diazepam and lormetazepam

diazepam has been researched along with lormetazepam in 33 studies

Research

Studies (33)

TimeframeStudies, this research(%)All Research%
pre-199019 (57.58)18.7374
1990's3 (9.09)18.2507
2000's7 (21.21)29.6817
2010's3 (9.09)24.3611
2020's1 (3.03)2.80

Authors

AuthorsStudies
Babbini, M; Barbaro, AM; Bartoletti, M; Biagi, GL; Borea, PA; Gaiardi, M; Guerra, MC1
Abraham, MH; Gao, F; Lombardo, F; Shalaeva, MY; Tupper, KA1
Gao, F; Lombardo, F; Shalaeva, MY; Tupper, KA1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY2
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Campillo, NE; Guerra, A; Páez, JA1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Doyle, D; Kragie, L1
Andrews, JS; Jensen, LH; Kehr, W; Petersen, EN; Rettig, KJ; Schmiechen, R; Schneider, HH; Stephens, DN; Turner, JD; Turski, L1
Doenicke, A; Greim, M; Juhl, G; Rampf, U; Suttmann, H1
Schneider, HH; Stephens, DN; Weidmann, R; Zimmermann, L1
Schneider, HH; Stephens, DN2
Wildmann, J1
Vernay, A; Vu Duc, T1
Grabe, N; Hansen, W; Jakobsen, CJ; Jensen, JJ1
Ceccarelli, G; de Leo, D1
Groves, ND; Rees, JL; Rosen, M1
Barry, H; Bewley, A; Fox, E; McCreary, C; O'Boyle, CA1
Benkert, O; Heuser, I; Wetzel, H1
Jung, M; Kappa, E; Manegold, BC; Müller, HP; Schratzer, M; Tolksdorf, W1
Fichte, K; Hentschel, HD; Sastre y Hernández, M1
Fichte, K; Hentschel, HD; Sastre y Hernández, MS1
Dorow, RG; Schneider, HH; Seidler, J1
Dorow, R; Horowski, R1
Fichte, K; Hemmerling, KG; Neubert, W; Ott, H; Schratzer, M; Willumeit, HP1
Ott, H1
Neubert, W; Ott, H; Willumeit, HP1
Kamei, C; Nishino, T; Takechi, K; Takeuchi, T1
Andresen-Streichert, H; Froch-Cortis, J; Lehmann, S; Mercer-Chalmers-Bender, K; Rothschild, MA; Sczyslo, A; Thevis, M1
Falcon, M; Fernadez-Lopez, L; Luna, A; Mancini, R; Pellegrini, M; Rotolo, M1

Trials

9 trial(s) available for diazepam and lormetazepam

ArticleYear
[Beta activation following the intravenous administration of benzodiazepines and the specific antagonist flumazenil (Ro 15-1788)].
    EEG-EMG Zeitschrift fur Elektroenzephalographie, Elektromyographie und verwandte Gebiete, 1990, Volume: 21, Issue:1

    Topics: Adult; Anti-Anxiety Agents; Benzodiazepines; Beta Rhythm; Diazepam; Dose-Response Relationship, Drug; Electroencephalography; Flumazenil; Flunitrazepam; Humans; Injections, Intravenous; Lorazepam; Male; Midazolam; Prospective Studies; Randomized Controlled Trials as Topic; Stimulation, Chemical

1990
Oral lormetazepam in premedication. A comparison with diazepam.
    Anaesthesia, 1986, Volume: 41, Issue:8

    Topics: Administration, Oral; Adult; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Drug Evaluation; Female; Humans; Lorazepam; Male; Preanesthetic Medication

1986
Antianxiety properties of lormetazepam. A double-blind crossover trial versus diazepam.
    The Journal of international medical research, 1986, Volume: 14, Issue:6

    Topics: Adult; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Humans; Lorazepam; Male; Middle Aged

1986
Controlled comparison of a new sublingual lormetazepam formulation and i.v. diazepam in outpatient minor oral surgery.
    British journal of anaesthesia, 1988, Volume: 60, Issue:4

    Topics: Administration, Sublingual; Adult; Ambulatory Surgical Procedures; Anesthesia, Dental; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Drug Evaluation; Hemodynamics; Humans; Infusions, Intravenous; Lorazepam; Memory; Patient Acceptance of Health Care; Preanesthetic Medication; Tooth, Impacted

1988
[Intravenous sedation before endoscopic interventions. Comparative study of lormetazepam and diazepam in oil].
    Fortschritte der Medizin, 1985, Mar-07, Volume: 103, Issue:9

    Topics: Adult; Aged; Anti-Anxiety Agents; Benzodiazepines; Cholangiopancreatography, Endoscopic Retrograde; Diazepam; Female; Humans; Hypnotics and Sedatives; Injections, Intravenous; Lorazepam; Male; Middle Aged; Premedication

1985
[Lormetazepam in the treatment of sleep disorders in a medical practice; double-blind test on 100 patients (author's transl)].
    Deutsche medizinische Wochenschrift (1946), 1981, May-29, Volume: 106, Issue:22

    Topics: Adult; Aged; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Double-Blind Method; Female; Humans; Lorazepam; Male; Middle Aged; Sleep Wake Disorders

1981
Comparative efficacy of lormetazepam (Noctamid) and diazepam (Valium) in 100 out-patients with insomnia.
    The Journal of international medical research, 1981, Volume: 9, Issue:3

    Topics: Adult; Aged; Anti-Anxiety Agents; Benzodiazepines; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Humans; Lorazepam; Male; Middle Aged; Sleep Initiation and Maintenance Disorders

1981
A radioreceptor assay to study the affinity of benzodiazepines and their receptor binding activity in human plasma including their active metabolites.
    British journal of clinical pharmacology, 1982, Volume: 13, Issue:4

    Topics: Adult; Anti-Anxiety Agents; Benzodiazepines; Biotransformation; Blood Proteins; Diazepam; Female; Humans; Lorazepam; Male; Nitrazepam; Nordazepam; Protein Binding; Radioligand Assay; Receptors, Drug; Receptors, GABA-A

1982
Are electroencephalographic and psychomotor measures sensitive in detecting residual sequelae of benzodiazepine hypnotics?
    Psychopharmacology. Supplementum, 1984, Volume: 1

    Topics: Adult; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Double-Blind Method; Electroencephalography; Female; Flunitrazepam; Half-Life; Humans; Hypnotics and Sedatives; Lorazepam; Male; Middle Aged; Psychomotor Performance; Radioligand Assay; Sleep

1984

Other Studies

24 other study(ies) available for diazepam and lormetazepam

ArticleYear
Rm values and structure-activity relationship of benzodiazepines.
    Journal of medicinal chemistry, 1980, Volume: 23, Issue:2

    Topics: Animals; Benzodiazepines; Chromatography, Thin Layer; Conflict, Psychological; Exploratory Behavior; Models, Biological; Rats; Solubility; Structure-Activity Relationship

1980
ElogPoct: a tool for lipophilicity determination in drug discovery.
    Journal of medicinal chemistry, 2000, Jul-27, Volume: 43, Issue:15

    Topics: 1-Octanol; Chromatography, High Pressure Liquid; Pharmaceutical Preparations; Solubility; Solvents

2000
ElogD(oct): a tool for lipophilicity determination in drug discovery. 2. Basic and neutral compounds.
    Journal of medicinal chemistry, 2001, Jul-19, Volume: 44, Issue:15

    Topics: 1-Octanol; Chromatography, High Pressure Liquid; Pharmaceutical Preparations; Solubility; Water

2001
Prediction of volume of distribution values in humans for neutral and basic drugs using physicochemical measurements and plasma protein binding data.
    Journal of medicinal chemistry, 2002, Jun-20, Volume: 45, Issue:13

    Topics: Blood Proteins; Chemical Phenomena; Chemistry, Physical; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding

2002
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Benzodiazepines inhibit temperature-dependent L-[125I]triiodothyronine accumulation into human liver, human neuroblast, and rat pituitary cell lines.
    Endocrinology, 1992, Volume: 130, Issue:3

    Topics: Adenoma; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Cell Line; Convulsants; Diazepam; Dose-Response Relationship, Drug; Humans; Iodine Radioisotopes; Liver; Lorazepam; Neuroblastoma; Pituitary Neoplasms; Rats; Receptors, Thyroid Hormone; Temperature; Triazolam; Triiodothyronine; Tritium; Tumor Cells, Cultured

1992
Abecarnil, a metabolically stable, anxioselective beta-carboline acting at benzodiazepine receptors.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Diazepam; Female; Lorazepam; Male; Mice; Motor Activity; Punishment; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
Decreased sensitivity to benzodiazepine receptor agonists and increased sensitivity to inverse agonists following chronic treatments: evidence for separate mechanisms.
    Advances in biochemical psychopharmacology, 1988, Volume: 45

    Topics: Animals; Anti-Anxiety Agents; Appetite Depressants; Benzodiazepines; Carbolines; Chlorides; Diazepam; Drug Interactions; Drug Tolerance; Exploratory Behavior; Ion Channels; Kindling, Neurologic; Locomotion; Lorazepam; Mice; Muscimol; Pentylenetetrazole; Rats; Receptors, GABA-A

1988
Co-existence of kindling induced by the beta-carboline, FG 7142, and tolerance to diazepam following chronic treatment in mice.
    European journal of pharmacology, 1988, Sep-01, Volume: 154, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Carbolines; Diazepam; Drug Tolerance; Female; Kindling, Neurologic; Lorazepam; Mice; Motor Activity; Punishment; Receptors, GABA-A; Seizures

1988
Increase of natural benzodiazepines in wheat and potato during germination.
    Biochemical and biophysical research communications, 1988, Dec-30, Volume: 157, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Brain; Cell Membrane; Chromatography, High Pressure Liquid; Diazepam; Gas Chromatography-Mass Spectrometry; Lorazepam; Plant Development; Plants; Rats; Receptors, GABA-A; Solanum tuberosum; Triticum

1988
[Validation of a method for detecting benzodiazepines in the urine by acid extraction of their benzophenones and thin layer chromatography].
    Annales de biologie clinique, 1985, Volume: 43, Issue:3

    Topics: Anti-Anxiety Agents; Benzodiazepines; Benzophenones; Bromazepam; Chromatography, Gas; Chromatography, Thin Layer; Clonazepam; Diazepam; Humans; Hydrogen-Ion Concentration; Hydrolysis; Lorazepam; Nitrazepam

1985
Effects of benzodiazepines on laryngeal reflexes. Comparison of lormetazepam and Diazemuls.
    Anaesthesia, 1987, Volume: 42, Issue:8

    Topics: Adolescent; Adult; Ammonia; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Humans; Larynx; Lorazepam; Psychomotor Performance; Reflex; Time Factors

1987
Benzodiazepines for catatonic symptoms, stupor, and mutism.
    Pharmacopsychiatry, 1988, Volume: 21, Issue:6

    Topics: Anti-Anxiety Agents; Benzodiazepines; Catatonia; Depressive Disorder; Diazepam; Female; Flumazenil; Humans; Lorazepam; Mutism

1988
Tolerance to the benzodiazepine diazepam in an animal model of anxiolytic activity.
    Psychopharmacology, 1985, Volume: 87, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Diazepam; Drug Tolerance; Female; gamma-Aminobutyric Acid; Lorazepam; Male; Mice; Punishment; Receptors, GABA-A

1985
[Significance of pharmacokinetic findings for the clinical effect of benzodiazepines].
    Der Internist, 1982, Volume: 23, Issue:11

    Topics: Anti-Anxiety Agents; Benzodiazepines; Biological Availability; Chemical Phenomena; Chemistry; Diazepam; Half-Life; Humans; Kinetics; Lorazepam

1982
Alcohol interaction of lormetazepam, mepindolol sulphate and diazepam measured by performance on the driving simulator.
    Pharmacopsychiatry, 1984, Volume: 17, Issue:2

    Topics: Adult; Anti-Anxiety Agents; Automobile Driving; Benzodiazepines; Diazepam; Double-Blind Method; Drug Interactions; Ethanol; Female; Humans; Lorazepam; Male; Pindolol; Placebos; Psychomotor Performance; Pulse; Reaction Time

1984
Simulated car driving as a useful technique for the determination of residual effects and alcohol interaction after short- and long-acting benzodiazepines.
    Psychopharmacology. Supplementum, 1984, Volume: 1

    Topics: Anti-Anxiety Agents; Automobile Driving; Benzodiazepines; Diazepam; Double-Blind Method; Drug Interactions; Ethanol; Flurazepam; Heart Rate; Humans; Hypnotics and Sedatives; Lorazepam; Pindolol; Psychomotor Performance; Reaction Time

1984
Evaluation of anxiolytic-like effects of some short-acting benzodiazepine hypnotics in mice.
    Journal of pharmacological sciences, 2008, Volume: 107, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Azepines; Benzodiazepines; Diazepam; Hypnotics and Sedatives; Lorazepam; Male; Maze Learning; Mice; Mice, Inbred ICR; Motor Activity; Triazolam

2008
Organ distribution of diclazepam, pyrazolam and 3-fluorophenmetrazine.
    Forensic science international, 2019, Volume: 303

    Topics: Adult; Benzodiazepines; Bile; Body Fluids; Brain Chemistry; Designer Drugs; Diazepam; Forensic Toxicology; Gastrointestinal Contents; Humans; Kidney; Liver; Lorazepam; Lung; Male; Nordazepam; Pericardial Fluid; Phenmetrazine; Postmortem Changes; Psoas Muscles; Tandem Mass Spectrometry

2019
Postmortem Analysis of Benzodiazepines in Human Bone by Gas Chromatography-Mass Spectrometry.
    Journal of analytical toxicology, 2021, Jan-21, Volume: 44, Issue:9

    Topics: Alprazolam; Autopsy; Benzodiazepines; Chromatography, Liquid; Clonazepam; Diazepam; Forensic Toxicology; Gas Chromatography-Mass Spectrometry; Humans; Liquid-Liquid Extraction; Lorazepam; Nordazepam; Oxazepam; Tandem Mass Spectrometry

2021