diazoxide and hydroflumethiazide

diazoxide has been researched along with hydroflumethiazide in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19905 (38.46)18.7374
1990's1 (7.69)18.2507
2000's1 (7.69)29.6817
2010's6 (46.15)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Gozalbes, R; Pineda-Lucena, A1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Blayac, JP; Loubatières-Mariani, MM; Manteghetti, M; Petit, P1
Cross, RB; Thornton, WM1
Gulbenkian, A; Tabachnick, II; Yannell, A1
Blayac, JP; Buys, D; Loubatieres-Mariani, MM; Puech, R; Ribes, G1
Blayac, JP; Loubatieres-Mariani, MM; Manteghetti, M; Puech, R; Ribes, G1
GILLENWATER, JY1

Reviews

1 review(s) available for diazoxide and hydroflumethiazide

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

12 other study(ies) available for diazoxide and hydroflumethiazide

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
QSAR-based solubility model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2010, Oct-01, Volume: 18, Issue:19

    Topics: Databases, Factual; Models, Molecular; Pharmaceutical Preparations; Quantitative Structure-Activity Relationship; Solubility; Water

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Comparative effects of LN 5330 and diazoxide on insulin release and 86Rb+ permeability in perifused rat islets of Langerhans.
    Biochemical pharmacology, 1991, Jul-25, Volume: 42, Issue:4

    Topics: Animals; Calcium; Cell Membrane Permeability; Diazoxide; Glucose; Hydroflumethiazide; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Male; Perfusion; Rats; Rats, Inbred Strains; Rubidium; Rubidium Radioisotopes

1991
The effect of benzothiadiazine diuretics on the renal concentrating mechanism of the sheep.
    Quarterly journal of experimental physiology and cognate medical sciences, 1966, Volume: 51, Issue:4

    Topics: Absorption; Animals; Bendroflumethiazide; Chlorides; Chlorothiazide; Diazoxide; Hydrochlorothiazide; Hydroflumethiazide; Kidney Tubules; Natriuresis; Potassium; Sheep; Vasopressins; Water-Electrolyte Balance

1966
The hyperglycemic activity of benzothiadiazine and other diuretics.
    Life sciences, 1965, Volume: 4, Issue:20

    Topics: Animals; Bendroflumethiazide; Benzothiadiazines; Chlorothiazide; Chlorthalidone; Diazoxide; Diuretics; Ethacrynic Acid; Hydroflumethiazide; Hyperglycemia; Methyclothiazide; Polythiazide; Rats; Sulfonamides; Trichlormethiazide

1965
Effects of a new benzothiadiazine derivative, LN 5330, on insulin secretion.
    Archives internationales de pharmacodynamie et de therapie, 1981, Volume: 253, Issue:1

    Topics: Animals; Diazoxide; Female; Glucose; Hydroflumethiazide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Perfusion; Rats; Rats, Inbred Strains; Somatostatin; Time Factors

1981
Effect of LN 5330 on insulin release and calcium uptake by isolated rat islets of Langerhans. Comparison with diazoxide.
    Archives internationales de pharmacodynamie et de therapie, 1984, Volume: 272, Issue:1

    Topics: Animals; Calcium; Calcium Radioisotopes; Diazoxide; Hydroflumethiazide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Rats; Rats, Inbred Strains

1984
THE ANTIDIURETIC PROPERTIES OF CHLOROTHIAZIDE IN DIABETES INSIPIDUS DOGS. I. EFFECT ON SOLUTE, WATER, AND ELECTROLYTE EXCRETION. REP 582.
    Report. Army Medical Research Laboratory (U.S.), 1963, Jul-15

    Topics: Animals; Bendroflumethiazide; Blood Volume; Body Fluids; Chlorothiazide; Chlorthalidone; Diabetes Insipidus; Diazoxide; Diuresis; Diuretics; Dogs; Electrolytes; Hydroflumethiazide; Kidney Function Tests; Pharmacology; Research; Urine; Water

1963