diazepam and imidazenil

diazepam has been researched along with imidazenil in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's12 (54.55)18.2507
2000's9 (40.91)29.6817
2010's1 (4.55)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Biggio, G; Dazzi, L; Gessa, GL; Imperato, A; Motzo, C; Serra, M1
Auta, J; Costa, E; Giusti, P; Guidotti, A1
Arban, R; Costa, E; Ducić, I; Giusti, P; Guidotti, A; Puia, G; Walser, A1
Biggio, G; Dazzi, L; Maira, G; Motzo, C; Sanna, A; Serra, M1
Biggio, G; Ghiani, CA; Motzo, C; Porceddu, ML; Serra, M1
Caruncho, H; Costa, E; Fritschy, JM; Guidotti, A; Impagnatiello, F; Longone, P; Pesold, C1
Contarino, A; Giusti, P; Lipartiti, M; Mariot, R; Zanotti, A1
Benke, D; Benson, JA; Carter, DB; Hamilton, BJ; Knoflach, F; Lüddens, H; Mohler, H; Scheurer, L; Wang, Y1
Costa, E; Guidotti, A; Impagnatiello, F; Longone, P1
Biggio, G; Dazzi, L; Motzo, C; Porceddu, ML; Sanna, A; Serra, M1
Appel, SB; Brodie, MS; Costa, E; Davis, JM; Giorgetti, M; Guidotti, A; Javaid, JI1
Contarino, A; Giusti, P; Lipartiti, M; Natolino, F; Zanotti, A1
Ator, NA; Kautz, MA1
Crain, BJ; Evenson, DA; Miller, KA; Nadler, JV; Schwartz-Bloom, RD1
Biggio, F; Biggio, G; Busonero, F; Cagetti, E; Carta, M; Desole, MS; Follesa, P; Maciocco, E; Manca, A; Mancuso, L; Massa, F; Sanna, E1
Auta, J; Costa, E; Grayson, DR; Guidotti, A; Matsumoto, K; Pappas, GD; Zhang, X1
Auta, J; Costa, E; Davis, J; Guidotti, A1
Auta, J; Costa, E; Davis, JM; Guidotti, A1
Agis-Balboa, RC; Costa, E; Grayson, DR; Guidotti, A; Matsumoto, K; Pinna, G; Zhubi, A1
Auta, J; Costa, E; Guidotti, A; Impagnatiello, F; Kadriu, B1
Auta, J; Costa, E; Guidotti, A; Kadriu, B1
Auta, J; Davis, JM; Gocel, J; Guidotti, A; Kadriu, B; Larson, J; Nambiar, MP1

Reviews

1 review(s) available for diazepam and imidazenil

ArticleYear
GABAA receptors and benzodiazepines: a role for dendritic resident subunit mRNAs.
    Neuropharmacology, 2002, Volume: 43, Issue:6

    Topics: Allosteric Regulation; Animals; Benzodiazepines; Binding, Competitive; Chloride Channels; Dendrites; Diazepam; Drug Tolerance; GABA Modulators; Glutamate Decarboxylase; Humans; Imidazoles; Isoenzymes; Models, Biological; Neocortex; Pharmacokinetics; Protein Subunits; Receptors, GABA-A; Recombinant Proteins; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Substance Withdrawal Syndrome

2002

Other Studies

21 other study(ies) available for diazepam and imidazenil

ArticleYear
Modulation of basal and stress-induced release of acetylcholine and dopamine in rat brain by abecarnil and imidazenil, two anxioselective gamma-aminobutyric acidA receptor modulators.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 273, Issue:1

    Topics: Acetylcholine; Animals; Anti-Anxiety Agents; Benzodiazepines; Carbolines; Diazepam; Dopamine; Ethanol; GABA Modulators; Hippocampus; Imidazoles; Male; Midazolam; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Stress, Physiological

1995
Imidazenil, a partial positive allosteric modulator of GABAA receptors, exhibits low tolerance and dependence liabilities in the rat.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:3

    Topics: Allosteric Regulation; Animals; Anticonvulsants; Benzodiazepines; Benzodiazepinones; Brain; Diazepam; Drug Interactions; Drug Tolerance; GABA Modulators; Imidazoles; Male; Rats; Rats, Sprague-Dawley; Substance-Related Disorders; Triazolam

1994
Imidazenil: a new partial positive allosteric modulator of gamma-aminobutyric acid (GABA) action at GABAA receptors.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:2

    Topics: Allosteric Regulation; Animals; Benzodiazepines; Benzodiazepinones; Chloride Channels; Conflict, Psychological; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Imidazoles; Male; Membrane Proteins; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Reflex; Seizures

1993
Enhancement of acetylcholine release by flumazenil in the hippocampus of rats chronically treated with diazepam but not with imidazenil or abecarnil.
    Psychopharmacology, 1995, Volume: 121, Issue:2

    Topics: Acetylcholine; Animals; Anticonvulsants; Benzodiazepines; Carbolines; Diazepam; Flumazenil; GABA Modulators; Hippocampus; Imidazoles; Male; Microdialysis; Rats; Rats, Sprague-Dawley; Time Factors

1995
Antagonism of isoniazid-induced convulsions by abecarnil in mice tolerant to diazepam.
    Pharmacology, biochemistry, and behavior, 1995, Volume: 52, Issue:2

    Topics: Animals; Anticonvulsants; Benzodiazepines; Carbolines; Convulsants; Diazepam; Dose-Response Relationship, Drug; Drug Tolerance; GABA Modulators; Imidazoles; Isoniazid; Male; Mice; Seizures

1995
Modifications of gamma-aminobutyric acidA receptor subunit expression in rat neocortex during tolerance to diazepam.
    Molecular pharmacology, 1996, Volume: 49, Issue:5

    Topics: Animals; Base Sequence; Benzodiazepines; Brain Mapping; Cerebral Cortex; Diazepam; DNA Primers; Drug Tolerance; GABA Modulators; Gene Expression; Imidazoles; Male; Molecular Sequence Data; Radioligand Assay; Rats; Receptors, GABA-A; RNA, Messenger; Time Factors

1996
Lack of anticonvulsant tolerance and benzodiazepine receptor down regulation with imidazenil in rats.
    British journal of pharmacology, 1996, Volume: 117, Issue:4

    Topics: Animals; Anticonvulsants; Benzodiazepines; Bicuculline; Diazepam; Down-Regulation; Drug Tolerance; Flumazenil; GABA Modulators; Imidazoles; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Seizures; Tritium

1996
Pharmacological modulation of the diazepam-insensitive recombinant gamma-aminobutyric acidA receptors alpha 4 beta 2 gamma 2 and alpha 6 beta 2 gamma 2.
    Molecular pharmacology, 1996, Volume: 50, Issue:5

    Topics: Animals; Azides; Benzodiazepines; Benzodiazepinones; Binding Sites; Carbolines; Diazepam; Furosemide; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Imidazoles; Kinetics; Membrane Potentials; Radioligand Assay; Rats; Receptors, GABA-A; Recombinant Proteins; Sensitivity and Specificity; Zinc

1996
Reversible modification of GABAA receptor subunit mRNA expression during tolerance to diazepam-induced cognition dysfunction.
    Neuropharmacology, 1996, Volume: 35, Issue:9-10

    Topics: Animals; Anticonvulsants; Benzodiazepines; Cognition Disorders; Diazepam; Drug Tolerance; GABA Modulators; Imidazoles; Male; Motor Activity; Polymerase Chain Reaction; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; RNA; RNA, Messenger

1996
Enhancement by flumazenil of dopamine release in the nucleus accumbens of rats repeatedly exposed to diazepam or imidazenil.
    Psychopharmacology, 1997, Volume: 131, Issue:1

    Topics: Animals; Benzodiazepines; Diazepam; Dopamine; Drug Synergism; Flumazenil; GABA Modulators; Imidazoles; Male; Nucleus Accumbens; Rats; Rats, Sprague-Dawley

1997
Imidazenil, a positive allosteric GABAA receptor modulator, inhibits the effects of cocaine on locomotor activity and extracellular dopamine in the nucleus accumbens shell without tolerance liability.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 287, Issue:1

    Topics: Allosteric Regulation; Animals; Benzodiazepines; Cocaine; Corpus Striatum; Diazepam; Dopamine; Drug Tolerance; GABA Modulators; gamma-Aminobutyric Acid; Imidazoles; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred F344; Receptors, GABA-A; Ventral Tegmental Area

1998
Abecarnil enhances recovery from diazepam tolerance.
    Neuropharmacology, 1999, Volume: 38, Issue:9

    Topics: Animals; Anticonvulsants; Benzodiazepines; Bicuculline; Carbolines; Cell Membrane; Cerebral Cortex; Clonazepam; Diazepam; Drug Interactions; Drug Tolerance; Flumazenil; Imidazoles; Ligands; Male; Mice; Receptors, GABA-A; Seizures; Tritium

1999
Differentiating benzodiazepine- and barbiturate-like discriminative stimulus effects of lorazepam, diazepam, pentobarbital, imidazenil and zaleplon in two- versus three-lever procedures.
    Behavioural pharmacology, 2000, Volume: 11, Issue:1

    Topics: Acetamides; Animals; Anti-Anxiety Agents; Benzodiazepines; Conditioning, Operant; Diazepam; Discrimination Learning; Discrimination, Psychological; GABA Modulators; Hypnotics and Sedatives; Imidazoles; Lorazepam; Pentobarbital; Pyrimidines; Rats; Rats, Long-Evans

2000
Benzodiazepines protect hippocampal neurons from degeneration after transient cerebral ischemia: an ultrastructural study.
    Neuroscience, 2000, Volume: 98, Issue:3

    Topics: Animals; Apoptosis; Benzodiazepines; Diazepam; DNA Fragmentation; GABA Modulators; Gerbillinae; Imidazoles; In Situ Nick-End Labeling; Ischemic Attack, Transient; Male; Microscopy, Electron; Nerve Degeneration; Neuroprotective Agents; Pyramidal Cells; Receptors, GABA-A

2000
Increase in expression of the GABA(A) receptor alpha(4) subunit gene induced by withdrawal of, but not by long-term treatment with, benzodiazepine full or partial agonists.
    Brain research. Molecular brain research, 2001, Aug-15, Volume: 92, Issue:1-2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Cell Membrane; Cells, Cultured; Cerebellum; Chloride Channels; Chlorides; Diazepam; Drug Tolerance; Female; Flumazenil; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Imidazoles; Ion Transport; Membrane Potentials; Microinjections; Nerve Tissue Proteins; Neurons; Oocytes; Protein Subunits; Rats; Receptors, GABA-A; RNA, Messenger; Substance Withdrawal Syndrome; Substance-Related Disorders; Up-Regulation; Xenopus laevis

2001
Imidazenil: a potent and safe protective agent against diisopropyl fluorophosphate toxicity.
    Neuropharmacology, 2004, Volume: 46, Issue:3

    Topics: Animals; Benzodiazepines; Diazepam; Imidazoles; Isoflurophate; Male; Neuroprotective Agents; Rats; Rats, Inbred F344; Seizures

2004
Imidazenil: an antagonist of the sedative but not the anticonvulsant action of diazepam.
    Neuropharmacology, 2005, Volume: 49, Issue:3

    Topics: Animals; Anticonvulsants; Benzodiazepines; Bicuculline; Convulsants; Diazepam; Dose-Response Relationship, Drug; GABA Antagonists; GABA Modulators; Hypnotics and Sedatives; Imidazoles; Male; Motor Activity; Rats; Rats, Inbred F344

2005
Imidazenil and diazepam increase locomotor activity in mice exposed to protracted social isolation.
    Proceedings of the National Academy of Sciences of the United States of America, 2006, Mar-14, Volume: 103, Issue:11

    Topics: Animals; Benzodiazepines; Diazepam; Frontal Lobe; GABA Modulators; Gene Expression; Hippocampus; Imidazoles; In Vitro Techniques; Male; Mice; Motor Activity; Protein Subunits; Pyridines; Receptors, GABA-A; RNA, Messenger; Social Isolation; Zolpidem

2006
Imidazenil: a low efficacy agonist at alpha1- but high efficacy at alpha5-GABAA receptors fail to show anticonvulsant cross tolerance to diazepam or zolpidem.
    Neuropharmacology, 2008, Volume: 55, Issue:2

    Topics: Animals; Anticonvulsants; Behavior, Animal; Benzodiazepines; Bicuculline; Diazepam; Differential Threshold; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Tolerance; GABA Modulators; Imidazoles; Male; Pyridines; Rats; Rats, Inbred F344; Seizures; Zolpidem

2008
Imidazenil, a non-sedating anticonvulsant benzodiazepine, is more potent than diazepam in protecting against DFP-induced seizures and neuronal damage.
    Toxicology, 2009, Feb-27, Volume: 256, Issue:3

    Topics: Animals; Anticonvulsants; Behavior, Animal; Benzodiazepines; Brain; Cholinesterase Inhibitors; Diazepam; DNA Fragmentation; Electroencephalography; Imidazoles; In Situ Nick-End Labeling; Isoflurophate; Male; Neurons; Rats; Rats, Inbred F344; Seizures; Status Epilepticus; Telemetry

2009
Absence of tolerance to the anticonvulsant and neuroprotective effects of imidazenil against DFP-induced seizure and neuronal damage.
    Neuropharmacology, 2011, Volume: 61, Issue:8

    Topics: Animals; Anticonvulsants; Benzodiazepines; Cholinesterase Inhibitors; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Fluoresceins; Imidazoles; Isoflurophate; Male; Neurons; Neuroprotective Agents; Organic Chemicals; Rats; Rats, Inbred F344; Seizures; Statistics, Nonparametric

2011