Page last updated: 2024-09-05

diazipine and dihydropyridines

diazipine has been researched along with dihydropyridines in 14 studies

Compound Research Comparison

Studies
(diazipine)
Trials
(diazipine)
Recent Studies (post-2010)
(diazipine)
Studies
(dihydropyridines)
Trials
(dihydropyridines)
Recent Studies (post-2010) (dihydropyridines)
14055,022529969

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (21.43)18.2507
2000's4 (28.57)29.6817
2010's7 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kanaoka, Y; Nakayama, H; Taki, M1
Catterall, WA; Glossmann, H; Kanaoka, Y; Nakayama, H; Striessnig, J; Taki, M1
Kanaoka, Y; Kuniyasu, A; Nakayama, H; Taki, M1
Kidwai, M; Misra, P; Sapra, P; Saxena, RK; Singh, M1
Caldwell, CG; Chen, P; Donnelly, KL; Grant, SK; Hagmann, WK; Humes, JL; Kelly, TM; Maccoss, M; Pacholok, SG; Shah, SK; Shankaran, K; Wong, KK1
Drewry, DH; Gray, DW; Hoekstra, WJ; Mehbob, A; Stewart, EL; Wiethe, RW1
Arami, M; Gharanjig, K; Limaee, NY; Mahmoodi, NM1
Bradner, JE; Cameron, MJ; Christie, AL; Fedorov, O; Felletar, I; Filippakopoulos, P; French, CA; Heightman, TD; Hickman, TT; Keates, T; Knapp, S; Kung, AL; La Thangue, N; McKeown, MR; Morse, EM; Munro, S; Philpott, M; Picaud, S; Qi, J; Schwartz, B; Shen, Y; Smith, WB; Wang, Y; West, N; Wiest, O1
Chung, TW; Sun, CM; Yellol, GS1
Hada, J; Hada, N; Higuchi, M; Kakiuchi, N; Ohtsuka, I; Sadakane, Y; Sakushima, A1
Liu, JT; Luo, JZ; Miao, JY; Shao, JH; Shen, SL; Zhao, BX1
Banotai, C; Baum, H; Beidler, D; Bove, S; Braden, T; Cornicelli, J; Goodman, A; Gowan, R; Hicks, J; Lightle, S; Lu, XK; Miller, H; Ogden, A; Pandit, J; Plummer, MS; Roark, H; Sadagopan, N; Sanchez, B; Sarver, R; Shahripour, A; Shen, XQ; Skalitzky, DJ; Spessard, C; Stankovic, CJ; Welch, K; Whitehead, C2
Baas, J; Dunbar, M; Rambohul, J; Spurgeon, D; Svendsen, C; van 't Zelfde, M; Vijver, M1

Other Studies

14 other study(ies) available for diazipine and dihydropyridines

ArticleYear
Diazipine, a novel photoaffinity probe for dihydropyridine receptors of calcium channels.
    FEBS letters, 1991, Jun-03, Volume: 283, Issue:2

    Topics: Affinity Labels; Animals; Azides; Azirines; Calcium Channel Blockers; Calcium Channels; Chromatography, Affinity; Dihydropyridines; Kinetics; Molecular Weight; Muscles; Rabbits; Receptors, Nicotinic

1991
Identification of 1,4-dihydropyridine binding regions within the alpha 1 subunit of skeletal muscle Ca2+ channels by photoaffinity labeling with diazipine.
    Proceedings of the National Academy of Sciences of the United States of America, 1991, Oct-15, Volume: 88, Issue:20

    Topics: Affinity Labels; Amino Acid Sequence; Animals; Antibodies; Azirines; Calcium Channels; Cell Membrane; Dihydropyridines; Lipid Bilayers; Macromolecular Substances; Models, Structural; Molecular Sequence Data; Muscles; Peptides; Protein Conformation; Rabbits; Receptors, Nicotinic

1991
Synthesis of diazipine and [3H]diazipine: novel dihydropyridines as photoaffinity probes of calcium channels.
    Chemical & pharmaceutical bulletin, 1991, Volume: 39, Issue:7

    Topics: Affinity Labels; Animals; Azirines; Calcium Channels; Dihydropyridines; In Vitro Techniques; Isotope Labeling; Myocardium; Swine

1991
Microwave assisted solid support synthesis of novel 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazepines as potent antimicrobial agents.
    Bioorganic & medicinal chemistry, 2001, Volume: 9, Issue:2

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Antifungal Agents; Aspergillus; Azirines; Bacillus; Combinatorial Chemistry Techniques; Dihydropyridines; Gram-Negative Bacteria; Microbial Sensitivity Tests; Microwaves; Structure-Activity Relationship; Triazoles

2001
Synthesis of analogs of (1,4)-3- and 5-imino oxazepane, thiazepane, and diazepane as inhibitors of nitric oxide synthases.
    Bioorganic & medicinal chemistry letters, 2004, Dec-06, Volume: 14, Issue:23

    Topics: Azirines; Dihydropyridines; Enzyme Inhibitors; Humans; Nitric Oxide Synthase; Oxazepines; Thiazepines

2004
Array synthesis of progesterone receptor antagonists: 3-aryl-1,2-diazepines.
    Bioorganic & medicinal chemistry letters, 2006, Jul-15, Volume: 16, Issue:14

    Topics: Azepines; Azirines; Binding Sites; Cells, Cultured; Dihydropyridines; Humans; Ligands; Models, Chemical; Receptors, Progesterone

2006
Photocatalytic degradation of agricultural N-heterocyclic organic pollutants using immobilized nanoparticles of titania.
    Journal of hazardous materials, 2007, Jun-25, Volume: 145, Issue:1-2

    Topics: Agrochemicals; Azirines; Catalysis; Dihydropyridines; Imidazoles; Metal Nanoparticles; Neonicotinoids; Nitro Compounds; Photochemistry; Titanium; Ultraviolet Rays; Water Pollutants, Chemical; Water Purification

2007
Selective inhibition of BET bromodomains.
    Nature, 2010, Dec-23, Volume: 468, Issue:7327

    Topics: Amino Acid Sequence; Animals; Azirines; Binding Sites; Carcinoma, Squamous Cell; Cell Cycle Proteins; Cell Differentiation; Cell Line, Tumor; Cell Proliferation; Chromatin; Dihydropyridines; Female; Humans; Mice; Mice, Nude; Models, Molecular; Molecular Sequence Data; Nuclear Proteins; Protein Binding; Protein Structure, Tertiary; Recombinant Proteins; Sequence Alignment; Skin Neoplasms; Stereoisomerism; Transcription Factors

2010
Novel cyclization of bis-Boc-guanidines: expeditive traceless synthesis of 1,3,5-oxadiazinones under microwave conditions.
    Chemical communications (Cambridge, England), 2010, Dec-28, Volume: 46, Issue:48

    Topics: Amines; Azirines; Cyclization; Dihydropyridines; Guanidines; Microwaves; Polyethylene Glycols

2010
The effect of structural differences in the reducing terminus of sugars on the binding affinity of carbohydrates and proteins analyzed using photoaffinity labeling.
    Bioorganic & medicinal chemistry, 2011, Jan-15, Volume: 19, Issue:2

    Topics: Azirines; Carbohydrates; Dihydropyridines; Lectins; Ligands; Microscopy, Atomic Force; Photoaffinity Labels; Protein Binding

2011
Novel chiral ferrocenylpyrazolo[1,5-a][1,4]diazepin-4-one derivatives--synthesis, characterization and inhibition against lung cancer cells.
    European journal of medicinal chemistry, 2013, Volume: 63

    Topics: Apoptosis; Azepines; Azirines; Cell Cycle Checkpoints; Cell Line, Tumor; Cell Proliferation; Crystallography, X-Ray; Dihydropyridines; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Electrochemical Techniques; Ferrous Compounds; Flow Cytometry; Humans; Hydrogen Bonding; Lung Neoplasms; Microscopy, Fluorescence; Models, Chemical; Molecular Structure; Pyrazoles; Stereoisomerism

2013
Discovery of potent, selective, bioavailable phosphodiesterase 2 (PDE2) inhibitors active in an osteoarthritis pain model, part I: transformation of selective pyrazolodiazepinone phosphodiesterase 4 (PDE4) inhibitors into selective PDE2 inhibitors.
    Bioorganic & medicinal chemistry letters, 2013, Jun-01, Volume: 23, Issue:11

    Topics: Animals; Azirines; Binding Sites; Catalytic Domain; Crystallography, X-Ray; Cyclic Nucleotide Phosphodiesterases, Type 2; Cyclic Nucleotide Phosphodiesterases, Type 4; Dihydropyridines; Disease Models, Animal; Drug Evaluation, Preclinical; Osteoarthritis; Phosphodiesterase 4 Inhibitors; Phosphodiesterase Inhibitors; Protein Binding; Structure-Activity Relationship

2013
Discovery of potent selective bioavailable phosphodiesterase 2 (PDE2) inhibitors active in an osteoarthritis pain model. Part II: optimization studies and demonstration of in vivo efficacy.
    Bioorganic & medicinal chemistry letters, 2013, Jun-01, Volume: 23, Issue:11

    Topics: Analgesics; Animals; Azepines; Azirines; Binding Sites; Catalytic Domain; Crystallography, X-Ray; Cyclic Nucleotide Phosphodiesterases, Type 2; Dihydropyridines; Disease Models, Animal; Drug Evaluation, Preclinical; Half-Life; Osteoarthritis; Phosphodiesterase 4 Inhibitors; Phosphodiesterase Inhibitors; Protein Binding; Pyrazoles; Rats; Structure-Activity Relationship

2013
Comparison and evaluation of pesticide monitoring programs using a process-based mixture model.
    Environmental toxicology and chemistry, 2016, Volume: 35, Issue:12

    Topics: Animals; Azirines; Chlorfenvinphos; Daphnia; Dihydropyridines; Environmental Monitoring; Europe; Lethal Dose 50; Limit of Detection; Models, Theoretical; Pesticide Residues; Program Evaluation

2016