diazepam and triazolam

diazepam has been researched along with triazolam in 121 studies

Research

Studies (121)

TimeframeStudies, this research(%)All Research%
pre-199044 (36.36)18.7374
1990's37 (30.58)18.2507
2000's28 (23.14)29.6817
2010's11 (9.09)24.3611
2020's1 (0.83)2.80

Authors

AuthorsStudies
Gall, M; Hester, JB; Lahti, RA; Rudzik, AD1
Chidester, C; Duchamp, DJ; Gall, M; Lahti, RA; Rudzik, AD; Scahill, T1
Collins, RJ; Gall, M; Kamdar, BV1
Hester, JB; Von Voigtlander, P1
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S1
Topliss, JG; Yoshida, F1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Andricopulo, AD; Moda, TL; Montanari, CA1
Lombardo, F; Obach, RS; Waters, NJ1
Clayton, T; Cook, J; DeLorey, TM; Furtmüller, R; Halliwell, RF; Harris, D; Huck, S; Sahbaie, P; Sieghart, W1
Kamide, T; Lee, S; Natsugari, H; Shiro, M; Tabata, H; Takahashi, H1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Alelyunas, YW; Bui, K; Empfield, JR; McCarthy, D; Pelosi-Kilby, L; Shen, C; Spreen, RC1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Araki, H; Fujiwara, M; Ohmori, K; Ueki, S; Watanabe, S; Yamamoto, T1
Gomita, H; Gomita, Y; Kataoka, Y; Nakaebisu, H; Ueki, S1
Nicholson, AN1
Gottschalk, LA1
Sellers, EM; Sullivan, JT1
Facklam, M; Haefely, WE; Schoch, P1
Bonetti, EP; Facklam, M; Haefely, WE; Jenck, F; Martin, JR; Moreau, JL; Schoch, P1
Loeffler, PM1
del Cerro, S; Jung, M; Lynch, G1
Ator, NA; Griffiths, RR2
Ishizu, H; Moriya, F1
Doyle, D; Kragie, L1
Franklin, SR; Tang, AH1
Lewis, DC; Sullivan, JT; Swift, RM1
Bickel, WK; Higgins, ST; Hughes, JR1
Haefely, WE; Jenck, F; Martin, JR; Moreau, JL; Pieri, L; Schoch, P1
Betschart, J; Blanchard, JC; Piot, O; Stutzmann, JM1
Ator, NA; Nierenberg, J1
Covington, EC; Rapport, DJ1
Griffiths, RR; Roache, JD2
Abenstein, JP; Baughman, VL; Becker, GL; Glaser, M; Ryan, CM1
Dunton, AW; Hendler, J; McGrath, J; Pitman, V; Schwam, E; Siegel, J1
Griffiths, RR; Lamb, RJ1
Griffith, JL1
Fell, D; Hunt, PC; Miller, R; Pinnock, CA; Smith, G1
Lynn, EJ1
Castleden, M; Fancourt, G1
Ellinwood, EH; Heatherly, DG; Nikaido, AM1
Pawluczyk, S; Schneider, LS; Syapin, PJ1
Albeck, JH1
Markin, RS; Murray, WJ1
Michenfelder, JD; Roald, OK; Stangland, K; Steen, PA1
Patterson, WM1
Cagen, LM; Chesney, CM; Pifer, DD1
Akane, A; Fukui, Y; Hama, K; Maseda, C; Matsubara, K; Tanabe, K1
Etienne, PE; Ilmoniemi, RJ; McCullough, JR; Sinton, CM1
Forrest, P; Galletly, DC; Yee, P1
Fleming, JA; Isomura, T; McMillan, MJ; Rungta, K1
Kuhn, FJ1
Stockhaus, K1
Ator, NA; Griffiths, RR; Lamb, RJ; Roache, JD1
Brady, JV; Hienz, RD; Lukas, SE1
Nicholson, AN; Pascoe, PA; Stone, BM1
Harris, DW; Sethy, VH1
Ator, NA; Brady, JV; Griffiths, RR; Lamb, RJ; Lukas, SE1
Swift, CG1
Gonzalez, JP; McCulloch, AJ; Nicholls, PJ; Sewell, RD; Tekle, A1
Ochs, HR1
Cole, NM; Cox, EB; Riefkohl, R1
Bonetti, EP; Cumin, R; Haefely, WE; Scherschlicht, R1
Ladewig, D1
Bickel, WK; Higgins, ST; Hughes, JR; Kamien, JB; Oliveto, AH1
Blaney, FE; Edge, C; Phippen, RW1
Zuber, TJ1
Needleman, SB; Porvaznik, M1
Gandolfo, G; Gottesmann, C; Scherschlicht, R1
Auta, J; Costa, E; Giusti, P; Guidotti, A1
Costa, E; Ducić, I; Puia, G; Vicini, S1
Kontinen, VK; Maunuksela, EL; Sarvela, J1
Dionne, RA; Hargreaves, KM; Kaufman, E1
Herink, J1
Kiviluoma, KT; Nuutinen, LS; Partanen, AM; Penttilä, HJ1
Okuyama, T; Tomita, M1
Ghosh, S; Kant, GJ; Vasilakis, AA; Wylie, RM1
Misawa, S; Tanaka, E; Terada, M; Wakasugi, C1
Kulkarni, SK; Reddy, DS1
Franko, T; Mendelson, WB; Thompson, C1
Asahi, T; Kuribara, H1
Bolognesi, R; Conti, M; Manca, C; Tsialtas, D; Vasini, P1
Dionne, RA; Ehrich, DG; Hutter, JW; Lundgren, JP; Nicoll, BK1
Kulkarni, SK; Shaji, AV1
Dionne, R1
Carter, RB; Gee, KW; Huber, M; Lan, NC; Robledo, S; Suruki, M; Vanover, KE; Wieland, S; Wood, PL1
Augustijns, P; Kinget, R; Van den Mooter, G1
Lelas, S; Rowlett, JK; Spealman, RD1
Cook, JM; Ma, C; Miczek, KA; Rowlett, JK; Tornatzky, W1
France, CP; McMahon, LR1
Gomez, TH; Meisch, RA; Roache, JD1
Feck, AS; Goodchild, JH; Silverman, MD1
Kishore, K; Saraf, MK; Sharma, A; Singh, M; Thomas, KM1
Hori, Y; Kudo, K; Kuroki, Y; Yamaguchi, Y; Yashiki, M1
Nakamura, J; Nakashima, M; Nishida, K; Sasaki, H; Shiota, H; Taniyama, K; Terazono, H1
Condouris, GA; Gries, DA; Houpt, M; Shey, Z1
Houston, JB; Jones, HM; Nicholls, G1
Dickson, SJ; Irving, RC1
Lu, DP; Lu, WI1
Galetin, A; Hallifax, D; Houston, JB1
Kamei, C; Nishino, T; Takechi, K; Takeuchi, T1
Hirase, M; Ishida, T; Kamei, C1
Mandrioli, R; Mercolini, L; Raggi, MA1
Koerner, KR1
Chronister, CW; Goldberger, BA; Merves, ML1
Buchbinder, R; Richards, BL; Whittle, SL1
Buchbinder, R; Richards, BL; van der Heijde, DM; Whittle, SL1
Ator, NA; Biawat, P; Clayton, T; Cook, JM; Rallapalli, SK; Soto, PL; Weed, MR1
Darnell, SB; Huizenga, MN; Licata, SC; Rowlett, JK; Rudolph, U; Sadri-Vakili, G; Sangrey, GR; Shinday, NM1
Arima, Y; Nagao, M; Namera, A; Shiraishi, H; Tajima, T; Torikoshi, A; Toubou, H1
Ishikawa, A; Kakehashi, H; Kamata, T; Katagi, M; Nakano-Fujii, S; Nitta, A; Sasaki, K; Sato, T; Shima, N; Wada, M1

Reviews

10 review(s) available for diazepam and triazolam

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Oral benzodiazepines and conscious sedation: a review.
    Journal of oral and maxillofacial surgery : official journal of the American Association of Oral and Maxillofacial Surgeons, 1992, Volume: 50, Issue:9

    Topics: Administration, Oral; Alprazolam; Ambulatory Surgical Procedures; Anti-Anxiety Agents; Conscious Sedation; Diazepam; Flurazepam; Humans; Lorazepam; Midazolam; Oxazepam; Premedication; Receptors, GABA-A; Temazepam; Triazolam

1992
Flumazenil: US clinical pharmacology studies.
    European journal of anaesthesiology. Supplement, 1988, Volume: 2

    Topics: Adult; Diazepam; Double-Blind Method; Drug Interactions; Female; Flumazenil; Humans; Lorazepam; Male; Memory; Receptors, GABA-A; Triazolam

1988
Withdrawal and detoxification from benzodiazepine dependence: a potential role for clonazepam.
    The Journal of clinical psychiatry, 1987, Volume: 48 Suppl

    Topics: Adolescent; Adult; Aged; Alprazolam; Anti-Anxiety Agents; Clonazepam; Diazepam; Drug Tolerance; Humans; Male; Middle Aged; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam

1987
Postural instability as a measure of sedative drug response.
    British journal of clinical pharmacology, 1984, Volume: 18 Suppl 1

    Topics: Adult; Aged; Amitriptyline; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Chlormethiazole; Diazepam; Dose-Response Relationship, Drug; Humans; Hypnotics and Sedatives; Nitrazepam; Posture; Temazepam; Time Factors; Triazolam

1984
[Benzodiazepines: significance of kinetics for therapy].
    Klinische Wochenschrift, 1983, Mar-01, Volume: 61, Issue:5

    Topics: Age Factors; Aged; Benzodiazepines; Diazepam; Humans; Kinetics; Metabolic Clearance Rate; Nordazepam; Sex Factors; Triazolam

1983
[Practical analysis of toxic substances useful for clinical toxicology--10--benzodiazepine].
    Chudoku kenkyu : Chudoku Kenkyukai jun kikanshi = The Japanese journal of toxicology, 2004, Volume: 17, Issue:2

    Topics: Anti-Anxiety Agents; Benzodiazepines; Diazepam; Gas Chromatography-Mass Spectrometry; Humans; Immunoassay; Toxicology; Triazolam

2004
Benzodiazepine metabolism: an analytical perspective.
    Current drug metabolism, 2008, Volume: 9, Issue:8

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Azepines; Benzodiazepines; Bromazepam; Chromatography, High Pressure Liquid; Diazepam; Humans; Lorazepam; Mass Spectrometry; Midazolam; Triazolam

2008
Muscle relaxants for pain management in rheumatoid arthritis.
    The Cochrane database of systematic reviews, 2012, Jan-18, Volume: 1

    Topics: Adult; Anti-Inflammatory Agents, Non-Steroidal; Arthralgia; Arthritis, Rheumatoid; Azabicyclo Compounds; Diazepam; Humans; Indomethacin; Muscle Relaxants, Central; Pain Management; Piperazines; Randomized Controlled Trials as Topic; Sulindac; Triazolam

2012
The efficacy and safety of muscle relaxants in inflammatory arthritis: a Cochrane systematic review.
    The Journal of rheumatology. Supplement, 2012, Volume: 90

    Topics: Analgesics; Arthritis, Rheumatoid; Diazepam; Drug Therapy, Combination; Humans; Muscle Relaxants, Central; Pain; Pain Management; Randomized Controlled Trials as Topic; Treatment Outcome; Triazolam

2012

Trials

14 trial(s) available for diazepam and triazolam

ArticleYear
Effects of certain benzodiazepine derivatives on disorganization of thought as manifested in speech.
    Current therapeutic research, clinical and experimental, 1977, Volume: 21, Issue:2

    Topics: Adult; Benzodiazepines; Chlordiazepoxide; Diazepam; Flurazepam; Humans; Lorazepam; Speech; Thinking; Time Factors; Triazolam

1977
The effects of diazepam and triazolam on repeated acquisition and performance of response sequences with an observing response.
    Journal of the experimental analysis of behavior, 1991, Volume: 56, Issue:2

    Topics: Adult; Arousal; Attention; Diazepam; Double-Blind Method; Female; Humans; Male; Psychomotor Performance; Reinforcement Schedule; Serial Learning; Triazolam

1991
Diazepam and triazolam self-administration in sedative abusers: concordance of subject ratings, performance and drug self-administration.
    Psychopharmacology, 1989, Volume: 99, Issue:3

    Topics: Adult; Diazepam; Double-Blind Method; Humans; Hypnotics and Sedatives; Male; Middle Aged; Psychomotor Performance; Reinforcement, Psychology; Self Administration; Substance-Related Disorders; Triazolam

1989
Effectiveness of triazolam, diazepam, and placebo as preanesthetic medications.
    Anesthesiology, 1989, Volume: 71, Issue:2

    Topics: Adult; Anxiety; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Humans; Hypnotics and Sedatives; Male; Mental Recall; Middle Aged; Placebos; Preanesthetic Medication; Random Allocation; Triazolam

1989
Flumazenil: US clinical pharmacology studies.
    European journal of anaesthesiology. Supplement, 1988, Volume: 2

    Topics: Adult; Diazepam; Double-Blind Method; Drug Interactions; Female; Flumazenil; Humans; Lorazepam; Male; Memory; Receptors, GABA-A; Triazolam

1988
A comparison of triazolam and diazepam as premedication agents for minor gynaecological surgery.
    Anaesthesia, 1985, Volume: 40, Issue:4

    Topics: Adult; Anti-Anxiety Agents; Anxiety; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Humans; Middle Aged; Preanesthetic Medication; Pregnancy; Psychomotor Performance; Triazolam

1985
Placebo controlled comparison of midazolam, triazolam and diazepam as oral premedicants for outpatient anaesthesia.
    Anaesthesia and intensive care, 1987, Volume: 15, Issue:3

    Topics: Administration, Oral; Adult; Anesthesia Recovery Period; Anesthesia, General; Diazepam; Double-Blind Method; Humans; Midazolam; Middle Aged; Pain Measurement; Preanesthetic Medication; Random Allocation; Surveys and Questionnaires; Triazolam; Urologic Diseases

1987
Repeated administration of diazepam and triazolam to subjects with histories of drug abuse.
    Drug and alcohol dependence, 1986, Volume: 17, Issue:1

    Topics: Adult; Diazepam; Dose-Response Relationship, Drug; Drug Tolerance; Humans; Male; Psychomotor Performance; Substance-Related Disorders; Triazolam

1986
Efficacy of some benzodiazepines for day-time sleep.
    British journal of clinical pharmacology, 1980, Volume: 10, Issue:5

    Topics: Adolescent; Adult; Anti-Anxiety Agents; Diazepam; Electroencephalography; Female; Flunitrazepam; Humans; Male; Ovum; Placebos; Sleep; Time Factors; Triazolam

1980
Effects of diazepam and hydromorphone in triazolam-trained humans under a novel-response drug discrimination procedure.
    Psychopharmacology, 1994, Volume: 114, Issue:3

    Topics: Adult; Diazepam; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Female; Humans; Hydromorphone; Male; Psychomotor Performance; Triazolam

1994
Premedication with sublingual triazolam compared with oral diazepam.
    Canadian journal of anaesthesia = Journal canadien d'anesthesie, 1993, Volume: 40, Issue:9

    Topics: Administration, Oral; Administration, Sublingual; Adult; Age Factors; Aged; Anesthesia, Local; Anxiety; Conscious Sedation; Diazepam; Double-Blind Method; Female; Humans; Male; Middle Aged; Ophthalmologic Surgical Procedures; Pilot Projects; Placebos; Preanesthetic Medication; Tablets; Time Factors; Triazolam

1993
Comparison of oral triazolam and nitrous oxide with placebo and intravenous diazepam for outpatient premedication.
    Oral surgery, oral medicine, and oral pathology, 1993, Volume: 75, Issue:2

    Topics: Administration, Oral; Analysis of Variance; Anesthesia Recovery Period; Anesthesia, Dental; Anesthesia, Intravenous; Chi-Square Distribution; Cognition; Conscious Sedation; Dental Anxiety; Diazepam; Dose-Response Relationship, Drug; Humans; Manifest Anxiety Scale; Memory; Nitrous Oxide; Pain Measurement; Preanesthetic Medication; Psychomotor Performance; Regression Analysis; Triazolam

1993
Sublingual triazolam versus peroral diazepam as a premedication for general anaesthesia.
    Canadian journal of anaesthesia = Journal canadien d'anesthesie, 1995, Volume: 42, Issue:10

    Topics: Administration, Oral; Administration, Sublingual; Adolescent; Adult; Aged; Anesthesia, General; Blood Pressure; Diazepam; Double-Blind Method; Female; Heart Rate; Humans; Hypnotics and Sedatives; Male; Middle Aged; Preanesthetic Medication; Triazolam

1995
Comparison of triazolam, diazepam, and placebo as outpatient oral premedication for endodontic patients.
    Journal of endodontics, 1997, Volume: 23, Issue:3

    Topics: Adjuvants, Anesthesia; Anesthesia, Dental; Anti-Anxiety Agents; Chi-Square Distribution; Conscious Sedation; Dental Anxiety; Diazepam; Double-Blind Method; Humans; Hypnotics and Sedatives; Preanesthetic Medication; Root Canal Therapy; Statistics, Nonparametric; Triazolam

1997

Other Studies

98 other study(ies) available for diazepam and triazolam

ArticleYear
Synthesis and pharmacology of novel anxiolytic agents derived from 2-[(dialkylamino)methyl-4H-triazol-4-yl] benzophenones and related heterocyclic benzophenones.
    Journal of medicinal chemistry, 1976, Volume: 19, Issue:8

    Topics: Animals; Anti-Anxiety Agents; Benzophenones; Drug Synergism; Electroshock; Ethanol; Male; Mice; Nicotine; Pentylenetetrazole; Semicarbazides; Strychnine; Triazoles

1976
Novel anxiolytic agents derived from alpha-amino-alpha-phenyl-o-tolyl-4H-triazoles and -imidazoles.
    Journal of medicinal chemistry, 1978, Volume: 21, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Brain; Crystallography; Hypnotics and Sedatives; Imidazoles; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Mice; Models, Molecular; Molecular Conformation; Muscle Relaxation; Nicotine; Pentylenetetrazole; Rats; Seizures; Semicarbazides; Triazoles

1978
Pharmacology of some metabolites of triazolam, alprazolam, and diazepam prepared by a simple, one-step oxidation of benzodiazepines.
    Journal of medicinal chemistry, 1978, Volume: 21, Issue:12

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Diazepam; Hydroxylation; Male; Methods; Mice; Oxidation-Reduction; Triazolam; Triazoles

1978
6-Aryl-4H-s-triazolo[4,3-a][1,4]benzodiazepines. Influence of 1-substitution on pharmacological activity.
    Journal of medicinal chemistry, 1979, Volume: 22, Issue:11

    Topics: Animals; Anti-Anxiety Agents; Apomorphine; Benzodiazepines; Body Temperature; Dextroamphetamine; Male; Mice; Motor Activity; Structure-Activity Relationship

1979
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship

2000
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Hologram QSAR model for the prediction of human oral bioavailability.
    Bioorganic & medicinal chemistry, 2007, Dec-15, Volume: 15, Issue:24

    Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Selective influence on contextual memory: physiochemical properties associated with selectivity of benzodiazepine ligands at GABAA receptors containing the alpha5 subunit.
    Journal of medicinal chemistry, 2008, Jul-10, Volume: 51, Issue:13

    Topics: Animals; Behavior, Animal; Benzodiazepines; Chemical Phenomena; Chemistry, Physical; Computer Simulation; Databases, Factual; Electrophysiology; Female; Ligands; Male; Memory; Mice; Models, Molecular; Molecular Structure; Oocytes; Protein Isoforms; Protein Subunits; Quantitative Structure-Activity Relationship; Receptors, GABA-A; Structure-Activity Relationship; Xenopus laevis

2008
Axial chirality and affinity at the GABA(A) receptor of pyrimido[1,2-a][1,4]benzodiazepines and related compounds.
    Bioorganic & medicinal chemistry, 2008, Nov-01, Volume: 16, Issue:21

    Topics: Benzodiazepines; Chromatography, High Pressure Liquid; Crystallography, X-Ray; gamma-Aminobutyric Acid; Humans; Molecular Structure; Protein Binding; Receptors, GABA-A; Stereoisomerism; Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Experimental solubility profiling of marketed CNS drugs, exploring solubility limit of CNS discovery candidate.
    Bioorganic & medicinal chemistry letters, 2010, Dec-15, Volume: 20, Issue:24

    Topics: Central Nervous System Agents; Drug Evaluation, Preclinical; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Solubility

2010
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
[Behavioral and EEG effects of triazolam in comparison with those of diazepam (author's transl)].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1978, Volume: 74, Issue:5

    Topics: Aggression; Agonistic Behavior; Animals; Anti-Anxiety Agents; Anticonvulsants; Diazepam; Electric Stimulation; Electroencephalography; Humans; Limbic System; Male; Mice; Motor Activity; Muscle Relaxants, Central; Olfactory Bulb; Rabbits; Rats; Septal Nuclei; Social Isolation; Triazolam

1978
[Effects of triazolam on conditioned behavior in rats (author's transl)].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1978, Volume: 74, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Conditioning, Psychological; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Hypothalamus; Male; Rats; Self Stimulation; Triazolam

1978
Hypnotics today.
    The Practitioner, 1979, Volume: 223, Issue:1336

    Topics: Aged; Anti-Anxiety Agents; Diazepam; Electroencephalography; Humans; Sleep; Sleep Initiation and Maintenance Disorders; Temazepam; Triazolam

1979
Detoxification for triazolam physical dependence.
    Journal of clinical psychopharmacology, 1992, Volume: 12, Issue:2

    Topics: Adult; Alcoholism; Diazepam; Dose-Response Relationship, Drug; Female; Half-Life; Hospitalization; Humans; Male; Middle Aged; Oxazepam; Substance Abuse Treatment Centers; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam

1992
Relationship between benzodiazepine receptor occupancy and potentiation of gamma-aminobutyric acid-stimulated chloride flux in vitro of four ligands of differing intrinsic efficacies.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:3

    Topics: Animals; Benzodiazepinones; Cell Membrane; Cerebral Cortex; Chlorides; Diazepam; Drug Synergism; Flumazenil; gamma-Aminobutyric Acid; Ligands; Male; Rats; Receptors, GABA-A; Triazolam

1992
Relationship between benzodiazepine receptor occupancy and functional effects in vivo of four ligands of differing intrinsic efficacies.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:3

    Topics: Administration, Oral; Animals; Benzodiazepinones; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Male; Mice; Mice, Inbred DBA; Motor Activity; Receptors, GABA-A; Seizures; Triazolam

1992
Benzodiazepines block long-term potentiation in slices of hippocampus and piriform cortex.
    Neuroscience, 1992, Volume: 49, Issue:1

    Topics: Analysis of Variance; Animals; Cerebral Cortex; Diazepam; Evoked Potentials; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Male; Organ Specificity; Rats; Rats, Wistar; Time Factors; Triazolam

1992
Oral self-administration of triazolam, diazepam and ethanol in the baboon: drug reinforcement and benzodiazepine physical dependence.
    Psychopharmacology, 1992, Volume: 108, Issue:3

    Topics: Animals; Conditioning, Operant; Diazepam; Drinking Behavior; Ethanol; Flumazenil; Food; Half-Life; Male; Papio; Reinforcement Schedule; Reward; Self Administration; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam

1992
Interactive effects of ethanol on benzodiazepines levels in blood and brain of rat.
    Arukoru kenkyu to yakubutsu izon = Japanese journal of alcohol studies & drug dependence, 1992, Volume: 27, Issue:3

    Topics: Administration, Oral; Animals; Benzodiazepines; Brain Chemistry; Chlordiazepoxide; Diazepam; Drug Interactions; Estazolam; Ethanol; Gas Chromatography-Mass Spectrometry; Male; Rats; Rats, Inbred Strains; Triazolam

1992
Benzodiazepines inhibit temperature-dependent L-[125I]triiodothyronine accumulation into human liver, human neuroblast, and rat pituitary cell lines.
    Endocrinology, 1992, Volume: 130, Issue:3

    Topics: Adenoma; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Cell Line; Convulsants; Diazepam; Dose-Response Relationship, Drug; Humans; Iodine Radioisotopes; Liver; Lorazepam; Neuroblastoma; Pituitary Neoplasms; Rats; Receptors, Thyroid Hormone; Temperature; Triazolam; Triiodothyronine; Tritium; Tumor Cells, Cultured

1992
The discriminative stimulus effects of diazepam in rats at two training doses.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:3

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Buspirone; Carbolines; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Flumazenil; Male; Morphine; Pentobarbital; Pyrazoles; Pyridazines; Rats; Rats, Inbred Strains; Triazolam

1991
Benzodiazepine requirements during alcohol withdrawal syndrome: clinical implications of using a standardized withdrawal scale.
    Journal of clinical psychopharmacology, 1991, Volume: 11, Issue:5

    Topics: Administration, Oral; Adult; Alcohol Withdrawal Delirium; Anti-Anxiety Agents; Chlordiazepoxide; Diazepam; Hospitalization; Humans; Length of Stay; Lorazepam; Neurologic Examination; Oxazepam; Retrospective Studies; Temazepam; Triazolam

1991
Physical dependence induced in DBA/2J mice by benzodiazepine receptor full agonists, but not by the partial agonist Ro 16-6028.
    European journal of pharmacology, 1990, Nov-06, Volume: 190, Issue:1-2

    Topics: Administration, Oral; Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepinones; Diazepam; Drug Implants; Mice; Mice, Inbred DBA; Receptors, GABA-A; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam

1990
Cyclopyrrolones, unlike some benzodiazepines, do not induce physical dependence in mice.
    Neuroscience letters, 1990, Sep-04, Volume: 117, Issue:1-2

    Topics: Animals; Azabicyclo Compounds; Carbolines; Convulsants; Diazepam; Disease Models, Animal; Flunitrazepam; Hypnotics and Sedatives; Lorazepam; Male; Mice; Mice, Inbred Strains; Naphthyridines; Piperazines; Seizures; Structure-Activity Relationship; Substance-Related Disorders; Sulfur Compounds; Triazolam

1990
Drug discrimination in rats successively trained to discriminate diazepam and pentobarbital.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 35, Issue:2

    Topics: Animals; Azabicyclo Compounds; Diazepam; Discrimination Learning; Discrimination, Psychological; Generalization, Stimulus; Male; Meprobamate; Pentobarbital; Piperazines; Rats; Rats, Inbred Strains; Triazolam

1990
Differential generalization to pentobarbital in rats trained to discriminate lorazepam, chlordiazepoxide, diazepam, or triazolam.
    Psychopharmacology, 1989, Volume: 98, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Chlordiazepoxide; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Generalization, Psychological; Humans; Lorazepam; Pentobarbital; Rats; Triazolam

1989
Motor phenomena in benzodiazepine withdrawal.
    Hospital & community psychiatry, 1989, Volume: 40, Issue:12

    Topics: Aged; Alprazolam; Anti-Anxiety Agents; Diagnosis, Differential; Diazepam; Drug Therapy, Combination; Female; Humans; Muscle Rigidity; Sleep Initiation and Maintenance Disorders; Substance Withdrawal Syndrome; Triazolam; Urinary Incontinence

1989
Effects of repeated RO 15-1788 administration in benzodiazepine-dependent baboons.
    European journal of pharmacology, 1985, Apr-02, Volume: 110, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Convulsants; Diazepam; Drug Tolerance; Flumazenil; Humans; Male; Papio; Posture; Substance Withdrawal Syndrome; Substance-Related Disorders; Tremor; Triazolam; Vomiting

1985
Treatment of episodic behavioral disorders with rapidly absorbed benzodiazepines.
    The Journal of nervous and mental disease, 1985, Volume: 173, Issue:5

    Topics: Administration, Oral; Adult; Aggression; Anger; Anti-Anxiety Agents; Clorazepate Dipotassium; Diazepam; Female; Humans; Kinetics; Male; Mental Disorders; Rage; Seizures; Triazolam

1985
Triazolam addiction.
    Hospital & community psychiatry, 1985, Volume: 36, Issue:7

    Topics: Adult; Anti-Anxiety Agents; Diazepam; Humans; Male; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam

1985
The use of benzodiazepines with particular reference to the elderly.
    British journal of hospital medicine, 1986, Volume: 35, Issue:5

    Topics: Aged; Anti-Anxiety Agents; Anxiety; Chlordiazepoxide; Diazepam; Humans; Infusions, Parenteral; Kinetics; Sleep Initiation and Maintenance Disorders; Temazepam; Triazolam

1986
Comparative pharmacodynamics of benzodiazepines.
    Psychopharmacology series, 1987, Volume: 3

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Humans; Kinetics; Lorazepam; Male; Psychomotor Performance; Triazolam

1987
Seizures following triazolam withdrawal despite benzodiazepine treatment.
    The Journal of clinical psychiatry, 1987, Volume: 48, Issue:10

    Topics: Anti-Anxiety Agents; Anxiety Disorders; Chlordiazepoxide; Diazepam; Humans; Male; Middle Aged; Receptors, GABA-A; Seizures; Substance Withdrawal Syndrome; Triazolam

1987
Searching for the endogenous benzodiazepine using the graph theoretical approach.
    Pharmaceutical research, 1988, Volume: 5, Issue:7

    Topics: Anti-Anxiety Agents; Carbolines; Diazepam; Models, Biological; Receptors, GABA-A; Triazolam

1988
The effects of triazolam on cerebral blood flow and metabolism in the dog.
    Acta anaesthesiologica Scandinavica, 1986, Volume: 30, Issue:3

    Topics: Animals; Benzodiazepines; Brain; Brain Chemistry; Cerebrovascular Circulation; Diazepam; Dogs; Electroencephalography; Energy Metabolism; Female; Male; Midazolam; Oxygen Consumption; Triazolam

1986
Triazolam withdrawal.
    The Journal of clinical psychiatry, 1988, Volume: 49, Issue:9

    Topics: Alprazolam; Diazepam; Drug Tolerance; Humans; Seizures; Substance Withdrawal Syndrome; Triazolam

1988
Triazolobenzodiazepines competitively inhibit the binding of platelet activating factor (PAF) to human platelets.
    Biochemical and biophysical research communications, 1987, Apr-14, Volume: 144, Issue:1

    Topics: Alprazolam; Binding, Competitive; Blood Platelets; Diazepam; Humans; In Vitro Techniques; Kinetics; Platelet Activating Factor; Platelet Aggregation; Triazolam

1987
[Analysis of etizolam, triazolam, nitrazepam and maprotiline in autopsy materials by high-performance liquid chromatography and gas chromatography].
    Nihon hoigaku zasshi = The Japanese journal of legal medicine, 1987, Volume: 41, Issue:1

    Topics: Anthracenes; Chromatography, Gas; Chromatography, High Pressure Liquid; Diazepam; Female; Forensic Medicine; Humans; Male; Maprotiline; Middle Aged; Nitrazepam; Triazolam

1987
Modulation of auditory evoked magnetic fields by benzodiazepines.
    Neuropsychobiology, 1986, Volume: 16, Issue:4

    Topics: Acoustic Stimulation; Auditory Cortex; Benzodiazepines; Diazepam; Humans; Magnetics; Triazolam

1986
Withdrawal regimen for triazolam-dependent patients.
    CMAJ : Canadian Medical Association journal = journal de l'Association medicale canadienne, 1986, Jun-01, Volume: 134, Issue:11

    Topics: Diazepam; Flurazepam; Humans; Sleep Initiation and Maintenance Disorders; Substance Withdrawal Syndrome; Triazolam

1986
Effects of brotizolam on the sleep-waking cycle of the cat.
    Arzneimittel-Forschung, 1986, Volume: 36, Issue:3A

    Topics: Animals; Azepines; Cats; Diazepam; Electrodes, Implanted; Electroencephalography; Female; Flurazepam; Hypnotics and Sedatives; Male; Nitrazepam; Sleep; Sleep, REM; Time Factors; Triazolam; Wakefulness

1986
Physical dependence capacity of brotizolam in rhesus monkeys. 2nd communication: primary dependence and barbital substitution.
    Arzneimittel-Forschung, 1986, Volume: 36, Issue:3A

    Topics: Animals; Azepines; Barbital; Barbiturates; Body Weight; Diazepam; Female; Hypnotics and Sedatives; Macaca mulatta; Male; Psychomotor Performance; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam

1986
Abuse liability of triazolam: experimental measurements in animals and humans.
    Psychopharmacology series, 1987, Volume: 3

    Topics: Animals; Diazepam; Drug Tolerance; Humans; Male; Papio; Pentobarbital; Psychomotor Performance; Self Administration; Substance-Related Disorders; Triazolam

1987
Effects of diazepam and triazolam on auditory and visual thresholds and reaction times in the baboon.
    Psychopharmacology, 1985, Volume: 87, Issue:2

    Topics: Animals; Auditory Threshold; Diazepam; Dogs; Male; Papio; Reaction Time; Sensory Thresholds; Time Factors; Triazolam; Vision, Ocular

1985
Determination of biological activity of alprazolam, triazolam and their metabolites.
    The Journal of pharmacy and pharmacology, 1982, Volume: 34, Issue:2

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Binding, Competitive; Brain; Diazepam; Flunitrazepam; Kinetics; Male; Membranes; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A; Triazolam

1982
Benzodiazepines: drug discrimination and physiological dependence.
    NIDA research monograph, 1984, Volume: 49

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Bromazepam; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Generalization, Stimulus; Humans; Lorazepam; Papio; Pentobarbital; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam

1984
Subacute benzodiazepine treatment: observations on behavioural tolerance and withdrawal.
    Alcohol and alcoholism (Oxford, Oxfordshire), 1984, Volume: 19, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Conditioning, Psychological; Diazepam; Drinking Behavior; Drug Tolerance; Humans; Male; Mice; Motor Activity; Oxazepam; Pentylenetetrazole; Rats; Seizures; Substance Withdrawal Syndrome; Triazolam

1984
The effectiveness of benzodiazepines and narcotics in outpatient surgery.
    Aesthetic plastic surgery, 1984, Volume: 8, Issue:4

    Topics: Ambulatory Surgical Procedures; Analgesics; Anesthesia, Local; Diazepam; Humans; Morphine; Preanesthetic Medication; Promethazine; Prospective Studies; Surgery, Plastic; Triazolam

1984
Use of the specific benzodiazepine antagonist, Ro 15-1788, in studies of physiological dependence on benzodiazepines.
    Experientia, 1982, Jul-15, Volume: 38, Issue:7

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Cats; Diazepam; Female; Flumazenil; Humans; Lorazepam; Male; Mice; Rats; Saimiri; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam

1982
Systematic review of the benzodiazepines. Guidelines for data sheets on diazepam, chlordiazepoxide, medazepam, clorazepate, lorazepam, oxazepam, temazepam, triazolam, nitrazepam, and flurazepam. Committee on the Review of Medicines.
    British medical journal, 1980, Mar-29, Volume: 280, Issue:6218

    Topics: Benzodiazepines; Chlordiazepoxide; Clorazepate Dipotassium; Diazepam; Flurazepam; Humans; Lorazepam; Medazepam; Nitrazepam; Oxazepam; Safety; Substance Withdrawal Syndrome; Substance-Related Disorders; Temazepam; Triazolam

1980
[Does a rebound insomnia following benzodiazepine administration exist?].
    Deutsche medizinische Wochenschrift (1946), 1980, Oct-24, Volume: 105, Issue:43

    Topics: Benzodiazepines; Diazepam; Flunitrazepam; Flurazepam; Humans; Nitrazepam; Sleep Initiation and Maintenance Disorders; Substance Withdrawal Syndrome; Triazolam

1980
Molecular surface comparison. 2. Similarity of electrostatic vector fields in drug design.
    Journal of molecular graphics, 1995, Volume: 13, Issue:3

    Topics: Anti-Anxiety Agents; Benzamides; Benzazepines; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Diazepam; Drug Design; Electricity; GABA-A Receptor Agonists; Granisetron; Indoles; Isomerism; Molecular Conformation; Ondansetron; Pharmaceutical Preparations; Protein Binding; Pyrazoles; Pyridazines; Receptors, Drug; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Structure-Activity Relationship; Surface Properties; Triazolam; Tropisetron

1995
A pilot project in office-based diagnostic esophagogastroduodenoscopy comparing two nonintravenous methods of sedation and anesthesia.
    Archives of family medicine, 1995, Volume: 4, Issue:7

    Topics: Administration, Intranasal; Administration, Oral; Adolescent; Adult; Aged; Aged, 80 and over; Analgesics; Butorphanol; Conscious Sedation; Diazepam; Drug Combinations; Endoscopy, Digestive System; Female; Humans; Injections, Intramuscular; Ketorolac Tromethamine; Male; Middle Aged; Office Visits; Patient Satisfaction; Pilot Projects; Surveys and Questionnaires; Tolmetin; Triazolam; Tromethamine

1995
Identification of parent benzodiazepines by gas chromotography/mass spectroscopy (GC/MS) from urinary extracts treated with B-glucuronidase.
    Forensic science international, 1995, May-09, Volume: 73, Issue:1

    Topics: Alprazolam; Benzodiazepines; Chlordiazepoxide; Clonazepam; Diazepam; Gas Chromatography-Mass Spectrometry; Glucuronidase; Humans; Lorazepam; Oxazepam; Triazolam

1995
Benzodiazepines promote the intermediate stage at the expense of paradoxical sleep in the rat.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 49, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Diazepam; Electroencephalography; Epilepsy; Eye Movements; Heart Rate; Male; Midazolam; Rats; Rats, Inbred Strains; Rats, Wistar; Sleep Stages; Sleep, REM; Species Specificity; Theta Rhythm; Triazolam

1994
Imidazenil, a partial positive allosteric modulator of GABAA receptors, exhibits low tolerance and dependence liabilities in the rat.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:3

    Topics: Allosteric Regulation; Animals; Anticonvulsants; Benzodiazepines; Benzodiazepinones; Brain; Diazepam; Drug Interactions; Drug Tolerance; GABA Modulators; Imidazoles; Male; Rats; Rats, Sprague-Dawley; Substance-Related Disorders; Triazolam

1994
Triazolam is more efficacious than diazepam in a broad spectrum of recombinant GABAA receptors.
    European journal of pharmacology, 1993, Jan-04, Volume: 244, Issue:1

    Topics: Animals; Cells, Cultured; Cerebral Cortex; Chloride Channels; Chlorides; Diazepam; Humans; Kidney; Membrane Proteins; Neurons; Rats; Receptors, GABA-A; Recombinant Proteins; Transfection; Triazolam

1993
Convulsive properties of N-(3,5-dimethoxy-4-propoxyphenyl-ethyl) aziridine and their influencing by diazepam and triazolam.
    Sbornik vedeckych praci Lekarske fakulty Karlovy university v Hradci Kralove, 1995, Volume: 38, Issue:2

    Topics: Animals; Anticonvulsants; Aziridines; Diazepam; Male; Rats; Rats, Wistar; Seizures; Triazolam

1995
Application of capillary electrophoresis to the simultaneous screening and quantitation of benzodiazepines.
    Journal of chromatography. B, Biomedical applications, 1996, Apr-12, Volume: 678, Issue:2

    Topics: Autoanalysis; Benzodiazepines; Bromazepam; Buffers; Diazepam; Electrophoresis, Capillary; Estazolam; Flurazepam; Humans; Hydrogen-Ion Concentration; Nitrazepam; Reproducibility of Results; Sensitivity and Specificity; Triazolam

1996
Effects of triazolam and diazepam on learning and memory as assessed using a water maze.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 53, Issue:2

    Topics: Animals; Diazepam; GABA Modulators; Male; Maze Learning; Memory; Rats; Rats, Sprague-Dawley; Triazolam

1996
Simultaneous determination of twelve benzodiazepines in human serum using a new reversed-phase chromatographic column on a 2-microns porous microspherical silica gel.
    Journal of chromatography. B, Biomedical applications, 1996, Jun-28, Volume: 682, Issue:1

    Topics: Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Bromazepam; Chlordiazepoxide; Chromatography, High Pressure Liquid; Clonazepam; Diazepam; Estazolam; Humans; Linear Models; Lorazepam; Microspheres; Nitrazepam; Reproducibility of Results; Silicon Dioxide; Spectrophotometry, Ultraviolet; Triazolam

1996
Role of GABA-A and mitochondrial diazepam binding inhibitor receptors in the anti-stress activity of neurosteroids in mice.
    Psychopharmacology, 1996, Volume: 128, Issue:3

    Topics: Analysis of Variance; Animals; Ascorbic Acid; Behavior, Animal; Binding Sites; Cerebellum; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Antagonists; GABA Modulators; Isoquinolines; Male; Mice; Mitochondria; Motor Activity; Pain Measurement; Picrotoxin; Progesterone; Receptors, GABA-A; RNA; Stress, Psychological; Triazolam

1996
Adverse reactions to sedative/hypnotics: three years' experience.
    Sleep, 1996, Volume: 19, Issue:9

    Topics: Accidental Falls; Adult; Aged; Diazepam; Female; Hospital Departments; Hospitalization; Hospitals, Teaching; Humans; Hypnotics and Sedatives; Lorazepam; Male; Middle Aged; Patient Care Team; Psychotropic Drugs; Triazolam

1996
Assessment of the anxiolytic and amnesic effects of three benzodiazepines, diazepam, alprazolam and triazolam, by conflict and non-matching to sample tests in mice.
    Nihon shinkei seishin yakurigaku zasshi = Japanese journal of psychopharmacology, 1997, Volume: 17, Issue:1

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Conflict, Psychological; Diazepam; Male; Maze Learning; Memory; Mice; Triazolam

1997
Abnormal ventricular repolarization mimicking myocardial infarction after heterocyclic antidepressant overdose.
    The American journal of cardiology, 1997, Jan-15, Volume: 79, Issue:2

    Topics: Adult; Amitriptyline; Anti-Anxiety Agents; Antidepressive Agents; Antidepressive Agents, Tricyclic; Antipsychotic Agents; Benzodiazepines; Bundle-Branch Block; Diagnosis, Differential; Diazepam; Electrocardiography; Female; Heart Ventricles; Humans; Hypnotics and Sedatives; Long QT Syndrome; Maprotiline; Myocardial Infarction; Nordazepam; Perphenazine; Triazolam

1997
Evidence of GABAergic modulation in melatonin-induced short-term memory deficits and food consumption.
    Methods and findings in experimental and clinical pharmacology, 1998, Volume: 20, Issue:4

    Topics: Animals; Antioxidants; Diazepam; Eating; Female; Flumazenil; GABA Modulators; Latency Period, Psychological; Male; Maze Learning; Melatonin; Memory Disorders; Memory, Short-Term; Mice; Muscarinic Antagonists; Rats; Rats, Wistar; Receptors, GABA; Scopolamine; Triazolam

1998
Oral sedation.
    Compendium of continuing education in dentistry (Jamesburg, N.J. : 1995), 1998, Volume: 19, Issue:9

    Topics: Administration, Oral; Algorithms; Anesthesia, Dental; Anti-Anxiety Agents; Chloral Hydrate; Conscious Sedation; Dental Anxiety; Diazepam; Histamine H1 Antagonists; Humans; Hydroxyzine; Hypnotics and Sedatives; Midazolam; Mutagens; Premedication; Triazolam

1998
Positive allosteric modulators of the GABA(A) receptor: differential interaction of benzodiazepines and neuroactive steroids with ethanol.
    Psychopharmacology, 1999, Volume: 141, Issue:1

    Topics: Allosteric Regulation; Animals; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; GABA-A Receptor Agonists; Male; Mice; Motor Activity; Neuroprotective Agents; Pregnanolone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sleep; Triazolam

1999
Stability prediction of amorphous benzodiazepines by calculation of the mean relaxation time constant using the Williams-Watts decay function.
    European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V, 1999, Volume: 48, Issue:1

    Topics: Benzodiazepines; Calorimetry, Differential Scanning; Chemical Phenomena; Chemistry, Physical; Crystallization; Diazepam; Drug Stability; Temazepam; Thermodynamics; Time Factors; Triazolam

1999
Transduction of the discriminative stimulus effects of zolpidem by GABA(A)/alpha1 receptors.
    European journal of pharmacology, 2000, Oct-06, Volume: 406, Issue:1

    Topics: Acetamides; Animals; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; Male; Protein Subunits; Pyridines; Pyrimidines; Reinforcement Schedule; Saimiri; Triazolam; Zolpidem

2000
Zolpidem, triazolam, and diazepam decrease distress vocalizations in mouse pups: differential antagonism by flumazenil and beta-Carboline-3-carboxylate-t-butyl ester (beta-CCt).
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 297, Issue:1

    Topics: Animals; Animals, Newborn; Anti-Anxiety Agents; Body Temperature; Carbolines; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Antagonists; Mice; Pyridines; Receptors, GABA-A; Triazolam; Vocalization, Animal; Zolpidem

2001
Daily treatment with diazepam differentially modifies sensitivity to the effects of gamma-aminobutyric acid(A) modulators on schedule-controlled responding in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 300, Issue:3

    Topics: Animals; Azides; Benzodiazepines; Carbolines; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Electroshock; Food; GABA Agonists; GABA Antagonists; GABA Modulators; Macaca mulatta; Male; Pentobarbital; Pregnanolone; Receptors, GABA-A; Reinforcement Schedule; Triazolam

2002
Orally delivered alprazolam, diazepam, and triazolam as reinforcers in rhesus monkeys.
    Psychopharmacology, 2002, Volume: 161, Issue:1

    Topics: Administration, Oral; Alprazolam; Animals; Anti-Anxiety Agents; Diazepam; Macaca mulatta; Male; Reinforcement, Psychology; Self Administration; Triazolam

2002
Anxiolysis in general dental practice.
    Dentistry today, 2003, Volume: 22, Issue:3

    Topics: Acetamides; Adjuvants, Anesthesia; Anesthesia, Dental; Anesthetics, Inhalation; Anti-Anxiety Agents; Clinical Protocols; Conscious Sedation; Dental Anxiety; Diazepam; GABA Modulators; General Practice, Dental; Humans; Hydroxyzine; Hypnotics and Sedatives; Lorazepam; Midazolam; Nitrous Oxide; Pyrimidines; Triazolam

2003
Role of platelet activating factor in triazolobenzodiazepines-induced retrograde amnesia.
    Behavioural brain research, 2003, Jun-16, Volume: 142, Issue:1-2

    Topics: 1-Alkyl-2-acetylglycerophosphocholine Esterase; Amnesia, Anterograde; Amnesia, Retrograde; Animals; Anti-Anxiety Agents; Azepines; Diazepam; Diterpenes; Escape Reaction; Female; Flumazenil; Ginkgolides; Lactones; Learning; Male; Mice; Phospholipases A; Platelet Activating Factor; Platelet Membrane Glycoproteins; Reaction Time; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Receptors, GABA-A; Retention, Psychology; Triazolam

2003
Postmortem changes in tissue concentrations of triazolam and diazepam in rats.
    Legal medicine (Tokyo, Japan), 2004, Volume: 6, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Diazepam; Forensic Medicine; Gas Chromatography-Mass Spectrometry; Gastrointestinal Contents; Intestine, Small; Kidney; Liver; Lung; Male; Muscle, Skeletal; Myocardium; Postmortem Changes; Rats; Rats, Wistar; Tissue Distribution; Triazolam

2004
New drugs for local anesthesia and oral sedation.
    Dentistry today, 2004, Volume: 23, Issue:12

    Topics: Administration, Oral; Anesthetics, Combined; Anesthetics, Local; Anti-Anxiety Agents; Carticaine; Diazepam; Drug Combinations; Humans; Lidocaine; Lidocaine, Prilocaine Drug Combination; Lorazepam; Prilocaine; Triazolam

2004
Anxiolytic-like action in mice treated with nitrous oxide and oral triazolam or diazepam.
    Life sciences, 2005, Feb-25, Volume: 76, Issue:15

    Topics: Administration, Oral; Animals; Anti-Anxiety Agents; Diazepam; Male; Mice; Nitrous Oxide; Triazolam

2005
Impact of end-product inhibition on the determination of in vitro metabolic clearance.
    Xenobiotica; the fate of foreign compounds in biological systems, 2005, Volume: 35, Issue:5

    Topics: Alamethicin; Animals; Biotransformation; Diazepam; Hepatocytes; Kinetics; Metabolic Clearance Rate; Microsomes, Liver; Models, Biological; Phenytoin; Rats; Triazolam

2005
The detection of sedatives in hair and nail samples using tandem LC-MS-MS.
    Forensic science international, 2007, Feb-14, Volume: 166, Issue:1

    Topics: Adult; Aged; Aged, 80 and over; Alprazolam; Azabicyclo Compounds; Benzodiazepines; Chromatography, Liquid; Clobazam; Clonazepam; Diazepam; Female; Forensic Pathology; Hair; Humans; Hypnotics and Sedatives; Male; Mass Spectrometry; Midazolam; Middle Aged; Nails; Oxazepam; Piperazines; Predictive Value of Tests; Rape; Temazepam; Triazolam

2007
Practical oral sedation in dentistry. Part II--Clinical application of various oral sedatives and discussion.
    Compendium of continuing education in dentistry (Jamesburg, N.J. : 1995), 2006, Volume: 27, Issue:9

    Topics: Administration, Oral; Adult; Age Factors; Aged; Aged, 80 and over; Anesthesia, Dental; Child; Child, Preschool; Chloral Hydrate; Conscious Sedation; Diazepam; Fentanyl; Humans; Hypnotics and Sedatives; Meperidine; Midazolam; Nausea; Promethazine; Triazolam; Vomiting

2006
Prediction of metabolic clearance using fresh human hepatocytes: comparison with cryopreserved hepatocytes and hepatic microsomes for five benzodiazepines.
    Xenobiotica; the fate of foreign compounds in biological systems, 2008, Volume: 38, Issue:4

    Topics: Alprazolam; Benzodiazepines; Cell Survival; Cells, Cultured; Cryopreservation; Cytochrome P-450 CYP3A; Diazepam; Flunitrazepam; Hepatocytes; Humans; Metabolic Clearance Rate; Microsomes, Liver; Midazolam; Substrate Specificity; Triazolam

2008
Evaluation of anxiolytic-like effects of some short-acting benzodiazepine hypnotics in mice.
    Journal of pharmacological sciences, 2008, Volume: 107, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Azepines; Benzodiazepines; Diazepam; Hypnotics and Sedatives; Lorazepam; Male; Maze Learning; Mice; Mice, Inbred ICR; Motor Activity; Triazolam

2008
Rebound insomnia induced by abrupt withdrawal of hypnotics in sleep-disturbed rats.
    European journal of pharmacology, 2008, Nov-12, Volume: 597, Issue:1-3

    Topics: Animals; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Hypnotics and Sedatives; Isoindoles; Male; Piperazines; Pyrimidines; Rats; Rats, Wistar; Sleep Initiation and Maintenance Disorders; Sleep Stages; Time Factors; Triazolam; Wakefulness

2008
Oral sedation for the apprehensive dental patient.
    Dentistry today, 2000, Volume: 19, Issue:4

    Topics: Administration, Oral; Adolescent; Anti-Anxiety Agents; Biological Availability; Conscious Sedation; Dental Anxiety; Diazepam; Female; Humans; Male; Safety; Therapeutic Equivalency; Triazolam; Young Adult

2000
Quantitation of benzodiazepines in blood and urine using gas chromatography-mass spectrometry (GC-MS).
    Methods in molecular biology (Clifton, N.J.), 2010, Volume: 603

    Topics: Alprazolam; Benzodiazepines; Diazepam; Gas Chromatography-Mass Spectrometry; Humans; Lorazepam; Nordazepam; Oxazepam; Solid Phase Extraction; Triazolam

2010
Allosteric modulation of GABA(A) receptor subtypes:effects on visual recognition and visuospatial working memory in rhesus monkeys [corrected].
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2013, Volume: 38, Issue:11

    Topics: Acetamides; Allosteric Regulation; Animals; Benzodiazepines; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Imidazoles; Macaca mulatta; Male; Memory, Short-Term; Pyridazines; Pyridines; Pyrimidines; Receptors, GABA-A; Recognition, Psychology; Triazolam; Triazoles; Zolpidem

2013
Alterations in brain-derived neurotrophic factor in the mouse hippocampus following acute but not repeated benzodiazepine treatment.
    PloS one, 2013, Volume: 8, Issue:12

    Topics: Analysis of Variance; Animals; Benzodiazepines; Blotting, Western; Brain-Derived Neurotrophic Factor; Chromatin Immunoprecipitation; Cyclic AMP Response Element-Binding Protein; Diazepam; Enzyme-Linked Immunosorbent Assay; Gene Expression Regulation; Genes, Immediate-Early; Hippocampus; Male; Mice; Mice, Inbred C57BL; Proto-Oncogene Proteins c-fos; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; Triazolam; Zolpidem

2013
[Cross-reactivity of Instant-View M-1 for detection of benzodiazepine-related drugs and their metabolites in urine].
    Chudoku kenkyu : Chudoku Kenkyukai jun kikanshi = The Japanese journal of toxicology, 2014, Volume: 27, Issue:1

    Topics: Alprazolam; Benzodiazepines; Biomarkers; Cross Reactions; Diazepam; Humans; Immunoassay; Nitrazepam; Reagent Kits, Diagnostic; Sensitivity and Specificity; Structure-Activity Relationship; Substance Abuse Detection; Triazolam

2014
Incorporation of five common hypnotics into hair after a single dose and application to a forensic case of drug facilitated crimes.
    Forensic science international, 2021, Volume: 325

    Topics: Adult; Asian People; Chromatography, Liquid; Crime; Diazepam; Female; Flunitrazepam; Forensic Toxicology; Hair; Humans; Hypnotics and Sedatives; Male; Mass Spectrometry; Nitrazepam; Substance Abuse Detection; Triazolam; Zolpidem

2021