diazepam has been researched along with triazolam in 121 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 44 (36.36) | 18.7374 |
1990's | 37 (30.58) | 18.2507 |
2000's | 28 (23.14) | 29.6817 |
2010's | 11 (9.09) | 24.3611 |
2020's | 1 (0.83) | 2.80 |
Authors | Studies |
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Gall, M; Hester, JB; Lahti, RA; Rudzik, AD | 1 |
Chidester, C; Duchamp, DJ; Gall, M; Lahti, RA; Rudzik, AD; Scahill, T | 1 |
Collins, RJ; Gall, M; Kamdar, BV | 1 |
Hester, JB; Von Voigtlander, P | 1 |
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S | 1 |
Topliss, JG; Yoshida, F | 1 |
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY | 1 |
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL | 1 |
Andricopulo, AD; Moda, TL; Montanari, CA | 1 |
Lombardo, F; Obach, RS; Waters, NJ | 1 |
Clayton, T; Cook, J; DeLorey, TM; Furtmüller, R; Halliwell, RF; Harris, D; Huck, S; Sahbaie, P; Sieghart, W | 1 |
Kamide, T; Lee, S; Natsugari, H; Shiro, M; Tabata, H; Takahashi, H | 1 |
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV | 1 |
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W | 1 |
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV | 1 |
García-Mera, X; González-Díaz, H; Prado-Prado, FJ | 1 |
Alelyunas, YW; Bui, K; Empfield, JR; McCarthy, D; Pelosi-Kilby, L; Shen, C; Spreen, RC | 1 |
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR | 1 |
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K | 1 |
Araki, H; Fujiwara, M; Ohmori, K; Ueki, S; Watanabe, S; Yamamoto, T | 1 |
Gomita, H; Gomita, Y; Kataoka, Y; Nakaebisu, H; Ueki, S | 1 |
Nicholson, AN | 1 |
Gottschalk, LA | 1 |
Sellers, EM; Sullivan, JT | 1 |
Facklam, M; Haefely, WE; Schoch, P | 1 |
Bonetti, EP; Facklam, M; Haefely, WE; Jenck, F; Martin, JR; Moreau, JL; Schoch, P | 1 |
Loeffler, PM | 1 |
del Cerro, S; Jung, M; Lynch, G | 1 |
Ator, NA; Griffiths, RR | 2 |
Ishizu, H; Moriya, F | 1 |
Doyle, D; Kragie, L | 1 |
Franklin, SR; Tang, AH | 1 |
Lewis, DC; Sullivan, JT; Swift, RM | 1 |
Bickel, WK; Higgins, ST; Hughes, JR | 1 |
Haefely, WE; Jenck, F; Martin, JR; Moreau, JL; Pieri, L; Schoch, P | 1 |
Betschart, J; Blanchard, JC; Piot, O; Stutzmann, JM | 1 |
Ator, NA; Nierenberg, J | 1 |
Covington, EC; Rapport, DJ | 1 |
Griffiths, RR; Roache, JD | 2 |
Abenstein, JP; Baughman, VL; Becker, GL; Glaser, M; Ryan, CM | 1 |
Dunton, AW; Hendler, J; McGrath, J; Pitman, V; Schwam, E; Siegel, J | 1 |
Griffiths, RR; Lamb, RJ | 1 |
Griffith, JL | 1 |
Fell, D; Hunt, PC; Miller, R; Pinnock, CA; Smith, G | 1 |
Lynn, EJ | 1 |
Castleden, M; Fancourt, G | 1 |
Ellinwood, EH; Heatherly, DG; Nikaido, AM | 1 |
Pawluczyk, S; Schneider, LS; Syapin, PJ | 1 |
Albeck, JH | 1 |
Markin, RS; Murray, WJ | 1 |
Michenfelder, JD; Roald, OK; Stangland, K; Steen, PA | 1 |
Patterson, WM | 1 |
Cagen, LM; Chesney, CM; Pifer, DD | 1 |
Akane, A; Fukui, Y; Hama, K; Maseda, C; Matsubara, K; Tanabe, K | 1 |
Etienne, PE; Ilmoniemi, RJ; McCullough, JR; Sinton, CM | 1 |
Forrest, P; Galletly, DC; Yee, P | 1 |
Fleming, JA; Isomura, T; McMillan, MJ; Rungta, K | 1 |
Kuhn, FJ | 1 |
Stockhaus, K | 1 |
Ator, NA; Griffiths, RR; Lamb, RJ; Roache, JD | 1 |
Brady, JV; Hienz, RD; Lukas, SE | 1 |
Nicholson, AN; Pascoe, PA; Stone, BM | 1 |
Harris, DW; Sethy, VH | 1 |
Ator, NA; Brady, JV; Griffiths, RR; Lamb, RJ; Lukas, SE | 1 |
Swift, CG | 1 |
Gonzalez, JP; McCulloch, AJ; Nicholls, PJ; Sewell, RD; Tekle, A | 1 |
Ochs, HR | 1 |
Cole, NM; Cox, EB; Riefkohl, R | 1 |
Bonetti, EP; Cumin, R; Haefely, WE; Scherschlicht, R | 1 |
Ladewig, D | 1 |
Bickel, WK; Higgins, ST; Hughes, JR; Kamien, JB; Oliveto, AH | 1 |
Blaney, FE; Edge, C; Phippen, RW | 1 |
Zuber, TJ | 1 |
Needleman, SB; Porvaznik, M | 1 |
Gandolfo, G; Gottesmann, C; Scherschlicht, R | 1 |
Auta, J; Costa, E; Giusti, P; Guidotti, A | 1 |
Costa, E; Ducić, I; Puia, G; Vicini, S | 1 |
Kontinen, VK; Maunuksela, EL; Sarvela, J | 1 |
Dionne, RA; Hargreaves, KM; Kaufman, E | 1 |
Herink, J | 1 |
Kiviluoma, KT; Nuutinen, LS; Partanen, AM; Penttilä, HJ | 1 |
Okuyama, T; Tomita, M | 1 |
Ghosh, S; Kant, GJ; Vasilakis, AA; Wylie, RM | 1 |
Misawa, S; Tanaka, E; Terada, M; Wakasugi, C | 1 |
Kulkarni, SK; Reddy, DS | 1 |
Franko, T; Mendelson, WB; Thompson, C | 1 |
Asahi, T; Kuribara, H | 1 |
Bolognesi, R; Conti, M; Manca, C; Tsialtas, D; Vasini, P | 1 |
Dionne, RA; Ehrich, DG; Hutter, JW; Lundgren, JP; Nicoll, BK | 1 |
Kulkarni, SK; Shaji, AV | 1 |
Dionne, R | 1 |
Carter, RB; Gee, KW; Huber, M; Lan, NC; Robledo, S; Suruki, M; Vanover, KE; Wieland, S; Wood, PL | 1 |
Augustijns, P; Kinget, R; Van den Mooter, G | 1 |
Lelas, S; Rowlett, JK; Spealman, RD | 1 |
Cook, JM; Ma, C; Miczek, KA; Rowlett, JK; Tornatzky, W | 1 |
France, CP; McMahon, LR | 1 |
Gomez, TH; Meisch, RA; Roache, JD | 1 |
Feck, AS; Goodchild, JH; Silverman, MD | 1 |
Kishore, K; Saraf, MK; Sharma, A; Singh, M; Thomas, KM | 1 |
Hori, Y; Kudo, K; Kuroki, Y; Yamaguchi, Y; Yashiki, M | 1 |
Nakamura, J; Nakashima, M; Nishida, K; Sasaki, H; Shiota, H; Taniyama, K; Terazono, H | 1 |
Condouris, GA; Gries, DA; Houpt, M; Shey, Z | 1 |
Houston, JB; Jones, HM; Nicholls, G | 1 |
Dickson, SJ; Irving, RC | 1 |
Lu, DP; Lu, WI | 1 |
Galetin, A; Hallifax, D; Houston, JB | 1 |
Kamei, C; Nishino, T; Takechi, K; Takeuchi, T | 1 |
Hirase, M; Ishida, T; Kamei, C | 1 |
Mandrioli, R; Mercolini, L; Raggi, MA | 1 |
Koerner, KR | 1 |
Chronister, CW; Goldberger, BA; Merves, ML | 1 |
Buchbinder, R; Richards, BL; Whittle, SL | 1 |
Buchbinder, R; Richards, BL; van der Heijde, DM; Whittle, SL | 1 |
Ator, NA; Biawat, P; Clayton, T; Cook, JM; Rallapalli, SK; Soto, PL; Weed, MR | 1 |
Darnell, SB; Huizenga, MN; Licata, SC; Rowlett, JK; Rudolph, U; Sadri-Vakili, G; Sangrey, GR; Shinday, NM | 1 |
Arima, Y; Nagao, M; Namera, A; Shiraishi, H; Tajima, T; Torikoshi, A; Toubou, H | 1 |
Ishikawa, A; Kakehashi, H; Kamata, T; Katagi, M; Nakano-Fujii, S; Nitta, A; Sasaki, K; Sato, T; Shima, N; Wada, M | 1 |
10 review(s) available for diazepam and triazolam
Article | Year |
---|---|
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk | 2016 |
Oral benzodiazepines and conscious sedation: a review.
Topics: Administration, Oral; Alprazolam; Ambulatory Surgical Procedures; Anti-Anxiety Agents; Conscious Sedation; Diazepam; Flurazepam; Humans; Lorazepam; Midazolam; Oxazepam; Premedication; Receptors, GABA-A; Temazepam; Triazolam | 1992 |
Flumazenil: US clinical pharmacology studies.
Topics: Adult; Diazepam; Double-Blind Method; Drug Interactions; Female; Flumazenil; Humans; Lorazepam; Male; Memory; Receptors, GABA-A; Triazolam | 1988 |
Withdrawal and detoxification from benzodiazepine dependence: a potential role for clonazepam.
Topics: Adolescent; Adult; Aged; Alprazolam; Anti-Anxiety Agents; Clonazepam; Diazepam; Drug Tolerance; Humans; Male; Middle Aged; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam | 1987 |
Postural instability as a measure of sedative drug response.
Topics: Adult; Aged; Amitriptyline; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Chlormethiazole; Diazepam; Dose-Response Relationship, Drug; Humans; Hypnotics and Sedatives; Nitrazepam; Posture; Temazepam; Time Factors; Triazolam | 1984 |
[Benzodiazepines: significance of kinetics for therapy].
Topics: Age Factors; Aged; Benzodiazepines; Diazepam; Humans; Kinetics; Metabolic Clearance Rate; Nordazepam; Sex Factors; Triazolam | 1983 |
[Practical analysis of toxic substances useful for clinical toxicology--10--benzodiazepine].
Topics: Anti-Anxiety Agents; Benzodiazepines; Diazepam; Gas Chromatography-Mass Spectrometry; Humans; Immunoassay; Toxicology; Triazolam | 2004 |
Benzodiazepine metabolism: an analytical perspective.
Topics: Alprazolam; Animals; Anti-Anxiety Agents; Azepines; Benzodiazepines; Bromazepam; Chromatography, High Pressure Liquid; Diazepam; Humans; Lorazepam; Mass Spectrometry; Midazolam; Triazolam | 2008 |
Muscle relaxants for pain management in rheumatoid arthritis.
Topics: Adult; Anti-Inflammatory Agents, Non-Steroidal; Arthralgia; Arthritis, Rheumatoid; Azabicyclo Compounds; Diazepam; Humans; Indomethacin; Muscle Relaxants, Central; Pain Management; Piperazines; Randomized Controlled Trials as Topic; Sulindac; Triazolam | 2012 |
The efficacy and safety of muscle relaxants in inflammatory arthritis: a Cochrane systematic review.
Topics: Analgesics; Arthritis, Rheumatoid; Diazepam; Drug Therapy, Combination; Humans; Muscle Relaxants, Central; Pain; Pain Management; Randomized Controlled Trials as Topic; Treatment Outcome; Triazolam | 2012 |
14 trial(s) available for diazepam and triazolam
Article | Year |
---|---|
Effects of certain benzodiazepine derivatives on disorganization of thought as manifested in speech.
Topics: Adult; Benzodiazepines; Chlordiazepoxide; Diazepam; Flurazepam; Humans; Lorazepam; Speech; Thinking; Time Factors; Triazolam | 1977 |
The effects of diazepam and triazolam on repeated acquisition and performance of response sequences with an observing response.
Topics: Adult; Arousal; Attention; Diazepam; Double-Blind Method; Female; Humans; Male; Psychomotor Performance; Reinforcement Schedule; Serial Learning; Triazolam | 1991 |
Diazepam and triazolam self-administration in sedative abusers: concordance of subject ratings, performance and drug self-administration.
Topics: Adult; Diazepam; Double-Blind Method; Humans; Hypnotics and Sedatives; Male; Middle Aged; Psychomotor Performance; Reinforcement, Psychology; Self Administration; Substance-Related Disorders; Triazolam | 1989 |
Effectiveness of triazolam, diazepam, and placebo as preanesthetic medications.
Topics: Adult; Anxiety; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Humans; Hypnotics and Sedatives; Male; Mental Recall; Middle Aged; Placebos; Preanesthetic Medication; Random Allocation; Triazolam | 1989 |
Flumazenil: US clinical pharmacology studies.
Topics: Adult; Diazepam; Double-Blind Method; Drug Interactions; Female; Flumazenil; Humans; Lorazepam; Male; Memory; Receptors, GABA-A; Triazolam | 1988 |
A comparison of triazolam and diazepam as premedication agents for minor gynaecological surgery.
Topics: Adult; Anti-Anxiety Agents; Anxiety; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Humans; Middle Aged; Preanesthetic Medication; Pregnancy; Psychomotor Performance; Triazolam | 1985 |
Placebo controlled comparison of midazolam, triazolam and diazepam as oral premedicants for outpatient anaesthesia.
Topics: Administration, Oral; Adult; Anesthesia Recovery Period; Anesthesia, General; Diazepam; Double-Blind Method; Humans; Midazolam; Middle Aged; Pain Measurement; Preanesthetic Medication; Random Allocation; Surveys and Questionnaires; Triazolam; Urologic Diseases | 1987 |
Repeated administration of diazepam and triazolam to subjects with histories of drug abuse.
Topics: Adult; Diazepam; Dose-Response Relationship, Drug; Drug Tolerance; Humans; Male; Psychomotor Performance; Substance-Related Disorders; Triazolam | 1986 |
Efficacy of some benzodiazepines for day-time sleep.
Topics: Adolescent; Adult; Anti-Anxiety Agents; Diazepam; Electroencephalography; Female; Flunitrazepam; Humans; Male; Ovum; Placebos; Sleep; Time Factors; Triazolam | 1980 |
Effects of diazepam and hydromorphone in triazolam-trained humans under a novel-response drug discrimination procedure.
Topics: Adult; Diazepam; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Female; Humans; Hydromorphone; Male; Psychomotor Performance; Triazolam | 1994 |
Premedication with sublingual triazolam compared with oral diazepam.
Topics: Administration, Oral; Administration, Sublingual; Adult; Age Factors; Aged; Anesthesia, Local; Anxiety; Conscious Sedation; Diazepam; Double-Blind Method; Female; Humans; Male; Middle Aged; Ophthalmologic Surgical Procedures; Pilot Projects; Placebos; Preanesthetic Medication; Tablets; Time Factors; Triazolam | 1993 |
Comparison of oral triazolam and nitrous oxide with placebo and intravenous diazepam for outpatient premedication.
Topics: Administration, Oral; Analysis of Variance; Anesthesia Recovery Period; Anesthesia, Dental; Anesthesia, Intravenous; Chi-Square Distribution; Cognition; Conscious Sedation; Dental Anxiety; Diazepam; Dose-Response Relationship, Drug; Humans; Manifest Anxiety Scale; Memory; Nitrous Oxide; Pain Measurement; Preanesthetic Medication; Psychomotor Performance; Regression Analysis; Triazolam | 1993 |
Sublingual triazolam versus peroral diazepam as a premedication for general anaesthesia.
Topics: Administration, Oral; Administration, Sublingual; Adolescent; Adult; Aged; Anesthesia, General; Blood Pressure; Diazepam; Double-Blind Method; Female; Heart Rate; Humans; Hypnotics and Sedatives; Male; Middle Aged; Preanesthetic Medication; Triazolam | 1995 |
Comparison of triazolam, diazepam, and placebo as outpatient oral premedication for endodontic patients.
Topics: Adjuvants, Anesthesia; Anesthesia, Dental; Anti-Anxiety Agents; Chi-Square Distribution; Conscious Sedation; Dental Anxiety; Diazepam; Double-Blind Method; Humans; Hypnotics and Sedatives; Preanesthetic Medication; Root Canal Therapy; Statistics, Nonparametric; Triazolam | 1997 |
98 other study(ies) available for diazepam and triazolam
Article | Year |
---|---|
Synthesis and pharmacology of novel anxiolytic agents derived from 2-[(dialkylamino)methyl-4H-triazol-4-yl] benzophenones and related heterocyclic benzophenones.
Topics: Animals; Anti-Anxiety Agents; Benzophenones; Drug Synergism; Electroshock; Ethanol; Male; Mice; Nicotine; Pentylenetetrazole; Semicarbazides; Strychnine; Triazoles | 1976 |
Novel anxiolytic agents derived from alpha-amino-alpha-phenyl-o-tolyl-4H-triazoles and -imidazoles.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Brain; Crystallography; Hypnotics and Sedatives; Imidazoles; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Mice; Models, Molecular; Molecular Conformation; Muscle Relaxation; Nicotine; Pentylenetetrazole; Rats; Seizures; Semicarbazides; Triazoles | 1978 |
Pharmacology of some metabolites of triazolam, alprazolam, and diazepam prepared by a simple, one-step oxidation of benzodiazepines.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Diazepam; Hydroxylation; Male; Methods; Mice; Oxidation-Reduction; Triazolam; Triazoles | 1978 |
6-Aryl-4H-s-triazolo[4,3-a][1,4]benzodiazepines. Influence of 1-substitution on pharmacological activity.
Topics: Animals; Anti-Anxiety Agents; Apomorphine; Benzodiazepines; Body Temperature; Dextroamphetamine; Male; Mice; Motor Activity; Structure-Activity Relationship | 1979 |
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship | 2000 |
QSAR model for drug human oral bioavailability.
Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship | 2000 |
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution | 2004 |
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration | 2004 |
Hologram QSAR model for the prediction of human oral bioavailability.
Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship | 2007 |
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding | 2008 |
Selective influence on contextual memory: physiochemical properties associated with selectivity of benzodiazepine ligands at GABAA receptors containing the alpha5 subunit.
Topics: Animals; Behavior, Animal; Benzodiazepines; Chemical Phenomena; Chemistry, Physical; Computer Simulation; Databases, Factual; Electrophysiology; Female; Ligands; Male; Memory; Mice; Models, Molecular; Molecular Structure; Oocytes; Protein Isoforms; Protein Subunits; Quantitative Structure-Activity Relationship; Receptors, GABA-A; Structure-Activity Relationship; Xenopus laevis | 2008 |
Axial chirality and affinity at the GABA(A) receptor of pyrimido[1,2-a][1,4]benzodiazepines and related compounds.
Topics: Benzodiazepines; Chromatography, High Pressure Liquid; Crystallography, X-Ray; gamma-Aminobutyric Acid; Humans; Molecular Structure; Protein Binding; Receptors, GABA-A; Stereoisomerism; Structure-Activity Relationship | 2008 |
Physicochemical determinants of human renal clearance.
Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight | 2009 |
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution | 2009 |
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations | 2010 |
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics | 2010 |
Experimental solubility profiling of marketed CNS drugs, exploring solubility limit of CNS discovery candidate.
Topics: Central Nervous System Agents; Drug Evaluation, Preclinical; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Solubility | 2010 |
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection | 2012 |
[Behavioral and EEG effects of triazolam in comparison with those of diazepam (author's transl)].
Topics: Aggression; Agonistic Behavior; Animals; Anti-Anxiety Agents; Anticonvulsants; Diazepam; Electric Stimulation; Electroencephalography; Humans; Limbic System; Male; Mice; Motor Activity; Muscle Relaxants, Central; Olfactory Bulb; Rabbits; Rats; Septal Nuclei; Social Isolation; Triazolam | 1978 |
[Effects of triazolam on conditioned behavior in rats (author's transl)].
Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Conditioning, Psychological; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Hypothalamus; Male; Rats; Self Stimulation; Triazolam | 1978 |
Hypnotics today.
Topics: Aged; Anti-Anxiety Agents; Diazepam; Electroencephalography; Humans; Sleep; Sleep Initiation and Maintenance Disorders; Temazepam; Triazolam | 1979 |
Detoxification for triazolam physical dependence.
Topics: Adult; Alcoholism; Diazepam; Dose-Response Relationship, Drug; Female; Half-Life; Hospitalization; Humans; Male; Middle Aged; Oxazepam; Substance Abuse Treatment Centers; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam | 1992 |
Relationship between benzodiazepine receptor occupancy and potentiation of gamma-aminobutyric acid-stimulated chloride flux in vitro of four ligands of differing intrinsic efficacies.
Topics: Animals; Benzodiazepinones; Cell Membrane; Cerebral Cortex; Chlorides; Diazepam; Drug Synergism; Flumazenil; gamma-Aminobutyric Acid; Ligands; Male; Rats; Receptors, GABA-A; Triazolam | 1992 |
Relationship between benzodiazepine receptor occupancy and functional effects in vivo of four ligands of differing intrinsic efficacies.
Topics: Administration, Oral; Animals; Benzodiazepinones; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Male; Mice; Mice, Inbred DBA; Motor Activity; Receptors, GABA-A; Seizures; Triazolam | 1992 |
Benzodiazepines block long-term potentiation in slices of hippocampus and piriform cortex.
Topics: Analysis of Variance; Animals; Cerebral Cortex; Diazepam; Evoked Potentials; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Male; Organ Specificity; Rats; Rats, Wistar; Time Factors; Triazolam | 1992 |
Oral self-administration of triazolam, diazepam and ethanol in the baboon: drug reinforcement and benzodiazepine physical dependence.
Topics: Animals; Conditioning, Operant; Diazepam; Drinking Behavior; Ethanol; Flumazenil; Food; Half-Life; Male; Papio; Reinforcement Schedule; Reward; Self Administration; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam | 1992 |
Interactive effects of ethanol on benzodiazepines levels in blood and brain of rat.
Topics: Administration, Oral; Animals; Benzodiazepines; Brain Chemistry; Chlordiazepoxide; Diazepam; Drug Interactions; Estazolam; Ethanol; Gas Chromatography-Mass Spectrometry; Male; Rats; Rats, Inbred Strains; Triazolam | 1992 |
Benzodiazepines inhibit temperature-dependent L-[125I]triiodothyronine accumulation into human liver, human neuroblast, and rat pituitary cell lines.
Topics: Adenoma; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Cell Line; Convulsants; Diazepam; Dose-Response Relationship, Drug; Humans; Iodine Radioisotopes; Liver; Lorazepam; Neuroblastoma; Pituitary Neoplasms; Rats; Receptors, Thyroid Hormone; Temperature; Triazolam; Triiodothyronine; Tritium; Tumor Cells, Cultured | 1992 |
The discriminative stimulus effects of diazepam in rats at two training doses.
Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Buspirone; Carbolines; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Flumazenil; Male; Morphine; Pentobarbital; Pyrazoles; Pyridazines; Rats; Rats, Inbred Strains; Triazolam | 1991 |
Benzodiazepine requirements during alcohol withdrawal syndrome: clinical implications of using a standardized withdrawal scale.
Topics: Administration, Oral; Adult; Alcohol Withdrawal Delirium; Anti-Anxiety Agents; Chlordiazepoxide; Diazepam; Hospitalization; Humans; Length of Stay; Lorazepam; Neurologic Examination; Oxazepam; Retrospective Studies; Temazepam; Triazolam | 1991 |
Physical dependence induced in DBA/2J mice by benzodiazepine receptor full agonists, but not by the partial agonist Ro 16-6028.
Topics: Administration, Oral; Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepinones; Diazepam; Drug Implants; Mice; Mice, Inbred DBA; Receptors, GABA-A; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam | 1990 |
Cyclopyrrolones, unlike some benzodiazepines, do not induce physical dependence in mice.
Topics: Animals; Azabicyclo Compounds; Carbolines; Convulsants; Diazepam; Disease Models, Animal; Flunitrazepam; Hypnotics and Sedatives; Lorazepam; Male; Mice; Mice, Inbred Strains; Naphthyridines; Piperazines; Seizures; Structure-Activity Relationship; Substance-Related Disorders; Sulfur Compounds; Triazolam | 1990 |
Drug discrimination in rats successively trained to discriminate diazepam and pentobarbital.
Topics: Animals; Azabicyclo Compounds; Diazepam; Discrimination Learning; Discrimination, Psychological; Generalization, Stimulus; Male; Meprobamate; Pentobarbital; Piperazines; Rats; Rats, Inbred Strains; Triazolam | 1990 |
Differential generalization to pentobarbital in rats trained to discriminate lorazepam, chlordiazepoxide, diazepam, or triazolam.
Topics: Animals; Anti-Anxiety Agents; Chlordiazepoxide; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Generalization, Psychological; Humans; Lorazepam; Pentobarbital; Rats; Triazolam | 1989 |
Motor phenomena in benzodiazepine withdrawal.
Topics: Aged; Alprazolam; Anti-Anxiety Agents; Diagnosis, Differential; Diazepam; Drug Therapy, Combination; Female; Humans; Muscle Rigidity; Sleep Initiation and Maintenance Disorders; Substance Withdrawal Syndrome; Triazolam; Urinary Incontinence | 1989 |
Effects of repeated RO 15-1788 administration in benzodiazepine-dependent baboons.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Convulsants; Diazepam; Drug Tolerance; Flumazenil; Humans; Male; Papio; Posture; Substance Withdrawal Syndrome; Substance-Related Disorders; Tremor; Triazolam; Vomiting | 1985 |
Treatment of episodic behavioral disorders with rapidly absorbed benzodiazepines.
Topics: Administration, Oral; Adult; Aggression; Anger; Anti-Anxiety Agents; Clorazepate Dipotassium; Diazepam; Female; Humans; Kinetics; Male; Mental Disorders; Rage; Seizures; Triazolam | 1985 |
Triazolam addiction.
Topics: Adult; Anti-Anxiety Agents; Diazepam; Humans; Male; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam | 1985 |
The use of benzodiazepines with particular reference to the elderly.
Topics: Aged; Anti-Anxiety Agents; Anxiety; Chlordiazepoxide; Diazepam; Humans; Infusions, Parenteral; Kinetics; Sleep Initiation and Maintenance Disorders; Temazepam; Triazolam | 1986 |
Comparative pharmacodynamics of benzodiazepines.
Topics: Adult; Alprazolam; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Humans; Kinetics; Lorazepam; Male; Psychomotor Performance; Triazolam | 1987 |
Seizures following triazolam withdrawal despite benzodiazepine treatment.
Topics: Anti-Anxiety Agents; Anxiety Disorders; Chlordiazepoxide; Diazepam; Humans; Male; Middle Aged; Receptors, GABA-A; Seizures; Substance Withdrawal Syndrome; Triazolam | 1987 |
Searching for the endogenous benzodiazepine using the graph theoretical approach.
Topics: Anti-Anxiety Agents; Carbolines; Diazepam; Models, Biological; Receptors, GABA-A; Triazolam | 1988 |
The effects of triazolam on cerebral blood flow and metabolism in the dog.
Topics: Animals; Benzodiazepines; Brain; Brain Chemistry; Cerebrovascular Circulation; Diazepam; Dogs; Electroencephalography; Energy Metabolism; Female; Male; Midazolam; Oxygen Consumption; Triazolam | 1986 |
Triazolam withdrawal.
Topics: Alprazolam; Diazepam; Drug Tolerance; Humans; Seizures; Substance Withdrawal Syndrome; Triazolam | 1988 |
Triazolobenzodiazepines competitively inhibit the binding of platelet activating factor (PAF) to human platelets.
Topics: Alprazolam; Binding, Competitive; Blood Platelets; Diazepam; Humans; In Vitro Techniques; Kinetics; Platelet Activating Factor; Platelet Aggregation; Triazolam | 1987 |
[Analysis of etizolam, triazolam, nitrazepam and maprotiline in autopsy materials by high-performance liquid chromatography and gas chromatography].
Topics: Anthracenes; Chromatography, Gas; Chromatography, High Pressure Liquid; Diazepam; Female; Forensic Medicine; Humans; Male; Maprotiline; Middle Aged; Nitrazepam; Triazolam | 1987 |
Modulation of auditory evoked magnetic fields by benzodiazepines.
Topics: Acoustic Stimulation; Auditory Cortex; Benzodiazepines; Diazepam; Humans; Magnetics; Triazolam | 1986 |
Withdrawal regimen for triazolam-dependent patients.
Topics: Diazepam; Flurazepam; Humans; Sleep Initiation and Maintenance Disorders; Substance Withdrawal Syndrome; Triazolam | 1986 |
Effects of brotizolam on the sleep-waking cycle of the cat.
Topics: Animals; Azepines; Cats; Diazepam; Electrodes, Implanted; Electroencephalography; Female; Flurazepam; Hypnotics and Sedatives; Male; Nitrazepam; Sleep; Sleep, REM; Time Factors; Triazolam; Wakefulness | 1986 |
Physical dependence capacity of brotizolam in rhesus monkeys. 2nd communication: primary dependence and barbital substitution.
Topics: Animals; Azepines; Barbital; Barbiturates; Body Weight; Diazepam; Female; Hypnotics and Sedatives; Macaca mulatta; Male; Psychomotor Performance; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam | 1986 |
Abuse liability of triazolam: experimental measurements in animals and humans.
Topics: Animals; Diazepam; Drug Tolerance; Humans; Male; Papio; Pentobarbital; Psychomotor Performance; Self Administration; Substance-Related Disorders; Triazolam | 1987 |
Effects of diazepam and triazolam on auditory and visual thresholds and reaction times in the baboon.
Topics: Animals; Auditory Threshold; Diazepam; Dogs; Male; Papio; Reaction Time; Sensory Thresholds; Time Factors; Triazolam; Vision, Ocular | 1985 |
Determination of biological activity of alprazolam, triazolam and their metabolites.
Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Binding, Competitive; Brain; Diazepam; Flunitrazepam; Kinetics; Male; Membranes; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A; Triazolam | 1982 |
Benzodiazepines: drug discrimination and physiological dependence.
Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Bromazepam; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Generalization, Stimulus; Humans; Lorazepam; Papio; Pentobarbital; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam | 1984 |
Subacute benzodiazepine treatment: observations on behavioural tolerance and withdrawal.
Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Conditioning, Psychological; Diazepam; Drinking Behavior; Drug Tolerance; Humans; Male; Mice; Motor Activity; Oxazepam; Pentylenetetrazole; Rats; Seizures; Substance Withdrawal Syndrome; Triazolam | 1984 |
The effectiveness of benzodiazepines and narcotics in outpatient surgery.
Topics: Ambulatory Surgical Procedures; Analgesics; Anesthesia, Local; Diazepam; Humans; Morphine; Preanesthetic Medication; Promethazine; Prospective Studies; Surgery, Plastic; Triazolam | 1984 |
Use of the specific benzodiazepine antagonist, Ro 15-1788, in studies of physiological dependence on benzodiazepines.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Cats; Diazepam; Female; Flumazenil; Humans; Lorazepam; Male; Mice; Rats; Saimiri; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam | 1982 |
Systematic review of the benzodiazepines. Guidelines for data sheets on diazepam, chlordiazepoxide, medazepam, clorazepate, lorazepam, oxazepam, temazepam, triazolam, nitrazepam, and flurazepam. Committee on the Review of Medicines.
Topics: Benzodiazepines; Chlordiazepoxide; Clorazepate Dipotassium; Diazepam; Flurazepam; Humans; Lorazepam; Medazepam; Nitrazepam; Oxazepam; Safety; Substance Withdrawal Syndrome; Substance-Related Disorders; Temazepam; Triazolam | 1980 |
[Does a rebound insomnia following benzodiazepine administration exist?].
Topics: Benzodiazepines; Diazepam; Flunitrazepam; Flurazepam; Humans; Nitrazepam; Sleep Initiation and Maintenance Disorders; Substance Withdrawal Syndrome; Triazolam | 1980 |
Molecular surface comparison. 2. Similarity of electrostatic vector fields in drug design.
Topics: Anti-Anxiety Agents; Benzamides; Benzazepines; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Diazepam; Drug Design; Electricity; GABA-A Receptor Agonists; Granisetron; Indoles; Isomerism; Molecular Conformation; Ondansetron; Pharmaceutical Preparations; Protein Binding; Pyrazoles; Pyridazines; Receptors, Drug; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Structure-Activity Relationship; Surface Properties; Triazolam; Tropisetron | 1995 |
A pilot project in office-based diagnostic esophagogastroduodenoscopy comparing two nonintravenous methods of sedation and anesthesia.
Topics: Administration, Intranasal; Administration, Oral; Adolescent; Adult; Aged; Aged, 80 and over; Analgesics; Butorphanol; Conscious Sedation; Diazepam; Drug Combinations; Endoscopy, Digestive System; Female; Humans; Injections, Intramuscular; Ketorolac Tromethamine; Male; Middle Aged; Office Visits; Patient Satisfaction; Pilot Projects; Surveys and Questionnaires; Tolmetin; Triazolam; Tromethamine | 1995 |
Identification of parent benzodiazepines by gas chromotography/mass spectroscopy (GC/MS) from urinary extracts treated with B-glucuronidase.
Topics: Alprazolam; Benzodiazepines; Chlordiazepoxide; Clonazepam; Diazepam; Gas Chromatography-Mass Spectrometry; Glucuronidase; Humans; Lorazepam; Oxazepam; Triazolam | 1995 |
Benzodiazepines promote the intermediate stage at the expense of paradoxical sleep in the rat.
Topics: Animals; Anti-Anxiety Agents; Diazepam; Electroencephalography; Epilepsy; Eye Movements; Heart Rate; Male; Midazolam; Rats; Rats, Inbred Strains; Rats, Wistar; Sleep Stages; Sleep, REM; Species Specificity; Theta Rhythm; Triazolam | 1994 |
Imidazenil, a partial positive allosteric modulator of GABAA receptors, exhibits low tolerance and dependence liabilities in the rat.
Topics: Allosteric Regulation; Animals; Anticonvulsants; Benzodiazepines; Benzodiazepinones; Brain; Diazepam; Drug Interactions; Drug Tolerance; GABA Modulators; Imidazoles; Male; Rats; Rats, Sprague-Dawley; Substance-Related Disorders; Triazolam | 1994 |
Triazolam is more efficacious than diazepam in a broad spectrum of recombinant GABAA receptors.
Topics: Animals; Cells, Cultured; Cerebral Cortex; Chloride Channels; Chlorides; Diazepam; Humans; Kidney; Membrane Proteins; Neurons; Rats; Receptors, GABA-A; Recombinant Proteins; Transfection; Triazolam | 1993 |
Convulsive properties of N-(3,5-dimethoxy-4-propoxyphenyl-ethyl) aziridine and their influencing by diazepam and triazolam.
Topics: Animals; Anticonvulsants; Aziridines; Diazepam; Male; Rats; Rats, Wistar; Seizures; Triazolam | 1995 |
Application of capillary electrophoresis to the simultaneous screening and quantitation of benzodiazepines.
Topics: Autoanalysis; Benzodiazepines; Bromazepam; Buffers; Diazepam; Electrophoresis, Capillary; Estazolam; Flurazepam; Humans; Hydrogen-Ion Concentration; Nitrazepam; Reproducibility of Results; Sensitivity and Specificity; Triazolam | 1996 |
Effects of triazolam and diazepam on learning and memory as assessed using a water maze.
Topics: Animals; Diazepam; GABA Modulators; Male; Maze Learning; Memory; Rats; Rats, Sprague-Dawley; Triazolam | 1996 |
Simultaneous determination of twelve benzodiazepines in human serum using a new reversed-phase chromatographic column on a 2-microns porous microspherical silica gel.
Topics: Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Bromazepam; Chlordiazepoxide; Chromatography, High Pressure Liquid; Clonazepam; Diazepam; Estazolam; Humans; Linear Models; Lorazepam; Microspheres; Nitrazepam; Reproducibility of Results; Silicon Dioxide; Spectrophotometry, Ultraviolet; Triazolam | 1996 |
Role of GABA-A and mitochondrial diazepam binding inhibitor receptors in the anti-stress activity of neurosteroids in mice.
Topics: Analysis of Variance; Animals; Ascorbic Acid; Behavior, Animal; Binding Sites; Cerebellum; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Antagonists; GABA Modulators; Isoquinolines; Male; Mice; Mitochondria; Motor Activity; Pain Measurement; Picrotoxin; Progesterone; Receptors, GABA-A; RNA; Stress, Psychological; Triazolam | 1996 |
Adverse reactions to sedative/hypnotics: three years' experience.
Topics: Accidental Falls; Adult; Aged; Diazepam; Female; Hospital Departments; Hospitalization; Hospitals, Teaching; Humans; Hypnotics and Sedatives; Lorazepam; Male; Middle Aged; Patient Care Team; Psychotropic Drugs; Triazolam | 1996 |
Assessment of the anxiolytic and amnesic effects of three benzodiazepines, diazepam, alprazolam and triazolam, by conflict and non-matching to sample tests in mice.
Topics: Alprazolam; Animals; Anti-Anxiety Agents; Conflict, Psychological; Diazepam; Male; Maze Learning; Memory; Mice; Triazolam | 1997 |
Abnormal ventricular repolarization mimicking myocardial infarction after heterocyclic antidepressant overdose.
Topics: Adult; Amitriptyline; Anti-Anxiety Agents; Antidepressive Agents; Antidepressive Agents, Tricyclic; Antipsychotic Agents; Benzodiazepines; Bundle-Branch Block; Diagnosis, Differential; Diazepam; Electrocardiography; Female; Heart Ventricles; Humans; Hypnotics and Sedatives; Long QT Syndrome; Maprotiline; Myocardial Infarction; Nordazepam; Perphenazine; Triazolam | 1997 |
Evidence of GABAergic modulation in melatonin-induced short-term memory deficits and food consumption.
Topics: Animals; Antioxidants; Diazepam; Eating; Female; Flumazenil; GABA Modulators; Latency Period, Psychological; Male; Maze Learning; Melatonin; Memory Disorders; Memory, Short-Term; Mice; Muscarinic Antagonists; Rats; Rats, Wistar; Receptors, GABA; Scopolamine; Triazolam | 1998 |
Oral sedation.
Topics: Administration, Oral; Algorithms; Anesthesia, Dental; Anti-Anxiety Agents; Chloral Hydrate; Conscious Sedation; Dental Anxiety; Diazepam; Histamine H1 Antagonists; Humans; Hydroxyzine; Hypnotics and Sedatives; Midazolam; Mutagens; Premedication; Triazolam | 1998 |
Positive allosteric modulators of the GABA(A) receptor: differential interaction of benzodiazepines and neuroactive steroids with ethanol.
Topics: Allosteric Regulation; Animals; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; GABA-A Receptor Agonists; Male; Mice; Motor Activity; Neuroprotective Agents; Pregnanolone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sleep; Triazolam | 1999 |
Stability prediction of amorphous benzodiazepines by calculation of the mean relaxation time constant using the Williams-Watts decay function.
Topics: Benzodiazepines; Calorimetry, Differential Scanning; Chemical Phenomena; Chemistry, Physical; Crystallization; Diazepam; Drug Stability; Temazepam; Thermodynamics; Time Factors; Triazolam | 1999 |
Transduction of the discriminative stimulus effects of zolpidem by GABA(A)/alpha1 receptors.
Topics: Acetamides; Animals; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; Male; Protein Subunits; Pyridines; Pyrimidines; Reinforcement Schedule; Saimiri; Triazolam; Zolpidem | 2000 |
Zolpidem, triazolam, and diazepam decrease distress vocalizations in mouse pups: differential antagonism by flumazenil and beta-Carboline-3-carboxylate-t-butyl ester (beta-CCt).
Topics: Animals; Animals, Newborn; Anti-Anxiety Agents; Body Temperature; Carbolines; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Antagonists; Mice; Pyridines; Receptors, GABA-A; Triazolam; Vocalization, Animal; Zolpidem | 2001 |
Daily treatment with diazepam differentially modifies sensitivity to the effects of gamma-aminobutyric acid(A) modulators on schedule-controlled responding in rhesus monkeys.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Electroshock; Food; GABA Agonists; GABA Antagonists; GABA Modulators; Macaca mulatta; Male; Pentobarbital; Pregnanolone; Receptors, GABA-A; Reinforcement Schedule; Triazolam | 2002 |
Orally delivered alprazolam, diazepam, and triazolam as reinforcers in rhesus monkeys.
Topics: Administration, Oral; Alprazolam; Animals; Anti-Anxiety Agents; Diazepam; Macaca mulatta; Male; Reinforcement, Psychology; Self Administration; Triazolam | 2002 |
Anxiolysis in general dental practice.
Topics: Acetamides; Adjuvants, Anesthesia; Anesthesia, Dental; Anesthetics, Inhalation; Anti-Anxiety Agents; Clinical Protocols; Conscious Sedation; Dental Anxiety; Diazepam; GABA Modulators; General Practice, Dental; Humans; Hydroxyzine; Hypnotics and Sedatives; Lorazepam; Midazolam; Nitrous Oxide; Pyrimidines; Triazolam | 2003 |
Role of platelet activating factor in triazolobenzodiazepines-induced retrograde amnesia.
Topics: 1-Alkyl-2-acetylglycerophosphocholine Esterase; Amnesia, Anterograde; Amnesia, Retrograde; Animals; Anti-Anxiety Agents; Azepines; Diazepam; Diterpenes; Escape Reaction; Female; Flumazenil; Ginkgolides; Lactones; Learning; Male; Mice; Phospholipases A; Platelet Activating Factor; Platelet Membrane Glycoproteins; Reaction Time; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Receptors, GABA-A; Retention, Psychology; Triazolam | 2003 |
Postmortem changes in tissue concentrations of triazolam and diazepam in rats.
Topics: Animals; Anti-Anxiety Agents; Diazepam; Forensic Medicine; Gas Chromatography-Mass Spectrometry; Gastrointestinal Contents; Intestine, Small; Kidney; Liver; Lung; Male; Muscle, Skeletal; Myocardium; Postmortem Changes; Rats; Rats, Wistar; Tissue Distribution; Triazolam | 2004 |
New drugs for local anesthesia and oral sedation.
Topics: Administration, Oral; Anesthetics, Combined; Anesthetics, Local; Anti-Anxiety Agents; Carticaine; Diazepam; Drug Combinations; Humans; Lidocaine; Lidocaine, Prilocaine Drug Combination; Lorazepam; Prilocaine; Triazolam | 2004 |
Anxiolytic-like action in mice treated with nitrous oxide and oral triazolam or diazepam.
Topics: Administration, Oral; Animals; Anti-Anxiety Agents; Diazepam; Male; Mice; Nitrous Oxide; Triazolam | 2005 |
Impact of end-product inhibition on the determination of in vitro metabolic clearance.
Topics: Alamethicin; Animals; Biotransformation; Diazepam; Hepatocytes; Kinetics; Metabolic Clearance Rate; Microsomes, Liver; Models, Biological; Phenytoin; Rats; Triazolam | 2005 |
The detection of sedatives in hair and nail samples using tandem LC-MS-MS.
Topics: Adult; Aged; Aged, 80 and over; Alprazolam; Azabicyclo Compounds; Benzodiazepines; Chromatography, Liquid; Clobazam; Clonazepam; Diazepam; Female; Forensic Pathology; Hair; Humans; Hypnotics and Sedatives; Male; Mass Spectrometry; Midazolam; Middle Aged; Nails; Oxazepam; Piperazines; Predictive Value of Tests; Rape; Temazepam; Triazolam | 2007 |
Practical oral sedation in dentistry. Part II--Clinical application of various oral sedatives and discussion.
Topics: Administration, Oral; Adult; Age Factors; Aged; Aged, 80 and over; Anesthesia, Dental; Child; Child, Preschool; Chloral Hydrate; Conscious Sedation; Diazepam; Fentanyl; Humans; Hypnotics and Sedatives; Meperidine; Midazolam; Nausea; Promethazine; Triazolam; Vomiting | 2006 |
Prediction of metabolic clearance using fresh human hepatocytes: comparison with cryopreserved hepatocytes and hepatic microsomes for five benzodiazepines.
Topics: Alprazolam; Benzodiazepines; Cell Survival; Cells, Cultured; Cryopreservation; Cytochrome P-450 CYP3A; Diazepam; Flunitrazepam; Hepatocytes; Humans; Metabolic Clearance Rate; Microsomes, Liver; Midazolam; Substrate Specificity; Triazolam | 2008 |
Evaluation of anxiolytic-like effects of some short-acting benzodiazepine hypnotics in mice.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Azepines; Benzodiazepines; Diazepam; Hypnotics and Sedatives; Lorazepam; Male; Maze Learning; Mice; Mice, Inbred ICR; Motor Activity; Triazolam | 2008 |
Rebound insomnia induced by abrupt withdrawal of hypnotics in sleep-disturbed rats.
Topics: Animals; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Hypnotics and Sedatives; Isoindoles; Male; Piperazines; Pyrimidines; Rats; Rats, Wistar; Sleep Initiation and Maintenance Disorders; Sleep Stages; Time Factors; Triazolam; Wakefulness | 2008 |
Oral sedation for the apprehensive dental patient.
Topics: Administration, Oral; Adolescent; Anti-Anxiety Agents; Biological Availability; Conscious Sedation; Dental Anxiety; Diazepam; Female; Humans; Male; Safety; Therapeutic Equivalency; Triazolam; Young Adult | 2000 |
Quantitation of benzodiazepines in blood and urine using gas chromatography-mass spectrometry (GC-MS).
Topics: Alprazolam; Benzodiazepines; Diazepam; Gas Chromatography-Mass Spectrometry; Humans; Lorazepam; Nordazepam; Oxazepam; Solid Phase Extraction; Triazolam | 2010 |
Allosteric modulation of GABA(A) receptor subtypes:effects on visual recognition and visuospatial working memory in rhesus monkeys [corrected].
Topics: Acetamides; Allosteric Regulation; Animals; Benzodiazepines; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Imidazoles; Macaca mulatta; Male; Memory, Short-Term; Pyridazines; Pyridines; Pyrimidines; Receptors, GABA-A; Recognition, Psychology; Triazolam; Triazoles; Zolpidem | 2013 |
Alterations in brain-derived neurotrophic factor in the mouse hippocampus following acute but not repeated benzodiazepine treatment.
Topics: Analysis of Variance; Animals; Benzodiazepines; Blotting, Western; Brain-Derived Neurotrophic Factor; Chromatin Immunoprecipitation; Cyclic AMP Response Element-Binding Protein; Diazepam; Enzyme-Linked Immunosorbent Assay; Gene Expression Regulation; Genes, Immediate-Early; Hippocampus; Male; Mice; Mice, Inbred C57BL; Proto-Oncogene Proteins c-fos; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; Triazolam; Zolpidem | 2013 |
[Cross-reactivity of Instant-View M-1 for detection of benzodiazepine-related drugs and their metabolites in urine].
Topics: Alprazolam; Benzodiazepines; Biomarkers; Cross Reactions; Diazepam; Humans; Immunoassay; Nitrazepam; Reagent Kits, Diagnostic; Sensitivity and Specificity; Structure-Activity Relationship; Substance Abuse Detection; Triazolam | 2014 |
Incorporation of five common hypnotics into hair after a single dose and application to a forensic case of drug facilitated crimes.
Topics: Adult; Asian People; Chromatography, Liquid; Crime; Diazepam; Female; Flunitrazepam; Forensic Toxicology; Hair; Humans; Hypnotics and Sedatives; Male; Mass Spectrometry; Nitrazepam; Substance Abuse Detection; Triazolam; Zolpidem | 2021 |