diazepam and piperidines

diazepam has been researched along with piperidines in 116 studies

Research

Studies (116)

TimeframeStudies, this research(%)All Research%
pre-199047 (40.52)18.7374
1990's23 (19.83)18.2507
2000's28 (24.14)29.6817
2010's17 (14.66)24.3611
2020's1 (0.86)2.80

Authors

AuthorsStudies
Hüther, KJ; Koch-Weser, J; Lundt, PV; Moser, L1
Dicsó, F; Dolinay, T; Hankovszky, E1
Lehmann, K; Schmidt, J1
Bjerkenstedt, L; Gullberg, B; Härnryd, C; Sedvall, G1
Leander, JD1
Gol'dovskaia, IL1
Nose, T; Takemoto, H1
Spiess, W1
Braestrup, C; Falch, E; Krogsgaard-Larsen, P; Nielsen, M2
Duvhök, C; Molander, L1
Baron, BM; Chi, EM; Harrison, BL; Kehne, JH; McCloskey, TC; Palfreyman, MG; Whitten, JP1
Almeida, SS; de Oliveira, LM; Graeff, FG2
Bakker, MH; Foster, AC1
Budziszewska, B; Grochmal, A; Przegaliński, E1
Idzikowski, C; James, RJ; Mills, FJ1
Borsini, F; D'Aranno, V; Lecci, A; Mancinelli, A; Meli, A; Stasi, MA; Volterra, G1
Dubrovina, NI; Il'iuchenok, RIu; Parkhomenko, RI1
Bezek, S; Durisová, M; Kállay, Z; Kukan, M; Laginová, V; Scasnár, V; Svoboda, V; Trnovec, T1
Bannister, SJ; Houser, VP; Hulse, JD; Kisicki, JC; Rasmussen, JG1
D'Angio, M; Scatton, B; Serrano, A1
Hiltunen, AJ; Järbe, TU1
Byberg, JR; Curtis, DR; Falch, E; Gynther, BD; Hjeds, H; Krogsgaard-Larsen, P; Labouta, IM1
Le Bihan, C; Simon, P; Soubrié, P; Thiébot, MH1
Colpaert, FC; Janssen, PA; Meert, TF; Niemegeers, CJ1
Lu, MW; Peng, JZ; Tao, SC1
Bian, CF; Xing, SH; Xu, PC1
Badian, M; Hundt, HK; Joubert, AL; Luus, HG; Meyer, BH; Müller, FO1
Iversen, LL; Wong, EH1
Curtis, DR; Falch, E; Krogsgaard-Larsen, P; Nielsen, L1
Creveling, CR; Daly, JW; Hollingsworth, EB; Lewandowski, G; Waters, JA1
Nomikos, GG; Spyraki, C1
de Chaffoy de Courcelles, D; Leysen, JE; Niemegeers, CJ; Van Gompel, P1
Bateman, DN1
Curtis, DR; Falch, E; Jacobsen, P; Krogsgaard-Larsen, P1
Kimishima, K; Ogura, C1
Dencker, SJ; Frankenberg, K; Malm, U; Zell, B1
Bjelke, E; Stovner, J; Theodorsen, L1
Clarke, SW; Kendall, MJ1
Ban, TA; Lehmann, HE1
Vinar, O1
Bartůnková, Z; Cerný, L; Drtilová, J; Sturma, J1
Kalff, G1
Linford, W1
Dobkin, AB; Evers, W; Ghanooni, S; Levy, AA; Thomas, ET1
Harthoorn, AM; Harthoorn, S; Sayer, PD1
Perez de Francisco, C1
Roth, F1
Laduron, PM; Luabeya, MK; Maloteaux, JM1
Gotsadze, GG; Kipiani, ZV; Nemsadze, NO; Shariia, RP1
Collins, RC; de Gubareff, T; Fuller, TA; Olney, JW1
Baggio, P; Danda, R; Fumiani, G1
Conway, PC; Corbett, R; Dunn, RW; Hartman, H; Helsley, GC; Kerman, LL; Strupczewski, JT; Woods, AT1
Bickerdike, MJ; Dourish, CT; Fletcher, A; Marsden, CA1
Aranko, K; Kuitunen, T; Mattila, MJ1
Lewander, P; Nordvall, M; Stenhammar, L; Wärngård, O1
Kluger, MT; McLean, C; Owen, H; Plummer, JL1
Fernández, AG; Palacios, JM; Silvestre, JS1
Misawa, M; Suzuki, T; Tsuda, M2
Griebel, G; Perrault, G; Sanger, DJ1
File, SE1
Baubichon, D; Burckhart, MF; Clarençon, D; Galonnier, M; Lallement, G; Masqueliez, C; Mestries, JC; Peoc'h, M1
Li, P; Tabibi, SE; Vishnuvajjala, R; Yalkowsky, SH1
Baubichon, D; Burckhart, MF; Clarençon, D; Galonnier, M; Lallement, G; Peoc'h, M1
Martin, BR; Wiley, JL1
Carlson, EC; de Felipe, C; Harrison, T; Hunt, S; Oates, B; Owen, S; Rupniak, NM; Seward, E; Wheeldon, A1
Griebel, G; Perrault, G; Rodgers, RJ; Sanger, DJ1
Ballard, TM; Higgins, GA; Sänger, S1
Almerigi, P; Antolini, F; Caporaloni, M; Di Mauro, L; Melloni, C; Urso, G1
Gasparini, F; Gentsch, C; Kuhn, R; Schoeffter, P; Spooren, WP1
Cecil, A; Crites, G; Goldenberg, R; Knapp, RJ; Malatynska, E; Miller, C; Shuck, C; Watkins, J1
Biedler, A; Kreuer, S; Larsen, R; Molter, G; Schoth, S; Wilhelm, W1
FUKUCHI, G1
FELLNER, CH1
Felouzis, E; Gustorff, B; Hoechtl, K; Kress, HG; Lehr, S; Sycha, T1
Bourin, M; Clénet, F; Fillion, G; Galons, H; Hascoët, M1
Griebel, G; Scatton, B; Stemmelin, J1
Bernöster, K; Dost, R; Egerland, U; Langen, B; Rundfeldt, C; Unverferth, K1
Biba, A; Christodoulou, A; Chrysikakou, S; Giannou, H; Kontis, D; Maillis, A; Pallidi, S; Rabavilas, A; Tsaltas, E1
Deprest, JA; Jani, JC; Lewi, LE; Marcus, MA; Missant, C; Teunkens, A; Van de Velde, M; Van Schoubroeck, D1
Bhagat, YA; Hamilton, MG; Kendall, EJ; Mikler, J; Obenaus, A1
Bahamonde, JA; Belda, C; Belda, J; Ferrandis, R; Llau, JV1
Kronbach, C; Lüddens, H; Rabe, H; Rundfeldt, C1
Krishna, DR; Kumar, KV; Palit, G1
Bocchi, A; Candini, M; Carrer, S; Donegà, L; Tartari, S1
Alizadeh, AM; Haghparast, A; Khani, A; Motamedi, F; Naderi, N; Rezaii, N; Saber-Tehrani, A1
Hayashi, S; Hirao, A; Imai, A; Sugie, Y; Toide, K; Yamada, Y1
Brocco, M; Dekeyne, A; Di Cara, B; Gobert, A; Millan, MJ; Ortuno, JC; Panayi, F; Rivet, JM1
Drago, F; Leggio, GM; Li Volsi, V; Mazzola, C; Micale, V; Tamburella, A1
Kitahara, M; Kitahara, T; Kubo, T; Okumura, S1
Cristino, L; Di Marzo, V; Drago, F; Leggio, GM; Micale, V; Petrosino, S; Tamburella, A2
Choi, DY; Kang, SH; Platt, B; Riedel, G1
Jain, NS; Manna, SS; Umathe, SN; Utturwar, KS1
Baarendse, PJ; Trezza, V; Vanderschuren, LJ1
Casarotto, PC; Gomes, FV; Guimarães, FS; Resstel, LB1
Ko, MC; Podlesnik, CA; Prinssen, EP; Wichmann, J; Winger, G; Woods, JH1
Cravatt, BF; Kinsey, SG; Lichtman, AH; Long, JZ; O'Neal, ST1
Hohmann, AG; Sciolino, NR; Zhou, W1
Gielen, MC; Lumb, MJ; Smart, TG1
Brito, GA; Cavalheiro, EA; da Costa, MA; da Cruz, GM; da Graça Naffah-Mazzacoratti, M; de Andrade, GM; de Barros Viana, GS; Felipe, CF; Leal, LK; Menezes, ML; Scorza, FA; Tavares, AF1
Binns, J; Bowlby, MR; Brunner, J; Cannon, CE; Coleman, PJ; Eddins, DM; Fox, SV; Garson, SL; Gotter, AL; Hodgson, R; Kuduk, SD; Mcdonald, TP; Renger, JJ; Savitz, AT; Stevens, J; Tannenbaum, PL; Tye, SJ; Uslaner, JM; Wang, X; Winrow, CJ; Yao, L1
Bègue, L; Bell, R; Duke, AA; Gilmore, PE; Page, D1
Dhingra, D; Gilhotra, N1
Austin, AT; Banks, CN; Bruun, DA; Hammock, BD; Inceoglu, B; Lein, PJ; Rogawski, MA; Tancredi, DJ; Vito, ST; Zolkowska, D1
Alderson, P; Kenth, JJ; Lewis, SR; Nicholson, A; Reed, SS; Smith, AF1
Jang, HJ; Joo, K; Kim, MJ; Lee, C; Rhie, DJ1
Lindsey, AM; Prinssen, EP; Rice, KC; Saccone, PA; Sulima, A; Wichmann, J; Woods, JH; Zelenock, KA1
Coleman, PJ; Fox, SV; Gotter, AL; Hargreaves, R; Kuduk, SD; Renger, JJ; Savitz, AT; Stevens, J; Tannenbaum, PL; Tye, SJ; Uslaner, JM; Winrow, CJ1
Alcorn, J; Benmansour, P; Billinsky, J; Duke-Novakovski, T1
Genewsky, A; Heinz, DE; Wotjak, CT1
Butler, CR; Guilmette, E; Pauletti, A; Piro, JR; Porcu, L; Rizzi, M; Salamone, A; Samad, TA; Sheehan, MJ; Terrone, G; Vezzani, A; Villa, BR1
Ito, S; Iwamoto, K; Kamimura, H; Mizunaga, M; Nakayama, K; Negoro, T; Nishiwaki, M; Nomura, Y; Suemizu, H; Yamazaki, H; Yoneda, N1

Reviews

3 review(s) available for diazepam and piperidines

ArticleYear
[Psychotropic therapy and intraocular pressure].
    Oftalmologicheskii zhurnal, 1975, Volume: 30, Issue:1

    Topics: Amitriptyline; Analgesics; Antidepressive Agents; Chlorpromazine; Diazepam; Diphenhydramine; Eye Diseases; Glaucoma; Histamine H1 Antagonists; Humans; Imipramine; Intraocular Pressure; Lithium; Mental Disorders; Mephenesin; Meprobamate; Piperidines; Psychotropic Drugs; Secologanin Tryptamine Alkaloids; Tranquilizing Agents; Trihexyphenidyl

1975
[Psychopharmaca in modern medicine].
    Ceskoslovenska farmacie, 1968, Volume: 17, Issue:10

    Topics: Amphetamine; Antidepressive Agents; Barbiturates; Butyrophenones; Chlordiazepoxide; Chlorprothixene; Diazepam; Dibenzazepines; Guaifenesin; Hallucinogens; Humans; Hypnotics and Sedatives; Imipramine; Lithium; Lysergic Acid Diethylamide; Methylphenidate; Monoamine Oxidase Inhibitors; Oxazepam; Phenmetrazine; Phenothiazines; Phytotherapy; Piperidines; Plants, Medicinal; Psilocybin; Psychopharmacology; Rauwolfia; Reserpine; Tranquilizing Agents; Xanthenes

1968
Anaesthetic and sedative agents used for electrical cardioversion.
    The Cochrane database of systematic reviews, 2015, Mar-22, Issue:3

    Topics: Anesthetics; Apnea; Diazepam; Electric Countershock; Etomidate; Fentanyl; Humans; Hypnotics and Sedatives; Hypotension; Mental Recall; Methyl Ethers; Midazolam; Piperidines; Propofol; Randomized Controlled Trials as Topic; Remifentanil; Sevoflurane; Thiopental

2015

Trials

16 trial(s) available for diazepam and piperidines

ArticleYear
Effects of terfenadine and diphenhydramine alone or in combination with diazepam or alcohol on psychomotor performance and subjective feelings.
    European journal of clinical pharmacology, 1978, Dec-18, Volume: 14, Issue:6

    Topics: Adult; Benzhydryl Compounds; Diazepam; Diphenhydramine; Double-Blind Method; Drug Interactions; Emotions; Ethanol; Female; Flicker Fusion; Histamine H1 Antagonists; Humans; Male; Motor Skills; Piperidines; Reaction Time

1978
[R 33812 (domperidon) i.v. and orally as antiemetic adjuvans for short anaesthetics induced with etomidate. A comparative study (author's transl)].
    Der Anaesthesist, 1979, Volume: 28, Issue:4

    Topics: Adjuvants, Anesthesia; Administration, Oral; Antiemetics; Benzimidazoles; Diazepam; Dilatation and Curettage; Drug Interactions; Etomidate; Female; Humans; Injections, Intravenous; Piperidines; Premedication

1979
A dose-response study examining the effects of ritanserin on human slow wave sleep.
    British journal of clinical pharmacology, 1991, Volume: 31, Issue:2

    Topics: Adolescent; Adult; Diazepam; Dose-Response Relationship, Drug; Double-Blind Method; Electroencephalography; Electromyography; Female; Humans; Male; Piperidines; Ritanserin; Sleep Stages; Sleep, REM

1991
Effects of HOE 760 (histamine H2-receptor antagonist) on diazepam pharmacokinetics.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1988, Apr-02, Volume: 73, Issue:7

    Topics: Adult; Clinical Trials as Topic; Diazepam; Double-Blind Method; Half-Life; Histamine H2 Antagonists; Humans; Male; Nordazepam; Piperidines; Time Factors

1988
The action of cisapride on gastric emptying and the pharmacodynamics and pharmacokinetics of oral diazepam.
    European journal of clinical pharmacology, 1986, Volume: 30, Issue:2

    Topics: Adult; Blood Pressure; Chromatography, Gas; Cisapride; Diazepam; Double-Blind Method; Drug Interactions; Gastric Emptying; Heart Rate; Humans; Intestinal Absorption; Kinetics; Piperidines; Random Allocation

1986
A controlled one-year study of pipotiazine palmitate and fluphenazine decanoate in chronic schizophrenic syndromes. Evaluation of results at 6 and 12 months' trial.
    Acta psychiatrica Scandinavica. Supplementum, 1973, Volume: 241

    Topics: Adult; Aged; Antiparkinson Agents; Antipsychotic Agents; Basal Ganglia Diseases; Clinical Trials as Topic; Diazepam; Drug Evaluation; Female; Fluphenazine; Humans; Imipramine; Injections; Male; Middle Aged; Palmitic Acids; Piperidines; Psychiatric Status Rating Scales; Schizophrenia; Sulfonamides; Time Factors

1973
Studies with new drugs in the treatment of convulsive disorders.
    Internationale Zeitschrift fur klinische Pharmakologie, Therapie, und Toxikologie. International journal of clinical pharmacology, therapy, and toxicology, 1968, Volume: 1, Issue:3

    Topics: Adult; Aggression; Anticonvulsants; Anxiety; Carbamazepine; Clinical Trials as Topic; Diazepam; Dibenzazepines; Epilepsy; Frustration; Hallucinations; Humans; Intellectual Disability; Middle Aged; Nitriles; Object Attachment; Perceptual Disorders; Phenothiazines; Piperidines; Psychiatric Status Rating Scales; Psychopathology; Schizophrenia; Thiazines; Tranquilizing Agents

1968
Propericiazin, diazepam, chlorpromazine and placebo in a doubleblind trial in pedopsychiatric therapy.
    Activitas nervosa superior, 1972, Volume: 14, Issue:2

    Topics: Adolescent; Aggression; Child; Child Behavior Disorders; Chlorpromazine; Clinical Trials as Topic; Diazepam; Evaluation Studies as Topic; Female; Humans; Male; Mental Disorders; Motor Activity; Nitriles; Phenothiazines; Piperidines; Placebos; Tranquilizing Agents

1972
Diazepam effects on the performance of healthy subjects are not enhanced by treatment with the antihistamine ebastine.
    British journal of clinical pharmacology, 1993, Volume: 35, Issue:3

    Topics: Administration, Oral; Adult; Analysis of Variance; Butyrophenones; Chromatography, High Pressure Liquid; Diazepam; Double-Blind Method; Drug Interactions; Female; Histamine H1 Antagonists; Humans; Male; Piperidines; Psychomotor Performance

1993
The effect of oral cisapride premedication on fasting gastric volumes.
    Anaesthesia and intensive care, 1995, Volume: 23, Issue:6

    Topics: Adjuvants, Anesthesia; Administration, Oral; Adolescent; Adult; Aged; Anesthesia, General; Cisapride; Diazepam; Double-Blind Method; Elective Surgical Procedures; Fasting; Gastric Emptying; Gastrointestinal Contents; Humans; Hydrogen-Ion Concentration; Hypnotics and Sedatives; Intubation, Gastrointestinal; Middle Aged; Piperidines; Placebos; Premedication; Serotonin Antagonists; Suction

1995
[Narcotrend stages and end-tidal desflurane concentrations. An investigation during recovery from desflurane/remifentanil anaesthesia].
    Der Anaesthesist, 2002, Volume: 51, Issue:10

    Topics: Adult; Anesthesia Recovery Period; Anesthetics, Inhalation; Anesthetics, Intravenous; Desflurane; Diazepam; Electroencephalography; Female; Humans; Isoflurane; Male; Middle Aged; Monitoring, Intraoperative; Piperidines; Preanesthetic Medication; Remifentanil

2002
The effects of remifentanil and gabapentin on hyperalgesia in a new extended inflammatory skin pain model in healthy volunteers.
    Anesthesia and analgesia, 2004, Volume: 98, Issue:2

    Topics: Acetates; Adult; Amines; Analgesics, Opioid; Cross-Over Studies; Cyclohexanecarboxylic Acids; Diazepam; Double-Blind Method; Drug Synergism; Excitatory Amino Acid Antagonists; Female; GABA Modulators; Gabapentin; gamma-Aminobutyric Acid; Humans; Hyperalgesia; Inflammation; Male; Pain Measurement; Pain Threshold; Physical Stimulation; Piperidines; Reaction Time; Remifentanil; Skin; Sunburn; Treatment Outcome

2004
Remifentanil for fetal immobilization and maternal sedation during fetoscopic surgery: a randomized, double-blind comparison with diazepam.
    Anesthesia and analgesia, 2005, Volume: 101, Issue:1

    Topics: Adult; Anesthetics, Intravenous; Blood Gas Analysis; Conscious Sedation; Diazepam; Double-Blind Method; Female; Fetal Movement; Fetoscopy; Heart Rate, Fetal; Humans; Hypnotics and Sedatives; Immobilization; Injections, Intravenous; Laser Coagulation; Monitoring, Intraoperative; Piperidines; Pregnancy; Remifentanil; Respiratory Mechanics; Spinal Cord

2005
Short term analgesia based sedation in the Intensive Care Unit: morphine vs remifentanil + morphine.
    Minerva anestesiologica, 2007, Volume: 73, Issue:6

    Topics: Aged; Analgesia; Analgesics, Opioid; Blood Pressure; Conscious Sedation; Critical Care; Diazepam; Female; Humans; Hypnotics and Sedatives; Infusions, Intravenous; Male; Middle Aged; Morphine; Piperidines; Prospective Studies; Remifentanil; Respiration, Artificial

2007
Effects of endolymphatic sac drainage with steroids for intractable Meniere's disease: a long-term follow-up and randomized controlled study.
    The Laryngoscope, 2008, Volume: 118, Issue:5

    Topics: Anti-Inflammatory Agents; Antidepressive Agents; Dexamethasone; Diazepam; Dimenhydrinate; Diuretics; Endolymphatic Sac; Female; Follow-Up Studies; Histamine H1 Antagonists; Humans; Male; Meniere Disease; Middle Aged; Piperidines; Prospective Studies

2008
Blood concentrations of remifentanil during and after infusion in horses anesthetized with isoflurane and dexmedetomidine.
    Research in veterinary science, 2016, Volume: 107

    Topics: Analgesics, Opioid; Anesthetics, Inhalation; Animals; Dexmedetomidine; Diazepam; Drug Interactions; Female; Half-Life; Horses; Isoflurane; Ketamine; Male; Piperidines; Remifentanil; Xylazine

2016

Other Studies

97 other study(ies) available for diazepam and piperidines

ArticleYear
[Sandosten poisoning in childhood].
    Orvosi hetilap, 1979, Feb-18, Volume: 120, Issue:7

    Topics: Child, Preschool; Diazepam; Drug Therapy, Combination; Female; Furosemide; Gastric Lavage; Histamine H1 Antagonists; Humans; Piperidines; Poisoning; Thiophenes

1979
[Effect of psychotropic drugs on somatosensory evoked cortical potentials].
    Acta biologica et medica Germanica, 1979, Volume: 38, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Desipramine; Diazepam; Evoked Potentials; Female; Haloperidol; Hexobarbital; Medazepam; Piperidines; Rats; Somatosensory Cortex

1979
Relationships between clinical and biochemical effects of melperone and thiothixene in psychotic women.
    Archiv fur Psychiatrie und Nervenkrankheiten, 1979, Volume: 227, Issue:3

    Topics: Butyrophenones; Diazepam; Female; Homovanillic Acid; Humans; Hydroxyindoleacetic Acid; Methoxyhydroxyphenylglycol; Paranoid Disorders; Piperidines; Prolactin; Schizophrenia; Therapeutic Equivalency; Thiothixene

1979
Attenuating the rate-decreasing effects of phenylpiperidine analgesics by pentobarbital.
    Psychopharmacology, 1979, May-08, Volume: 63, Issue:1

    Topics: Analgesics; Animals; Chlorpromazine; Columbidae; Conditioning, Operant; Diazepam; Male; Meperidine; Pentobarbital; Piperidines; Reinforcement Schedule

1979
The effect of penfluridol and some psychotropic drugs on monoamine metabolism in central nervous system.
    European journal of pharmacology, 1975, Volume: 31, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Biogenic Amines; Brain; Brain Chemistry; Chlordiazepoxide; Chlorpromazine; Diazepam; Dopamine; Haloperidol; Homovanillic Acid; Hydroxyindoleacetic Acid; Male; Mice; Norepinephrine; Penfluridol; Pimozide; Piperazines; Piperidines; Psychotropic Drugs; Rats; Serotonin

1975
Partial agonists for brain GABA/benzodiazepine receptor complex.
    Nature, 1979, Jul-26, Volume: 280, Issue:5720

    Topics: Animals; Benzodiazepines; Bicuculline; Brain; Crotonates; Diazepam; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Isoxazoles; Muscimol; Piperidines; Rats; Receptors, Drug; Sulfonic Acids

1979
Acute effects of oxazepam, diazepam and methylperone, alone and in combination with alcohol on sedation, coordination and mood.
    Acta pharmacologica et toxicologica, 1976, Volume: 38, Issue:2

    Topics: Adult; Attention; Butyrophenones; Diazepam; Drug Interactions; Emotions; Ethanol; Flicker Fusion; Humans; Male; Middle Aged; Motor Skills; Oxazepam; Piperidines; Tranquilizing Agents

1976
NMDA receptor complex antagonists have potential anxiolytic effects as measured with separation-induced ultrasonic vocalizations.
    European journal of pharmacology, 1991, Feb-14, Volume: 193, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Anxiety, Separation; Behavior, Animal; Buspirone; Diazepam; Dioxins; Dizocilpine Maleate; Dose-Response Relationship, Drug; Indoles; Kynurenic Acid; Maternal Deprivation; Mephenesin; Piperidines; Quinolizines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Serotonin Antagonists; Spiro Compounds; Valine; Vocalization, Animal

1991
Early life protein malnutrition changes exploration of the elevated plus-maze and reactivity to anxiolytics.
    Psychopharmacology, 1991, Volume: 103, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Male; Piperidines; Propanolamines; Protein-Energy Malnutrition; Pyrimidines; Rats; Rats, Inbred Strains; Ritanserin

1991
An investigation of the mechanisms of delayed neurodegeneration caused by direct injection of quinolinate into the rat striatum in vivo.
    Neuroscience, 1991, Volume: 42, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Anticonvulsants; Convulsants; Corpus Striatum; Dialysis; Diazepam; Dizocilpine Maleate; Glutamate Decarboxylase; Haloperidol; Ibotenic Acid; Injections; Male; Nerve Degeneration; Pipecolic Acids; Piperazines; Piperidines; Quinolinic Acid; Quinolinic Acids; Rats; Rats, Inbred Strains; Stereotaxic Techniques

1991
Oxaprotiline enantiomers stimulate ACTH and corticosterone secretion in the rat.
    Journal of neural transmission. General section, 1991, Volume: 85, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenocorticotropic Hormone; Animals; Antidepressive Agents; Benzylamines; Corticosterone; Dexamethasone; Diazepam; Dose-Response Relationship, Drug; Male; Maprotiline; Metergoline; Naloxone; Piperidines; Pyrimidines; Radioimmunoassay; Rats; Rats, Inbred Strains; Serotonin Antagonists; Stereoisomerism; Sulpiride; Sympathomimetics

1991
Decreased reactivity to anxiolytics caused by early protein malnutrition in rats.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Body Weight; Diazepam; Diet; Dose-Response Relationship, Drug; Hypertonic Solutions; Lactation; Male; Piperidines; Propanolamines; Protein-Energy Malnutrition; Pyrimidines; Rats; Rats, Inbred Strains; Ritanserin

1990
Effect of serotoninergic drugs on stress-induced hyperthermia (SIH) in mice.
    Journal of neural transmission. General section, 1990, Volume: 82, Issue:3

    Topics: 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Body Temperature Regulation; Buspirone; Diazepam; Ergolines; Fenclonine; Fever; Flumazenil; Imidazoles; Male; Mice; Ondansetron; Piperazines; Piperidines; Ritanserin; Serotonin; Serotonin Antagonists; Stress, Psychological; Tetrahydronaphthalenes

1990
[GABAergic modulation of amnesic trace reproduction by activation of the dopaminergic system].
    Biulleten' eksperimental'noi biologii i meditsiny, 1990, Volume: 110, Issue:12

    Topics: Animals; Avoidance Learning; Bupropion; Diazepam; Dopamine Agents; Ergolines; Male; Mice; Mice, Inbred BALB C; Piperidines; Propiophenones; Quinpirole; Receptors, GABA-A

1990
Irradiation of the head by 60Co opens the blood-brain barrier for drugs in rats.
    Experientia, 1990, Oct-15, Volume: 46, Issue:10

    Topics: Animals; Aspirin; Blood-Brain Barrier; Brain; Carbamates; Chloramphenicol; Cobalt Radioisotopes; Cranial Irradiation; Diazepam; Etimizol; Male; Piperidines; Rats; Rats, Inbred Strains; Regression Analysis

1990
Evaluation of the potential for interactions of paroxetine with diazepam, cimetidine, warfarin, and digoxin.
    Acta psychiatrica Scandinavica. Supplementum, 1989, Volume: 350

    Topics: Adult; Antidepressive Agents; Biological Availability; Cimetidine; Diazepam; Digoxin; Drug Interactions; Humans; Male; Paroxetine; Piperidines; Serotonin Antagonists; Warfarin

1989
NMDA antagonists block restraint-induced increase in extracellular DOPAC in rat nucleus accumbens.
    European journal of pharmacology, 1989, Mar-14, Volume: 162, Issue:1

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adrenergic alpha-Antagonists; Animals; Aspartic Acid; Carbolines; Convulsants; Diazepam; Male; N-Methylaspartate; Nucleus Accumbens; Phenylacetates; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Restraint, Physical; Riluzole; Septal Nuclei; Thiazoles

1989
Limited stimulus generalization between delta 9-THC and diazepam in pigeons and gerbils.
    Psychopharmacology, 1988, Volume: 94, Issue:3

    Topics: Animals; Benzodiazepinones; Columbidae; Diazepam; Discrimination, Psychological; Dronabinol; Generalization, Stimulus; Gerbillinae; Male; Piperidines; Receptors, GABA-A

1988
Synthesis and biological activity of a GABAA agonist which has no effect on benzodiazepine binding and of structurally related glycine antagonists.
    Drug design and delivery, 1987, Volume: 1, Issue:4

    Topics: Animals; Bicuculline; Brain Chemistry; Chemical Phenomena; Chemistry; Diazepam; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Isoxazoles; Oxazoles; Piperidines; Pyrrolidines; Rats; Receptors, GABA-A; Synaptic Membranes

1987
Benzodiazepines reduce the tolerance to reward delay in rats.
    Psychopharmacology, 1985, Volume: 86, Issue:1-2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Choice Behavior; Diazepam; Flumazenil; Male; Piperidines; Rats; Rats, Inbred Strains; Reward; Serotonin Antagonists; Synaptic Transmission; Zimeldine

1985
Behavioral and 5-HT antagonist effects of ritanserin: a pure and selective antagonist of LSD discrimination in rat.
    Psychopharmacology, 1985, Volume: 86, Issue:1-2

    Topics: 5-Hydroxytryptophan; Animals; Anti-Anxiety Agents; Anxiety; Chlordiazepoxide; Diazepam; Disease Models, Animal; Histamine H2 Antagonists; Humans; Lysergic Acid Diethylamide; Male; Motor Activity; Piperidines; Pyrimidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists

1985
[Central convulsive action of l-securinine].
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1986, Volume: 7, Issue:1

    Topics: Alkaloids; Animals; Azepines; Central Nervous System Stimulants; Diazepam; Drug Synergism; gamma-Aminobutyric Acid; Heterocyclic Compounds, 4 or More Rings; Heterocyclic Compounds, Bridged-Ring; Humans; Lactones; Male; Mice; Piperidines; Seizures

1986
[The interactions between dihydroetorphine, L-tetrahydropalmatine, B-7601 and diazepam].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1986, Volume: 21, Issue:8

    Topics: Alkaloids; Anesthesia, General; Anesthesia, Intravenous; Animals; Antipsychotic Agents; Benzilates; Berberine Alkaloids; Diazepam; Dogs; Drug Interactions; Etorphine; Female; Male; Mice; Morphinans; Piperidines; Rabbits

1986
Modulation of [3H]diazepam binding in rat cortical membranes by GABAA agonists.
    Journal of neurochemistry, 1985, Volume: 44, Issue:4

    Topics: Androstanes; Animals; Azasteroids; Bicuculline; Cell Membrane; Cerebral Cortex; Diazepam; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Isonicotinic Acids; Isoxazoles; Muscimol; Piperidines; Rats; Receptors, GABA-A; Taurine

1985
GABA agonists. Resolution, absolute stereochemistry, and enantioselectivity of (S)-(+)- and (R)-(-)-dihydromuscimol.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:11

    Topics: Animals; Bicuculline; Brain; Cats; Chemical Phenomena; Chemistry; Diazepam; gamma-Aminobutyric Acid; Isoxazoles; Molecular Conformation; Muscimol; Neurons; Oxazolidinones; Piperidines; Rats; Receptors, GABA-A; Spinal Cord; Stereoisomerism; Structure-Activity Relationship; Synaptic Membranes

1985
Anticonvulsant activity of piperidinol and (dialkylamino)alkanol esters.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:8

    Topics: Amino Alcohols; Animals; Anticonvulsants; Ataxia; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Diazepam; Electroshock; Esters; Muscimol; Pentylenetetrazole; Phenytoin; Piperidines; Rats; Receptors, GABA-A; Structure-Activity Relationship

1986
Effects of ritanserin on the rewarding properties of d-amphetamine, morphine and diazepam revealed by conditioned place preference in rats.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:4

    Topics: Analgesia; Animals; Conditioning, Operant; Dextroamphetamine; Diazepam; Exploratory Behavior; Male; Morphine; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Reference Values; Reinforcement, Psychology; Reward; Ritanserin; Serotonin Antagonists

1988
Opposite regulation of serotonin-S2 and dopamine-D2 receptors in rat brain following chronic receptor blockade.
    Journal of receptor research, 1987, Volume: 7, Issue:1-4

    Topics: Animals; Apomorphine; Behavior, Animal; Corpus Striatum; Diazepam; Dopamine Antagonists; Frontal Lobe; Gene Expression Regulation; Ketanserin; Male; Models, Biological; Piperidines; Pyrimidinones; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Serotonin Antagonists; Tryptamines

1987
GABA-mimetic activity and effects on diazepam binding of aminosulphonic acids structurally related to piperidine-4-sulphonic acid.
    Journal of neurochemistry, 1985, Volume: 44, Issue:1

    Topics: Animals; Binding Sites; Brain; Diazepam; gamma-Aminobutyric Acid; Piperidines; Pyridines; Pyrrolidines; Rats; Structure-Activity Relationship; Synaptic Membranes

1985
Central nervous actions and screening methods of antidepressants.
    Folia psychiatrica et neurologica japonica, 1972, Volume: 26, Issue:4

    Topics: Acetylcholine; Amitriptyline; Animals; Antidepressive Agents; Behavior, Animal; Biogenic Amines; Blood Pressure; Brain Chemistry; Central Nervous System; Diazepam; Electroshock; Ethanol; Hexobarbital; Hypertension; Hypothermia, Induced; Imipramine; Iproniazid; Methamphetamine; Mice; Nialamide; Physostigmine; Piperidines; Reserpine; Tremorine

1972
[Experimental studies on prevention of muscular cramps caused by 2 F-type schistosomicides].
    Zhonghua yi xue za zhi, 1974, Volume: 1

    Topics: Acrylamides; Animals; Anthelmintics; Cats; Chlordiazepoxide; Diazepam; Mice; Muscle Cramp; Nitrofurans; Piperidines; Rabbits; Schistosomiasis; Schistosomicides

1974
Sensitivity to gallamine and pancuronium with special reference to serum proteins.
    British journal of anaesthesia, 1971, Volume: 43, Issue:10

    Topics: Androstanes; Anesthesia, General; Blood Proteins; Body Surface Area; Diazepam; Female; Gallamine Triethiodide; Humans; Injections, Intramuscular; Neuromuscular Nondepolarizing Agents; Piperidines; Serum Albumin; Thiopental

1971
Prolonged coma after tetanus.
    British medical journal, 1972, Feb-05, Volume: 1, Issue:5796

    Topics: Aged; Androstanes; Coma; Diazepam; Female; Humans; Neuromuscular Nondepolarizing Agents; Piperidines; Respiration, Artificial; Tetanus

1972
Diazepam combination-anesthesia.
    Acta anaesthesiologica Belgica, 1974, Volume: 25, Issue:3

    Topics: Animals; Blood Circulation; Blood Pressure; Cardiac Output; Diazepam; Dogs; Drug Synergism; Fentanyl; Heart Rate; Humans; Isonipecotic Acids; Morphine; Piperidines; Vascular Resistance

1974
New horizons in psychopharmacology.
    Proceedings of the Royal Society of Medicine, 1972, Volume: 65, Issue:9

    Topics: Animals; Anthracenes; Antidepressive Agents; Anxiety; Benzamides; Benzazepines; Butyrophenones; Chlordiazepoxide; Chlorprothixene; Diazepam; Dibenzothiazepines; Humans; Monoamine Oxidase Inhibitors; Nitrazepam; Oxazepam; Pharmacogenetics; Phenothiazines; Piperidines; Plants, Medicinal; Psychopharmacology; Rauwolfia; Sleep; Tranquilizing Agents

1972
Pancuronium bromide (Pavulon) evaluation of its clinical pharmacology.
    Canadian Anaesthetists' Society journal, 1971, Volume: 18, Issue:5

    Topics: Androstanes; Anesthesia, Inhalation; Atropine; Blood Pressure; Body Temperature; Carbon Dioxide; Diazepam; Electrocardiography; Female; Fentanyl; Halothane; Histamine; Humans; Hydrogen-Ion Concentration; Intubation, Intratracheal; Male; Meperidine; Methoxyflurane; Middle Aged; Neostigmine; Nitrous Oxide; Oxygen; Piperidines; Potassium; Pulse; Respiration; Surgical Procedures, Operative; Thiopental; Urination

1971
Two field operations on the African lion (Felis leo).
    The Veterinary record, 1971, Aug-07, Volume: 89, Issue:6

    Topics: Anesthesia, Intravenous; Animals; Antisepsis; Carnivora; Chlorpromazine; Diazepam; Eye Foreign Bodies; Fracture Fixation, Intramedullary; Humeral Fractures; Male; Piperidines; Thiopental

1971
[Psychopharmacological treatment of anxiety].
    La Prensa medica mexicana, 1971, Volume: 36, Issue:9

    Topics: Adult; Amitriptyline; Anxiety; Benzazepines; Carbamates; Chlordiazepoxide; Diazepam; Dibenzazepines; Female; Humans; Ketones; Meprobamate; Methotrimeprazine; Nitro Compounds; Oxazepam; Piperidines; Thioridazine

1971
[Anesthesia in cardioversion].
    Schweizerische medizinische Wochenschrift, 1969, Oct-25, Volume: 99, Issue:43

    Topics: Anesthesia, General; Anesthetics; Arrhythmias, Cardiac; Diazepam; Electric Countershock; Humans; Methods; Nitrous Oxide; Piperidines; Preanesthetic Medication; Thiopental

1969
Regional and cortical laminar distributions of serotonin S2, benzodiazepine, muscarinic, and dopamine D2 receptors in human brain.
    Journal of neurochemistry, 1984, Volume: 43, Issue:4

    Topics: Adult; Aged; Brain; Cerebral Cortex; Diazepam; Humans; Ketanserin; Male; Middle Aged; Piperidines; Quinuclidinyl Benzilate; Receptors, Cell Surface; Receptors, Dopamine; Receptors, GABA-A; Receptors, Muscarinic; Receptors, Serotonin; Spiperone; Tissue Distribution

1984
Two or more conformations of benzodiazepine receptors depending on GABA receptors and other variables.
    Advances in biochemical psychopharmacology, 1980, Volume: 21

    Topics: Animals; Benzodiazepines; Bicuculline; Brain; Diazepam; gamma-Aminobutyric Acid; Macromolecular Substances; Male; Muscimol; Piperidines; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Structure-Activity Relationship; Synaptic Membranes

1980
[Functional state of the fetus during labor with the use of spasmoanalgesic and tranquilizing agents].
    Akusherstvo i ginekologiia, 1983, Issue:5

    Topics: Anesthesia, Obstetrical; Benzophenones; Butylscopolammonium Bromide; Diazepam; Dipyrone; Drug Combinations; Female; Fetus; Humans; Infant, Newborn; Labor, Obstetric; Parasympatholytics; Piperidines; Pregnancy

1983
Systemic dipiperidinoethane mimics the convulsant and neurotoxic actions of kainic acid.
    Brain research, 1980, Oct-27, Volume: 200, Issue:1

    Topics: Animals; Behavior, Animal; Diazepam; Hippocampus; Kainic Acid; Male; Piperidines; Pyrrolidines; Rats; Seizures

1980
[Tipepidine poisoning].
    Minerva pediatrica, 1980, Jun-30, Volume: 32, Issue:12

    Topics: Akathisia, Drug-Induced; Child, Preschool; Diazepam; Female; Humans; Medication Errors; Piperidines; Psychomotor Agitation

1980
Effects of atypical antipsychotic agents on social behavior in rodents.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 45, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Apomorphine; Benzazepines; Catalepsy; Chlorpromazine; Clozapine; Diazepam; Haloperidol; Isoxazoles; Male; Mice; Mice, Inbred Strains; Piperidines; Raclopride; Radioligand Assay; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Serotonin; Risperidone; Salicylamides; Social Behavior

1993
The influence of 5-hydroxytryptamine re-uptake blockade on CCK receptor antagonist effects in the rat elevated zero-maze.
    European journal of pharmacology, 1994, Dec-27, Volume: 271, Issue:2-3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Devazepide; Diazepam; Indoles; Male; Maze Learning; Meglumine; Niacinamide; Phenylurea Compounds; Piperazines; Piperidines; Rats; Receptors, Cholecystokinin; Selective Serotonin Reuptake Inhibitors; Zimeldine

1994
Oral versus intravenous premedication for small bowel biopsy in children: effect on procedure and fluoroscopy times.
    Acta paediatrica (Oslo, Norway : 1992), 1993, Volume: 82, Issue:1

    Topics: Administration, Oral; Adolescent; Biopsy; Celiac Disease; Child; Child, Preschool; Cisapride; Diazepam; Fluoroscopy; Humans; Infant; Infusions, Intravenous; Intestine, Small; Metoclopramide; Midazolam; Piperidines; Premedication; Serotonin Antagonists; Trimeprazine

1993
Effects of 5-HT4 receptor antagonists on rat behaviour in the elevated plus-maze test.
    European journal of pharmacology, 1996, Aug-15, Volume: 309, Issue:3

    Topics: Animals; Behavior, Animal; Diazepam; Dioxanes; Dose-Response Relationship, Drug; Granisetron; Indoles; Male; Maze Learning; Piperidines; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Sulfonamides

1996
Recovery of decreased seizure threshold for pentylenetetrazole during diazepam withdrawal by NMDA receptor antagonists.
    European journal of pharmacology, 1997, Apr-11, Volume: 324, Issue:1

    Topics: Animals; Anticonvulsants; Convulsants; Diazepam; Disease Models, Animal; Dizocilpine Maleate; Drug Interactions; Excitatory Amino Acid Antagonists; Infusions, Intravenous; Injections, Intraperitoneal; Injections, Subcutaneous; Kynurenic Acid; Male; Mice; Neuroprotective Agents; Pentylenetetrazole; Piperidines; Receptors, N-Methyl-D-Aspartate; Seizures; Substance Withdrawal Syndrome

1997
A comparative study of the effects of selective and non-selective 5-HT2 receptor subtype antagonists in rat and mouse models of anxiety.
    Neuropharmacology, 1997, Volume: 36, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Diazepam; Drinking; Fluorobenzenes; Indoles; Male; Maze Learning; Mianserin; Mice; Mice, Inbred BALB C; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists

1997
Anxiolytic action of a neurokinin1 receptor antagonist in the social interaction test.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 58, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Diazepam; Drug Tolerance; Handling, Psychological; Interpersonal Relations; Lighting; Male; Motor Activity; Neurokinin-1 Receptor Antagonists; Piperidines; Quinolines; Rats; Stress, Psychological

1997
Nerve agent poisoning in primates: antilethal, anti-epileptic and neuroprotective effects of GK-11.
    Archives of toxicology, 1998, Volume: 72, Issue:2

    Topics: Animals; Anticonvulsants; Atropine; Brain; Chemical Warfare Agents; Cholinesterase Inhibitors; Cholinesterase Reactivators; Cyclohexanes; Cyclohexenes; Diazepam; Drug Combinations; Excitatory Amino Acid Antagonists; Injections, Intravenous; Macaca fascicularis; Male; Muscarinic Antagonists; Neuroprotective Agents; Piperidines; Pralidoxime Compounds; Seizures; Soman; Staining and Labeling; Time Factors

1998
Evaluation of in vitro precipitation methods.
    Journal of pharmaceutical sciences, 1998, Volume: 87, Issue:2

    Topics: Antineoplastic Agents; Chemical Precipitation; Chemistry, Pharmaceutical; Diazepam; Flavonoids; Injections; Piperidines; Solubility; Solutions; Time Factors

1998
NMDA receptor antagonists potently suppress the spontaneous withdrawal signs induced by discontinuation of long-term diazepam treatment in Fischer 344 rats.
    Brain research, 1998, Apr-20, Volume: 790, Issue:1-2

    Topics: Administration, Oral; Animals; Anorexia; Anti-Anxiety Agents; Behavior, Animal; Diazepam; Dizocilpine Maleate; Eating; Emotions; Excitatory Amino Acid Antagonists; Male; Motor Activity; Piperidines; Rats; Rats, Inbred F344; Receptors, N-Methyl-D-Aspartate; Substance Withdrawal Syndrome; Time Factors; Weight Loss

1998
Acute soman poisoning in primates neither pretreated nor receiving immediate therapy: value of gacyclidine (GK-11) in delayed medical support.
    Archives of toxicology, 1999, Volume: 73, Issue:2

    Topics: Animals; Anticonvulsants; Antidotes; Atropine; Brain; Cerebellum; Cerebral Cortex; Chemical Warfare Agents; Cholinesterase Reactivators; Cyclohexanes; Cyclohexenes; Diazepam; Drug Therapy, Combination; Electrocardiography; Excitatory Amino Acid Antagonists; Haplorhini; Macaca fascicularis; Male; Piperidines; Poisoning; Pralidoxime Compounds; Seizures; Soman; Time Factors

1999
Effects of SR141716A on diazepam substitution for delta9-tetrahydrocannabinol in rat drug discrimination.
    Pharmacology, biochemistry, and behavior, 1999, Volume: 64, Issue:3

    Topics: Animals; Cannabinoids; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Dronabinol; GABA Modulators; Generalization, Psychological; Hallucinogens; Male; Piperidines; Pyrazoles; Rats; Rats, Long-Evans; Rats, Sprague-Dawley; Rimonabant

1999
Pharmacological blockade or genetic deletion of substance P (NK(1)) receptors attenuates neonatal vocalisation in guinea-pigs and mice.
    Neuropharmacology, 2000, Jun-08, Volume: 39, Issue:8

    Topics: Animals; Animals, Newborn; Anti-Anxiety Agents; Antidepressive Agents; Behavior, Animal; Buspirone; Diazepam; Dose-Response Relationship, Drug; Female; Fluoxetine; Gene Deletion; Guinea Pigs; Imipramine; Injections, Intraventricular; Male; Mice; Mice, Inbred Strains; Motor Activity; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Social Isolation; Stress, Psychological; Substance P; Tetrazoles; Vocalization, Animal

2000
The effects of compounds varying in selectivity as 5-HT(1A) receptor antagonists in three rat models of anxiety.
    Neuropharmacology, 2000, Jul-24, Volume: 39, Issue:10

    Topics: Aminopyridines; Animals; Anxiety; Cyclohexane Monoterpenes; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drinking Behavior; Isoquinolines; Male; Maze Learning; Motor Activity; Pindolol; Piperazines; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Succinimides

2000
Inhibition of shock-induced foot tapping behaviour in the gerbil by a tachykinin NK1 receptor antagonist.
    European journal of pharmacology, 2001, Feb-02, Volume: 412, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Antidepressive Agents, Second-Generation; Aprepitant; Conditioning, Operant; Diazepam; Female; Fluoxetine; Gerbillinae; Humans; Male; Morpholines; Motor Activity; Neurokinin-1 Receptor Antagonists; Piperidines; Receptors, Neurokinin-1

2001
[Propofol and remifentanil in day surgery].
    Minerva anestesiologica, 2000, Volume: 66, Issue:10

    Topics: Adult; Ambulatory Surgical Procedures; Anesthesia Recovery Period; Anesthesia, General; Anesthetics, Intravenous; Conscious Sedation; Diazepam; Humans; Midazolam; Piperidines; Preanesthetic Medication; Propofol; Remifentanil

2000
Pharmacological and endocrinological characterisation of stress-induced hyperthermia in singly housed mice using classical and candidate anxiolytics (LY314582, MPEP and NKP608).
    European journal of pharmacology, 2002, Jan-25, Volume: 435, Issue:2-3

    Topics: Adrenocorticotropic Hormone; Analysis of Variance; Animals; Anti-Anxiety Agents; Benzodiazepines; Body Temperature; Bridged Bicyclo Compounds; Buspirone; Chlordiazepoxide; Clobazam; Corticosterone; Diazepam; Ethanol; Hyperthermia, Induced; Male; Mice; Mice, Inbred ICR; Oxazepam; Piperidines; Pyridines; Quinolines; Reproducibility of Results; Stress, Physiological

2002
Antidepressant activity of memory-enhancing drugs in the reduction of submissive behavior model.
    European journal of pharmacology, 2002, Apr-05, Volume: 440, Issue:1

    Topics: Animals; Antidepressive Agents; Competitive Behavior; Desipramine; Diazepam; Dioxoles; Dose-Response Relationship, Drug; Fluoxetine; Injections, Intraperitoneal; Male; Maze Learning; Models, Animal; Nootropic Agents; Piperidines; Piracetam; Pyrrolidinones; Rats; Rats, Sprague-Dawley

2002
[DRUGS ACTING ON THE NERVOUS SYSTEM. (2). WITH SPECIAL REFERENCE TO TRANQUILIZERS AND ANTIDEPRESSIVE AGENTS].
    [Chiryo] [Therapy], 1963, Volume: 45

    Topics: Amides; Amitriptyline; Antidepressive Agents; Benactyzine; Chemical Phenomena; Chemistry; Chlordiazepoxide; Desipramine; Diazepam; Haloperidol; Humans; Hydroxyzine; Hypnotics and Sedatives; Imipramine; Isocarboxazid; Meprobamate; Methylphenidate; Monoamine Oxidase Inhibitors; Nervous System; Nialamide; Pharmacology; Phenelzine; Piperidines; Tranquilizing Agents; Tranylcypromine; Tryptamines

1963
EARLY RECOGNITION OF DEPRESSION.
    Geriatrics, 1964, Volume: 19

    Topics: Amitriptyline; Amphetamine; Amphetamines; Barbiturates; Benactyzine; Chlordiazepoxide; Deanol; Depression; Depressive Disorder; Diagnosis; Diazepam; Drug Therapy; Geriatrics; Humans; Imipramine; Meprobamate; Methylphenidate; Monoamine Oxidase Inhibitors; Phenmetrazine; Piperidines; Psychotherapy; Toxicology

1964
Anxiolytic profile of HG1, a 5-HT-moduline antagonist, in three mouse models of anxiety.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2004, Volume: 14, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Dose-Response Relationship, Drug; Electroshock; Light; Male; Mice; Motor Activity; Neuropeptides; Oligopeptides; Piperidines; Serotonin Antagonists

2004
Effects of the cannabinoid CB1 receptor antagonist rimonabant in models of emotional reactivity in rodents.
    Biological psychiatry, 2005, Feb-01, Volume: 57, Issue:3

    Topics: Aggression; Analysis of Variance; Animals; Anti-Anxiety Agents; Antidepressive Agents, Second-Generation; Behavior, Animal; Depression; Diazepam; Dose-Response Relationship, Drug; Electroshock; Emotions; Fluoxetine; Gerbillinae; Immobility Response, Tonic; Male; Maze Learning; Mice; Models, Animal; Neuropsychological Tests; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Rimonabant

2005
Characterization in rats of the anxiolytic potential of ELB139 [1-(4-chlorophenyl)-4-piperidin-1-yl-1,5-dihydro-imidazol-2-on], a new agonist at the benzodiazepine binding site of the GABAA receptor.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Binding Sites; Binding, Competitive; Conflict, Psychological; Diazepam; Drug Tolerance; Flumazenil; Flunitrazepam; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Imidazoles; Light; Male; Membrane Potentials; Patch-Clamp Techniques; Piperidines; Rats; Rats, Wistar

2005
Reinforced spatial alternation as an animal model of obsessive-compulsive disorder (OCD): investigation of 5-HT2C and 5-HT1D receptor involvement in OCD pathophysiology.
    Biological psychiatry, 2005, May-15, Volume: 57, Issue:10

    Topics: Animals; Anti-Anxiety Agents; Antidepressive Agents, Tricyclic; Desipramine; Diazepam; Disease Models, Animal; Fluoxetine; Indoles; Male; Maze Learning; Obsessive-Compulsive Disorder; Piperazines; Piperidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2C; Reinforcement, Psychology; Selective Serotonin Reuptake Inhibitors; Serotonin Receptor Agonists; Tryptamines

2005
Neuroprotection from soman-induced seizures in the rodent: evaluation with diffusion- and T2-weighted magnetic resonance imaging.
    Neurotoxicology, 2005, Volume: 26, Issue:6

    Topics: Animals; Anticonvulsants; Brain; Cell Death; Cyclohexanes; Cyclohexenes; Diazepam; Diffusion Magnetic Resonance Imaging; Magnetic Resonance Imaging; Male; Neuroprotective Agents; Piperidines; Rats; Rats, Sprague-Dawley; Seizures; Soman; Status Epilepticus

2005
Anesthesia for cardiac surgery on a patient with stiff person syndrome.
    Journal of cardiothoracic and vascular anesthesia, 2005, Volume: 19, Issue:3

    Topics: Adult; Analgesics, Opioid; Anesthesia; Anesthetics, Intravenous; Anticonvulsants; Cardiopulmonary Bypass; Diazepam; Etomidate; Female; Fentanyl; Heart Valve Diseases; Heparin; Humans; Midazolam; Morphine; Neuromuscular Nondepolarizing Agents; Pain, Postoperative; Pancuronium; Piperidines; Propofol; Remifentanil; Stiff-Person Syndrome

2005
The novel anxiolytic ELB139 displays selectivity to recombinant GABA(A) receptors different from diazepam.
    Neuropharmacology, 2007, Volume: 52, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Cell Line, Transformed; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; GABA-A Receptor Agonists; Humans; Imidazoles; Membrane Potentials; Patch-Clamp Techniques; Piperidines; Rats; Receptors, GABA-A; Transfection

2007
Histaminergic H1 receptors mediate L-histidine-induced anxiety in elevated plus-maze test in mice.
    Behavioural pharmacology, 2007, Volume: 18, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzothiazoles; Diazepam; Dose-Response Relationship, Drug; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Male; Mice; Phenoxypropanolamines; Piperidines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H3

2007
Interaction between cannabinoid compounds and diazepam on anxiety-like behaviour of mice.
    Pharmacology, biochemistry, and behavior, 2008, Volume: 89, Issue:1

    Topics: Amidohydrolases; Animals; Anxiety; Arachidonic Acids; Behavior, Animal; Benzamides; Benzoxazines; Cannabinoids; Carbamates; Data Interpretation, Statistical; Diazepam; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Enzyme Inhibitors; GABA Modulators; Hypnotics and Sedatives; Male; Mice; Morpholines; Naphthalenes; Piperidines; Postural Balance; Pyrazoles; Receptor, Cannabinoid, CB1

2008
Pharmacological characterization of the newly synthesized nociceptin/orphanin FQ-receptor agonist 1-[1-(1-methylcyclooctyl)-4-piperidinyl]-2-[(3R)-3-piperidinyl]-1H-benzimidazole as an anxiolytic agent.
    Journal of pharmacological sciences, 2008, Volume: 106, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzimidazoles; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Ethanol; Humans; Male; Memory; Mice; Motor Activity; Nociceptin Receptor; Piperidines; Receptors, Opioid

2008
The melanin-concentrating hormone1 receptor antagonists, SNAP-7941 and GW3430, enhance social recognition and dialysate levels of acetylcholine in the frontal cortex of rats.
    The international journal of neuropsychopharmacology, 2008, Volume: 11, Issue:8

    Topics: Acetylcholine; Aggression; Animals; Anxiety; Ataxia; Brain Chemistry; Conflict, Psychological; Data Interpretation, Statistical; Depression; Diazepam; Hypnotics and Sedatives; Microdialysis; Motor Activity; Muscarinic Antagonists; Piperidines; Prefrontal Cortex; Pyrimidines; Rats; Rats, Wistar; Receptors, Somatostatin; Recognition, Psychology; Scopolamine; Social Behavior; Swimming

2008
Behavioral effects of saredutant, a tachykinin NK2 receptor antagonist, in experimental models of mood disorders under basal and stress-related conditions.
    Pharmacology, biochemistry, and behavior, 2008, Volume: 90, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Antidepressive Agents, Tricyclic; Anxiety; Behavior, Animal; Benzamides; Clomipramine; Depressive Disorder; Diazepam; Electroshock; Grooming; Male; Mice; Mood Disorders; Motor Activity; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Stress, Psychological; Swimming

2008
Anxiolytic effects in mice of a dual blocker of fatty acid amide hydrolase and transient receptor potential vanilloid type-1 channels.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2009, Volume: 34, Issue:3

    Topics: Amidohydrolases; Anilides; Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Benzamides; Brain; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Cinnamates; Diazepam; Exploratory Behavior; Male; Mice; Mice, Inbred C57BL; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Serotonin; TRPV Cation Channels

2009
Scopolamine-induced deficits in social memory in mice: reversal by donepezil.
    Behavioural brain research, 2009, Dec-01, Volume: 204, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Cholinesterase Inhibitors; Diazepam; Donepezil; Dose-Response Relationship, Drug; Exploratory Behavior; Female; Indans; Memory; Memory Disorders; Mice; Mice, Inbred C57BL; Muscarinic Antagonists; Neuropsychological Tests; Nootropic Agents; Piperidines; Random Allocation; Scopolamine; Social Behavior; Time Factors

2009
Endocannabinoids mediate anxiolytic-like effect of acetaminophen via CB1 receptors.
    Progress in neuro-psychopharmacology & biological psychiatry, 2009, Oct-01, Volume: 33, Issue:7

    Topics: Acetaminophen; Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Behavior, Animal; Cannabinoid Receptor Modulators; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drinking; Endocannabinoids; Injections, Intraventricular; Interpersonal Relations; Male; Mice; Motor Activity; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1

2009
Altered responses of dopamine D3 receptor null mice to excitotoxic or anxiogenic stimuli: Possible involvement of the endocannabinoid and endovanilloid systems.
    Neurobiology of disease, 2009, Volume: 36, Issue:1

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Anti-Inflammatory Agents, Non-Steroidal; Anxiety; Arachidonic Acids; Brain; Cannabinoid Receptor Modulators; Capsaicin; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Endocannabinoids; Epilepsy; GABA Antagonists; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Knockout; Picrotoxin; Piperidines; Pyrazoles; Reaction Time; Receptor, Cannabinoid, CB1; Receptors, Dopamine D3; Serotonin; TRPV Cation Channels

2009
Prosocial effects of nicotine and ethanol in adolescent rats through partially dissociable neurobehavioral mechanisms.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2009, Volume: 34, Issue:12

    Topics: Aging; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Central Nervous System Depressants; Diazepam; Dopamine Antagonists; Ethanol; Exploratory Behavior; Flupenthixol; Locomotion; Male; Naloxone; Narcotic Antagonists; Nicotine; Nicotinic Agonists; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Rimonabant; Social Behavior

2009
Cannabidiol inhibitory effect on marble-burying behaviour: involvement of CB1 receptors.
    Behavioural pharmacology, 2010, Volume: 21, Issue:4

    Topics: Animals; Behavior, Animal; Cannabidiol; Diazepam; Dose-Response Relationship, Drug; Hypnotics and Sedatives; Male; Mice; Mice, Inbred C57BL; Motor Activity; Paroxetine; Piperazines; Piperidines; Pyrazoles; Pyridines; Receptor, Cannabinoid, CB1; Receptor, Serotonin, 5-HT1A; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Synaptic Transmission

2010
The effects of nociceptin/orphanin FQ receptor agonist Ro 64-6198 and diazepam on antinociception and remifentanil self-administration in rhesus monkeys.
    Psychopharmacology, 2011, Volume: 213, Issue:1

    Topics: Animals; Benzimidazoles; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Female; Imidazoles; Macaca mulatta; Male; Narcotic Antagonists; Nociceptin Receptor; Pain Measurement; Piperidines; Receptors, Opioid; Remifentanil; Self Administration; Spiro Compounds

2011
Inhibition of endocannabinoid catabolic enzymes elicits anxiolytic-like effects in the marble burying assay.
    Pharmacology, biochemistry, and behavior, 2011, Volume: 98, Issue:1

    Topics: Amidohydrolases; Animals; Anti-Anxiety Agents; Anxiety Disorders; Benzodioxoles; Cannabinoid Receptor Modulators; Diazepam; Disease Models, Animal; Dronabinol; Endocannabinoids; Enzyme Inhibitors; Male; Mice; Mice, Inbred C57BL; Monoacylglycerol Lipases; Obsessive-Compulsive Disorder; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant

2011
Enhancement of endocannabinoid signaling with JZL184, an inhibitor of the 2-arachidonoylglycerol hydrolyzing enzyme monoacylglycerol lipase, produces anxiolytic effects under conditions of high environmental aversiveness in rats.
    Pharmacological research, 2011, Volume: 64, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Benzodioxoles; Cannabinoid Receptor Modulators; Catalepsy; Diazepam; Endocannabinoids; Glycerides; Male; Monoacylglycerol Lipases; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; Signal Transduction

2011
Benzodiazepines modulate GABAA receptors by regulating the preactivation step after GABA binding.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Apr-25, Volume: 32, Issue:17

    Topics: Animals; Benzodiazepines; Binding Sites; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Ion Channel Gating; Isoxazoles; Larva; Membrane Potentials; Models, Biological; Mutation; Oocytes; Patch-Clamp Techniques; Piperidines; Protein Binding; Protein Subunits; Receptors, GABA-A; Xenopus

2012
Piperine decreases pilocarpine-induced convulsions by GABAergic mechanisms.
    Pharmacology, biochemistry, and behavior, 2013, Volume: 104

    Topics: Alkaloids; Amino Acids; Animals; Anticonvulsants; Antioxidants; Atropine; Benzodioxoles; Biogenic Monoamines; Brain; Diazepam; Disease Models, Animal; Epilepsy; Flumazenil; gamma-Aminobutyric Acid; Humans; Male; Memantine; Mice; Nimodipine; Nitrites; Pilocarpine; Piperidines; Polyunsaturated Alkamides; Seizures; Tumor Necrosis Factor-alpha

2013
Orexin receptor antagonists differ from standard sleep drugs by promoting sleep at doses that do not disrupt cognition.
    Science translational medicine, 2013, Apr-03, Volume: 5, Issue:179

    Topics: Administration, Oral; Animals; Attention; Azabicyclo Compounds; Choice Behavior; Cognition; Cytoskeletal Proteins; Diazepam; Eszopiclone; gamma-Aminobutyric Acid; Hippocampus; Hypnotics and Sedatives; Macaca mulatta; Male; Memory, Short-Term; Nerve Tissue Proteins; Orexin Receptors; Piperazines; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Recognition, Psychology; Sleep; Task Performance and Analysis; Time Factors; Triazoles; Zolpidem

2013
Anxiolytic-like effects observed in rats exposed to the elevated zero-maze following treatment with 5-HT2/5-HT3/5-HT4 ligands.
    Scientific reports, 2014, Jan-24, Volume: 4

    Topics: Aniline Compounds; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Male; Maze Learning; Oxazines; Piperidines; Propane; Pyrazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sulfonamides

2014
Possible involvement of GABAergic and nitriergic systems for antianxiety-like activity of piperine in unstressed and stressed mice.
    Pharmacological reports : PR, 2014, Volume: 66, Issue:5

    Topics: Alkaloids; Animals; Anti-Anxiety Agents; Anxiety; Benzodioxoles; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Guanidines; Indazoles; Male; Maze Learning; Mice; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type II; Nitrites; Piperidines; Polyunsaturated Alkamides; Stress, Psychological

2014
Post-exposure administration of diazepam combined with soluble epoxide hydrolase inhibition stops seizures and modulates neuroinflammation in a murine model of acute TETS intoxication.
    Toxicology and applied pharmacology, 2014, Dec-01, Volume: 281, Issue:2

    Topics: Animals; Anti-Inflammatory Agents; Anticonvulsants; Brain; Brain Waves; Bridged-Ring Compounds; Diazepam; Disease Models, Animal; Drug Administration Schedule; Drug Therapy, Combination; Electroencephalography; Encephalitis; Enzyme Inhibitors; Epoxide Hydrolases; GABA Modulators; Male; Mice; Phenylurea Compounds; Piperidines; Seizures; Time Factors

2014
GluN2B-containing N-methyl-D-aspartate receptors compensate for the inhibitory control of synaptic plasticity during the early critical period in the rat visual cortex.
    Journal of neuroscience research, 2015, Volume: 93, Issue:9

    Topics: 2-Amino-5-phosphonovalerate; Age Factors; Animals; Animals, Newborn; Bicuculline; Diazepam; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA Modulators; GABA-A Receptor Antagonists; Gene Expression Regulation, Developmental; Long-Term Potentiation; Male; Neural Inhibition; Piperidines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, N-Methyl-D-Aspartate; Visual Cortex

2015
Characterization of the Discriminative Stimulus Effects of a NOP Receptor Agonist Ro 64-6198 in Rhesus Monkeys.
    The Journal of pharmacology and experimental therapeutics, 2016, Volume: 357, Issue:1

    Topics: Analgesics, Opioid; Animals; Benzimidazoles; Conditioning, Operant; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Female; Fentanyl; GABA Modulators; Imidazoles; Macaca mulatta; Male; Naltrexone; Narcotic Antagonists; Nociceptin Receptor; Pain Measurement; Piperidines; Receptors, Opioid; Spiro Compounds

2016
Inhibition of Orexin Signaling Promotes Sleep Yet Preserves Salient Arousability in Monkeys.
    Sleep, 2016, Mar-01, Volume: 39, Issue:3

    Topics: Animals; Arousal; Conditioning, Classical; Cross-Over Studies; Diazepam; Eszopiclone; GABA Agents; Hypnotics and Sedatives; Macaca mulatta; Male; Orexin Receptor Antagonists; Orexins; Piperidines; Polysomnography; Signal Transduction; Sleep; Sleep Stages; Triazoles; Wakefulness

2016
Enhanced anandamide signaling reduces flight behavior elicited by an approaching robo-beetle.
    Neuropharmacology, 2017, Volume: 126

    Topics: Amidohydrolases; Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Avoidance Learning; Behavior, Animal; Benzamides; Benzodioxoles; Cannabinoid Receptor Agonists; Carbamates; Diazepam; Endocannabinoids; Fear; Male; Mice, Inbred C57BL; Monoacylglycerol Lipases; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant

2017
Inhibition of monoacylglycerol lipase terminates diazepam-resistant status epilepticus in mice and its effects are potentiated by a ketogenic diet.
    Epilepsia, 2018, Volume: 59, Issue:1

    Topics: Animals; Brain; Brain Waves; Carbamates; Cognition Disorders; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Resistant Epilepsy; Electroencephalography; Excitatory Amino Acid Agonists; Fluoresceins; Kainic Acid; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Monoacylglycerol Lipases; Neurons; Piperidines; Random Allocation; Receptor, Cannabinoid, CB1; Recognition, Psychology; Status Epilepticus; Sulfonamides; Time Factors

2018
Predicted values for human total clearance of a variety of typical compounds with differently humanized-liver mouse plasma data.
    Drug metabolism and pharmacokinetics, 2020, Volume: 35, Issue:4

    Topics: Acetamides; Albuterol; Animals; Carbamates; Chromatography, Liquid; Diazepam; Diclofenac; Digitoxin; Humans; Itraconazole; Ketoprofen; Liver; Metabolic Clearance Rate; Mice; Mice, Transgenic; Naproxen; Pharmaceutical Preparations; Phenytoin; Piperidines; Pravastatin; Pyrimidines; Quinidine; Tandem Mass Spectrometry; Telmisartan; Terfenadine; Verapamil

2020