diazepam has been researched along with piperidines in 116 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 47 (40.52) | 18.7374 |
1990's | 23 (19.83) | 18.2507 |
2000's | 28 (24.14) | 29.6817 |
2010's | 17 (14.66) | 24.3611 |
2020's | 1 (0.86) | 2.80 |
Authors | Studies |
---|---|
Hüther, KJ; Koch-Weser, J; Lundt, PV; Moser, L | 1 |
Dicsó, F; Dolinay, T; Hankovszky, E | 1 |
Lehmann, K; Schmidt, J | 1 |
Bjerkenstedt, L; Gullberg, B; Härnryd, C; Sedvall, G | 1 |
Leander, JD | 1 |
Gol'dovskaia, IL | 1 |
Nose, T; Takemoto, H | 1 |
Spiess, W | 1 |
Braestrup, C; Falch, E; Krogsgaard-Larsen, P; Nielsen, M | 2 |
Duvhök, C; Molander, L | 1 |
Baron, BM; Chi, EM; Harrison, BL; Kehne, JH; McCloskey, TC; Palfreyman, MG; Whitten, JP | 1 |
Almeida, SS; de Oliveira, LM; Graeff, FG | 2 |
Bakker, MH; Foster, AC | 1 |
Budziszewska, B; Grochmal, A; Przegaliński, E | 1 |
Idzikowski, C; James, RJ; Mills, FJ | 1 |
Borsini, F; D'Aranno, V; Lecci, A; Mancinelli, A; Meli, A; Stasi, MA; Volterra, G | 1 |
Dubrovina, NI; Il'iuchenok, RIu; Parkhomenko, RI | 1 |
Bezek, S; Durisová, M; Kállay, Z; Kukan, M; Laginová, V; Scasnár, V; Svoboda, V; Trnovec, T | 1 |
Bannister, SJ; Houser, VP; Hulse, JD; Kisicki, JC; Rasmussen, JG | 1 |
D'Angio, M; Scatton, B; Serrano, A | 1 |
Hiltunen, AJ; Järbe, TU | 1 |
Byberg, JR; Curtis, DR; Falch, E; Gynther, BD; Hjeds, H; Krogsgaard-Larsen, P; Labouta, IM | 1 |
Le Bihan, C; Simon, P; Soubrié, P; Thiébot, MH | 1 |
Colpaert, FC; Janssen, PA; Meert, TF; Niemegeers, CJ | 1 |
Lu, MW; Peng, JZ; Tao, SC | 1 |
Bian, CF; Xing, SH; Xu, PC | 1 |
Badian, M; Hundt, HK; Joubert, AL; Luus, HG; Meyer, BH; Müller, FO | 1 |
Iversen, LL; Wong, EH | 1 |
Curtis, DR; Falch, E; Krogsgaard-Larsen, P; Nielsen, L | 1 |
Creveling, CR; Daly, JW; Hollingsworth, EB; Lewandowski, G; Waters, JA | 1 |
Nomikos, GG; Spyraki, C | 1 |
de Chaffoy de Courcelles, D; Leysen, JE; Niemegeers, CJ; Van Gompel, P | 1 |
Bateman, DN | 1 |
Curtis, DR; Falch, E; Jacobsen, P; Krogsgaard-Larsen, P | 1 |
Kimishima, K; Ogura, C | 1 |
Dencker, SJ; Frankenberg, K; Malm, U; Zell, B | 1 |
Bjelke, E; Stovner, J; Theodorsen, L | 1 |
Clarke, SW; Kendall, MJ | 1 |
Ban, TA; Lehmann, HE | 1 |
Vinar, O | 1 |
Bartůnková, Z; Cerný, L; Drtilová, J; Sturma, J | 1 |
Kalff, G | 1 |
Linford, W | 1 |
Dobkin, AB; Evers, W; Ghanooni, S; Levy, AA; Thomas, ET | 1 |
Harthoorn, AM; Harthoorn, S; Sayer, PD | 1 |
Perez de Francisco, C | 1 |
Roth, F | 1 |
Laduron, PM; Luabeya, MK; Maloteaux, JM | 1 |
Gotsadze, GG; Kipiani, ZV; Nemsadze, NO; Shariia, RP | 1 |
Collins, RC; de Gubareff, T; Fuller, TA; Olney, JW | 1 |
Baggio, P; Danda, R; Fumiani, G | 1 |
Conway, PC; Corbett, R; Dunn, RW; Hartman, H; Helsley, GC; Kerman, LL; Strupczewski, JT; Woods, AT | 1 |
Bickerdike, MJ; Dourish, CT; Fletcher, A; Marsden, CA | 1 |
Aranko, K; Kuitunen, T; Mattila, MJ | 1 |
Lewander, P; Nordvall, M; Stenhammar, L; Wärngård, O | 1 |
Kluger, MT; McLean, C; Owen, H; Plummer, JL | 1 |
Fernández, AG; Palacios, JM; Silvestre, JS | 1 |
Misawa, M; Suzuki, T; Tsuda, M | 2 |
Griebel, G; Perrault, G; Sanger, DJ | 1 |
File, SE | 1 |
Baubichon, D; Burckhart, MF; Clarençon, D; Galonnier, M; Lallement, G; Masqueliez, C; Mestries, JC; Peoc'h, M | 1 |
Li, P; Tabibi, SE; Vishnuvajjala, R; Yalkowsky, SH | 1 |
Baubichon, D; Burckhart, MF; Clarençon, D; Galonnier, M; Lallement, G; Peoc'h, M | 1 |
Martin, BR; Wiley, JL | 1 |
Carlson, EC; de Felipe, C; Harrison, T; Hunt, S; Oates, B; Owen, S; Rupniak, NM; Seward, E; Wheeldon, A | 1 |
Griebel, G; Perrault, G; Rodgers, RJ; Sanger, DJ | 1 |
Ballard, TM; Higgins, GA; Sänger, S | 1 |
Almerigi, P; Antolini, F; Caporaloni, M; Di Mauro, L; Melloni, C; Urso, G | 1 |
Gasparini, F; Gentsch, C; Kuhn, R; Schoeffter, P; Spooren, WP | 1 |
Cecil, A; Crites, G; Goldenberg, R; Knapp, RJ; Malatynska, E; Miller, C; Shuck, C; Watkins, J | 1 |
Biedler, A; Kreuer, S; Larsen, R; Molter, G; Schoth, S; Wilhelm, W | 1 |
FUKUCHI, G | 1 |
FELLNER, CH | 1 |
Felouzis, E; Gustorff, B; Hoechtl, K; Kress, HG; Lehr, S; Sycha, T | 1 |
Bourin, M; Clénet, F; Fillion, G; Galons, H; Hascoët, M | 1 |
Griebel, G; Scatton, B; Stemmelin, J | 1 |
Bernöster, K; Dost, R; Egerland, U; Langen, B; Rundfeldt, C; Unverferth, K | 1 |
Biba, A; Christodoulou, A; Chrysikakou, S; Giannou, H; Kontis, D; Maillis, A; Pallidi, S; Rabavilas, A; Tsaltas, E | 1 |
Deprest, JA; Jani, JC; Lewi, LE; Marcus, MA; Missant, C; Teunkens, A; Van de Velde, M; Van Schoubroeck, D | 1 |
Bhagat, YA; Hamilton, MG; Kendall, EJ; Mikler, J; Obenaus, A | 1 |
Bahamonde, JA; Belda, C; Belda, J; Ferrandis, R; Llau, JV | 1 |
Kronbach, C; Lüddens, H; Rabe, H; Rundfeldt, C | 1 |
Krishna, DR; Kumar, KV; Palit, G | 1 |
Bocchi, A; Candini, M; Carrer, S; Donegà, L; Tartari, S | 1 |
Alizadeh, AM; Haghparast, A; Khani, A; Motamedi, F; Naderi, N; Rezaii, N; Saber-Tehrani, A | 1 |
Hayashi, S; Hirao, A; Imai, A; Sugie, Y; Toide, K; Yamada, Y | 1 |
Brocco, M; Dekeyne, A; Di Cara, B; Gobert, A; Millan, MJ; Ortuno, JC; Panayi, F; Rivet, JM | 1 |
Drago, F; Leggio, GM; Li Volsi, V; Mazzola, C; Micale, V; Tamburella, A | 1 |
Kitahara, M; Kitahara, T; Kubo, T; Okumura, S | 1 |
Cristino, L; Di Marzo, V; Drago, F; Leggio, GM; Micale, V; Petrosino, S; Tamburella, A | 2 |
Choi, DY; Kang, SH; Platt, B; Riedel, G | 1 |
Jain, NS; Manna, SS; Umathe, SN; Utturwar, KS | 1 |
Baarendse, PJ; Trezza, V; Vanderschuren, LJ | 1 |
Casarotto, PC; Gomes, FV; Guimarães, FS; Resstel, LB | 1 |
Ko, MC; Podlesnik, CA; Prinssen, EP; Wichmann, J; Winger, G; Woods, JH | 1 |
Cravatt, BF; Kinsey, SG; Lichtman, AH; Long, JZ; O'Neal, ST | 1 |
Hohmann, AG; Sciolino, NR; Zhou, W | 1 |
Gielen, MC; Lumb, MJ; Smart, TG | 1 |
Brito, GA; Cavalheiro, EA; da Costa, MA; da Cruz, GM; da Graça Naffah-Mazzacoratti, M; de Andrade, GM; de Barros Viana, GS; Felipe, CF; Leal, LK; Menezes, ML; Scorza, FA; Tavares, AF | 1 |
Binns, J; Bowlby, MR; Brunner, J; Cannon, CE; Coleman, PJ; Eddins, DM; Fox, SV; Garson, SL; Gotter, AL; Hodgson, R; Kuduk, SD; Mcdonald, TP; Renger, JJ; Savitz, AT; Stevens, J; Tannenbaum, PL; Tye, SJ; Uslaner, JM; Wang, X; Winrow, CJ; Yao, L | 1 |
Bègue, L; Bell, R; Duke, AA; Gilmore, PE; Page, D | 1 |
Dhingra, D; Gilhotra, N | 1 |
Austin, AT; Banks, CN; Bruun, DA; Hammock, BD; Inceoglu, B; Lein, PJ; Rogawski, MA; Tancredi, DJ; Vito, ST; Zolkowska, D | 1 |
Alderson, P; Kenth, JJ; Lewis, SR; Nicholson, A; Reed, SS; Smith, AF | 1 |
Jang, HJ; Joo, K; Kim, MJ; Lee, C; Rhie, DJ | 1 |
Lindsey, AM; Prinssen, EP; Rice, KC; Saccone, PA; Sulima, A; Wichmann, J; Woods, JH; Zelenock, KA | 1 |
Coleman, PJ; Fox, SV; Gotter, AL; Hargreaves, R; Kuduk, SD; Renger, JJ; Savitz, AT; Stevens, J; Tannenbaum, PL; Tye, SJ; Uslaner, JM; Winrow, CJ | 1 |
Alcorn, J; Benmansour, P; Billinsky, J; Duke-Novakovski, T | 1 |
Genewsky, A; Heinz, DE; Wotjak, CT | 1 |
Butler, CR; Guilmette, E; Pauletti, A; Piro, JR; Porcu, L; Rizzi, M; Salamone, A; Samad, TA; Sheehan, MJ; Terrone, G; Vezzani, A; Villa, BR | 1 |
Ito, S; Iwamoto, K; Kamimura, H; Mizunaga, M; Nakayama, K; Negoro, T; Nishiwaki, M; Nomura, Y; Suemizu, H; Yamazaki, H; Yoneda, N | 1 |
3 review(s) available for diazepam and piperidines
Article | Year |
---|---|
[Psychotropic therapy and intraocular pressure].
Topics: Amitriptyline; Analgesics; Antidepressive Agents; Chlorpromazine; Diazepam; Diphenhydramine; Eye Diseases; Glaucoma; Histamine H1 Antagonists; Humans; Imipramine; Intraocular Pressure; Lithium; Mental Disorders; Mephenesin; Meprobamate; Piperidines; Psychotropic Drugs; Secologanin Tryptamine Alkaloids; Tranquilizing Agents; Trihexyphenidyl | 1975 |
[Psychopharmaca in modern medicine].
Topics: Amphetamine; Antidepressive Agents; Barbiturates; Butyrophenones; Chlordiazepoxide; Chlorprothixene; Diazepam; Dibenzazepines; Guaifenesin; Hallucinogens; Humans; Hypnotics and Sedatives; Imipramine; Lithium; Lysergic Acid Diethylamide; Methylphenidate; Monoamine Oxidase Inhibitors; Oxazepam; Phenmetrazine; Phenothiazines; Phytotherapy; Piperidines; Plants, Medicinal; Psilocybin; Psychopharmacology; Rauwolfia; Reserpine; Tranquilizing Agents; Xanthenes | 1968 |
Anaesthetic and sedative agents used for electrical cardioversion.
Topics: Anesthetics; Apnea; Diazepam; Electric Countershock; Etomidate; Fentanyl; Humans; Hypnotics and Sedatives; Hypotension; Mental Recall; Methyl Ethers; Midazolam; Piperidines; Propofol; Randomized Controlled Trials as Topic; Remifentanil; Sevoflurane; Thiopental | 2015 |
16 trial(s) available for diazepam and piperidines
Article | Year |
---|---|
Effects of terfenadine and diphenhydramine alone or in combination with diazepam or alcohol on psychomotor performance and subjective feelings.
Topics: Adult; Benzhydryl Compounds; Diazepam; Diphenhydramine; Double-Blind Method; Drug Interactions; Emotions; Ethanol; Female; Flicker Fusion; Histamine H1 Antagonists; Humans; Male; Motor Skills; Piperidines; Reaction Time | 1978 |
[R 33812 (domperidon) i.v. and orally as antiemetic adjuvans for short anaesthetics induced with etomidate. A comparative study (author's transl)].
Topics: Adjuvants, Anesthesia; Administration, Oral; Antiemetics; Benzimidazoles; Diazepam; Dilatation and Curettage; Drug Interactions; Etomidate; Female; Humans; Injections, Intravenous; Piperidines; Premedication | 1979 |
A dose-response study examining the effects of ritanserin on human slow wave sleep.
Topics: Adolescent; Adult; Diazepam; Dose-Response Relationship, Drug; Double-Blind Method; Electroencephalography; Electromyography; Female; Humans; Male; Piperidines; Ritanserin; Sleep Stages; Sleep, REM | 1991 |
Effects of HOE 760 (histamine H2-receptor antagonist) on diazepam pharmacokinetics.
Topics: Adult; Clinical Trials as Topic; Diazepam; Double-Blind Method; Half-Life; Histamine H2 Antagonists; Humans; Male; Nordazepam; Piperidines; Time Factors | 1988 |
The action of cisapride on gastric emptying and the pharmacodynamics and pharmacokinetics of oral diazepam.
Topics: Adult; Blood Pressure; Chromatography, Gas; Cisapride; Diazepam; Double-Blind Method; Drug Interactions; Gastric Emptying; Heart Rate; Humans; Intestinal Absorption; Kinetics; Piperidines; Random Allocation | 1986 |
A controlled one-year study of pipotiazine palmitate and fluphenazine decanoate in chronic schizophrenic syndromes. Evaluation of results at 6 and 12 months' trial.
Topics: Adult; Aged; Antiparkinson Agents; Antipsychotic Agents; Basal Ganglia Diseases; Clinical Trials as Topic; Diazepam; Drug Evaluation; Female; Fluphenazine; Humans; Imipramine; Injections; Male; Middle Aged; Palmitic Acids; Piperidines; Psychiatric Status Rating Scales; Schizophrenia; Sulfonamides; Time Factors | 1973 |
Studies with new drugs in the treatment of convulsive disorders.
Topics: Adult; Aggression; Anticonvulsants; Anxiety; Carbamazepine; Clinical Trials as Topic; Diazepam; Dibenzazepines; Epilepsy; Frustration; Hallucinations; Humans; Intellectual Disability; Middle Aged; Nitriles; Object Attachment; Perceptual Disorders; Phenothiazines; Piperidines; Psychiatric Status Rating Scales; Psychopathology; Schizophrenia; Thiazines; Tranquilizing Agents | 1968 |
Propericiazin, diazepam, chlorpromazine and placebo in a doubleblind trial in pedopsychiatric therapy.
Topics: Adolescent; Aggression; Child; Child Behavior Disorders; Chlorpromazine; Clinical Trials as Topic; Diazepam; Evaluation Studies as Topic; Female; Humans; Male; Mental Disorders; Motor Activity; Nitriles; Phenothiazines; Piperidines; Placebos; Tranquilizing Agents | 1972 |
Diazepam effects on the performance of healthy subjects are not enhanced by treatment with the antihistamine ebastine.
Topics: Administration, Oral; Adult; Analysis of Variance; Butyrophenones; Chromatography, High Pressure Liquid; Diazepam; Double-Blind Method; Drug Interactions; Female; Histamine H1 Antagonists; Humans; Male; Piperidines; Psychomotor Performance | 1993 |
The effect of oral cisapride premedication on fasting gastric volumes.
Topics: Adjuvants, Anesthesia; Administration, Oral; Adolescent; Adult; Aged; Anesthesia, General; Cisapride; Diazepam; Double-Blind Method; Elective Surgical Procedures; Fasting; Gastric Emptying; Gastrointestinal Contents; Humans; Hydrogen-Ion Concentration; Hypnotics and Sedatives; Intubation, Gastrointestinal; Middle Aged; Piperidines; Placebos; Premedication; Serotonin Antagonists; Suction | 1995 |
[Narcotrend stages and end-tidal desflurane concentrations. An investigation during recovery from desflurane/remifentanil anaesthesia].
Topics: Adult; Anesthesia Recovery Period; Anesthetics, Inhalation; Anesthetics, Intravenous; Desflurane; Diazepam; Electroencephalography; Female; Humans; Isoflurane; Male; Middle Aged; Monitoring, Intraoperative; Piperidines; Preanesthetic Medication; Remifentanil | 2002 |
The effects of remifentanil and gabapentin on hyperalgesia in a new extended inflammatory skin pain model in healthy volunteers.
Topics: Acetates; Adult; Amines; Analgesics, Opioid; Cross-Over Studies; Cyclohexanecarboxylic Acids; Diazepam; Double-Blind Method; Drug Synergism; Excitatory Amino Acid Antagonists; Female; GABA Modulators; Gabapentin; gamma-Aminobutyric Acid; Humans; Hyperalgesia; Inflammation; Male; Pain Measurement; Pain Threshold; Physical Stimulation; Piperidines; Reaction Time; Remifentanil; Skin; Sunburn; Treatment Outcome | 2004 |
Remifentanil for fetal immobilization and maternal sedation during fetoscopic surgery: a randomized, double-blind comparison with diazepam.
Topics: Adult; Anesthetics, Intravenous; Blood Gas Analysis; Conscious Sedation; Diazepam; Double-Blind Method; Female; Fetal Movement; Fetoscopy; Heart Rate, Fetal; Humans; Hypnotics and Sedatives; Immobilization; Injections, Intravenous; Laser Coagulation; Monitoring, Intraoperative; Piperidines; Pregnancy; Remifentanil; Respiratory Mechanics; Spinal Cord | 2005 |
Short term analgesia based sedation in the Intensive Care Unit: morphine vs remifentanil + morphine.
Topics: Aged; Analgesia; Analgesics, Opioid; Blood Pressure; Conscious Sedation; Critical Care; Diazepam; Female; Humans; Hypnotics and Sedatives; Infusions, Intravenous; Male; Middle Aged; Morphine; Piperidines; Prospective Studies; Remifentanil; Respiration, Artificial | 2007 |
Effects of endolymphatic sac drainage with steroids for intractable Meniere's disease: a long-term follow-up and randomized controlled study.
Topics: Anti-Inflammatory Agents; Antidepressive Agents; Dexamethasone; Diazepam; Dimenhydrinate; Diuretics; Endolymphatic Sac; Female; Follow-Up Studies; Histamine H1 Antagonists; Humans; Male; Meniere Disease; Middle Aged; Piperidines; Prospective Studies | 2008 |
Blood concentrations of remifentanil during and after infusion in horses anesthetized with isoflurane and dexmedetomidine.
Topics: Analgesics, Opioid; Anesthetics, Inhalation; Animals; Dexmedetomidine; Diazepam; Drug Interactions; Female; Half-Life; Horses; Isoflurane; Ketamine; Male; Piperidines; Remifentanil; Xylazine | 2016 |
97 other study(ies) available for diazepam and piperidines
Article | Year |
---|---|
[Sandosten poisoning in childhood].
Topics: Child, Preschool; Diazepam; Drug Therapy, Combination; Female; Furosemide; Gastric Lavage; Histamine H1 Antagonists; Humans; Piperidines; Poisoning; Thiophenes | 1979 |
[Effect of psychotropic drugs on somatosensory evoked cortical potentials].
Topics: Animals; Anti-Anxiety Agents; Desipramine; Diazepam; Evoked Potentials; Female; Haloperidol; Hexobarbital; Medazepam; Piperidines; Rats; Somatosensory Cortex | 1979 |
Relationships between clinical and biochemical effects of melperone and thiothixene in psychotic women.
Topics: Butyrophenones; Diazepam; Female; Homovanillic Acid; Humans; Hydroxyindoleacetic Acid; Methoxyhydroxyphenylglycol; Paranoid Disorders; Piperidines; Prolactin; Schizophrenia; Therapeutic Equivalency; Thiothixene | 1979 |
Attenuating the rate-decreasing effects of phenylpiperidine analgesics by pentobarbital.
Topics: Analgesics; Animals; Chlorpromazine; Columbidae; Conditioning, Operant; Diazepam; Male; Meperidine; Pentobarbital; Piperidines; Reinforcement Schedule | 1979 |
The effect of penfluridol and some psychotropic drugs on monoamine metabolism in central nervous system.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Biogenic Amines; Brain; Brain Chemistry; Chlordiazepoxide; Chlorpromazine; Diazepam; Dopamine; Haloperidol; Homovanillic Acid; Hydroxyindoleacetic Acid; Male; Mice; Norepinephrine; Penfluridol; Pimozide; Piperazines; Piperidines; Psychotropic Drugs; Rats; Serotonin | 1975 |
Partial agonists for brain GABA/benzodiazepine receptor complex.
Topics: Animals; Benzodiazepines; Bicuculline; Brain; Crotonates; Diazepam; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Isoxazoles; Muscimol; Piperidines; Rats; Receptors, Drug; Sulfonic Acids | 1979 |
Acute effects of oxazepam, diazepam and methylperone, alone and in combination with alcohol on sedation, coordination and mood.
Topics: Adult; Attention; Butyrophenones; Diazepam; Drug Interactions; Emotions; Ethanol; Flicker Fusion; Humans; Male; Middle Aged; Motor Skills; Oxazepam; Piperidines; Tranquilizing Agents | 1976 |
NMDA receptor complex antagonists have potential anxiolytic effects as measured with separation-induced ultrasonic vocalizations.
Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Anxiety, Separation; Behavior, Animal; Buspirone; Diazepam; Dioxins; Dizocilpine Maleate; Dose-Response Relationship, Drug; Indoles; Kynurenic Acid; Maternal Deprivation; Mephenesin; Piperidines; Quinolizines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Serotonin Antagonists; Spiro Compounds; Valine; Vocalization, Animal | 1991 |
Early life protein malnutrition changes exploration of the elevated plus-maze and reactivity to anxiolytics.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Male; Piperidines; Propanolamines; Protein-Energy Malnutrition; Pyrimidines; Rats; Rats, Inbred Strains; Ritanserin | 1991 |
An investigation of the mechanisms of delayed neurodegeneration caused by direct injection of quinolinate into the rat striatum in vivo.
Topics: Adrenergic alpha-Antagonists; Animals; Anticonvulsants; Convulsants; Corpus Striatum; Dialysis; Diazepam; Dizocilpine Maleate; Glutamate Decarboxylase; Haloperidol; Ibotenic Acid; Injections; Male; Nerve Degeneration; Pipecolic Acids; Piperazines; Piperidines; Quinolinic Acid; Quinolinic Acids; Rats; Rats, Inbred Strains; Stereotaxic Techniques | 1991 |
Oxaprotiline enantiomers stimulate ACTH and corticosterone secretion in the rat.
Topics: Adrenergic alpha-Antagonists; Adrenocorticotropic Hormone; Animals; Antidepressive Agents; Benzylamines; Corticosterone; Dexamethasone; Diazepam; Dose-Response Relationship, Drug; Male; Maprotiline; Metergoline; Naloxone; Piperidines; Pyrimidines; Radioimmunoassay; Rats; Rats, Inbred Strains; Serotonin Antagonists; Stereoisomerism; Sulpiride; Sympathomimetics | 1991 |
Decreased reactivity to anxiolytics caused by early protein malnutrition in rats.
Topics: Animals; Anti-Anxiety Agents; Body Weight; Diazepam; Diet; Dose-Response Relationship, Drug; Hypertonic Solutions; Lactation; Male; Piperidines; Propanolamines; Protein-Energy Malnutrition; Pyrimidines; Rats; Rats, Inbred Strains; Ritanserin | 1990 |
Effect of serotoninergic drugs on stress-induced hyperthermia (SIH) in mice.
Topics: 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Body Temperature Regulation; Buspirone; Diazepam; Ergolines; Fenclonine; Fever; Flumazenil; Imidazoles; Male; Mice; Ondansetron; Piperazines; Piperidines; Ritanserin; Serotonin; Serotonin Antagonists; Stress, Psychological; Tetrahydronaphthalenes | 1990 |
[GABAergic modulation of amnesic trace reproduction by activation of the dopaminergic system].
Topics: Animals; Avoidance Learning; Bupropion; Diazepam; Dopamine Agents; Ergolines; Male; Mice; Mice, Inbred BALB C; Piperidines; Propiophenones; Quinpirole; Receptors, GABA-A | 1990 |
Irradiation of the head by 60Co opens the blood-brain barrier for drugs in rats.
Topics: Animals; Aspirin; Blood-Brain Barrier; Brain; Carbamates; Chloramphenicol; Cobalt Radioisotopes; Cranial Irradiation; Diazepam; Etimizol; Male; Piperidines; Rats; Rats, Inbred Strains; Regression Analysis | 1990 |
Evaluation of the potential for interactions of paroxetine with diazepam, cimetidine, warfarin, and digoxin.
Topics: Adult; Antidepressive Agents; Biological Availability; Cimetidine; Diazepam; Digoxin; Drug Interactions; Humans; Male; Paroxetine; Piperidines; Serotonin Antagonists; Warfarin | 1989 |
NMDA antagonists block restraint-induced increase in extracellular DOPAC in rat nucleus accumbens.
Topics: 3,4-Dihydroxyphenylacetic Acid; Adrenergic alpha-Antagonists; Animals; Aspartic Acid; Carbolines; Convulsants; Diazepam; Male; N-Methylaspartate; Nucleus Accumbens; Phenylacetates; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Restraint, Physical; Riluzole; Septal Nuclei; Thiazoles | 1989 |
Limited stimulus generalization between delta 9-THC and diazepam in pigeons and gerbils.
Topics: Animals; Benzodiazepinones; Columbidae; Diazepam; Discrimination, Psychological; Dronabinol; Generalization, Stimulus; Gerbillinae; Male; Piperidines; Receptors, GABA-A | 1988 |
Synthesis and biological activity of a GABAA agonist which has no effect on benzodiazepine binding and of structurally related glycine antagonists.
Topics: Animals; Bicuculline; Brain Chemistry; Chemical Phenomena; Chemistry; Diazepam; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Isoxazoles; Oxazoles; Piperidines; Pyrrolidines; Rats; Receptors, GABA-A; Synaptic Membranes | 1987 |
Benzodiazepines reduce the tolerance to reward delay in rats.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Choice Behavior; Diazepam; Flumazenil; Male; Piperidines; Rats; Rats, Inbred Strains; Reward; Serotonin Antagonists; Synaptic Transmission; Zimeldine | 1985 |
Behavioral and 5-HT antagonist effects of ritanserin: a pure and selective antagonist of LSD discrimination in rat.
Topics: 5-Hydroxytryptophan; Animals; Anti-Anxiety Agents; Anxiety; Chlordiazepoxide; Diazepam; Disease Models, Animal; Histamine H2 Antagonists; Humans; Lysergic Acid Diethylamide; Male; Motor Activity; Piperidines; Pyrimidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists | 1985 |
[Central convulsive action of l-securinine].
Topics: Alkaloids; Animals; Azepines; Central Nervous System Stimulants; Diazepam; Drug Synergism; gamma-Aminobutyric Acid; Heterocyclic Compounds, 4 or More Rings; Heterocyclic Compounds, Bridged-Ring; Humans; Lactones; Male; Mice; Piperidines; Seizures | 1986 |
[The interactions between dihydroetorphine, L-tetrahydropalmatine, B-7601 and diazepam].
Topics: Alkaloids; Anesthesia, General; Anesthesia, Intravenous; Animals; Antipsychotic Agents; Benzilates; Berberine Alkaloids; Diazepam; Dogs; Drug Interactions; Etorphine; Female; Male; Mice; Morphinans; Piperidines; Rabbits | 1986 |
Modulation of [3H]diazepam binding in rat cortical membranes by GABAA agonists.
Topics: Androstanes; Animals; Azasteroids; Bicuculline; Cell Membrane; Cerebral Cortex; Diazepam; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Isonicotinic Acids; Isoxazoles; Muscimol; Piperidines; Rats; Receptors, GABA-A; Taurine | 1985 |
GABA agonists. Resolution, absolute stereochemistry, and enantioselectivity of (S)-(+)- and (R)-(-)-dihydromuscimol.
Topics: Animals; Bicuculline; Brain; Cats; Chemical Phenomena; Chemistry; Diazepam; gamma-Aminobutyric Acid; Isoxazoles; Molecular Conformation; Muscimol; Neurons; Oxazolidinones; Piperidines; Rats; Receptors, GABA-A; Spinal Cord; Stereoisomerism; Structure-Activity Relationship; Synaptic Membranes | 1985 |
Anticonvulsant activity of piperidinol and (dialkylamino)alkanol esters.
Topics: Amino Alcohols; Animals; Anticonvulsants; Ataxia; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Diazepam; Electroshock; Esters; Muscimol; Pentylenetetrazole; Phenytoin; Piperidines; Rats; Receptors, GABA-A; Structure-Activity Relationship | 1986 |
Effects of ritanserin on the rewarding properties of d-amphetamine, morphine and diazepam revealed by conditioned place preference in rats.
Topics: Analgesia; Animals; Conditioning, Operant; Dextroamphetamine; Diazepam; Exploratory Behavior; Male; Morphine; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Reference Values; Reinforcement, Psychology; Reward; Ritanserin; Serotonin Antagonists | 1988 |
Opposite regulation of serotonin-S2 and dopamine-D2 receptors in rat brain following chronic receptor blockade.
Topics: Animals; Apomorphine; Behavior, Animal; Corpus Striatum; Diazepam; Dopamine Antagonists; Frontal Lobe; Gene Expression Regulation; Ketanserin; Male; Models, Biological; Piperidines; Pyrimidinones; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Serotonin Antagonists; Tryptamines | 1987 |
GABA-mimetic activity and effects on diazepam binding of aminosulphonic acids structurally related to piperidine-4-sulphonic acid.
Topics: Animals; Binding Sites; Brain; Diazepam; gamma-Aminobutyric Acid; Piperidines; Pyridines; Pyrrolidines; Rats; Structure-Activity Relationship; Synaptic Membranes | 1985 |
Central nervous actions and screening methods of antidepressants.
Topics: Acetylcholine; Amitriptyline; Animals; Antidepressive Agents; Behavior, Animal; Biogenic Amines; Blood Pressure; Brain Chemistry; Central Nervous System; Diazepam; Electroshock; Ethanol; Hexobarbital; Hypertension; Hypothermia, Induced; Imipramine; Iproniazid; Methamphetamine; Mice; Nialamide; Physostigmine; Piperidines; Reserpine; Tremorine | 1972 |
[Experimental studies on prevention of muscular cramps caused by 2 F-type schistosomicides].
Topics: Acrylamides; Animals; Anthelmintics; Cats; Chlordiazepoxide; Diazepam; Mice; Muscle Cramp; Nitrofurans; Piperidines; Rabbits; Schistosomiasis; Schistosomicides | 1974 |
Sensitivity to gallamine and pancuronium with special reference to serum proteins.
Topics: Androstanes; Anesthesia, General; Blood Proteins; Body Surface Area; Diazepam; Female; Gallamine Triethiodide; Humans; Injections, Intramuscular; Neuromuscular Nondepolarizing Agents; Piperidines; Serum Albumin; Thiopental | 1971 |
Prolonged coma after tetanus.
Topics: Aged; Androstanes; Coma; Diazepam; Female; Humans; Neuromuscular Nondepolarizing Agents; Piperidines; Respiration, Artificial; Tetanus | 1972 |
Diazepam combination-anesthesia.
Topics: Animals; Blood Circulation; Blood Pressure; Cardiac Output; Diazepam; Dogs; Drug Synergism; Fentanyl; Heart Rate; Humans; Isonipecotic Acids; Morphine; Piperidines; Vascular Resistance | 1974 |
New horizons in psychopharmacology.
Topics: Animals; Anthracenes; Antidepressive Agents; Anxiety; Benzamides; Benzazepines; Butyrophenones; Chlordiazepoxide; Chlorprothixene; Diazepam; Dibenzothiazepines; Humans; Monoamine Oxidase Inhibitors; Nitrazepam; Oxazepam; Pharmacogenetics; Phenothiazines; Piperidines; Plants, Medicinal; Psychopharmacology; Rauwolfia; Sleep; Tranquilizing Agents | 1972 |
Pancuronium bromide (Pavulon) evaluation of its clinical pharmacology.
Topics: Androstanes; Anesthesia, Inhalation; Atropine; Blood Pressure; Body Temperature; Carbon Dioxide; Diazepam; Electrocardiography; Female; Fentanyl; Halothane; Histamine; Humans; Hydrogen-Ion Concentration; Intubation, Intratracheal; Male; Meperidine; Methoxyflurane; Middle Aged; Neostigmine; Nitrous Oxide; Oxygen; Piperidines; Potassium; Pulse; Respiration; Surgical Procedures, Operative; Thiopental; Urination | 1971 |
Two field operations on the African lion (Felis leo).
Topics: Anesthesia, Intravenous; Animals; Antisepsis; Carnivora; Chlorpromazine; Diazepam; Eye Foreign Bodies; Fracture Fixation, Intramedullary; Humeral Fractures; Male; Piperidines; Thiopental | 1971 |
[Psychopharmacological treatment of anxiety].
Topics: Adult; Amitriptyline; Anxiety; Benzazepines; Carbamates; Chlordiazepoxide; Diazepam; Dibenzazepines; Female; Humans; Ketones; Meprobamate; Methotrimeprazine; Nitro Compounds; Oxazepam; Piperidines; Thioridazine | 1971 |
[Anesthesia in cardioversion].
Topics: Anesthesia, General; Anesthetics; Arrhythmias, Cardiac; Diazepam; Electric Countershock; Humans; Methods; Nitrous Oxide; Piperidines; Preanesthetic Medication; Thiopental | 1969 |
Regional and cortical laminar distributions of serotonin S2, benzodiazepine, muscarinic, and dopamine D2 receptors in human brain.
Topics: Adult; Aged; Brain; Cerebral Cortex; Diazepam; Humans; Ketanserin; Male; Middle Aged; Piperidines; Quinuclidinyl Benzilate; Receptors, Cell Surface; Receptors, Dopamine; Receptors, GABA-A; Receptors, Muscarinic; Receptors, Serotonin; Spiperone; Tissue Distribution | 1984 |
Two or more conformations of benzodiazepine receptors depending on GABA receptors and other variables.
Topics: Animals; Benzodiazepines; Bicuculline; Brain; Diazepam; gamma-Aminobutyric Acid; Macromolecular Substances; Male; Muscimol; Piperidines; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Structure-Activity Relationship; Synaptic Membranes | 1980 |
[Functional state of the fetus during labor with the use of spasmoanalgesic and tranquilizing agents].
Topics: Anesthesia, Obstetrical; Benzophenones; Butylscopolammonium Bromide; Diazepam; Dipyrone; Drug Combinations; Female; Fetus; Humans; Infant, Newborn; Labor, Obstetric; Parasympatholytics; Piperidines; Pregnancy | 1983 |
Systemic dipiperidinoethane mimics the convulsant and neurotoxic actions of kainic acid.
Topics: Animals; Behavior, Animal; Diazepam; Hippocampus; Kainic Acid; Male; Piperidines; Pyrrolidines; Rats; Seizures | 1980 |
[Tipepidine poisoning].
Topics: Akathisia, Drug-Induced; Child, Preschool; Diazepam; Female; Humans; Medication Errors; Piperidines; Psychomotor Agitation | 1980 |
Effects of atypical antipsychotic agents on social behavior in rodents.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Apomorphine; Benzazepines; Catalepsy; Chlorpromazine; Clozapine; Diazepam; Haloperidol; Isoxazoles; Male; Mice; Mice, Inbred Strains; Piperidines; Raclopride; Radioligand Assay; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Serotonin; Risperidone; Salicylamides; Social Behavior | 1993 |
The influence of 5-hydroxytryptamine re-uptake blockade on CCK receptor antagonist effects in the rat elevated zero-maze.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Devazepide; Diazepam; Indoles; Male; Maze Learning; Meglumine; Niacinamide; Phenylurea Compounds; Piperazines; Piperidines; Rats; Receptors, Cholecystokinin; Selective Serotonin Reuptake Inhibitors; Zimeldine | 1994 |
Oral versus intravenous premedication for small bowel biopsy in children: effect on procedure and fluoroscopy times.
Topics: Administration, Oral; Adolescent; Biopsy; Celiac Disease; Child; Child, Preschool; Cisapride; Diazepam; Fluoroscopy; Humans; Infant; Infusions, Intravenous; Intestine, Small; Metoclopramide; Midazolam; Piperidines; Premedication; Serotonin Antagonists; Trimeprazine | 1993 |
Effects of 5-HT4 receptor antagonists on rat behaviour in the elevated plus-maze test.
Topics: Animals; Behavior, Animal; Diazepam; Dioxanes; Dose-Response Relationship, Drug; Granisetron; Indoles; Male; Maze Learning; Piperidines; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Sulfonamides | 1996 |
Recovery of decreased seizure threshold for pentylenetetrazole during diazepam withdrawal by NMDA receptor antagonists.
Topics: Animals; Anticonvulsants; Convulsants; Diazepam; Disease Models, Animal; Dizocilpine Maleate; Drug Interactions; Excitatory Amino Acid Antagonists; Infusions, Intravenous; Injections, Intraperitoneal; Injections, Subcutaneous; Kynurenic Acid; Male; Mice; Neuroprotective Agents; Pentylenetetrazole; Piperidines; Receptors, N-Methyl-D-Aspartate; Seizures; Substance Withdrawal Syndrome | 1997 |
A comparative study of the effects of selective and non-selective 5-HT2 receptor subtype antagonists in rat and mouse models of anxiety.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Diazepam; Drinking; Fluorobenzenes; Indoles; Male; Maze Learning; Mianserin; Mice; Mice, Inbred BALB C; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists | 1997 |
Anxiolytic action of a neurokinin1 receptor antagonist in the social interaction test.
Topics: Animals; Anti-Anxiety Agents; Diazepam; Drug Tolerance; Handling, Psychological; Interpersonal Relations; Lighting; Male; Motor Activity; Neurokinin-1 Receptor Antagonists; Piperidines; Quinolines; Rats; Stress, Psychological | 1997 |
Nerve agent poisoning in primates: antilethal, anti-epileptic and neuroprotective effects of GK-11.
Topics: Animals; Anticonvulsants; Atropine; Brain; Chemical Warfare Agents; Cholinesterase Inhibitors; Cholinesterase Reactivators; Cyclohexanes; Cyclohexenes; Diazepam; Drug Combinations; Excitatory Amino Acid Antagonists; Injections, Intravenous; Macaca fascicularis; Male; Muscarinic Antagonists; Neuroprotective Agents; Piperidines; Pralidoxime Compounds; Seizures; Soman; Staining and Labeling; Time Factors | 1998 |
Evaluation of in vitro precipitation methods.
Topics: Antineoplastic Agents; Chemical Precipitation; Chemistry, Pharmaceutical; Diazepam; Flavonoids; Injections; Piperidines; Solubility; Solutions; Time Factors | 1998 |
NMDA receptor antagonists potently suppress the spontaneous withdrawal signs induced by discontinuation of long-term diazepam treatment in Fischer 344 rats.
Topics: Administration, Oral; Animals; Anorexia; Anti-Anxiety Agents; Behavior, Animal; Diazepam; Dizocilpine Maleate; Eating; Emotions; Excitatory Amino Acid Antagonists; Male; Motor Activity; Piperidines; Rats; Rats, Inbred F344; Receptors, N-Methyl-D-Aspartate; Substance Withdrawal Syndrome; Time Factors; Weight Loss | 1998 |
Acute soman poisoning in primates neither pretreated nor receiving immediate therapy: value of gacyclidine (GK-11) in delayed medical support.
Topics: Animals; Anticonvulsants; Antidotes; Atropine; Brain; Cerebellum; Cerebral Cortex; Chemical Warfare Agents; Cholinesterase Reactivators; Cyclohexanes; Cyclohexenes; Diazepam; Drug Therapy, Combination; Electrocardiography; Excitatory Amino Acid Antagonists; Haplorhini; Macaca fascicularis; Male; Piperidines; Poisoning; Pralidoxime Compounds; Seizures; Soman; Time Factors | 1999 |
Effects of SR141716A on diazepam substitution for delta9-tetrahydrocannabinol in rat drug discrimination.
Topics: Animals; Cannabinoids; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Dronabinol; GABA Modulators; Generalization, Psychological; Hallucinogens; Male; Piperidines; Pyrazoles; Rats; Rats, Long-Evans; Rats, Sprague-Dawley; Rimonabant | 1999 |
Pharmacological blockade or genetic deletion of substance P (NK(1)) receptors attenuates neonatal vocalisation in guinea-pigs and mice.
Topics: Animals; Animals, Newborn; Anti-Anxiety Agents; Antidepressive Agents; Behavior, Animal; Buspirone; Diazepam; Dose-Response Relationship, Drug; Female; Fluoxetine; Gene Deletion; Guinea Pigs; Imipramine; Injections, Intraventricular; Male; Mice; Mice, Inbred Strains; Motor Activity; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Social Isolation; Stress, Psychological; Substance P; Tetrazoles; Vocalization, Animal | 2000 |
The effects of compounds varying in selectivity as 5-HT(1A) receptor antagonists in three rat models of anxiety.
Topics: Aminopyridines; Animals; Anxiety; Cyclohexane Monoterpenes; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drinking Behavior; Isoquinolines; Male; Maze Learning; Motor Activity; Pindolol; Piperazines; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Succinimides | 2000 |
Inhibition of shock-induced foot tapping behaviour in the gerbil by a tachykinin NK1 receptor antagonist.
Topics: Animals; Anti-Anxiety Agents; Antidepressive Agents, Second-Generation; Aprepitant; Conditioning, Operant; Diazepam; Female; Fluoxetine; Gerbillinae; Humans; Male; Morpholines; Motor Activity; Neurokinin-1 Receptor Antagonists; Piperidines; Receptors, Neurokinin-1 | 2001 |
[Propofol and remifentanil in day surgery].
Topics: Adult; Ambulatory Surgical Procedures; Anesthesia Recovery Period; Anesthesia, General; Anesthetics, Intravenous; Conscious Sedation; Diazepam; Humans; Midazolam; Piperidines; Preanesthetic Medication; Propofol; Remifentanil | 2000 |
Pharmacological and endocrinological characterisation of stress-induced hyperthermia in singly housed mice using classical and candidate anxiolytics (LY314582, MPEP and NKP608).
Topics: Adrenocorticotropic Hormone; Analysis of Variance; Animals; Anti-Anxiety Agents; Benzodiazepines; Body Temperature; Bridged Bicyclo Compounds; Buspirone; Chlordiazepoxide; Clobazam; Corticosterone; Diazepam; Ethanol; Hyperthermia, Induced; Male; Mice; Mice, Inbred ICR; Oxazepam; Piperidines; Pyridines; Quinolines; Reproducibility of Results; Stress, Physiological | 2002 |
Antidepressant activity of memory-enhancing drugs in the reduction of submissive behavior model.
Topics: Animals; Antidepressive Agents; Competitive Behavior; Desipramine; Diazepam; Dioxoles; Dose-Response Relationship, Drug; Fluoxetine; Injections, Intraperitoneal; Male; Maze Learning; Models, Animal; Nootropic Agents; Piperidines; Piracetam; Pyrrolidinones; Rats; Rats, Sprague-Dawley | 2002 |
[DRUGS ACTING ON THE NERVOUS SYSTEM. (2). WITH SPECIAL REFERENCE TO TRANQUILIZERS AND ANTIDEPRESSIVE AGENTS].
Topics: Amides; Amitriptyline; Antidepressive Agents; Benactyzine; Chemical Phenomena; Chemistry; Chlordiazepoxide; Desipramine; Diazepam; Haloperidol; Humans; Hydroxyzine; Hypnotics and Sedatives; Imipramine; Isocarboxazid; Meprobamate; Methylphenidate; Monoamine Oxidase Inhibitors; Nervous System; Nialamide; Pharmacology; Phenelzine; Piperidines; Tranquilizing Agents; Tranylcypromine; Tryptamines | 1963 |
EARLY RECOGNITION OF DEPRESSION.
Topics: Amitriptyline; Amphetamine; Amphetamines; Barbiturates; Benactyzine; Chlordiazepoxide; Deanol; Depression; Depressive Disorder; Diagnosis; Diazepam; Drug Therapy; Geriatrics; Humans; Imipramine; Meprobamate; Methylphenidate; Monoamine Oxidase Inhibitors; Phenmetrazine; Piperidines; Psychotherapy; Toxicology | 1964 |
Anxiolytic profile of HG1, a 5-HT-moduline antagonist, in three mouse models of anxiety.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Dose-Response Relationship, Drug; Electroshock; Light; Male; Mice; Motor Activity; Neuropeptides; Oligopeptides; Piperidines; Serotonin Antagonists | 2004 |
Effects of the cannabinoid CB1 receptor antagonist rimonabant in models of emotional reactivity in rodents.
Topics: Aggression; Analysis of Variance; Animals; Anti-Anxiety Agents; Antidepressive Agents, Second-Generation; Behavior, Animal; Depression; Diazepam; Dose-Response Relationship, Drug; Electroshock; Emotions; Fluoxetine; Gerbillinae; Immobility Response, Tonic; Male; Maze Learning; Mice; Models, Animal; Neuropsychological Tests; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Rimonabant | 2005 |
Characterization in rats of the anxiolytic potential of ELB139 [1-(4-chlorophenyl)-4-piperidin-1-yl-1,5-dihydro-imidazol-2-on], a new agonist at the benzodiazepine binding site of the GABAA receptor.
Topics: Animals; Anti-Anxiety Agents; Binding Sites; Binding, Competitive; Conflict, Psychological; Diazepam; Drug Tolerance; Flumazenil; Flunitrazepam; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Imidazoles; Light; Male; Membrane Potentials; Patch-Clamp Techniques; Piperidines; Rats; Rats, Wistar | 2005 |
Reinforced spatial alternation as an animal model of obsessive-compulsive disorder (OCD): investigation of 5-HT2C and 5-HT1D receptor involvement in OCD pathophysiology.
Topics: Animals; Anti-Anxiety Agents; Antidepressive Agents, Tricyclic; Desipramine; Diazepam; Disease Models, Animal; Fluoxetine; Indoles; Male; Maze Learning; Obsessive-Compulsive Disorder; Piperazines; Piperidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2C; Reinforcement, Psychology; Selective Serotonin Reuptake Inhibitors; Serotonin Receptor Agonists; Tryptamines | 2005 |
Neuroprotection from soman-induced seizures in the rodent: evaluation with diffusion- and T2-weighted magnetic resonance imaging.
Topics: Animals; Anticonvulsants; Brain; Cell Death; Cyclohexanes; Cyclohexenes; Diazepam; Diffusion Magnetic Resonance Imaging; Magnetic Resonance Imaging; Male; Neuroprotective Agents; Piperidines; Rats; Rats, Sprague-Dawley; Seizures; Soman; Status Epilepticus | 2005 |
Anesthesia for cardiac surgery on a patient with stiff person syndrome.
Topics: Adult; Analgesics, Opioid; Anesthesia; Anesthetics, Intravenous; Anticonvulsants; Cardiopulmonary Bypass; Diazepam; Etomidate; Female; Fentanyl; Heart Valve Diseases; Heparin; Humans; Midazolam; Morphine; Neuromuscular Nondepolarizing Agents; Pain, Postoperative; Pancuronium; Piperidines; Propofol; Remifentanil; Stiff-Person Syndrome | 2005 |
The novel anxiolytic ELB139 displays selectivity to recombinant GABA(A) receptors different from diazepam.
Topics: Animals; Anti-Anxiety Agents; Cell Line, Transformed; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; GABA-A Receptor Agonists; Humans; Imidazoles; Membrane Potentials; Patch-Clamp Techniques; Piperidines; Rats; Receptors, GABA-A; Transfection | 2007 |
Histaminergic H1 receptors mediate L-histidine-induced anxiety in elevated plus-maze test in mice.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzothiazoles; Diazepam; Dose-Response Relationship, Drug; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Male; Mice; Phenoxypropanolamines; Piperidines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H3 | 2007 |
Interaction between cannabinoid compounds and diazepam on anxiety-like behaviour of mice.
Topics: Amidohydrolases; Animals; Anxiety; Arachidonic Acids; Behavior, Animal; Benzamides; Benzoxazines; Cannabinoids; Carbamates; Data Interpretation, Statistical; Diazepam; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Enzyme Inhibitors; GABA Modulators; Hypnotics and Sedatives; Male; Mice; Morpholines; Naphthalenes; Piperidines; Postural Balance; Pyrazoles; Receptor, Cannabinoid, CB1 | 2008 |
Pharmacological characterization of the newly synthesized nociceptin/orphanin FQ-receptor agonist 1-[1-(1-methylcyclooctyl)-4-piperidinyl]-2-[(3R)-3-piperidinyl]-1H-benzimidazole as an anxiolytic agent.
Topics: Animals; Anti-Anxiety Agents; Benzimidazoles; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Ethanol; Humans; Male; Memory; Mice; Motor Activity; Nociceptin Receptor; Piperidines; Receptors, Opioid | 2008 |
The melanin-concentrating hormone1 receptor antagonists, SNAP-7941 and GW3430, enhance social recognition and dialysate levels of acetylcholine in the frontal cortex of rats.
Topics: Acetylcholine; Aggression; Animals; Anxiety; Ataxia; Brain Chemistry; Conflict, Psychological; Data Interpretation, Statistical; Depression; Diazepam; Hypnotics and Sedatives; Microdialysis; Motor Activity; Muscarinic Antagonists; Piperidines; Prefrontal Cortex; Pyrimidines; Rats; Rats, Wistar; Receptors, Somatostatin; Recognition, Psychology; Scopolamine; Social Behavior; Swimming | 2008 |
Behavioral effects of saredutant, a tachykinin NK2 receptor antagonist, in experimental models of mood disorders under basal and stress-related conditions.
Topics: Animals; Anti-Anxiety Agents; Antidepressive Agents, Tricyclic; Anxiety; Behavior, Animal; Benzamides; Clomipramine; Depressive Disorder; Diazepam; Electroshock; Grooming; Male; Mice; Mood Disorders; Motor Activity; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Stress, Psychological; Swimming | 2008 |
Anxiolytic effects in mice of a dual blocker of fatty acid amide hydrolase and transient receptor potential vanilloid type-1 channels.
Topics: Amidohydrolases; Anilides; Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Benzamides; Brain; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Cinnamates; Diazepam; Exploratory Behavior; Male; Mice; Mice, Inbred C57BL; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Serotonin; TRPV Cation Channels | 2009 |
Scopolamine-induced deficits in social memory in mice: reversal by donepezil.
Topics: Animals; Anti-Anxiety Agents; Cholinesterase Inhibitors; Diazepam; Donepezil; Dose-Response Relationship, Drug; Exploratory Behavior; Female; Indans; Memory; Memory Disorders; Mice; Mice, Inbred C57BL; Muscarinic Antagonists; Neuropsychological Tests; Nootropic Agents; Piperidines; Random Allocation; Scopolamine; Social Behavior; Time Factors | 2009 |
Endocannabinoids mediate anxiolytic-like effect of acetaminophen via CB1 receptors.
Topics: Acetaminophen; Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Behavior, Animal; Cannabinoid Receptor Modulators; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drinking; Endocannabinoids; Injections, Intraventricular; Interpersonal Relations; Male; Mice; Motor Activity; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1 | 2009 |
Altered responses of dopamine D3 receptor null mice to excitotoxic or anxiogenic stimuli: Possible involvement of the endocannabinoid and endovanilloid systems.
Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Anti-Inflammatory Agents, Non-Steroidal; Anxiety; Arachidonic Acids; Brain; Cannabinoid Receptor Modulators; Capsaicin; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Endocannabinoids; Epilepsy; GABA Antagonists; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Knockout; Picrotoxin; Piperidines; Pyrazoles; Reaction Time; Receptor, Cannabinoid, CB1; Receptors, Dopamine D3; Serotonin; TRPV Cation Channels | 2009 |
Prosocial effects of nicotine and ethanol in adolescent rats through partially dissociable neurobehavioral mechanisms.
Topics: Aging; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Central Nervous System Depressants; Diazepam; Dopamine Antagonists; Ethanol; Exploratory Behavior; Flupenthixol; Locomotion; Male; Naloxone; Narcotic Antagonists; Nicotine; Nicotinic Agonists; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Rimonabant; Social Behavior | 2009 |
Cannabidiol inhibitory effect on marble-burying behaviour: involvement of CB1 receptors.
Topics: Animals; Behavior, Animal; Cannabidiol; Diazepam; Dose-Response Relationship, Drug; Hypnotics and Sedatives; Male; Mice; Mice, Inbred C57BL; Motor Activity; Paroxetine; Piperazines; Piperidines; Pyrazoles; Pyridines; Receptor, Cannabinoid, CB1; Receptor, Serotonin, 5-HT1A; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Synaptic Transmission | 2010 |
The effects of nociceptin/orphanin FQ receptor agonist Ro 64-6198 and diazepam on antinociception and remifentanil self-administration in rhesus monkeys.
Topics: Animals; Benzimidazoles; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Female; Imidazoles; Macaca mulatta; Male; Narcotic Antagonists; Nociceptin Receptor; Pain Measurement; Piperidines; Receptors, Opioid; Remifentanil; Self Administration; Spiro Compounds | 2011 |
Inhibition of endocannabinoid catabolic enzymes elicits anxiolytic-like effects in the marble burying assay.
Topics: Amidohydrolases; Animals; Anti-Anxiety Agents; Anxiety Disorders; Benzodioxoles; Cannabinoid Receptor Modulators; Diazepam; Disease Models, Animal; Dronabinol; Endocannabinoids; Enzyme Inhibitors; Male; Mice; Mice, Inbred C57BL; Monoacylglycerol Lipases; Obsessive-Compulsive Disorder; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant | 2011 |
Enhancement of endocannabinoid signaling with JZL184, an inhibitor of the 2-arachidonoylglycerol hydrolyzing enzyme monoacylglycerol lipase, produces anxiolytic effects under conditions of high environmental aversiveness in rats.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Benzodioxoles; Cannabinoid Receptor Modulators; Catalepsy; Diazepam; Endocannabinoids; Glycerides; Male; Monoacylglycerol Lipases; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; Signal Transduction | 2011 |
Benzodiazepines modulate GABAA receptors by regulating the preactivation step after GABA binding.
Topics: Animals; Benzodiazepines; Binding Sites; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Ion Channel Gating; Isoxazoles; Larva; Membrane Potentials; Models, Biological; Mutation; Oocytes; Patch-Clamp Techniques; Piperidines; Protein Binding; Protein Subunits; Receptors, GABA-A; Xenopus | 2012 |
Piperine decreases pilocarpine-induced convulsions by GABAergic mechanisms.
Topics: Alkaloids; Amino Acids; Animals; Anticonvulsants; Antioxidants; Atropine; Benzodioxoles; Biogenic Monoamines; Brain; Diazepam; Disease Models, Animal; Epilepsy; Flumazenil; gamma-Aminobutyric Acid; Humans; Male; Memantine; Mice; Nimodipine; Nitrites; Pilocarpine; Piperidines; Polyunsaturated Alkamides; Seizures; Tumor Necrosis Factor-alpha | 2013 |
Orexin receptor antagonists differ from standard sleep drugs by promoting sleep at doses that do not disrupt cognition.
Topics: Administration, Oral; Animals; Attention; Azabicyclo Compounds; Choice Behavior; Cognition; Cytoskeletal Proteins; Diazepam; Eszopiclone; gamma-Aminobutyric Acid; Hippocampus; Hypnotics and Sedatives; Macaca mulatta; Male; Memory, Short-Term; Nerve Tissue Proteins; Orexin Receptors; Piperazines; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Recognition, Psychology; Sleep; Task Performance and Analysis; Time Factors; Triazoles; Zolpidem | 2013 |
Anxiolytic-like effects observed in rats exposed to the elevated zero-maze following treatment with 5-HT2/5-HT3/5-HT4 ligands.
Topics: Aniline Compounds; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Male; Maze Learning; Oxazines; Piperidines; Propane; Pyrazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sulfonamides | 2014 |
Possible involvement of GABAergic and nitriergic systems for antianxiety-like activity of piperine in unstressed and stressed mice.
Topics: Alkaloids; Animals; Anti-Anxiety Agents; Anxiety; Benzodioxoles; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Guanidines; Indazoles; Male; Maze Learning; Mice; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type II; Nitrites; Piperidines; Polyunsaturated Alkamides; Stress, Psychological | 2014 |
Post-exposure administration of diazepam combined with soluble epoxide hydrolase inhibition stops seizures and modulates neuroinflammation in a murine model of acute TETS intoxication.
Topics: Animals; Anti-Inflammatory Agents; Anticonvulsants; Brain; Brain Waves; Bridged-Ring Compounds; Diazepam; Disease Models, Animal; Drug Administration Schedule; Drug Therapy, Combination; Electroencephalography; Encephalitis; Enzyme Inhibitors; Epoxide Hydrolases; GABA Modulators; Male; Mice; Phenylurea Compounds; Piperidines; Seizures; Time Factors | 2014 |
GluN2B-containing N-methyl-D-aspartate receptors compensate for the inhibitory control of synaptic plasticity during the early critical period in the rat visual cortex.
Topics: 2-Amino-5-phosphonovalerate; Age Factors; Animals; Animals, Newborn; Bicuculline; Diazepam; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA Modulators; GABA-A Receptor Antagonists; Gene Expression Regulation, Developmental; Long-Term Potentiation; Male; Neural Inhibition; Piperidines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, N-Methyl-D-Aspartate; Visual Cortex | 2015 |
Characterization of the Discriminative Stimulus Effects of a NOP Receptor Agonist Ro 64-6198 in Rhesus Monkeys.
Topics: Analgesics, Opioid; Animals; Benzimidazoles; Conditioning, Operant; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Female; Fentanyl; GABA Modulators; Imidazoles; Macaca mulatta; Male; Naltrexone; Narcotic Antagonists; Nociceptin Receptor; Pain Measurement; Piperidines; Receptors, Opioid; Spiro Compounds | 2016 |
Inhibition of Orexin Signaling Promotes Sleep Yet Preserves Salient Arousability in Monkeys.
Topics: Animals; Arousal; Conditioning, Classical; Cross-Over Studies; Diazepam; Eszopiclone; GABA Agents; Hypnotics and Sedatives; Macaca mulatta; Male; Orexin Receptor Antagonists; Orexins; Piperidines; Polysomnography; Signal Transduction; Sleep; Sleep Stages; Triazoles; Wakefulness | 2016 |
Enhanced anandamide signaling reduces flight behavior elicited by an approaching robo-beetle.
Topics: Amidohydrolases; Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Avoidance Learning; Behavior, Animal; Benzamides; Benzodioxoles; Cannabinoid Receptor Agonists; Carbamates; Diazepam; Endocannabinoids; Fear; Male; Mice, Inbred C57BL; Monoacylglycerol Lipases; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant | 2017 |
Inhibition of monoacylglycerol lipase terminates diazepam-resistant status epilepticus in mice and its effects are potentiated by a ketogenic diet.
Topics: Animals; Brain; Brain Waves; Carbamates; Cognition Disorders; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Resistant Epilepsy; Electroencephalography; Excitatory Amino Acid Agonists; Fluoresceins; Kainic Acid; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Monoacylglycerol Lipases; Neurons; Piperidines; Random Allocation; Receptor, Cannabinoid, CB1; Recognition, Psychology; Status Epilepticus; Sulfonamides; Time Factors | 2018 |
Predicted values for human total clearance of a variety of typical compounds with differently humanized-liver mouse plasma data.
Topics: Acetamides; Albuterol; Animals; Carbamates; Chromatography, Liquid; Diazepam; Diclofenac; Digitoxin; Humans; Itraconazole; Ketoprofen; Liver; Metabolic Clearance Rate; Mice; Mice, Transgenic; Naproxen; Pharmaceutical Preparations; Phenytoin; Piperidines; Pravastatin; Pyrimidines; Quinidine; Tandem Mass Spectrometry; Telmisartan; Terfenadine; Verapamil | 2020 |