Page last updated: 2024-08-17

dichloroacetic acid and monorden

dichloroacetic acid has been researched along with monorden in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chuang, DT; Chuang, JL; Gui, WJ; Morlock, LK; Owens, KR; Qi, X; Scherer, PE; Tambar, UK; Tso, SC; Wernstedt-Asterholm, I; Williams, NS; Wu, CY; Wynn, RM1
Geng, M; Hilpert, K; Huang, M; Meng, T; Regenass, U; Shen, J; Wu, S; Wyder, L; Xie, Z; Yu, T; Zhang, D1
Chuang, DT; Chuang, JL; Kato, M; Li, J1

Other Studies

3 other study(ies) available for dichloroacetic acid and monorden

ArticleYear
Structure-guided development of specific pyruvate dehydrogenase kinase inhibitors targeting the ATP-binding pocket.
    The Journal of biological chemistry, 2014, Feb-14, Volume: 289, Issue:7

    Topics: Animals; Diabetes Mellitus, Type 2; Drug Delivery Systems; Drug Design; Enzyme Inhibitors; Fatty Liver; HSP90 Heat-Shock Proteins; Humans; Isoenzymes; Isoindoles; Male; Mice; Mice, Obese; Obesity; Protein Serine-Threonine Kinases; Pyruvate Dehydrogenase Acetyl-Transferring Kinase; Sulfones

2014
Discovery and optimization of 4,5-diarylisoxazoles as potent dual inhibitors of pyruvate dehydrogenase kinase and heat shock protein 90.
    Journal of medicinal chemistry, 2014, Dec-11, Volume: 57, Issue:23

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; HSP90 Heat-Shock Proteins; Humans; Isoxazoles; Piperazines; Protein Serine-Threonine Kinases; Pyruvate Dehydrogenase Acetyl-Transferring Kinase; Structure-Activity Relationship

2014
Distinct structural mechanisms for inhibition of pyruvate dehydrogenase kinase isoforms by AZD7545, dichloroacetate, and radicicol.
    Structure (London, England : 1993), 2007, Volume: 15, Issue:8

    Topics: Amino Acid Motifs; Amino Acid Sequence; Anilides; Binding Sites; Crystallography, X-Ray; Dichloroacetic Acid; Dimerization; Dose-Response Relationship, Drug; Humans; Hydrogen Bonding; Inhibitory Concentration 50; Isoenzymes; Macrolides; Models, Molecular; Molecular Structure; Protein Binding; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Protein Structure, Tertiary; Pyruvate Dehydrogenase Acetyl-Transferring Kinase; Solubility; Spectrum Analysis, Raman

2007