diazepam and quercetin

diazepam has been researched along with quercetin in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (7.69)18.2507
2000's1 (7.69)29.6817
2010's7 (53.85)24.3611
2020's4 (30.77)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, S; Han, J; Li, Z; Liu, T; Wang, M; Wu, M1
Chen, S; Du, J; Li, R; Li, Z; Liu, T; Xing, S1
Ardenghi, P; Dias, M; Ferreira, MB; Izquierdo, I; Medina, JH; Salgueiro, JB1
Chen, BM; Dai, LL; Jia, SJ; Li, J; Liu, SK; Yang, GP; Yuan, H; Zhang, BK; Zhang, J; Zhou, LY; Zuo, XC1
Butterweck, V; Kelber, O; Nieber, K; Vissiennon, C1
Bernardi, MM; Díaz, IE; Estork, DM; Gusmão, DF; Montero, EF; Paciencia, ML; Reis, LF; Suffredini, IB; Varella, AD; Younes, RN1
Ghorbanihaghjo, A; Kosari-Nasab, M; Mesgari-Abbasi, M; Salari, AA; Shokouhi, G1
Amirabadizadeh, A; Askari, M; Brent, J; Farrokhfall, K; Foadoddini, M; Megarbane, B; Mehrpour, O; Miri-Moghaddam, E; Nakhaee, S1
Ahmed, T; Al-Khafaji, K; Araújo, IM; Bappi, MH; Coutinho, HDM; de Andrade, EM; Hanif, MA; Hossain, R; Islam, MS; Islam, MT; Khan, RA; Kowalska, G; Kowalski, R; Rahaman, MM; Sarkar, C1

Other Studies

13 other study(ies) available for diazepam and quercetin

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Design and synthesis of 3-(4-pyridyl)-5-(4-sulfamido-phenyl)-1,2,4-oxadiazole derivatives as novel GSK-3β inhibitors and evaluation of their potential as multifunctional anti-Alzheimer agents.
    European journal of medicinal chemistry, 2021, Jan-01, Volume: 209

    Topics: Alzheimer Disease; Animals; Cognition; Drug Design; Enzyme Inhibitors; Glucose; Glycogen Synthase Kinase 3 beta; Hep G2 Cells; Humans; Male; Mice, Inbred C57BL; Molecular Docking Simulation; Oxadiazoles; Reactive Oxygen Species

2021
Design, synthesis, and biological evaluation of novel (4-(1,2,4-oxadiazol-5-yl)phenyl)-2-aminoacetamide derivatives as multifunctional agents for the treatment of Alzheimer's disease.
    European journal of medicinal chemistry, 2022, Jan-05, Volume: 227

    Topics: Acetamides; Alzheimer Disease; Amyloid beta-Peptides; Antioxidants; Biphenyl Compounds; Butyrylcholinesterase; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Drug Design; Humans; Molecular Structure; Neuroprotective Agents; Oxadiazoles; Picrates; Protein Aggregates; Structure-Activity Relationship

2022
Anxiolytic natural and synthetic flavonoid ligands of the central benzodiazepine receptor have no effect on memory tasks in rats.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 58, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Chamomile; Diazepam; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Ligands; Male; Memory; Oils, Volatile; Plants, Medicinal; Psychomotor Performance; Quercetin; Rats; Rats, Wistar; Reaction Time; Receptors, GABA-A

1997
Effects of Ginkgo biloba extracts on diazepam metabolism: a pharmacokinetic study in healthy Chinese male subjects.
    European journal of clinical pharmacology, 2010, Volume: 66, Issue:5

    Topics: Asian People; Diazepam; Ginkgo biloba; Herb-Drug Interactions; Humans; Hydrocortisone; Male; Plant Extracts; Quercetin; Young Adult

2010
Route of administration determines the anxiolytic activity of the flavonols kaempferol, quercetin and myricetin--are they prodrugs?
    The Journal of nutritional biochemistry, 2012, Volume: 23, Issue:7

    Topics: 3,4-Dihydroxyphenylacetic Acid; Administration, Oral; Animals; Anti-Anxiety Agents; Diazepam; Dose-Response Relationship, Drug; Flavonoids; Injections, Intraperitoneal; Kaempferols; Male; Mice; Mice, Inbred C57BL; Phenylacetates; Prodrugs; Quercetin

2012
First chemical evaluation and toxicity of Casinga-cheirosa to Balb-c male mice.
    Molecules (Basel, Switzerland), 2014, Apr-02, Volume: 19, Issue:4

    Topics: alpha-Tocopherol; Animals; Body Weight; Diazepam; Gastrointestinal Hemorrhage; Humans; Lethal Dose 50; Male; Mice; Mice, Inbred BALB C; Organ Size; Piloerection; Plant Extracts; Quercetin; Quinic Acid; Respiration; Salicaceae; Sitosterols

2014
Quercetin mitigates anxiety-like behavior and normalizes hypothalamus-pituitary-adrenal axis function in a mouse model of mild traumatic brain injury.
    Behavioural pharmacology, 2019, Volume: 30, Issue:2 and 3-Sp

    Topics: Adrenocorticotropic Hormone; Animals; Anxiety; Anxiety Disorders; Brain Concussion; Corticosterone; Corticotropin-Releasing Hormone; Depression; Diazepam; Disease Models, Animal; Hypothalamo-Hypophyseal System; Male; Mice; Pituitary-Adrenal System; Quercetin; Stress, Psychological

2019
The effects of naloxone, diazepam, and quercetin on seizure and sedation in acute on chronic tramadol administration: an experimental study.
    Behavioral and brain functions : BBF, 2021, May-29, Volume: 17, Issue:1

    Topics: Animals; Diazepam; Male; Naloxone; Quercetin; Rats; Rats, Wistar; Seizures; Tramadol

2021
Anxiolytic-like Effect of Quercetin Possibly through GABA Receptor Interaction Pathway: In Vivo and In Silico Studies.
    Molecules (Basel, Switzerland), 2022, Oct-22, Volume: 27, Issue:21

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Diazepam; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Maze Learning; Mice; Quercetin; Receptors, GABA; Receptors, GABA-A

2022