diazepam and thiazoles

diazepam has been researched along with thiazoles in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-199010 (43.48)18.7374
1990's1 (4.35)18.2507
2000's10 (43.48)29.6817
2010's2 (8.70)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
D'Angio, M; Scatton, B; Serrano, A1
Arvela, P; Klotz, U; Rosenkranz, B1
Greenblatt, DJ; Harmatz, JS; Locniskar, A; Shader, RI; Zinny, MA1
Arvela, P; Klotz, U; Pasanen, M; Pelkonen, O; Sotaniemi, E1
Dammann, HG; Gottlieb, W; Keohane, PP; Klotz, U1
Klotz, U1
Benavides, J; Camelin, JC; Flamand, F; Gueremy, C; Le Fur, G; Legrand, JJ; Mitrani, N; Uzan, A1
Dammann, HG; Gottlieb, WR; Keohane, P; Klotz, U; Walter, TA1
Helmchen, H1
Matsumoto, K; Nakamura, M; Ohno, Y; Sakamoto, H1
Anziano, RJ; Fricke, JR; Johnson, AC; Miceli, JJ; Titus, CK; Wilner, KD1
Harper, EA; Morton, MF; Shankley, NP; Tavares, IA1
HABER, J; HERZKA, H1
Chojnacka-Wójcik, E; Cosford, ND; Klodzinska, A; Nowak, G; Pilc, A; Tatarczyńska, E1
Cryan, JF; Gasparini, F; Page, ME; Szeliga, P1
Bespalov, AY; Danysz, W; Gravius, A; Maciejak, P; Pietraszek, M; Płaźnik, A; Sukhanov, I; Szyndler, J; Wisłowska, A1
Barberi, C; Danysz, W; Gravius, A; Schäfer, D; Schmidt, WJ1
Cansel, N; Herken, H; Ozen, ME; Savas, HA; Yumru, M1
Cleveland, NR; Heard, K; Krier, S1
Klein, S; Nicolas, LB; Prinssen, EP1
Hoffman, RS; Manini, AF; Pearl-Davis, MS; Wu, S1
Cao, L; Chen, J; Hu, J; Lin, J; Lin, S; Mao, L; Ouyang, Y; Yan, G; Yang, X; Zhang, H; Zhou, Y; Zhu, W1
Baur, R; Maldifassi, MC; Middendorp, SJ; Sigel, E1

Trials

4 trial(s) available for diazepam and thiazoles

ArticleYear
Famotidine, a new H2-receptor antagonist, does not affect hepatic elimination of diazepam or tubular secretion of procainamide.
    European journal of clinical pharmacology, 1985, Volume: 28, Issue:6

    Topics: Adult; Cimetidine; Diazepam; Famotidine; Histamine H2 Antagonists; Humans; In Vitro Techniques; Kidney Tubules; Kinetics; Liver; Male; Microsomes, Liver; Middle Aged; Procainamide; Random Allocation; Thiazoles

1985
Nocturnal doses of ranitidine and nizatidine do not affect the disposition of diazepam.
    Journal of clinical pharmacology, 1987, Volume: 27, Issue:3

    Topics: Adult; Diazepam; Drug Interactions; Histamine H2 Antagonists; Humans; Male; Nizatidine; Nordazepam; Ranitidine; Thiazoles

1987
Nizatidine (300 mg nocte) does not interfere with diazepam pharmacokinetics in man.
    British journal of clinical pharmacology, 1987, Volume: 23, Issue:1

    Topics: Adult; Diazepam; Drug Interactions; Humans; Kinetics; Male; Nizatidine; Thiazoles

1987
The anxiolytic effect of the novel antipsychotic ziprasidone compared with diazepam in subjects anxious before dental surgery.
    Journal of clinical psychopharmacology, 2002, Volume: 22, Issue:2

    Topics: Adolescent; Adult; Anti-Anxiety Agents; Antipsychotic Agents; Arousal; Dental Anxiety; Diazepam; Double-Blind Method; Female; Humans; Male; Middle Aged; Piperazines; Premedication; Thiazoles; Treatment Outcome

2002

Other Studies

19 other study(ies) available for diazepam and thiazoles

ArticleYear
NMDA antagonists block restraint-induced increase in extracellular DOPAC in rat nucleus accumbens.
    European journal of pharmacology, 1989, Mar-14, Volume: 162, Issue:1

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adrenergic alpha-Antagonists; Animals; Aspartic Acid; Carbolines; Convulsants; Diazepam; Male; N-Methylaspartate; Nucleus Accumbens; Phenylacetates; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Restraint, Physical; Riluzole; Septal Nuclei; Thiazoles

1989
Interaction of diazepam with famotidine and cimetidine, two H2-receptor antagonists.
    Journal of clinical pharmacology, 1986, Volume: 26, Issue:4

    Topics: Adult; Biotransformation; Cimetidine; Diazepam; Drug Interactions; Famotidine; Half-Life; Histamine H2 Antagonists; Humans; Infusions, Parenteral; Kinetics; Male; Metabolic Clearance Rate; Middle Aged; Nordazepam; Thiazoles

1986
Effect of five structurally diverse H2-receptor antagonists on drug metabolism.
    Biochemical pharmacology, 1986, Dec-15, Volume: 35, Issue:24

    Topics: 7-Alkoxycoumarin O-Dealkylase; Animals; Aryl Hydrocarbon Hydroxylases; Biotransformation; Cimetidine; Cytochrome P-450 CYP1A1; Cytochrome P-450 Enzyme System; Diazepam; Famotidine; Histamine H2 Antagonists; Humans; Imidazoles; Kinetics; Male; Microsomes, Liver; Nizatidine; Oxidoreductases; Oxygenases; Pharmaceutical Preparations; Ranitidine; Rats; Rats, Inbred Strains; Thiazoles

1986
Lack of effect of nizatidine on drug metabolism.
    Scandinavian journal of gastroenterology. Supplement, 1987, Volume: 136

    Topics: Adult; Animals; Cytochrome P-450 Enzyme System; Diazepam; Double-Blind Method; Drug Interactions; Histamine H2 Antagonists; Humans; In Vitro Techniques; Male; Microsomes, Liver; Nizatidine; Pharmaceutical Preparations; Random Allocation; Rats; Rats, Inbred Strains; Thiazoles

1987
2-Amino-6-trifluoromethoxy benzothiazole, a possible antagonist of excitatory amino acid neurotransmission--II. Biochemical properties.
    Neuropharmacology, 1985, Volume: 24, Issue:11

    Topics: Acetylcholine; Amino Acids; Animals; Anticonvulsants; Apomorphine; Cerebellum; Chlordiazepoxide; Cyclic GMP; Diazepam; gamma-Aminobutyric Acid; Harmaline; In Vitro Techniques; Injections, Intraventricular; Isoniazid; Male; Rats; Rats, Inbred Strains; Riluzole; Synaptic Transmission; Thiazoles

1985
[Psychopharmacological agents in treatment of psychiatric emergencies].
    La Clinica terapeutica, 1971, Mar-31, Volume: 56, Issue:6

    Topics: Adult; Age Factors; Aged; Antidepressive Agents; Dementia; Diazepam; Haloperidol; Humans; Hypnotics and Sedatives; Mental Disorders; Middle Aged; Phenothiazines; Psychoses, Alcoholic; Suicide Prevention; Sulfonic Acids; Thiazoles; Tranquilizing Agents

1971
Anxiolytic-like effects of perospirone, a novel serotonin-2 and dopamine-2 antagonist (SDA)-type antipsychotic agent.
    Pharmacology, biochemistry, and behavior, 1998, Volume: 60, Issue:4

    Topics: Aggression; Animals; Anti-Anxiety Agents; Antipsychotic Agents; Diazepam; Dopamine Antagonists; Dose-Response Relationship, Drug; Haloperidol; Indoles; Interpersonal Relations; Isoindoles; Male; Rats; Serotonin Antagonists; Thiazoles

1998
Pharmacological evidence for putative CCK(1) receptor heterogeneity in human colon smooth muscle.
    British journal of pharmacology, 2002, Volume: 136, Issue:6

    Topics: Aspartic Acid; Binding Sites; Binding, Competitive; Colon; Devazepide; Diazepam; Gallbladder; Humans; Indoleacetic Acids; Kinetics; Membranes; Models, Biological; Muscle, Smooth; Naphthalenesulfonates; Organ Culture Techniques; Organ Specificity; Protease Inhibitors; Radioligand Assay; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Thiazoles; Time Factors

2002
[CLINICAL REPORT ON THE EFFECTIVENESS OF DAPTAZOLE (AMIPHENAZOLE) IN A CASE OF VALIUM POISONING].
    Schweizerische medizinische Wochenschrift, 1965, Mar-13, Volume: 95

    Topics: Antidotes; Child; Diazepam; Drug Therapy; Hypnotics and Sedatives; Poisoning; Thiazoles; Toxicology

1965
Anxiolytic-like effects of MTEP, a potent and selective mGlu5 receptor agonist does not involve GABA(A) signaling.
    Neuropharmacology, 2004, Volume: 47, Issue:3

    Topics: Animals; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Drinking; Drinking Behavior; Drug Interactions; Electroshock; Exploratory Behavior; Flumazenil; GABA Modulators; Male; Maze Learning; Mice; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, GABA-A; Receptors, Metabotropic Glutamate; Sensory Thresholds; Signal Transduction; Thiazoles

2004
Blockade of the mGlu5 receptor decreases basal and stress-induced cortical norepinephrine in rodents.
    Psychopharmacology, 2005, Volume: 179, Issue:1

    Topics: Animals; Diazepam; Excitatory Amino Acid Antagonists; Frontal Lobe; Male; Microdialysis; Norepinephrine; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Stress, Psychological; Thiazoles

2005
Anxiolytic-like effects of mGlu1 and mGlu5 receptor antagonists in rats.
    European journal of pharmacology, 2005, May-02, Volume: 514, Issue:1

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Chlordiazepoxide; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Male; Maze Learning; Midazolam; Punishment; Pyridines; Quinolines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Reflex, Startle; Thiazoles

2005
The role of group I metabotropic glutamate receptors in acquisition and expression of contextual and auditory fear conditioning in rats - a comparison.
    Neuropharmacology, 2006, Volume: 51, Issue:7-8

    Topics: Acoustic Stimulation; Animals; Avoidance Learning; Citalopram; Conditioning, Classical; Diazepam; Dizocilpine Maleate; Electroshock; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Fear; Freezing Reaction, Cataleptic; Hippocampus; Long-Term Potentiation; Male; Pyridines; Quinolines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Scopolamine; Thiazoles

2006
Neuroleptic malignant syndrome induced by ziprasidone on the second day of treatment.
    The world journal of biological psychiatry : the official journal of the World Federation of Societies of Biological Psychiatry, 2007, Volume: 8, Issue:1

    Topics: Adult; Antipsychotic Agents; Biperiden; Diagnosis, Differential; Diazepam; Drug Therapy, Combination; Humans; Infusions, Intravenous; Male; Neuroleptic Malignant Syndrome; Neurologic Examination; Parkinsonian Disorders; Piperazines; Schizophrenia; Thiazoles

2007
Ziprasidone, diazepam, or the combination for prevention of cocaine toxicity in a mouse model.
    Academic emergency medicine : official journal of the Society for Academic Emergency Medicine, 2007, Volume: 14, Issue:8

    Topics: Animals; Cocaine; Cocaine-Related Disorders; Confidence Intervals; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Therapy, Combination; Male; Mice; Mice, Inbred Strains; Piperazines; Random Allocation; Reference Values; Sensitivity and Specificity; Statistics, Nonparametric; Survival Rate; Thiazoles

2007
Defensive-like behaviors induced by ultrasound: further pharmacological characterization in Lister-hooded rats.
    Psychopharmacology, 2007, Volume: 194, Issue:2

    Topics: Amines; Analgesics, Opioid; Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Buspirone; Calcium Channel Blockers; Cyclohexanecarboxylic Acids; Diazepam; Dose-Response Relationship, Drug; Escape Reaction; Fear; Freezing Reaction, Cataleptic; Gabapentin; gamma-Aminobutyric Acid; Haloperidol; Imidazoles; Male; Morphine; Motor Activity; Nociceptin Receptor; Pregabalin; Pyridines; Rats; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, Opioid; Spiro Compounds; Thiazoles; Ultrasonics

2007
Use of antipsychotics to treat cocaine toxicity?
    Academic emergency medicine : official journal of the Society for Academic Emergency Medicine, 2008, Volume: 15, Issue:1

    Topics: Animals; Antipsychotic Agents; Cocaine; Cocaine-Related Disorders; Diazepam; Disease Models, Animal; Mice; Piperazines; Thiazoles; Treatment Outcome

2008
Diazepam inhibits proliferation of human glioblastoma cells through triggering a G0/G1 cell cycle arrest.
    Journal of neurosurgical anesthesiology, 2013, Volume: 25, Issue:3

    Topics: Antimetabolites; Benzimidazoles; Blotting, Western; Brain Neoplasms; Bromodeoxyuridine; Cell Cycle; Cell Cycle Proteins; Cell Line, Tumor; Cell Proliferation; Cell Survival; Coloring Agents; Diazepam; Fluorescent Dyes; G1 Phase; G1 Phase Cell Cycle Checkpoints; GABA Modulators; Glioblastoma; Humans; L-Lactate Dehydrogenase; Resting Phase, Cell Cycle; S Phase; Tetrazolium Salts; Thiazoles

2013
Positive modulation of synaptic and extrasynaptic GABAA receptors by an antagonist of the high affinity benzodiazepine binding site.
    Neuropharmacology, 2015, Volume: 95

    Topics: Allosteric Regulation; Animals; Benzodiazepines; Binding Sites; Diazepam; Flumazenil; GABA Agents; gamma-Aminobutyric Acid; HEK293 Cells; Humans; Membrane Potentials; Mutation; Neurons; Oocytes; Patch-Clamp Techniques; Protein Isoforms; Quinolines; Radioligand Assay; Receptors, GABA-A; Recombinant Proteins; Thiazoles; Transfection; Xenopus laevis

2015