diazoxide and colforsin

diazoxide has been researched along with colforsin in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-19901 (4.00)18.7374
1990's7 (28.00)18.2507
2000's16 (64.00)29.6817
2010's1 (4.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Ahrén, B; Lindskog, S1
Ashcroft, SJ; Niki, I1
Baró, I; Berthon, B; Escande, D; Hongre, AS1
Bégin-Heick, N; Fournier, L; Schwartz, JL; Whitfield, JF1
Detimary, P; Gao, ZY; Gembal, M; Gilon, P; Henquin, JC1
Abdel-Halim, SM; Berggren, PO; Efendić, S; Guenifi, A; Khan, A; Larsson, O; Ostenson, CG1
Aizawa, T; Hashizume, K; Kaneko, T; Komatsu, M; Nagai, M; Schermerhorn, T; Sharp, GW; Yajima, H1
Haynes, JM1
Asai, M; Iwasaki, Y; Morishita, M; Mutsuga, N; Nomura, A; Oiso, Y; Saito, H; Yamamori, E; Yoshida, M1
Björklund, A; Grill, VE1
Fujimoto, S; Hamamoto, Y; Ishida, H; Kajikawa, M; Mukai, E; Seino, Y; Takeda, T; Tsuji, K; Tsuura, Y; Yamada, Y1
García de Boto, MJ; Hidalgo, A; Martínez, C; Sánchez, M1
Cerasi, E; Efendic, S; Kaiser, N; Khan, A; Nesher, R; Warwar, N1
Aizawa, T; Hashizume, K; Komatsu, M; Sato, Y; Yamada, S; Yamauchi, K1
Greger, R; Herbst, M; Hescheler, J; Sasse, P; Ullrich, S; Yu, H1
da Silva Xavier, G; Holz, GG; Jouaville, LS; Rutter, GA; Thomas, AP; Tsuboi, T1
Göpel, SO; Holm, C; Olofsson, CS; Rorsman, P; Salehi, A1
Kwon, G; Marshall, CA; McDaniel, ML; Pappan, KL; Remedi, MS1
Nakaya, H; Saegusa, N; Saito, T; Sato, T1
Anwar, MR; Capito, K; Thams, P1
Philbrick, W; Yamazaki, H; Zawalich, KC; Zawalich, WS1
Araújo, PV; Clemente, CM; de Oliveira, RB; dos Santos, AA; Fernandes, GH; Magalhães, PJ; Palheta, RC; Ratts, ZM; Rola, FH1
Henquin, JC; Nenquin, M1

Reviews

1 review(s) available for diazoxide and colforsin

ArticleYear
Signaling elements involved in the metabolic regulation of mTOR by nutrients, incretins, and growth factors in islets.
    Diabetes, 2004, Volume: 53 Suppl 3

    Topics: Animals; Colforsin; Cyclic AMP; Diazoxide; Growth Substances; Humans; Insulin; Insulin Secretion; Islets of Langerhans; Nutritional Physiological Phenomena; Phosphorylation; Protein Kinases; Signal Transduction; TOR Serine-Threonine Kinases

2004

Other Studies

24 other study(ies) available for diazoxide and colforsin

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Studies on the mechanism by which galanin inhibits insulin secretion in islets.
    European journal of pharmacology, 1991, Nov-19, Volume: 205, Issue:1

    Topics: Animals; Bucladesine; Calcium Radioisotopes; Colforsin; Diazoxide; Galanin; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Mice; Mice, Inbred Strains; Neuropeptides; Peptides; Permeability; Rats; Rats, Inbred Strains; Rubidium Radioisotopes; Tetradecanoylphorbol Acetate

1991
Possible involvement of protein phosphorylation in the regulation of the sulphonylurea receptor of a pancreatic beta-cell line, HIT T15.
    Biochimica et biophysica acta, 1991, Dec-03, Volume: 1133, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Cell Line; Cell Membrane; Colforsin; Diazoxide; Glyburide; Humans; Insulin; Insulin Secretion; Islets of Langerhans; Isoquinolines; Phosphorylation; Piperazines; Potassium Channels; Potassium Channels, Inwardly Rectifying; Protein Kinase Inhibitors; Proteins; Receptors, Drug; Rubidium; Sulfonylurea Receptors; Tetradecanoylphorbol Acetate

1991
Effects of sulphonylureas on cAMP-stimulated Cl- transport via the cystic fibrosis gene product in human epithelial cells.
    Pflugers Archiv : European journal of physiology, 1994, Volume: 426, Issue:3-4

    Topics: Adenosine Triphosphate; Blood Proteins; Cell Line; Chloride Channels; Colforsin; Cyclic AMP; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Diazoxide; Electrophysiology; Glyburide; Humans; Sulfonylurea Compounds; Tolbutamide

1994
Cyclic AMP triggers large [Ca2+]i oscillations in glucose-stimulated beta-cells from ob/ob mice.
    The Journal of biological chemistry, 1994, Jan-14, Volume: 269, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Diazoxide; Glucose; In Vitro Techniques; Ion Channel Gating; Islets of Langerhans; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Obese; Potassium; Potassium Channels

1994
Mechanisms by which glucose can control insulin release independently from its action on adenosine triphosphate-sensitive K+ channels in mouse B cells.
    The Journal of clinical investigation, 1993, Volume: 91, Issue:3

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Diazoxide; Diterpenes; Glucose; Inositol Phosphates; Insulin; Insulin Secretion; Islets of Langerhans; Keto Acids; Kinetics; Male; Mice; Mice, Inbred Strains; Phorbol 12,13-Dibutyrate; Potassium; Potassium Channels; Protein Kinase C; Terpenes; Tetradecanoylphorbol Acetate

1993
Impaired coupling of glucose signal to the exocytotic machinery in diabetic GK rats: a defect ameliorated by cAMP.
    Diabetes, 1996, Volume: 45, Issue:7

    Topics: Animals; Arginine; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Diabetes Mellitus, Type 2; Diazoxide; Exocytosis; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Male; Membrane Potentials; Patch-Clamp Techniques; Rats; Rats, Mutant Strains; Reference Values

1996
cAMP enhances insulin secretion by an action on the ATP-sensitive K+ channel-independent pathway of glucose signaling in rat pancreatic islets.
    Diabetes, 1999, Volume: 48, Issue:5

    Topics: Adenosine Triphosphate; Animals; Calcium; Colforsin; Cyclic AMP; Diazoxide; Enzyme Activation; Glucose; Insulin; Insulin Secretion; Islets of Langerhans; Male; Potassium Channels; Potassium Chloride; Protein Kinase C; Rats; Rats, Wistar; Signal Transduction; Tetradecanoylphorbol Acetate

1999
A(2A) adenosine receptor mediated potassium channel activation in rat epididymal smooth muscle.
    British journal of pharmacology, 2000, Volume: 130, Issue:3

    Topics: Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Diazoxide; Enzyme Activation; Epididymis; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Phenylephrine; Potassium Channels; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Receptors, Purinergic P1; Vasoconstrictor Agents; Vasodilator Agents

2000
Antidiabetic sulfonylurea enhances secretagogue-induced adrenocorticotropin secretion and proopiomelanocortin gene expression in vitro.
    Endocrinology, 2000, Volume: 141, Issue:9

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenocorticotropic Hormone; Animals; Cell Line; Clone Cells; Colforsin; Diazoxide; Diuretics; Gene Expression; Glyburide; Hypoglycemic Agents; Plasmids; Pro-Opiomelanocortin; Promoter Regions, Genetic; Rats; Reverse Transcriptase Polymerase Chain Reaction; Sodium Chloride Symporter Inhibitors; Stimulation, Chemical; Sulfonylurea Compounds

2000
Relief from glucose-induced over-stimulation sensitizes the adenylate cyclase-cAMP system of rat pancreatic islets.
    The Journal of endocrinology, 2000, Volume: 166, Issue:3

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Diazoxide; Dichlororibofuranosylbenzimidazole; Dose-Response Relationship, Drug; Glucose; GTP-Binding Protein alpha Subunits, Gi-Go; Insulin; Insulin Secretion; Islets of Langerhans; Male; Pertussis Toxin; Potassium Channels; Rats; Rats, Sprague-Dawley; Stimulation, Chemical; Thionucleotides; Virulence Factors, Bordetella

2000
Augmentation of basal insulin release from rat islets by preexposure to a high concentration of glucose.
    American journal of physiology. Endocrinology and metabolism, 2000, Volume: 279, Issue:4

    Topics: Adenosine Triphosphate; Adrenergic alpha-Agonists; Animals; Calcium; Cell Membrane Permeability; Cells, Cultured; Clonidine; Colforsin; Diazoxide; Dose-Response Relationship, Drug; Electroporation; Glucose; Guanosine Diphosphate; Insulin; Insulin Secretion; Intracellular Fluid; Islets of Langerhans; Male; Mannoheptulose; Mycophenolic Acid; Oligomycins; Potassium; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate; Thionucleotides

2000
Involvement of K(ATP) channels in diethylstilbestrol-induced relaxation in rat aorta.
    European journal of pharmacology, 2001, Feb-09, Volume: 413, Issue:1

    Topics: Animals; Aorta; Colforsin; Cyclic AMP; Diazoxide; Diethylstilbestrol; Dose-Response Relationship, Drug; Eflornithine; Glyburide; In Vitro Techniques; Indoles; Male; Muscle, Smooth, Vascular; Norepinephrine; Papaverine; Potassium Channels; Rats; Rats, Wistar; Spermine; Tamoxifen; Tetraethylammonium; Vasoconstriction; Vasodilation; Vasodilator Agents

2001
Defective stimulus-secretion coupling in islets of Psammomys obesus, an animal model for type 2 diabetes.
    Diabetes, 2001, Volume: 50, Issue:2

    Topics: Animals; Colforsin; Diabetes Mellitus, Type 2; Diazoxide; Disease Models, Animal; Disease Susceptibility; Gerbillinae; Glucagon; Glucagon-Like Peptide 1; Glucose; Hyperglycemia; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Isoenzymes; Oxidation-Reduction; Peptide Fragments; Protein Kinase C; Protein Precursors; Rats; Rats, Sprague-Dawley; Reference Values; Signal Transduction; Tetradecanoylphorbol Acetate

2001
Triggering of insulin release by a combination of cAMP signal and nutrients: an ATP-sensitive K+ channel-independent phenomenon.
    Diabetes, 2002, Volume: 51 Suppl 1

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine Triphosphate; Animals; Calcium; Colforsin; Cyclic AMP; Diazoxide; Glucagon; Glucagon-Like Peptide 1; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Peptide Fragments; Phosphodiesterase Inhibitors; Potassium Channels; Protein Precursors; Rats; Rats, Wistar; Signal Transduction; Sodium Azide; Vasodilator Agents

2002
Membrane potential dependent modulations of calcium oscillations in insulin-secreting INS-1 cells.
    Cell calcium, 2002, Volume: 31, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Calcium Signaling; Cell Line; Clonidine; Colforsin; Diazoxide; Enzyme Inhibitors; Epinephrine; Fluorescent Dyes; Fura-2; Glucose; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Membrane Potentials; Mice; Patch-Clamp Techniques; Potassium Channels; Prazosin; Receptors, Adrenergic, alpha-2; Thapsigargin; Tolbutamide

2002
Glucagon-like peptide-1 mobilizes intracellular Ca2+ and stimulates mitochondrial ATP synthesis in pancreatic MIN6 beta-cells.
    The Biochemical journal, 2003, Jan-15, Volume: 369, Issue:Pt 2

    Topics: Adenosine Triphosphate; Animals; Calcium; Calcium Signaling; Carbachol; Cell Line; Chelating Agents; Cholinergic Agonists; Colforsin; Cyclic AMP; Diazoxide; Egtazic Acid; Enzyme Inhibitors; Glucagon; Glucagon-Like Peptide 1; Glucose; Homeostasis; Insulin; Insulin Secretion; Islets of Langerhans; Macrocyclic Compounds; Mitochondria; Oxazoles; Peptide Fragments; Protein Precursors; Ryanodine; Ryanodine Receptor Calcium Release Channel; Thionucleotides

2003
Palmitate stimulation of glucagon secretion in mouse pancreatic alpha-cells results from activation of L-type calcium channels and elevation of cytoplasmic calcium.
    Diabetes, 2004, Volume: 53, Issue:11

    Topics: Animals; Colforsin; Diazoxide; Glucagon; Islets of Langerhans; Isradipine; Kinetics; Membrane Potentials; Mice; Mice, Inbred Strains; Palmitic Acid; Potassium; Triazenes

2004
Mitochondrial Ca2+-activated K+ channels in cardiac myocytes: a mechanism of the cardioprotective effect and modulation by protein kinase A.
    Circulation, 2005, Jan-18, Volume: 111, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzimidazoles; Carbocyanines; Cell Death; Colforsin; Cyclic AMP-Dependent Protein Kinases; Decanoic Acids; Diazoxide; Fluorescent Dyes; Guinea Pigs; Heart Ventricles; Heterocyclic Compounds, 3-Ring; Hydroxy Acids; Indoles; Intracellular Membranes; Ion Transport; Membrane Potentials; Mitochondria, Heart; Myocytes, Cardiac; Ouabain; Potassium; Potassium Channels, Calcium-Activated; Second Messenger Systems; Tetradecanoylphorbol Acetate

2005
Glucose triggers protein kinase A-dependent insulin secretion in mouse pancreatic islets through activation of the K+ATP channel-dependent pathway.
    European journal of endocrinology, 2005, Volume: 152, Issue:4

    Topics: Adenosine Triphosphate; Adenylyl Cyclases; Animals; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Diazoxide; Enzyme Activation; Glucose; Insulin; Insulin Secretion; Intracellular Signaling Peptides and Proteins; Islets of Langerhans; Isoquinolines; Male; Mice; Ouabain; Potassium; Potassium Channels; Protein Kinase C; Sulfonamides

2005
Acute and chronic effects of glucose and carbachol on insulin secretion and phospholipase C activation: studies with diazoxide and atropine.
    American journal of physiology. Endocrinology and metabolism, 2006, Volume: 290, Issue:1

    Topics: Animals; Atropine; Carbachol; Colforsin; Diazoxide; Enzyme Activation; Glucose; Hyperglycemia; In Vitro Techniques; Inositol; Inositol Phosphates; Insulin; Insulin Secretion; Islets of Langerhans; Male; Rats; Rats, Sprague-Dawley; Type C Phospholipases

2006
Sildenafil inhibits duodenal contractility via activation of the NO-K+ channel pathway.
    Fundamental & clinical pharmacology, 2008, Volume: 22, Issue:1

    Topics: Animals; Colforsin; Diazoxide; Duodenum; In Vitro Techniques; Male; Muscle Contraction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Nitroprusside; Phosphodiesterase Inhibitors; Piperazines; Potassium Channel Blockers; Potassium Channels; Purines; Rats; Rats, Wistar; Sildenafil Citrate; Sulfones; Vasodilator Agents

2008
Dynamics and Regulation of Insulin Secretion in Pancreatic Islets from Normal Young Children.
    PloS one, 2016, Volume: 11, Issue:11

    Topics: Amino Acids; Calcium Chloride; Child, Preschool; Colforsin; Diazoxide; Female; Glucose; Humans; Infant; Insulin; Insulin Secretion; Islets of Langerhans; Male; Tolbutamide

2016