diazoxide and bms 191095

diazoxide has been researched along with bms 191095 in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (62.50)29.6817
2010's3 (37.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carroll, WA; Coghlan, MJ; Gopalakrishnan, M1
Balsamo, A; Bianucci, AM; Calderone, V; Coi, A; Digiacomo, M; Rapposelli, S; Testai, L1
Grover, GJ; Kolár, F; Koten, L; Neckár, J; Ost'ádal, B; Papousek, F; Szárszoi, O1
Bari, F; Busija, DW; Domoki, F; Grover, G; Katakam, P; Kis, B; Rajapakse, NC1
Ahmad, N; Ashraf, M; Haider, KH; Pasha, Z; Uzun, O; Wang, B; Wang, Y1
Busija, DW; Domoki, F; Gáspár, T; Grovenburg, SM; Institoris, A; Katakam, PV; Katz, PS; Rutkai, I; Snipes, JA; Wappler, EA1
Busija, DW; Gordon, AO; Katakam, PV; Rutkai, I; Sure, VN1
Busija, DW; Dutta, S; Gordon, AO; Grovenburg, SM; Katakam, PV; Peterson, NR; Rutkai, I; Sure, VN1

Reviews

1 review(s) available for diazoxide and bms 191095

ArticleYear
Recent developments in the biology and medicinal chemistry of potassium channel modulators: update from a decade of progress.
    Journal of medicinal chemistry, 2001, May-24, Volume: 44, Issue:11

    Topics: Adenosine Triphosphate; Angina Pectoris; Arrhythmias, Cardiac; Asthma; Calcium; Ion Channel Gating; Myocardial Ischemia; Potassium Channel Blockers; Potassium Channels; Urinary Incontinence

2001

Other Studies

7 other study(ies) available for diazoxide and bms 191095

ArticleYear
Predictive models, based on classification algorithms, for compounds potentially active as mitochondrial ATP-sensitive potassium channel openers.
    Bioorganic & medicinal chemistry, 2009, Aug-01, Volume: 17, Issue:15

    Topics: Algorithms; Benzopyrans; Cardiotonic Agents; KATP Channels; Models, Chemical; Molecular Structure; Quantitative Structure-Activity Relationship; Spiro Compounds

2009
Effects of mitochondrial K(ATP) modulators on cardioprotection induced by chronic high altitude hypoxia in rats.
    Cardiovascular research, 2002, Aug-15, Volume: 55, Issue:3

    Topics: Altitude; Analysis of Variance; Animals; Benzopyrans; Chronic Disease; Decanoic Acids; Diazoxide; Hydroxy Acids; Hypoxia; Imidazoles; Male; Mitochondria, Heart; Models, Animal; Myocardial Contraction; Myocardial Infarction; Myocardium; Perfusion; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Statistics, Nonparametric; Time Factors

2002
Effects of ATP-sensitive potassium channel activators diazoxide and BMS-191095 on membrane potential and reactive oxygen species production in isolated piglet mitochondria.
    Brain research bulletin, 2005, Jul-30, Volume: 66, Issue:2

    Topics: Adenosine Triphosphate; Analysis of Variance; Animals; Animals, Newborn; Benzopyrans; Decanoic Acids; Diazoxide; Dose-Response Relationship, Drug; Drug Interactions; Glyburide; Hydroxy Acids; Imidazoles; Membrane Potentials; Mitochondria; Organometallic Compounds; Potassium Channel Blockers; Potassium Channels; Reactive Oxygen Species; Swine; Time Factors

2005
Cardiac protection by mitoKATP channels is dependent on Akt translocation from cytosol to mitochondria during late preconditioning.
    American journal of physiology. Heart and circulatory physiology, 2006, Volume: 290, Issue:6

    Topics: Androstadienes; Animals; Apoptosis; Benzopyrans; Blotting, Western; Cardiotonic Agents; Cytosol; Diazoxide; Enzyme Inhibitors; Hemodynamics; Imidazoles; In Situ Nick-End Labeling; In Vitro Techniques; Ischemic Preconditioning, Myocardial; L-Lactate Dehydrogenase; Male; Mice; Mice, Inbred C57BL; Mitochondria, Heart; Myocardial Ischemia; Phosphorylation; Potassium Channels; Proto-Oncogene Proteins c-akt; Translocation, Genetic; Vasodilator Agents; Wortmannin

2006
Depolarization of mitochondria in endothelial cells promotes cerebral artery vasodilation by activation of nitric oxide synthase.
    Arteriosclerosis, thrombosis, and vascular biology, 2013, Volume: 33, Issue:4

    Topics: Animals; Benzopyrans; Blotting, Western; Calcium; Cells, Cultured; Cerebral Arteries; Cerebrovascular Circulation; Diazoxide; Dose-Response Relationship, Drug; Electron Spin Resonance Spectroscopy; Endothelial Cells; Enzyme Activation; Enzyme Inhibitors; Free Radical Scavengers; Imidazoles; Membrane Potential, Mitochondrial; Mitochondria; Nitric Oxide; Nitric Oxide Synthase Type III; Phosphatidylinositol 3-Kinase; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Potassium Channel Blockers; Potassium Channels; Proto-Oncogene Proteins c-akt; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Signal Transduction; Vasodilation; Vasodilator Agents

2013
Diversity of mitochondria-dependent dilator mechanisms in vascular smooth muscle of cerebral arteries from normal and insulin-resistant rats.
    American journal of physiology. Heart and circulatory physiology, 2014, Aug-15, Volume: 307, Issue:4

    Topics: Animals; Benzopyrans; Calcium Signaling; Cerebral Arteries; Diazoxide; Imidazoles; Insulin Resistance; Large-Conductance Calcium-Activated Potassium Channels; Membrane Potential, Mitochondrial; Mitochondria, Muscle; Muscle, Smooth, Vascular; Potassium Channels; Rats; Rats, Sprague-Dawley; Rats, Zucker; Reactive Oxygen Species; Vasodilation; Vasodilator Agents

2014
Depolarization of mitochondria in neurons promotes activation of nitric oxide synthase and generation of nitric oxide.
    American journal of physiology. Heart and circulatory physiology, 2016, 05-01, Volume: 310, Issue:9

    Topics: Animals; Benzopyrans; Cells, Cultured; Cerebral Arteries; Diazoxide; Enzyme Activation; Enzyme Inhibitors; Imidazoles; Indazoles; Male; Membrane Potential, Mitochondrial; Mitochondria; Nitrergic Neurons; Nitric Oxide; Nitric Oxide Synthase Type I; Paracrine Communication; Phosphorylation; Potassium Channels; Primary Cell Culture; Rats, Sprague-Dawley; Reactive Oxygen Species; Serine; Signal Transduction; Vasodilation

2016