diazoxide and prazosin

diazoxide has been researched along with prazosin in 47 studies

Research

Studies (47)

TimeframeStudies, this research(%)All Research%
pre-199036 (76.60)18.7374
1990's0 (0.00)18.2507
2000's5 (10.64)29.6817
2010's6 (12.77)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Nies, AS1
Pettinger, WA1
Oparil, S; Rick, JH1
Graham, RM; Oates, HF; Stoker, LM; Stokes, GS2
Gifford, RW; Tarazi, RC; Wollam, GL1
Sterz, H1
Sternon, J1
Romankiewicz, JA1
McKenzie, JK1
Collier, JG; Lorge, RE; Robinson, BF1
Graham, RM; Oates, HF; Stokes, GS1
Rubin, PC1
Kincaid-Smith, P1
Petrie, JC1
Fischer, E; Siegenthaler, W1
Anand, MP1
Andersson, O1
Plouin, PF1
Ram, CV1
Song, YC1
Barry, DI; Braendstrup, O; Graham, DI; Jarden, JO; Strandgaard, S; Svendsen, UG; Vorstrup, S2
Strandgaard, S1
Constantine, JW; Lebel, W; Weeks, R1
Julius, S; Osterziel, KJ1
White, SJ; Williamson, K1
Berkowitz, RL1
Freed, CR; Gerber, JG; Nies, AS1
Croveri, G; Lucignani, P1
Reisman, L; Selden, RV1
Pruitt, AW1
Bannan, LT; Beevers, DG; Wright, N1
Elkayam, U1
Lim, SK1
Greger, R; Herbst, M; Hescheler, J; Sasse, P; Ullrich, S; Yu, H1

Reviews

14 review(s) available for diazoxide and prazosin

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Clinical pharmacology of antihypertensive drugs.
    The Medical clinics of North America, 1977, Volume: 61, Issue:3

    Topics: Adrenergic alpha-Antagonists; Aldosterone; Angiotensin II; Antihypertensive Agents; Bethanidine; Blood Pressure; Clonidine; Diazoxide; Diuretics; Emergencies; Guanethidine; Humans; Hydralazine; Hypertension; Methyldopa; Minoxidil; Monoamine Oxidase Inhibitors; Nitroprusside; Prazosin; Propranolol; Renin; Reserpine; Sympathetic Nervous System; Trimethaphan

1977
Recent advances in the treatment of hypertension.
    Archives of internal medicine, 1977, Volume: 137, Issue:5

    Topics: Adrenergic beta-Antagonists; Antihypertensive Agents; Chronic Disease; Clonidine; Diazoxide; Drug Therapy, Combination; Humans; Hypertension; Prazosin; Propranolol; Renin; Vasodilator Agents

1977
Antihypertensive drugs: clinical pharmacology and therapeutic use.
    Drugs, 1977, Volume: 14, Issue:6

    Topics: Adrenergic beta-Antagonists; Angiotensin II; Angiotensin-Converting Enzyme Inhibitors; Antihypertensive Agents; Clonidine; Diazoxide; Diuretics; Ganglionic Blockers; Humans; Hydralazine; Hypertension; Labetalol; Methyldopa; Minoxidil; Monoamine Oxidase Inhibitors; Nitroprusside; Potassium; Prazosin; Secologanin Tryptamine Alkaloids; Sympatholytics

1977
[New aspects in the treatment of acute cardiac insufficiency].
    Wiener medizinische Wochenschrift (1946), 1978, May-15, Volume: 128, Issue:9

    Topics: Adrenergic beta-Antagonists; Clonidine; Diazoxide; Digitalis Glycosides; Diuretics; Droperidol; Fentanyl; Fibrinolytic Agents; Heart Failure; Humans; Hydralazine; Isosorbide Dinitrate; Microcirculation; Myocardial Contraction; Neuroleptanalgesia; Nitroprusside; Phentolamine; Prazosin; Respiration, Artificial; Vascular Resistance; Vasodilator Agents

1978
Acute and chronic therapy of hypertension with vasodilators.
    Clinical and investigative medicine. Medecine clinique et experimentale, 1978, Volume: 1, Issue:3-4

    Topics: Antihypertensive Agents; Diazoxide; Humans; Hypertension; Minoxidil; Nitroprusside; Prazosin; Time Factors; Vasodilator Agents

1978
Treatment of hypertension in pregnancy.
    Clinics in obstetrics and gynaecology, 1986, Volume: 13, Issue:2

    Topics: Adrenergic beta-Antagonists; Antihypertensive Agents; Diazoxide; Diuretics; Eclampsia; Female; Humans; Hydralazine; Hypertension; Methyldopa; Nitroprusside; Prazosin; Pre-Eclampsia; Pregnancy; Pregnancy Complications, Cardiovascular

1986
Vasodilator drugs in the treatment of hypertension.
    The Medical journal of Australia, 1985, Apr-15, Volume: 142, Issue:8

    Topics: Calcium Channel Blockers; Captopril; Cardiac Output; Diazoxide; Diuretics; Dose-Response Relationship, Drug; Drug Therapy, Combination; Hemodynamics; Humans; Hydralazine; Hypertension; Infusions, Parenteral; Minoxidil; Prazosin; Renal Circulation; Vasodilator Agents

1985
Hypertension--drug management.
    The Journal of the Association of Physicians of India, 1982, Volume: 30, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Calcium Channel Blockers; Captopril; Diazoxide; Humans; Hypertension; Indoramin; Labetalol; Minoxidil; Nifedipine; Nitroprusside; Prazosin; Sympatholytics; Vasodilator Agents; Verapamil

1982
Hypertensive crisis.
    Cardiology clinics, 1984, Volume: 2, Issue:2

    Topics: Antihypertensive Agents; Brain Diseases; Cerebrovascular Disorders; Clonidine; Coronary Disease; Diazoxide; Eclampsia; Emergencies; Female; Humans; Hydralazine; Hypertension; Hypertension, Malignant; Labetalol; Minoxidil; Nifedipine; Nitroprusside; Phentolamine; Prazosin; Pregnancy; Pulmonary Edema; Trimethaphan

1984
Anti-hypertensive drugs in the pregnant patient.
    Obstetrical & gynecological survey, 1980, Volume: 35, Issue:4

    Topics: Antihypertensive Agents; Chronic Disease; Clonidine; Diazoxide; Diuretics; Female; Fetus; Furosemide; Guanethidine; Humans; Hydralazine; Hypertension; Infant Mortality; Methyldopa; Nitroprusside; Prazosin; Pre-Eclampsia; Pregnancy; Pregnancy Complications, Cardiovascular; Propranolol; Secologanin Tryptamine Alkaloids; Sodium; Sodium Chloride Symporter Inhibitors

1980
Antihypertensive pharmacology.
    The Western journal of medicine, 1980, Volume: 132, Issue:5

    Topics: Adolescent; Adult; Antihypertensive Agents; Clonidine; Diazoxide; Diuretics; Guanethidine; Humans; Hydralazine; Hypertension; Methyldopa; Metoprolol; Minoxidil; Nitroprusside; Patient Compliance; Prazosin; Propranolol; Reserpine; Sodium Chloride Symporter Inhibitors

1980
[Arterial hypertension, III. Antihypertensive therapy (1). Diuretics].
    Minerva medica, 1980, Dec-15, Volume: 71, Issue:50

    Topics: Antihypertensive Agents; Diazoxide; Diuretics; Humans; Hydralazine; Hypertension; Mineralocorticoid Receptor Antagonists; Minoxidil; Prazosin; Sodium Chloride Symporter Inhibitors; Vasodilator Agents

1980
Management of systemic hypertension in children.
    Pediatric annals, 1982, Volume: 11, Issue:7

    Topics: Adolescent; Antihypertensive Agents; Child; Clonidine; Diazoxide; Diet, Sodium-Restricted; Diuretics; Humans; Hydralazine; Hypertension; Methyldopa; Minoxidil; Nitroprusside; Prazosin; Propranolol

1982

Other Studies

33 other study(ies) available for diazoxide and prazosin

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Drug treatment of hypertension.
    Comprehensive therapy, 1977, Volume: 3, Issue:5

    Topics: Clonidine; Diazoxide; Diuretics; Ganglionic Blockers; Guanethidine; Humans; Hydralazine; Hypertension; Mecamylamine; Methyldopa; Mineralocorticoid Receptor Antagonists; Minoxidil; Nitroprusside; Prazosin; Propranolol; Secologanin Tryptamine Alkaloids; Sodium Chloride Symporter Inhibitors; Spironolactone; Sympatholytics; Triamterene; Trimethaphan; Vasodilator Agents

1977
Alpha blocking action of the antihypertensive agent, prazosin.
    The Journal of pharmacology and experimental therapeutics, 1977, Volume: 201, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Diazoxide; Pentolinium Tartrate; Phentolamine; Prazosin; Quinazolines; Rats; Vasodilator Agents

1977
[The practitioner and drug-induced, predominantly orthostatic hypotension].
    Acta clinica Belgica, 1978, Volume: 33, Issue:6

    Topics: Adrenergic Agents; Adrenergic Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Antidepressive Agents, Tricyclic; Antihypertensive Agents; Antipsychotic Agents; Barbiturates; Butyrophenones; Clonidine; Debrisoquin; Diazoxide; Diuretics; Ganglionic Blockers; Humans; Hydralazine; Hypotension, Orthostatic; Levodopa; Meprobamate; Methyldopa; Mineralocorticoids; Monoamine Oxidase Inhibitors; Phenothiazines; Prazosin; Psychotropic Drugs; Reserpine; Vasodilator Agents

1978
Hypotensive agents. Part I: Vasodilators.
    The Journal of practical nursing, 1979, Volume: 29, Issue:6

    Topics: Diazoxide; Humans; Hydralazine; Hypertension; Prazosin; Quinazolines

1979
Comparison of effects of tolmesoxide (RX71107), diazoxide, hydrallazine, prazosin, glyceryl trinitrate and sodium nitroprusside on forearm arteries and dorsal hand veins of man.
    British journal of clinical pharmacology, 1978, Volume: 5, Issue:1

    Topics: Adult; Antihypertensive Agents; Arteries; Blood Vessels; Diazoxide; Female; Forearm; Hand; Humans; Hydralazine; Male; Middle Aged; Nitroglycerin; Nitroprusside; Prazosin; Regional Blood Flow; Sulfoxides; Toluene; Vasodilation; Veins

1978
When to use oral vasodilators for hypertension.
    Drug and therapeutics bulletin, 1979, Jul-20, Volume: 17, Issue:15

    Topics: Administration, Oral; Diazoxide; Humans; Hydralazine; Hypertension; Minoxidil; Prazosin; Vasodilator Agents

1979
Mechanism of the hypotensive action of prazosin.
    Archives internationales de pharmacodynamie et de therapie, 1977, Volume: 227, Issue:1

    Topics: Angiotensin II; Animals; Antihypertensive Agents; Blood Pressure; Diazoxide; Dose-Response Relationship, Drug; Drug Interactions; Epinephrine; Heart Rate; Hydralazine; Indoramin; Norepinephrine; Pentolinium Tartrate; Phentolamine; Prazosin; Quinazolines; Rats

1977
Haemodynamic effects of prazosin.
    Archives internationales de pharmacodynamie et de therapie, 1976, Volume: 224, Issue:2

    Topics: Animals; Atropine; Blood Cell Count; Blood Pressure; Diazoxide; Dose-Response Relationship, Drug; Drug Interactions; Heart Rate; Hemodynamics; Isoproterenol; Pentolinium Tartrate; Prazosin; Quinazolines; Rats; Renin; Timolol

1976
Current trends in the management of hypertension.
    Comprehensive therapy, 1980, Volume: 6, Issue:3

    Topics: Adrenergic beta-Antagonists; Aged; Diazoxide; Diuretics; Female; Humans; Hydralazine; Hypertension; Male; Methyldopa; Middle Aged; Minoxidil; Nitroprusside; Prazosin; Risk; Vasodilator Agents

1980
[Vasodilators in heart failure? Basic principles and its role in practice].
    Deutsche medizinische Wochenschrift (1946), 1981, Sep-25, Volume: 106, Issue:39

    Topics: Adrenergic alpha-Antagonists; Captopril; Diazoxide; Furosemide; Heart Failure; Humans; Hydralazine; Minoxidil; Phentolamine; Prazosin; Vasodilator Agents

1981
[Vasodilating agents in the treatment of hypertension - a review].
    Lakartidningen, 1981, Jan-28, Volume: 78, Issue:5

    Topics: Diazoxide; Humans; Hydralazine; Hypertension; Minoxidil; Nitroprusside; Prazosin; Synaptic Transmission; Vasodilator Agents

1981
[Antihypertensive vasodilators].
    La semaine des hopitaux : organe fonde par l'Association d'enseignement medical des hopitaux de Paris, 1983, Nov-17, Volume: 59, Issue:42

    Topics: Antihypertensive Agents; Chemical Phenomena; Chemistry; Diazoxide; Dihydralazine; Humans; Hydralazine; Minoxidil; Nitroprusside; Prazosin; Vasodilator Agents

1983
[Clinical use of new antihypertensives].
    Zhonghua yi xue za zhi, 1984, Volume: 64, Issue:8

    Topics: Alkaloids; Antihypertensive Agents; Benzylisoquinolines; Captopril; Diazoxide; Diterpenes; Humans; Hypertension; Labetalol; Minoxidil; Nifedipine; Nitroprusside; Prazosin

1984
Effects of antihypertensive drugs on the cerebral circulation.
    Acta medica Scandinavica. Supplementum, 1983, Volume: 677

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cerebrovascular Circulation; Diazoxide; Dihydralazine; Homeostasis; Prazosin; Rats; Reserpine

1983
Cerebral blood flow in hypertension.
    Acta medica Scandinavica. Supplementum, 1983, Volume: 678

    Topics: Antihypertensive Agents; Brain Ischemia; Cerebrovascular Circulation; Cerebrovascular Disorders; Diazoxide; Dihydralazine; Emergencies; Homeostasis; Humans; Hypertension; Nitroprusside; Phenoxybenzamine; Prazosin; Risk; Trimethaphan

1983
The effect of chronic hypertension and antihypertensive drugs on the cerebral circulation.
    Acta medica Scandinavica. Supplementum, 1983, Volume: 678

    Topics: Animals; Antihypertensive Agents; Cerebrovascular Circulation; Diazoxide; Dihydralazine; Homeostasis; Humans; Hypertension; Prazosin; Rats; Rats, Inbred Strains; Vasodilation

1983
Effects of trimazosin and prazosin on blood pressure and on pressor responses to phenylephrine in rats.
    American heart journal, 1983, Volume: 106, Issue:5 Pt 2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Diazoxide; Dose-Response Relationship, Drug; Heart Rate; Male; Phenylephrine; Piperazines; Prazosin; Pressoreceptors; Quinazolines; Rats; Solvents

1983
Vasodilators in the treatment of hypertension.
    Comprehensive therapy, 1982, Volume: 8, Issue:11

    Topics: Calcium Channel Blockers; Captopril; Diazoxide; Humans; Hydralazine; Hypertension; Minoxidil; Nitroprusside; Prazosin; Vasodilator Agents

1982
What to watch for with peripherally acting antihypertensives.
    RN, 1980, Volume: 43, Issue:1

    Topics: Antihypertensive Agents; Diazoxide; Drug Interactions; Humans; Hydralazine; Nitroprusside; Prazosin

1980
Pharmacologic approach to the management of childhood hypertension.
    Pediatric clinics of North America, 1981, Volume: 28, Issue:1

    Topics: Antihypertensive Agents; Autonomic Nervous System; Central Nervous System; Child; Diazoxide; Humans; Hydralazine; Hypertension; Minoxidil; Muscle, Smooth, Vascular; Nitroprusside; Prazosin; Receptors, Adrenergic

1981
Vasodilator drugs and resistant hypertension.
    British medical journal, 1980, Oct-18, Volume: 281, Issue:6247

    Topics: Antihypertensive Agents; Diazoxide; Drug Therapy, Combination; Humans; Hydralazine; Hypertension; Minoxidil; Prazosin; Vasodilator Agents

1980
Vasodilator therapy in primary pulmonary hypertension.
    Chest, 1981, Volume: 79, Issue:3

    Topics: Adult; Diazoxide; Female; Hemodynamics; Humans; Hydralazine; Hypertension, Pulmonary; Isoproterenol; Male; Phentolamine; Physical Exertion; Prazosin; Pulmonary Circulation; Vasodilator Agents

1981
Consequences of haemolysis without haptoglobin.
    Redox report : communications in free radical research, 2001, Volume: 6, Issue:6

    Topics: Aldehydes; Animals; Cysteine Proteinase Inhibitors; Diazoxide; Haptoglobins; Hemoglobins; Hemolysis; Kidney; Malondialdehyde; Mice; Mice, Knockout; Nitric Oxide; Orosomucoid; Oxidative Stress; Phenotype; Prazosin; Protein Binding; Vasodilator Agents

2001
Membrane potential dependent modulations of calcium oscillations in insulin-secreting INS-1 cells.
    Cell calcium, 2002, Volume: 31, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Calcium Signaling; Cell Line; Clonidine; Colforsin; Diazoxide; Enzyme Inhibitors; Epinephrine; Fluorescent Dyes; Fura-2; Glucose; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Membrane Potentials; Mice; Patch-Clamp Techniques; Potassium Channels; Prazosin; Receptors, Adrenergic, alpha-2; Thapsigargin; Tolbutamide

2002