diazepam and l 663581

diazepam has been researched along with l 663581 in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19901 (20.00)18.7374
1990's3 (60.00)18.2507
2000's1 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baker, R; Engelstoff, M; Herbert, R; Knight, A; MacLeod, A; Merchant, K; Moseley, J; Saunders, J; Swain, CJ; Watjen, F1
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S1
Honoré, T; Iversen, SD; Kemp, JA; Knight, AR; Marshall, GR; Rupniak, NM; Singh, L; Tricklebank, MD; Tye, S; Watjen, F1
Lin, JH; Lin, TH1
Jackson, A1

Other Studies

5 other study(ies) available for diazepam and l 663581

ArticleYear
Novel benzodiazepine receptor partial agonists: oxadiazolylimidazobenzodiazepines.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:10

    Topics: Animals; Benzodiazepines; Cell Membrane; Cerebral Cortex; Models, Molecular; Molecular Conformation; Molecular Structure; Oxadiazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Structure-Activity Relationship; X-Ray Diffraction

1989
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship

2000
The pharmacological properties of the imidazobenzodiazepine, FG 8205, a novel partial agonist at the benzodiazepine receptor.
    British journal of pharmacology, 1990, Volume: 101, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Brain; Conditioning, Psychological; Diazepam; In Vitro Techniques; Macaca fascicularis; Male; Mice; Rats; Receptors, GABA-A; Seizures

1990
Effects of protein binding and experimental disease states on brain uptake of benzodiazepines in rats.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Blood-Brain Barrier; Brain; Devazepide; Diabetes Mellitus, Experimental; Diazepam; Kidney Diseases; Liver Diseases; Male; Phenylurea Compounds; Protein Binding; Rats; Rats, Inbred Strains; Serum Albumin

1990
State-dependent effects of atypical benzodiazepine-receptor agonists.
    Psychopharmacology, 1995, Volume: 119, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; GABA-A Receptor Agonists; Hypnotics and Sedatives; Male; Pyridines; Rats; Rats, Wistar; Zolpidem

1995