diazepam and quinine

diazepam has been researched along with quinine in 38 studies

Research

Studies (38)

TimeframeStudies, this research(%)All Research%
pre-199010 (26.32)18.7374
1990's7 (18.42)18.2507
2000's13 (34.21)29.6817
2010's8 (21.05)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Andersson, K; Borg, P; Frostell-Karlsson, A; Hämäläinen, M; Karlsson, R; Remaeus, A; Roos, H1
Topliss, JG; Yoshida, F1
Johans, C; Kinnunen, PK; Söderlund, T; Suomalainen, P1
Caron, G; Ermondi, G1
Briand, X; Faller, B; Lázaro, E; Lowe, PJ1
Lombardo, F; Obach, RS; Waters, NJ1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Avdeef, A; Tam, KY1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Ahlin, G; Bergström, F; Bredberg, U; Fridén, M; Hammarlund-Udenaes, M; Rehngren, M; Wan, H1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Monforte, JR1
Aster, RH; Cimo, PL; Desai, RG; Pino, JL; Pisciotta, AV1
Tagashire, E; Yanaura, S1
Amabeoku, GJ; Chikuni, O1
Bhattacharya, SK; Mitra, SK1
Koley, KC; Roy, AK; Sinha, G1
Duff, HJ; Rahmberg, M; Sheldon, RS1
Berridge, KC; Treit, D1
Heyne, A; Wolffgramm, J1
Mitsumoto, Y; Mohri, T; Sato, K1
Uono, M1
McBay, AJ1
Esteban, A; Giménez-Roldán, S1
Bwibo, NO1
Brooke, OG; Evans, AN; West, RJ1
Barbotin-Larrieu, F; Clemessy, JL1
Fushiki, T; Hanai, K; Imaizumi, M; Inoue, K; Kuroda, K; Manabe, Y; Sako, N; Yamamoto, T1
Corrêa, FM; Peres-Polon, VL; Tavares, RF1
Sturm, JW; Townend, BS; Whyte, S1
Berridge, KC; Cooper, SJ; Reynolds, SM; Richardson, DK1

Reviews

4 review(s) available for diazepam and quinine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
[Treatment of myotonic dystrophy].
    Naika. Internal medicine, 1970, Volume: 25, Issue:4

    Topics: Adrenal Cortex Hormones; Adrenocorticotropic Hormone; Adult; Chlordiazepoxide; Chlormezanone; Diazepam; Female; Humans; Ion Exchange Resins; Male; Mephenesin; Methocarbamol; Myotonia; Phenytoin; Procainamide; Quinine; Thyroid Hormones; Zoxazolamine

1970
Toxicological findings in fatal poisonings.
    Clinical chemistry, 1973, Volume: 19, Issue:4

    Topics: 1-Propanol; Alcoholic Intoxication; Amphetamine; Carbon Monoxide Poisoning; Chloral Hydrate; Chlordiazepoxide; Dextropropoxyphene; Diazepam; Ethchlorvynol; Glutethimide; Heroin; Humans; Meprobamate; Methadone; Methanol; Morphine; Orphenadrine; Paraldehyde; Pentazocine; Phenothiazines; Phenytoin; Poisoning; Quinine; Salicylates; Toxicology; Tranquilizing Agents

1973
Quinine associated blindness.
    Australian family physician, 2004, Volume: 33, Issue:8

    Topics: Blindness; Diazepam; Family Practice; Humans; Male; Middle Aged; Muscle Relaxants, Central; Quinine; Sleep-Wake Transition Disorders; Suicide, Attempted; Treatment Outcome

2004

Other Studies

34 other study(ies) available for diazepam and quinine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Biosensor analysis of the interaction between immobilized human serum albumin and drug compounds for prediction of human serum albumin binding levels.
    Journal of medicinal chemistry, 2000, May-18, Volume: 43, Issue:10

    Topics: Binding Sites; Biosensing Techniques; Digitoxin; Drug Stability; Humans; Molecular Weight; Naproxen; Orosomucoid; Pharmaceutical Preparations; Protein Binding; Quinine; Rifampin; Ritonavir; Serum Albumin; Solvents; Warfarin

2000
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Surface activity profiling of drugs applied to the prediction of blood-brain barrier permeability.
    Journal of medicinal chemistry, 2004, Mar-25, Volume: 47, Issue:7

    Topics: Blood-Brain Barrier; Lipid Bilayers; Micelles; Permeability; Pharmaceutical Preparations; Structure-Activity Relationship; Surface Properties

2004
Calculating virtual log P in the alkane/water system (log P(N)(alk)) and its derived parameters deltalog P(N)(oct-alk) and log D(pH)(alk).
    Journal of medicinal chemistry, 2005, May-05, Volume: 48, Issue:9

    Topics: 1-Octanol; Alkanes; Hydrogen-Ion Concentration; Least-Squares Analysis; Mathematics; Models, Chemical; Models, Molecular; Solvents; Water

2005
New approach to measure protein binding based on a parallel artificial membrane assay and human serum albumin.
    Journal of medicinal chemistry, 2008, Apr-10, Volume: 51, Issue:7

    Topics: Humans; Kinetics; Membranes, Artificial; Permeability; Protein Binding; Serum Albumin

2008
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
How well can the Caco-2/Madin-Darby canine kidney models predict effective human jejunal permeability?
    Journal of medicinal chemistry, 2010, May-13, Volume: 53, Issue:9

    Topics: Animals; Disease Models, Animal; Dogs; Humans; Jejunal Diseases; Kidney Diseases; Models, Biological; Permeability; Porosity; Regression Analysis

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Measurement of unbound drug exposure in brain: modeling of pH partitioning explains diverging results between the brain slice and brain homogenate methods.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:3

    Topics: Animals; Biological Transport; Brain; Chemical Phenomena; Dialysis; Hydrogen-Ion Concentration; In Vitro Techniques; Lysosomes; Male; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Tissue Distribution

2011
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Some observations concerning blood morphine concentrations in narcotic addicts.
    Journal of forensic sciences, 1977, Volume: 22, Issue:4

    Topics: Diazepam; Ethanol; Heroin; Homicide; Humans; Morphine; Poisoning; Quinine; Substance-Related Disorders

1977
Detection of drug-dependent antibodies by the 51Cr platelet lysis test: documentation of immune thrombocytopenia induced by diphenylhydantoin, diazepam, and sulfisoxazole.
    American journal of hematology, 1977, Volume: 2, Issue:1

    Topics: Adolescent; Antibodies; Antibody Specificity; Blood Platelets; Chromium Radioisotopes; Diazepam; Female; Humans; Male; Middle Aged; Phenytoin; Quinidine; Quinine; Sulfisoxazole; Thrombocytopenia

1977
[Dependence on and preference for morphine (II). Comparison among morphine, phenobarbital and diazepam].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1975, Volume: 71, Issue:3

    Topics: Animals; Body Weight; Choice Behavior; Decision Making; Diazepam; Female; Humans; Male; Methods; Morphine; Morphine Dependence; Phenobarbital; Quinine; Rats; Statistics as Topic; Substance-Related Disorders; Time Factors

1975
Effects of some GABAergic agents on quinine-induced seizures in mice.
    Experientia, 1992, Jul-15, Volume: 48, Issue:7

    Topics: Aminobutyrates; Aminooxyacetic Acid; Animals; Baclofen; Bicuculline; Diazepam; Male; Mice; Mice, Inbred Strains; Muscimol; Phenobarbital; Phenytoin; Quinine; Receptors, GABA-A; Seizures

1992
Anxiogenic activity of quinine--an experimental study in rodents.
    Indian journal of experimental biology, 1992, Volume: 30, Issue:1

    Topics: Analysis of Variance; Animals; Anxiety; Diazepam; Dose-Response Relationship, Drug; Drinking Behavior; Interpersonal Relations; Male; Movement; Quinine; Rats; Rats, Inbred Strains; Yohimbine

1992
Neuromyotonia.
    Journal of the Indian Medical Association, 1992, Volume: 90, Issue:5

    Topics: Adult; Diazepam; Fasciculation; Humans; Male; Myotonia; Quinine

1992
Role of quinidine in the mexiletine-quinidine interaction: electrophysiologic correlates of enhanced antiarrhythmic efficacy.
    Journal of cardiovascular pharmacology, 1990, Volume: 16, Issue:5

    Topics: Action Potentials; Animals; Anti-Arrhythmia Agents; Diazepam; Dogs; Drug Combinations; Drug Interactions; Heart Conduction System; Mexiletine; Quinidine; Quinine; Refractory Period, Electrophysiological

1990
A comparison of benzodiazepine, serotonin, and dopamine agents in the taste-reactivity paradigm.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 37, Issue:3

    Topics: Amphetamine; Animals; Apomorphine; Benzodiazepines; Buspirone; Chlordiazepoxide; Diazepam; Dopamine Agents; Feeding Behavior; Haloperidol; Male; Pyrimidines; Quinine; Rats; Rats, Inbred Strains; Serotonin; Sucrose; Taste

1990
Social behavior, dominance, and social deprivation of rats determine drug choice.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 38, Issue:2

    Topics: Animals; Behavior, Animal; Body Weight; Diazepam; Drinking; Eating; Ethanol; Male; Quinine; Rats; Rats, Inbred Strains; Social Behavior; Social Dominance; Social Isolation

1991
Possible participation of calmodulin in stimulation of leucine transport by concanavalin A in human lymphocytes.
    Biochemical and biophysical research communications, 1988, Jun-16, Volume: 153, Issue:2

    Topics: Calcimycin; Calcium; Calmodulin; Chlorpromazine; Concanavalin A; Diazepam; Humans; In Vitro Techniques; Ion Channels; Leucine; Lymphocyte Activation; Lymphocytes; Membrane Potentials; Potassium; Quinine; Sulfonamides

1988
Orbicularis oculi "myotonia" in hypothyroid myopathy.
    European neurology, 1973, Volume: 9, Issue:1

    Topics: Cold Temperature; Diazepam; Electromyography; Humans; Hypothyroidism; Male; Middle Aged; Muscle Contraction; Neuromuscular Diseases; Oculomotor Muscles; Phenytoin; Quinine; Triiodothyronine

1973
Accidental poisoning in children in Uganda.
    British medical journal, 1969, Dec-06, Volume: 4, Issue:5683

    Topics: Amitriptyline; Aspirin; Barbiturates; Child; Child, Preschool; Chloroquine; Codeine; Dapsone; Diazepam; Ethanol; Female; Humans; Infant; Iron; Kerosene; Male; Pesticides; Poisoning; Quinine; Tetrachloroethylene; Uganda

1969
The ingestion by pregnant women of substances toxic to the foetus.
    The Practitioner, 1980, Volume: 224, Issue:1341

    Topics: Abnormalities, Drug-Induced; Barbiturates; Clitoris; Diazepam; Disorders of Sex Development; Doxylamine; Female; Fetal Alcohol Spectrum Disorders; Humans; Hydroxyprogesterones; Infant, Newborn; Infant, Newborn, Diseases; Male; Phenytoin; Pregnancy; Progesterone Congeners; Quinine; Substance Withdrawal Syndrome

1980
[Effect of diazepam in acute quinine poisoning?].
    Archives de pediatrie : organe officiel de la Societe francaise de pediatrie, 1994, Volume: 1, Issue:1

    Topics: Acute Disease; Child; Diazepam; Humans; Poisoning; Quinine

1994
Diazepam-binding inhibitor-like activity in rat cerebrospinal fluid after stimulation by an aversive quinine taste.
    Chemical senses, 2000, Volume: 25, Issue:6

    Topics: Animals; Cerebrospinal Fluid; Diazepam; Drinking; Flumazenil; GABA-A Receptor Antagonists; Glutathione; Hydra; Male; Mice; Peptide Fragments; Pronase; Quinine; Rats; Rats, Wistar; Sucrose; Taste

2000
Mechanisms involved in the water intake-related pressor response in the rat.
    Journal of hypertension, 2002, Volume: 20, Issue:2

    Topics: Animals; Antihypertensive Agents; Arteries; Blood Pressure; Brazil; Diazepam; Dose-Response Relationship, Drug; Drinking; Heart Rate; Idazoxan; Lidocaine; Losartan; Male; Mecamylamine; Models, Animal; Muscle Relaxants, Central; Prazosin; Quinine; Rats; Rats, Wistar; Sodium Chloride; Tropanes; Water

2002
Endogenous opioids are necessary for benzodiazepine palatability enhancement: naltrexone blocks diazepam-induced increase of sucrose-'liking'.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 81, Issue:3

    Topics: Analysis of Variance; Animals; Behavior, Animal; Benzodiazepines; Diazepam; Food Preferences; Male; Naltrexone; Narcotic Antagonists; Opioid Peptides; Quinine; Rats; Rats, Sprague-Dawley; Solutions; Sucrose; Taste; Taste Threshold; Time Factors

2005