diazepam and mannitol

diazepam has been researched along with mannitol in 38 studies

Research

Studies (38)

TimeframeStudies, this research(%)All Research%
pre-199012 (31.58)18.7374
1990's1 (2.63)18.2507
2000's13 (34.21)29.6817
2010's11 (28.95)24.3611
2020's1 (2.63)2.80

Authors

AuthorsStudies
Ghuloum, AM; Jain, AN; Sage, CR1
Duffy, EM; Jorgensen, WL1
Ertl, P; Rohde, B; Selzer, P1
Artursson, P; Luthman, K; Norinder, U; Stenberg, P1
Caron, G; Ermondi, G1
Baert, B; Beetens, J; Bodé, S; De Spiegeleer, B; Deconinck, E; Lambert, J; Slegers, G; Slodicka, M; Stoppie, P; Van Gele, M; Vander Heyden, Y1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Du-Cuny, L; Mash, EA; Meuillet, EJ; Moses, S; Powis, G; Song, Z; Zhang, S1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Campillo, NE; Guerra, A; Páez, JA1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Barber, S; Dew, TP; Farrell, TL; Poquet, L; Williamson, G1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Fieschi, C; Pappius, HM; Rapoport, SI; Savaki, HE; Sokoloff, L1
Kelly, JV1
Posner, JB1
Barkhatova, TP; Rasstrigin, NN; Sukhanova, LP1
Ono, T; Umemoto, S; Wada, O1
Brehm, R1
Cavazzuti, GB1
Anglin, C; Bannatyne, R; Fleming, P; Hsuen, J; Murray, JD; Weber, J1
Black, AM1
Haller, J1
Ferrero, A; Marzullo, C; Salmoiraghi, ML1
Fieschi, C; Lenzi, GL; Orzi, F; Passero, S; Zanette, E1
Charman, SA; Gibson, PR; Porter, CJ; Sinclair, AJ; Vine, DF1
Dey, S; Gunda, S; Mitra, AK1
Kansara, V; Mitra, AK1
Katragadda, S; Mitra, AK; Talluri, RS1
Abbate, M; Ferlazzo, E; Granata, F; Mazzù, I; Musolino, R; Narbone, MC1
Betto, G; Fan, Q; Fazio, V; Ghosh, C; Janigro, D; Machado, A; Marchi, N1
Freeman, DE; Graham, AS; Grosche, A; Morton, AJ; Polyak, MM1
Douville, NJ; ElSayed, M; Takayama, S; Wang, JD1
Broekhuis, J; Frijlink, HW; Grasmeijer, N; Hinrichs, WLJ; Kauppinen, A; Ketolainen, J; Tonnis, W1
Hansen, SE; Jacobsen, J; Janfelt, C; Marxen, E1
Aumann, M; Clabots, MF; Gaillard, E1
Nelson, KM; Rautiola, D; Siegel, RA; Updyke, JL1

Reviews

2 review(s) available for diazepam and mannitol

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
The continuing problem of purulent meningitis in infants and children.
    Pediatric clinics of North America, 1974, Volume: 21, Issue:4

    Topics: Bacterial Vaccines; Bicarbonates; Brain Edema; Diagnosis, Differential; Diazepam; Digoxin; Fever; Gastrointestinal Hemorrhage; Heparin; Humans; Hydrocortisone; Infant; Infant, Newborn; Isoproterenol; Mannitol; Meningitis; Meningitis, Meningococcal; Meningitis, Viral; Phenytoin; Seizures; Shock, Septic; Vitamin K

1974

Other Studies

36 other study(ies) available for diazepam and mannitol

ArticleYear
Molecular hashkeys: a novel method for molecular characterization and its application for predicting important pharmaceutical properties of molecules.
    Journal of medicinal chemistry, 1999, May-20, Volume: 42, Issue:10

    Topics: Drug Design; Intestinal Absorption; Models, Molecular; Pharmaceutical Preparations; Structure-Activity Relationship

1999
Prediction of drug solubility from Monte Carlo simulations.
    Bioorganic & medicinal chemistry letters, 2000, Jun-05, Volume: 10, Issue:11

    Topics: Monte Carlo Method; Pharmaceutical Preparations; Solubility

2000
Fast calculation of molecular polar surface area as a sum of fragment-based contributions and its application to the prediction of drug transport properties.
    Journal of medicinal chemistry, 2000, Oct-05, Volume: 43, Issue:20

    Topics: Biological Availability; Biological Transport; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Reproducibility of Results

2000
Experimental and computational screening models for the prediction of intestinal drug absorption.
    Journal of medicinal chemistry, 2001, Jun-07, Volume: 44, Issue:12

    Topics: Biological Transport; Carbon Radioisotopes; Cell Line; Cell Membrane; Cell Membrane Permeability; Ciprofloxacin; Computational Biology; Drug Design; Foscarnet; Humans; Hydrogen Bonding; Intestinal Absorption; Intestinal Mucosa; Lactulose; Mannitol; Models, Biological; Raffinose; Surface Properties; Tritium; Verapamil

2001
Calculating virtual log P in the alkane/water system (log P(N)(alk)) and its derived parameters deltalog P(N)(oct-alk) and log D(pH)(alk).
    Journal of medicinal chemistry, 2005, May-05, Volume: 48, Issue:9

    Topics: 1-Octanol; Alkanes; Hydrogen-Ion Concentration; Least-Squares Analysis; Mathematics; Models, Chemical; Models, Molecular; Solvents; Water

2005
Transdermal penetration behaviour of drugs: CART-clustering, QSPR and selection of model compounds.
    Bioorganic & medicinal chemistry, 2007, Nov-15, Volume: 15, Issue:22

    Topics: Anti-Inflammatory Agents; Cell Membrane Permeability; Cluster Analysis; Drug Evaluation, Preclinical; Humans; Models, Biological; Predictive Value of Tests; Quantitative Structure-Activity Relationship; Regression Analysis; Skin; Skin Absorption

2007
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Computational modeling of novel inhibitors targeting the Akt pleckstrin homology domain.
    Bioorganic & medicinal chemistry, 2009, Oct-01, Volume: 17, Issue:19

    Topics: Antineoplastic Agents; Blood Proteins; Caco-2 Cells; Cell Membrane Permeability; Computer Simulation; Drug Discovery; Drug Screening Assays, Antitumor; Humans; Models, Molecular; Phosphoproteins; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-akt; Quantitative Structure-Activity Relationship

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
Predicting phenolic acid absorption in Caco-2 cells: a theoretical permeability model and mechanistic study.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:2

    Topics: Artificial Intelligence; Caco-2 Cells; Cell Membrane Permeability; Cinnamates; Enterocytes; Humans; Hydrophobic and Hydrophilic Interactions; Intestinal Absorption; Kinetics; Models, Biological; Molecular Conformation; Osmolar Concentration; Phenols

2012
Osmotic opening of the blood-brain barrier and local cerebral glucose utilization.
    Annals of neurology, 1979, Volume: 5, Issue:3

    Topics: Animals; Autoradiography; Blood-Brain Barrier; Brain; Cerebrovascular Circulation; Deoxyglucose; Diazepam; Glucose; Hypertonic Solutions; Male; Mannitol; Rats

1979
Drugs used in the management of toxemia of pregnancy.
    Clinical obstetrics and gynecology, 1977, Volume: 20, Issue:2

    Topics: Anticonvulsants; Antihypertensive Agents; Barbiturates; Benzothiadiazines; Blood Volume; Diazepam; Diuretics; Ethacrynic Acid; Female; Furosemide; Heparin; Humans; Hydralazine; Magnesium; Mannitol; Methyldopa; Myometrium; Phytotherapy; Plants, Medicinal; Plants, Toxic; Pre-Eclampsia; Pregnancy; Ritodrine; Secologanin Tryptamine Alkaloids; Sodium Chloride Symporter Inhibitors; Veratrum

1977
The comatose patient.
    JAMA, 1975, Sep-22, Volume: 233, Issue:12

    Topics: Coma; Dexamethasone; Diazepam; Emergencies; Fever; Glucose; Humans; Hypothermia; Intracranial Pressure; Intubation, Intratracheal; Mannitol; Seizures

1975
[Use of droperidol in the complex treatment of severe forms of late pregnancy toxemias].
    Akusherstvo i ginekologiia, 1975, Issue:9

    Topics: Adolescent; Adult; Diazepam; Droperidol; Drug Therapy, Combination; Female; Humans; Injections, Intravenous; Mannitol; Pre-Eclampsia; Pregnancy

1975
Introduction of new indices into continuous avoidance test--a trial to detect the effects of sodium chloride and mannitol on avoidance behavior.
    The Journal of toxicological sciences, 1987, Volume: 12, Issue:4

    Topics: Animals; Avoidance Learning; Diazepam; Male; Mannitol; Mice; Mice, Inbred Strains; Microcomputers; Signal Processing, Computer-Assisted; Sodium Chloride

1987
[Therapy of late gestoses].
    Minerva ginecologica, 1973, Volume: 25, Issue:7

    Topics: Adult; Chlormethiazole; Diazepam; Diuretics; Eclampsia; Female; Heparinoids; Humans; Mannitol; Pre-Eclampsia; Pregnancy

1973
[Considerations and research on febrile convulsions].
    Minerva pediatrica, 1974, Apr-14, Volume: 26, Issue:13

    Topics: Anticonvulsants; Brain Diseases; Child, Preschool; Diagnosis, Differential; Diazepam; Electroencephalography; Epilepsy; Female; Fever; Humans; Infant; Male; Mannitol; Phenobarbital; Phenytoin; Primidone; Seizures

1974
Self poisoning with dieldrin: a case report and pharmacokinetic discussion.
    Anaesthesia and intensive care, 1974, Volume: 2, Issue:4

    Topics: Adult; Diazepam; Dieldrin; Electroencephalography; Humans; Male; Mannitol; Poisoning; Positive-Pressure Respiration; Suicide

1974
[Therapy of EPH gestosis].
    Deutsche medizinische Wochenschrift (1946), 1973, Jul-06, Volume: 98, Issue:27

    Topics: Chlorthalidone; Diazepam; Diet Therapy; Eclampsia; Edema; Female; Furosemide; Guanethidine; Humans; Hydralazine; Hydrochlorothiazide; Hypertension; Magnesium Sulfate; Mannitol; Phenobarbital; Phytotherapy; Plants, Medicinal; Pre-Eclampsia; Pregnancy; Proteinuria; Rauwolfia

1973
[Intensive therapy of gestoses. Our experience in the years 1969-1971].
    Annali di ostetricia, ginecologia, medicina perinatale, 1971, Volume: 92, Issue:12

    Topics: Betamethasone; Brain Edema; Diazepam; Ergoloid Mesylates; Female; Furosemide; Humans; Mannitol; Papaverine; Phytotherapy; Plants, Medicinal; Pre-Eclampsia; Pregnancy; Rauwolfia; Thiopental

1971
Effects on EEG of the osmotic opening of the blood-brain barrier in rats.
    Life sciences, 1980, Jul-21, Volume: 27, Issue:3

    Topics: Animals; Blood-Brain Barrier; Diazepam; Electroencephalography; Evans Blue; Male; Mannitol; Osmosis; Rats; Seizures

1980
Effect of dietary fatty acids on the intestinal permeability of marker drug compounds in excised rat jejunum.
    The Journal of pharmacy and pharmacology, 2002, Volume: 54, Issue:6

    Topics: Analysis of Variance; Animals; Biological Transport; Diazepam; Dietary Fats; Digoxin; Electrophysiology; Fatty Acids; Fatty Acids, Unsaturated; Glucose; In Vitro Techniques; Intestinal Absorption; Jejunum; Male; Mannitol; Microvilli; Permeability; Phospholipids; Rats; Rats, Sprague-Dawley

2002
Pharmacokinetics of erythromycin in rabbit corneas after single-dose infusion: role of P-glycoprotein as a barrier to in vivo ocular drug absorption.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 311, Issue:1

    Topics: Absorption; Amino Acid Sequence; Animals; Area Under Curve; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Carbon Radioisotopes; Cell Division; Cells, Cultured; Cornea; Diazepam; Dogs; Dose-Response Relationship, Drug; Erythromycin; Eye; Humans; Male; Mannitol; Molecular Sequence Data; Protein Biosynthesis; Protein Synthesis Inhibitors; Rabbits; Reverse Transcriptase Polymerase Chain Reaction; Sequence Homology, Amino Acid

2004
Evaluation of an ex vivo model implication for carrier-mediated retinal drug delivery.
    Current eye research, 2006, Volume: 31, Issue:5

    Topics: Animals; Biological Transport; Carrier Proteins; Cell Membrane Permeability; Cell Survival; Choroid; Diazepam; Diffusion Chambers, Culture; Drug Delivery Systems; Electric Conductivity; Folate Receptors, GPI-Anchored; Folic Acid; Hydrogen-Ion Concentration; Mannitol; Membrane Potentials; Methotrexate; Models, Biological; Pigment Epithelium of Eye; Rabbits; Receptors, Cell Surface; Retina; Sclera; Temperature; Tetrahydrofolates

2006
Simultaneous modulation of transport and metabolism of acyclovir prodrugs across rabbit cornea: An approach involving enzyme inhibitors.
    International journal of pharmaceutics, 2006, Aug-31, Volume: 320, Issue:1-2

    Topics: Acyclovir; Aminopeptidases; Animals; Antiviral Agents; Biological Transport; Carboxylic Ester Hydrolases; Cell Membrane Permeability; Cells, Cultured; Cornea; Diazepam; Dose-Response Relationship, Drug; Enzyme Inhibitors; Hydrolysis; Kinetics; Leucine; Male; Mannitol; p-Chloromercuribenzoic Acid; Peptides; Prodrugs; Rabbits; Valacyclovir; Valine

2006
PRES: posterior or potentially reversible encephalopathy syndrome?
    Neurological sciences : official journal of the Italian Neurological Society and of the Italian Society of Clinical Neurophysiology, 2006, Volume: 27, Issue:3

    Topics: Adult; Anti-Inflammatory Agents; Anticonvulsants; Antihypertensive Agents; Brain; Brain Diseases; Clonidine; Dexamethasone; Diazepam; Diuretics, Osmotic; Eclampsia; Female; Humans; Magnesium Sulfate; Magnetic Resonance Imaging; Mannitol; Nifedipine; Pregnancy; Seizures

2006
Blood-brain barrier damage and brain penetration of antiepileptic drugs: role of serum proteins and brain edema.
    Epilepsia, 2009, Volume: 50, Issue:4

    Topics: Analysis of Variance; Animals; Anticonvulsants; Blood Proteins; Blood-Brain Barrier; Brain; Brain Edema; Capillary Permeability; Carbon Isotopes; Chromatography, High Pressure Liquid; Deoxyglucose; Diazepam; Diuretics, Osmotic; Electrochemistry; Hippocampus; In Vitro Techniques; Male; Mannitol; Models, Biological; Phenytoin; Radioligand Assay; Rats; Rats, Sprague-Dawley; Sucrose; Time Factors; Tissue Distribution; Tritium

2009
In vitro and in vivo responses of mucosa from the large colon of horses to ischemia and reperfusion.
    American journal of veterinary research, 2011, Volume: 72, Issue:7

    Topics: Analysis of Variance; Anesthetics, Intravenous; Animals; Colon; Diazepam; Electric Impedance; Horse Diseases; Horses; Hypnotics and Sedatives; Intestinal Mucosa; Ischemia; Ketamine; Mannitol; Reperfusion Injury; Statistics, Nonparametric; Xylazine

2011
Quantitative analysis of molecular absorption into PDMS microfluidic channels.
    Annals of biomedical engineering, 2012, Volume: 40, Issue:9

    Topics: 1-Octanol; Absorption; Dexamethasone; Diazepam; Dimethylpolysiloxanes; Glass; Hydrophobic and Hydrophilic Interactions; Mannitol; Microfluidic Analytical Techniques; Phenytoin; Rhodamines; Titanium; Water

2012
Efficient production of solid dispersions by spray drying solutions of high solid content using a 3-fluid nozzle.
    European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V, 2018, Volume: 123

    Topics: Diazepam; Drug Carriers; Drug Compounding; Hydrophobic and Hydrophilic Interactions; Mannitol; Particle Size; Solubility; Solutions; Solvents; Water

2018
Buccal delivery of small molecules - Impact of levulinic acid, oleic acid, sodium dodecyl sulfate and hypotonicity on ex vivo permeability and spatial distribution in mucosa.
    European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V, 2018, Volume: 133

    Topics: Administration, Buccal; Animals; Caffeine; Diazepam; Epithelium; Levulinic Acids; Lipids; Mannitol; Micelles; Mouth Mucosa; Oleic Acid; Osmolar Concentration; Permeability; Propylene Glycol; Small Molecule Libraries; Sodium Dodecyl Sulfate; Swine

2018
Acute kidney injury, seizures, and hypertonic hyponatremia secondary to mannitol intoxication in a dog.
    Journal of veterinary emergency and critical care (San Antonio, Tex. : 2001), 2019, Volume: 29, Issue:6

    Topics: Acute Kidney Injury; Animals; Anticonvulsants; Creatinine; Diazepam; Dog Diseases; Dogs; Drug Overdose; Hypokalemia; Hyponatremia; Male; Mannitol; Osmolar Concentration; Seizures; Urinalysis

2019
Diazepam Prodrug Stabilizes Human Aminopeptidase B during Lyophilization.
    Molecular pharmaceutics, 2020, 02-03, Volume: 17, Issue:2

    Topics: Aminopeptidases; Biocatalysis; Diazepam; Dipeptides; Drug Stability; Enzyme Stability; Freeze Drying; Freezing; Humans; Mannitol; Prodrugs; Proteolysis; Trehalose

2020