprenolol binding and inhibition of histamine release.
Topics: Acetylcholine; Alprenolol; Animals; Cyclic AMP; Dihydroalprenolol; Epinephrine; Histamine Release; In Vitro Techniques; Male; Mast Cells; p-Methoxy-N-methylphenethylamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Sympathomimetics | 1982 |
Bromoacetylalprenololmenthane: a potent irreversible antagonist of beta adrenergic elicited protein exocytosis in rat parotid cells.
Topics: Adrenergic beta-Antagonists; Alprenolol; Amylases; Animals; Cyclohexane Monoterpenes; Depression, Chemical; Dihydroalprenolol; Exocytosis; Isoproterenol; Male; Microscopy, Electron; Parotid Gland; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1983 |
Hippocampal alpha- and beta-adrenergic receptors: comparison of [3H]dihydroalprenolol and [3H]WB 4101 binding with noradrenergic innervation in the rat.
Topics: Alprenolol; Animals; Binding Sites; Binding, Competitive; Dihydroalprenolol; Epinephrine; Hippocampus; Isoproterenol; Microscopy, Fluorescence; Norepinephrine; Radioligand Assay; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Synaptosomes | 1980 |
Effect of propranolol on beta-adrenoceptors in rat hearts.
Topics: Alprenolol; Animals; Dihydroalprenolol; Heart; Ligands; Male; Propranolol; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Cell metabolism affects the density of beta-adrenergic receptors in intact rat reticulocytes.
Topics: Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; Erythrocyte Membrane; Kinetics; Rabbits; Receptors, Adrenergic; Receptors, Adrenergic, beta; Reticulocytes | 1980 |
A ternary complex model explains the agonist-specific binding properties of the adenylate cyclase-coupled beta-adrenergic receptor.
Topics: Adenylyl Cyclases; Alprenolol; Animals; Anura; Binding Sites; Binding, Competitive; Dihydroalprenolol; Erythrocyte Membrane; Erythrocytes; Isoproterenol; Kinetics; Mathematics; Protein Binding; Receptors, Adrenergic; Receptors, Adrenergic, beta; Turkeys | 1980 |
[Characteristics of 3H-dihydroalprenolol binding to beta-receptors in the fat cells of rats and spontaneous genetic hypertension and in hypertensive disease].
Topics: Adipose Tissue; Adrenalectomy; Alprenolol; Animals; Binding Sites; Cell Membrane; Dihydroalprenolol; Humans; Hypertension; In Vitro Techniques; Male; Omentum; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Negative cooperativity of rat kidney beta-adrenergic receptors.
Topics: Alprenolol; Animals; Binding Sites; Cell Membrane; Dihydroalprenolol; Kidney; Kinetics; Mathematics; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
beta 1-Adrenergic receptors in kidney tubular cell membrane in the rat.
Topics: Alprenolol; Animals; Cell Membrane; Depression, Chemical; Dihydroalprenolol; Epinephrine; Isoproterenol; Kidney Tubules; Kinetics; Norepinephrine; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Decreased beta-adrenergic responses in the female rat brain are eliminated by ovariectomy: correlation of [3H]dihydroalprenolol binding and catecholamine stimulated cyclic AMP levels.
Topics: Alprenolol; Animals; Binding Sites; Castration; Cerebral Cortex; Cyclic AMP; Dihydroalprenolol; Estrogens; Estrus; Female; Isoproterenol; Male; Pregnancy; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Effects of phospholipids on the binding of [3H]dihydroalprenolol to the beta-adrenergic receptor of rabbit heart membranes.
Topics: Alprenolol; Animals; Dihydroalprenolol; In Vitro Techniques; Kinetics; Membranes; Myocardium; Phospholipids; Rabbits; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Myocardial beta-adrenergic receptors from adrenalectomized rats: impaired formation of high-affinity agonist-receptor complexes.
Topics: Adenylyl Cyclases; Adrenal Glands; Adrenalectomy; Alprenolol; Animals; Computers; Dihydroalprenolol; In Vitro Techniques; Isoproterenol; Male; Myocardium; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Down regulation of dihydroalprenolol and imipramine binding sites in brain of rats repeatedly treated with imipramine.
Topics: Alprenolol; Animals; Binding Sites; Brain; Dihydroalprenolol; Imipramine; In Vitro Techniques; Iprindole; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1980 |
Changes in ovarian beta-adrenergic receptors during the estrous cycle of the rat.
Topics: Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; Estrus; Female; Kinetics; Ovary; Pregnancy; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Alprenolol binding and cyclic AMP production in embryonic chick red cells during erythropoiesis.
Topics: Aging; Alprenolol; Animals; Chick Embryo; Cyclic AMP; Dihydroalprenolol; Epinephrine; Erythrocytes; Erythropoiesis; Filtration; Receptors, Adrenergic, beta | 1980 |
The influences of glucagon, epinephrine and alpha- and beta-adrenergic agents on glycogenolysis in isolated rabbit hepatocytes and perfused livers.
Topics: Alprenolol; Animals; Bucladesine; Cyclic AMP; Dihydroalprenolol; Epinephrine; Glucagon; In Vitro Techniques; Isoproterenol; Liver; Liver Glycogen; Male; Phentolamine; Phenylephrine; Rabbits | 1981 |
Beta-adrenoceptors of human lymphocytes: decrease in affinity of agonist for (-)3h-dihydroalprenolol binding sites by cytoplasmic fractions.
Topics: Alprenolol; Cytoplasm; Dihydroalprenolol; Humans; Lymphocytes; Receptors, Adrenergic; Receptors, Adrenergic, beta; Subcellular Fractions; Tritium | 1981 |
Binding of dihydroalprenolol and dihydroergocryptine to sheep myometrium.
Topics: Alprenolol; Animals; Binding Sites; Castration; Dihydroalprenolol; Dihydroergotoxine; Estradiol; Estrus; Female; Myometrium; Pregnancy; Progesterone; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Sheep; Uterus | 1981 |
Comparison of beta-adrenoceptors in bovine intracerebral microvessels and cerebral grey matter by [3H]dihydroalprenolol binding.
Topics: Alprenolol; Animals; Capillaries; Cattle; Cerebral Arteries; Cerebral Cortex; Dihydroalprenolol; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta; Stereoisomerism | 1981 |
Molecular pharmacology of adenylate cyclase-coupled alpha- and beta-adrenergic receptors.
Topics: Adenylyl Cyclases; Alprenolol; Animals; Blood Platelets; Cell Membrane; Dihydroalprenolol; Epinephrine; Erythrocyte Membrane; Erythrocytes; Guanosine Triphosphate; Isoproterenol; Kinetics; Ranidae; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1981 |
(-)-[3H]Dihydroalprenolol binding in subcellular fractions of rat cortex following noradrenergic denervation.
Topics: Alprenolol; Animals; Brain Neoplasms; Cerebral Cortex; Denervation; Dihydroalprenolol; Glioma; Kinetics; Male; Neoplasms, Experimental; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Synaptosomes | 1981 |
The effect of alprenolol on the beta-receptor and adenylate cyclase activity in rabbit heart membranes.
Topics: Adenylyl Cyclases; Alprenolol; Animals; Cell Membrane; Dihydroalprenolol; Guanine Nucleotides; Heart; In Vitro Techniques; Isoproterenol; Myocardium; Rabbits; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Aliphatic alcohols and the inhibition by thiol chelating agents of the binding of [3H[ dihydroalprenolol to myocardial beta-adrenoceptors.
Topics: 1-Butanol; Alcohols; Alprenolol; Animals; Butanols; Chelating Agents; Dihydroalprenolol; Ethylmaleimide; In Vitro Techniques; Myocardium; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Sheep; Sulfhydryl Compounds | 1981 |
Altered states of cardiac beta-adrenoreceptors.
Topics: Alprenolol; Animals; Ascorbic Acid; Chymotrypsin; Dihydroalprenolol; Dogs; Female; Hot Temperature; Isoproterenol; Male; Myocardium; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1981 |
Receptor binding sites for beta-adrenergic ligands on human erythrocytes.
Topics: Adult; Alprenolol; Binding, Competitive; Cyclic AMP; Dihydroalprenolol; Erythrocyte Membrane; Erythrocytes; Humans; Isoproterenol; Kinetics; Propranolol; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1982 |
Temperature dependence of [3H]dihydroalprenolol binding in rat myocardium.
Topics: Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; In Vitro Techniques; Male; Membranes; Myocardium; Rats; Receptors, Adrenergic, beta; Stereoisomerism; Sympathomimetics; Temperature; Time Factors | 1982 |
Binding of 3H-dihydroalprenolol to beta-adrenoceptors in adipocytes of spontaneously hypertensive rats and essentially hypertensive patients.
Topics: Adipose Tissue; Adult; Alprenolol; Animals; Cell Membrane; Dihydroalprenolol; Female; Humans; Hypertension; Male; Middle Aged; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1982 |
Uptake and displacement of [3H]dihydroalprenolol, [3H]epinephrine and [3H]clonidine in isolated perfused rabbit lung.
Topics: Alprenolol; Animals; Clonidine; Dihydroalprenolol; Epinephrine; In Vitro Techniques; Lung; Male; Perfusion; Phenoxybenzamine; Phentolamine; Rabbits; Receptors, Adrenergic, beta; Tritium | 1982 |
Binding of fluorescent and radiolabelled alprenolol to intact cultured brain cells and liposomes.
Topics: Alprenolol; Animals; Brain; Cells, Cultured; Chick Embryo; Dihydroalprenolol; Fluorescence; Liposomes; Receptors, Adrenergic; Receptors, Adrenergic, beta; Tritium | 1981 |
The (--)[3H]dihydroalprenolol binding to rat adipocyte membranes: an explanation of curvilinear Scatchard plots and implications for quantitation of beta-adrenergic sites.
Topics: Adipose Tissue; Alprenolol; Animals; Binding, Competitive; Cell Membrane; Dihydroalprenolol; Kinetics; Male; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Stereoisomerism; Tritium | 1982 |
Characterization of postsynaptic beta-adrenergic receptors and presynaptic muscarinic cholinergic receptors in the rat spleen.
Topics: Alprenolol; Animals; Dihydroalprenolol; Hydroxydopamines; In Vitro Techniques; Male; Norepinephrine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Receptors, Cholinergic; Receptors, Muscarinic; Spleen; Time Factors | 1982 |
Characterization of (-)-[3H]dihydroalprenolol binding to intact and broken cell preparations of human peripheral blood lymphocytes.
Topics: Alprenolol; Cell Membrane; Dihydroalprenolol; Guanine Nucleotides; Humans; In Vitro Techniques; Kinetics; Lymphocytes; Phentolamine; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta; Tritium | 1982 |
Beta-adrenergic receptors in early human placenta characterization of [3H]-dihydroalprenolol binding.
Topics: Alprenolol; Binding, Competitive; Dihydroalprenolol; Epinephrine; Female; Humans; Isoproterenol; Kinetics; Membranes; Norepinephrine; Placenta; Pregnancy; Pregnancy Trimester, First; Receptors, Adrenergic; Receptors, Adrenergic, beta; Substrate Specificity | 1983 |
Binding of [3H]-dihydroalprenolol and [3H]-acetobutolol to human blood platelets is not related to occupancy of beta-adrenoceptors.
Topics: Acebutolol; Alprenolol; Blood Platelets; Butoxamine; Dihydroalprenolol; Humans; Isoproterenol; Kinetics; Practolol; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1983 |
beta-2 adrenergic receptors on intact human erythrocytes.
Topics: Alprenolol; Binding, Competitive; Cyclic AMP; Dihydroalprenolol; Erythrocytes; Humans; In Vitro Techniques; Isoproterenol; Receptors, Adrenergic; Receptors, Adrenergic, beta | 1983 |
The interaction of triamterene at the myocardial beta receptor site.
Topics: Alprenolol; Animals; Binding, Competitive; Cell Membrane; Dihydroalprenolol; Guinea Pigs; Myocardial Contraction; Myocardium; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta; Triamterene | 1983 |
Binding characteristics of 3H-dihydroalprenolol to beta-adrenoceptors of rat heart treated with neuraminidase.
Topics: Alprenolol; Animals; Cell Membrane; Dihydroalprenolol; In Vitro Techniques; Kinetics; Male; Myocardium; Neuraminidase; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Sialic Acids; Stereoisomerism | 1983 |
Formation of complexes between avidin and beta-adrenergic receptors using biotinyl-alprenolol derivatives.
Topics: Alprenolol; Animals; Avidin; Binding, Competitive; Digitonin; Dihydroalprenolol; Ducks; Erythrocyte Membrane; Erythrocytes; Kinetics; Ovalbumin; Receptors, Adrenergic, beta | 1983 |
[Determination of beta-receptors on intact polymorphonuclear leukocytes in autologous plasma].
Topics: Alprenolol; Cell Membrane; Dihydroalprenolol; Humans; Kinetics; Male; Neutrophils; Physical Endurance; Physical Exertion; Receptors, Adrenergic, beta | 1983 |
[Effect of thyroid hormones on the beta-adrenergic receptor internalization in isolated rat hepatocytes].
Topics: Alprenolol; Animals; Cadaverine; Dihydroalprenolol; In Vitro Techniques; Isoproterenol; Liver; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Thyroidectomy; Thyroxine | 1983 |
Genetic variation in beta-adrenergic receptors in mice: a magnesium effect determined by a single gene.
Topics: Alprenolol; Animals; Dihydroalprenolol; Female; Genetic Variation; Magnesium; Male; Mice; Mice, Inbred Strains; Receptors, Adrenergic, beta | 1983 |
Tolbutamide and glyburide differ in effectiveness to displace alpha- and beta-adrenergic radioligands in pancreatic islet cells and membranes.
Topics: Alprenolol; Animals; Cell Membrane; Clonidine; Dihydroalprenolol; Epinephrine; Glyburide; Islets of Langerhans; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Tolbutamide | 1984 |
Postnatal development of the beta-adrenergic receptor complex in brown adipose tissue of the rat.
Topics: Adenylyl Cyclases; Adipose Tissue, Brown; Alprenolol; Animals; Animals, Newborn; Binding Sites; Dihydroalprenolol; Enzyme Activation; Female; Isoproterenol; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Sodium Fluoride | 1984 |
Methodological aspects of receptor research: problems in the assessment of specific and non-specific binding of 3H-dihydroalprenolol to bovine lung membranes.
Topics: Alprenolol; Animals; Binding Sites; Cattle; Dihydroalprenolol; Lung; Receptors, Adrenergic, beta; Tritium | 1984 |
Some characteristics of 3H-dihydroalprenolol binding to intact normal granulocytes, lymphocytes and membrane preparations of these cells.
Topics: Alprenolol; Cell Membrane; Dihydroalprenolol; Ethanolamines; Granulocytes; Humans; Lymphocytes; Practolol; Procaterol; Receptors, Adrenergic, beta; Tritium | 1984 |
Specific binding of [3H]WB 4101, [3H]clonidine and [3H]dihydroalprenolol in cerebral cortical membranes in developing, adult and old rats.
Topics: Aging; Alprenolol; Animals; Cerebral Cortex; Clonidine; Dihydroalprenolol; Dioxanes; Dioxins; Female; Male; Membranes; Rats; Rats, Inbred Strains; Synapses | 1984 |
Effects of pH and ascorbic acid on 3H-spiperone and 3H-dihydroalprenolol binding in rat forebrain homogenates.
Topics: Alprenolol; Animals; Ascorbic Acid; Butyrophenones; Diencephalon; Dihydroalprenolol; Hydrogen-Ion Concentration; In Vitro Techniques; Lipid Peroxides; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Telencephalon | 1984 |
Influences of isoproterenol pretreatment on cerebral cortical bindings of [3H]clonidine and [3H]dihydroalprenolol in infant and adult rats.
Topics: Alprenolol; Animals; Cerebral Cortex; Clonidine; Dihydroalprenolol; Female; Isoproterenol; Male; Rats; Rats, Inbred Strains; Tritium | 1983 |
Ascorbate-induced lipid peroxidation and the binding of [3H]dihydroalprenolol.
Topics: Alprenolol; Animals; Ascorbic Acid; Cerebral Cortex; Dihydroalprenolol; In Vitro Techniques; Iron; Kinetics; Lipid Peroxides; Male; Rats; Rats, Inbred Strains | 1983 |
[Specific binding of [3H]-dihydroalprenolol and [3H]-prazosin to kidney tubules].
Topics: Alprenolol; Animals; Dihydroalprenolol; Female; Kidney Tubules; Prazosin; Quinazolines; Rabbits; Tritium | 1983 |
Monoclonal antibodies specific for beta-adrenergic ligands.
Topics: Alprenolol; Animals; Antibodies, Monoclonal; Antibody Specificity; Binding Sites, Antibody; Binding, Competitive; Dihydroalprenolol; Mice; Mice, Inbred BALB C; Propranolol; Spectrometry, Fluorescence; Thermodynamics | 1984 |
Binding of [3H]dihydroalprenolol and [3H]quinuclidinyl benzilate to intact cells of cultured corneal epithelium.
Topics: Alprenolol; Animals; Binding, Competitive; Cells, Cultured; Cornea; Dihydroalprenolol; Epinephrine; Male; Parasympatholytics; Propranolol; Quinuclidines; Quinuclidinyl Benzilate; Rabbits; Receptors, Cholinergic | 1982 |
The uptake of amines by polymorphonuclear leukocytes.
Topics: Alprenolol; Animals; Binding, Competitive; Biological Transport; Brain; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Dihydroalprenolol; Humans; Hydrogen-Ion Concentration; Kinetics; Male; Myocardium; Neutrophils; Quinuclidines; Quinuclidinyl Benzilate; Rats; Valinomycin | 1981 |
Changes in catecholamine neuronal uptake and receptor binding in the brains of spontaneously hypertensive rats (SHR).
Topics: Aging; Alprenolol; Animals; Biological Transport; Brain; Dihydroalprenolol; Dopamine; Hypertension; Kinetics; Neurons; Norepinephrine; Organ Specificity; Rats; Rats, Inbred Strains | 1981 |
Rapid-eye-movement sleep deprivation decreases the density of 3H-dihydroalprenolol and 3H-imipramine binding sites in the rat cerebral cortex.
Topics: Alprenolol; Animals; Binding Sites; Cerebral Cortex; Dihydroalprenolol; Imipramine; Male; Rats; Sleep, REM; Time Factors | 1980 |
Beta-Adrenergic receptors in rat fat cells and their relationship with lipolysis.
Topics: Adipocytes; Adrenergic Agents; Adrenergic beta-Antagonists; Alprenolol; Animals; Binding Sites; Binding, Competitive; Dihydroalprenolol; Lipolysis; Male; Norepinephrine; Propranolol; Rats; Receptors, Adrenergic, beta; Sonication | 1996 |