diazepam has been researched along with flurazepam in 126 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 103 (81.75) | 18.7374 |
1990's | 15 (11.90) | 18.2507 |
2000's | 6 (4.76) | 29.6817 |
2010's | 2 (1.59) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Engel, J; Fleischhauer, I; Jakovlev, V; Johanson, CE; Kleemann, A; Kutscher, B; Nickel, B; Rauer, H; Szelenyi, I; Werner, U | 1 |
Aoyama, T; Ichikawa, H; Suzuki, Y | 1 |
Babbini, M; Barbaro, AM; Bartoletti, M; Biagi, GL; Borea, PA; Gaiardi, M; Guerra, MC | 1 |
Choi, SS; Contrera, JF; Hastings, KL; Kruhlak, NL; Sancilio, LF; Weaver, JL; Willard, JM | 1 |
Buttar, D; Colclough, N; Gerhardt, S; MacFaul, PA; Maskos, K; Phillips, SD; Plowright, A; Steinbacher, S; Steuber, H; Tam, K; Whittamore, P | 1 |
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K | 1 |
Overton, DA | 1 |
Aliverti, V; Mariani, L | 1 |
Dorrity, F; Linnoila, M | 1 |
Aalto, U; Linnoila, M; Viukari, M | 1 |
Ohmori, K | 1 |
Solomon, D | 1 |
Deinum, EJ; Ifabumuyi, OI; Kazarian, SS; Merskey, H; Tekatch, GM | 1 |
Chiu, TH; Rosenberg, HC | 4 |
Kaplan, SR; Murkofsky, C | 1 |
Davis, M | 1 |
Avant, GR; Berman, ML; Schenker, S; Speeg, KV; Wang, S | 1 |
Jensen, RA; Martinez, JL; McGaugh, JL; Vasquez, BJ | 1 |
Salzman, C; van der Kolk, BA | 1 |
Needle, M; Taclob, L | 1 |
Heiss, WD; Hoyer, J; Rappelsberger, P | 1 |
Becker, CE; Boerner, U; Luce, J; Roe, R; Scott, R; Tong, T | 1 |
Barsuhn, C; Lahti, RA | 1 |
Djojodibroto, RD; Groenewoud, ET; Leeuwin, RS | 1 |
MacPhail, I; Ogilvie, WA; Purvis, CR | 1 |
Gottschalk, LA | 1 |
Miller, RR | 1 |
Nicholson, AN | 1 |
Kopjak, L; Peat, MA | 1 |
Banerjee, U; Yeoh, PN | 1 |
Brand, SJ; Curtis, DR; Johnston, GA; Lodge, D | 1 |
Tietz, EI; Xie, XH | 1 |
Loeffler, PM | 1 |
Guentert, TW; Stebler, T | 1 |
Dittrich, P; Lenk, W; Pöch, G; Reiffenstein, RJ; Schuster, A | 1 |
Deutsch, SI; Huntzinger, JA; Mastropaolo, J; Novitzki, MR; Rosse, RB | 1 |
Haefely, W | 1 |
Chiu, TH; Rosenberg, HC; Tietz, EI | 1 |
Fillenz, M; Pei, Q; Zetterström, T | 1 |
Gallager, DW; Wilson, MA | 1 |
Booraem, CD; Flowers, JV; Gumbiner, J | 1 |
Kubota, K; Matsuda, I; Matsuoka, Y; Sugaya, K; Terawaki, Y | 1 |
Barclay, AM | 1 |
Namima, M; Sakai, Y | 1 |
Kubota, K; Matsuda, I; Sugaya, K; Uruno, T | 1 |
Alonso, R; Astier, H; Tapia-Arancibia, L | 1 |
Bouthillier, A; De Montigny, C | 1 |
Romstedt, K | 1 |
Abraham, CJ; De Blas, AL; Haney, SA; Park, D; Rayner, CA; Sangameswaran, L | 1 |
Fares, F; Gavish, M | 1 |
Hicks, TP; Jang, EK; Oka, JI | 1 |
Barnett, A; Ongini, E | 1 |
Busto, U; Cappell, H; Naranjo, CA; Sanchez-Craig, M; Sellers, EM; Sykora, K | 1 |
Chiu, TH; Rosenberg, HC; Yu, O | 1 |
Kawasaki, K; Matsushita, A; Satoh, M; Takagi, H | 1 |
Morrow, AL; Paul, SM | 1 |
Kawasaki, H; Nuki, C; Ohno, H; Takasaki, K; Urabe, M; Yamamoto, R | 1 |
Fleming, JA; Isomura, T; McMillan, MJ; Rungta, K | 1 |
Thomas, WA | 1 |
Kuhn, FJ | 1 |
Sanderson, G; Scholfield, CN | 1 |
Gyermek, L | 1 |
Greenblatt, DJ; Shader, RI | 1 |
Hailey, DM | 1 |
Nicholson, AN; Wright, CM | 1 |
Cereda, E; Domenichini, E; Fischetti, M; Pagnin, A | 1 |
Müller, W; Wollert, U | 1 |
Fryer, RI; Walser, A | 1 |
Fennessy, MR; Sawynok, J | 1 |
Ghisoni, T; Poggi, E | 1 |
Mendelson, WB | 1 |
Assié, MB; Briley, M; Charveron, M; Stenger, A | 1 |
Cohen, ES; Holman, RC | 1 |
Bender, AS; Phillis, JW; Wu, PH | 1 |
Forster, J; Patten, DW; Rosser, WW; Simms, JG | 1 |
Black, DB; Lawrence, RC; Lovering, EG; Watson, JR | 1 |
Kamp, CW; Morgan, WW | 1 |
Shader, RI | 1 |
Mariotti, M; Ongini, E | 1 |
Berlin, RM; Conell, LJ | 1 |
Ikeda, K; Kiyota, Y; Ohta, H; Sato, Y; Shibata, K; Shibata, S; Ueki, S; Watanabe, S; Yamamoto, T | 1 |
Neubert, W; Ott, H; Willumeit, HP | 1 |
Bichard, AR; Little, HJ | 1 |
Lader, M; Olajide, D | 1 |
Choi, DW; Farb, DH; Fischbach, GD | 1 |
Morin, AM; Tanaka, IA; Wasterlain, CG | 1 |
Chiu, TH; Rosenberg, HC; Smith, S | 1 |
Feil, P; Scharf, MB | 1 |
Abernethy, DR; Divoll, M; Greenblatt, DJ; Ochs, HR; Shader, RI | 1 |
Lloyd, HG; Morgan, PF; Stone, TW | 2 |
Minchin, MC; Nutt, DJ | 1 |
de Wit, H; Johanson, CE; Uhlenhuth, EH | 1 |
Moskowitz, H | 1 |
Gillin, JC; Kamgar-Parsi, B; Wehr, TA | 1 |
Pearlman, T | 1 |
Shannon, HE | 1 |
Meyer, BR | 1 |
Bittencourt, PR; Richens, A; Smith, AT; Wade, P | 1 |
Dixon, R | 1 |
Lee, EK; Ross, RJ; Walters, JR; Waszczak, BL | 1 |
Pristach, CA; Smith, CM; Whitney, RB | 1 |
Ando, J; Ishii, K; Kano, T | 1 |
Clarens, RD; Kuzel, RJ; Lindblom, ML; Seifert, RD; Sorensen, MD | 1 |
Akutagawa, M; Ando, J; Ishii, K; Kano, T; Makino, M; Tanaka, T | 1 |
Bamonte, F; Ongini, E; Parravicini, L | 1 |
Hertz, L; Mukerji, S | 1 |
Ladewig, D | 1 |
Bourn, WM; Reigel, CE | 1 |
Chiu, TH; Ramsey-Williams, V; Rosenberg, HC; Wu, Y | 1 |
Guo, XQ; Xu, NS; Zhang, JR | 1 |
Linsner, JP; Perlick, D; Pollak, CP | 1 |
Chiu, TH; Rosenberg, HC; Zhao, TJ | 1 |
Chiu, TH; Li, M; Rosenberg, HC | 1 |
Vieweg, WV | 1 |
Okuyama, T; Tomita, M | 1 |
Li, M; Rosenberg, HC; Szabo, A | 1 |
Abdel-Mottaleb, M; El-Sayed, AA; Kitamura, K; Omran, AA; Takegami, S | 1 |
Abdel-Mottaleb, M; El-Sayed, AA; Kitade, T; Kitamura, K; Mohamed, MH; Omran, AA; Takegami, S | 1 |
Downing, SS; Farb, DH; Gibbs, TT; Lee, YT | 1 |
Aller, MI; Korpi, ER; Leppä, E; Linden, AM; Rosenberg, PH; Wisden, W | 1 |
8 review(s) available for diazepam and flurazepam
Article | Year |
---|---|
Neural networks applied to quantitative structure-activity relationship analysis.
Topics: Animals; Azirines; Benzodiazepines; Carbazilquinone; Nerve Net; Nervous System; Regression Analysis; Structure-Activity Relationship | 1990 |
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk | 2016 |
Oral benzodiazepines and conscious sedation: a review.
Topics: Administration, Oral; Alprazolam; Ambulatory Surgical Procedures; Anti-Anxiety Agents; Conscious Sedation; Diazepam; Flurazepam; Humans; Lorazepam; Midazolam; Oxazepam; Premedication; Receptors, GABA-A; Temazepam; Triazolam | 1992 |
Time course for development of benzodiazepine tolerance and physical dependence.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Diazepam; Drug Tolerance; Flumazenil; Flurazepam; Humans; Hypnotics and Sedatives; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors | 1985 |
Drug therapy. Benzodiazepines (first of two parts).
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Antidepressive Agents; Behavior, Animal; Biotransformation; Blood Circulation; Carboxylic Acids; Chlordiazepoxide; Costs and Cost Analysis; Diazepam; Flurazepam; Humans; Limbic System; Muscles; Oxazepam; Respiration; Structure-Activity Relationship | 1974 |
Chromatography of the 1,4-benzodiazepines.
Topics: Anti-Anxiety Agents; Chlordiazepoxide; Chromatography; Diazepam; Flurazepam; Humans; Methylation; Nitrazepam; Oxazepam; Oxazoles; Prazepam; Solvents; Spectrometry, Fluorescence; Temperature | 1974 |
Benzodiazepine kinetics: implications for therapeutics and pharmacogeriatrics.
Topics: Adolescent; Adult; Age Factors; Aged; Benzodiazepines; Biotransformation; Child; Diazepam; Flurazepam; Half-Life; Humans; Kinetics; Middle Aged; Nordazepam; Oxidation-Reduction | 1983 |
Benzodiazepines in the elderly.
Topics: Adult; Aged; Aging; Benzodiazepines; Diazepam; Female; Flurazepam; Humans; Kinetics; Male; Middle Aged | 1982 |
7 trial(s) available for diazepam and flurazepam
Article | Year |
---|---|
Efficacy and side effects of flurazepam, fosazepam, and nitrazepam as sleeping aids in psychogeriatric patients.
Topics: Aged; Anti-Anxiety Agents; Clinical Trials as Topic; Diazepam; Drug Evaluation; Female; Flurazepam; Humans; Male; Memory; Mental Disorders; Motor Activity; Nitrazepam; Sleep Wake Disorders | 1978 |
Comparison of diazepam and flurazepam in the treatment of insomnia in general practice.
Topics: Administration, Oral; Adolescent; Adult; Aged; Capsules; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Flurazepam; Humans; Hypnotics and Sedatives; Male; Middle Aged; Sleep Initiation and Maintenance Disorders | 1979 |
Effects of certain benzodiazepine derivatives on disorganization of thought as manifested in speech.
Topics: Adult; Benzodiazepines; Chlordiazepoxide; Diazepam; Flurazepam; Humans; Lorazepam; Speech; Thinking; Time Factors; Triazolam | 1977 |
Withdrawal reaction after long-term therapeutic use of benzodiazepines.
Topics: Adolescent; Adult; Aged; Anxiety; Benzodiazepines; Diazepam; Double-Blind Method; Female; Flurazepam; Humans; Long-Term Care; Lorazepam; Male; Middle Aged; Oxazepam; Patient Compliance; Placebos; Substance Withdrawal Syndrome; Time Factors | 1986 |
Flurazepam versus diazepam in an anaesthesia: a clinical study.
Topics: Adolescent; Adult; Aged; Analgesics; Anesthesia, Intravenous; Blood Pressure; Clinical Trials as Topic; Diazepam; Drug Synergism; Female; Flurazepam; Halothane; Humans; Male; Middle Aged; Muscle Tonus; Preanesthetic Medication; Sleep; Time Factors | 1973 |
Lack of preference for flurazepam in normal volunteers.
Topics: Adult; Diazepam; Female; Flurazepam; Humans; Lorazepam; Male; Reinforcement, Psychology | 1984 |
The relationship between peak velocity of saccadic eye movements and serum benzodiazepine concentration.
Topics: Adult; Benzodiazepines; Diazepam; Double-Blind Method; Eye Movements; Flurazepam; Humans; Male; Nitrazepam; Nordazepam; Reticular Formation; Saccades; Temazepam | 1981 |
111 other study(ies) available for diazepam and flurazepam
Article | Year |
---|---|
Chemistry and pharmacology of the non-benzodiazepine anxiolytic enciprazine and related compounds.
Topics: Aggression; Animals; Anti-Anxiety Agents; Behavior, Animal; Chemical Phenomena; Chemistry; Exploratory Behavior; Female; Male; Mice; Molecular Structure; Piperazines; Rats; Self Administration; Structure-Activity Relationship; Substance-Related Disorders | 1990 |
Rm values and structure-activity relationship of benzodiazepines.
Topics: Animals; Benzodiazepines; Chromatography, Thin Layer; Conflict, Psychological; Exploratory Behavior; Models, Biological; Rats; Solubility; Structure-Activity Relationship | 1980 |
Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.
Topics: | 2008 |
A combined spectroscopic and crystallographic approach to probing drug-human serum albumin interactions.
Topics: Binding Sites; Crystallography, X-Ray; Drug Interactions; Humans; Pharmaceutical Preparations; Protein Binding; Protein Structure, Tertiary; Serum Albumin; Spectrometry, Fluorescence | 2010 |
Discriminable effects of benzodiazepines.
Topics: Anti-Anxiety Agents; Barbiturates; Chlordiazepoxide; Diazepam; Discrimination, Psychological; Flurazepam | 1976 |
[Therapeutic notes: benzodiazepines].
Topics: Anti-Anxiety Agents; Chemical Phenomena; Chemistry; Chlordiazepoxide; Clorazepate Dipotassium; Diazepam; Flurazepam; Humans; Lorazepam; Nitrazepam; Oxazepam | 1976 |
Rapid gas chromatographic assay of serum diazepam, N-desmethyldiazepam, and N-desalkylflurazepam.
Topics: Anti-Anxiety Agents; Chromatography, Gas; Diazepam; Flurazepam; Humans; Nordazepam; Time Factors | 1977 |
[Electroencephalographic effects of flurazepam in rabbits (author's transl)].
Topics: Animals; Anti-Anxiety Agents; Blood Pressure; Brain; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Electric Stimulation; Electrodes, Implanted; Electroencephalography; Evoked Potentials; Flurazepam; Male; Photic Stimulation; Physostigmine; Rabbits; Recruitment, Neurophysiological | 1977 |
High-dose benzodiazepines in the treatment of severe neurotic anxiety.
Topics: Adult; Aged; Anti-Anxiety Agents; Anxiety Disorders; Diazepam; Female; Flurazepam; Humans; Male; Oxazepam; Substance-Related Disorders | 1978 |
Effects of antianxiety agents on relaxation training: a preliminary investigation.
Topics: Adolescent; Adult; Aged; Anti-Anxiety Agents; Anxiety; Diazepam; Female; Flurazepam; Humans; Male; Mental Disorders; Middle Aged; Neurotic Disorders; Oxazepam; Personality Disorders; Phenobarbital; Relaxation Therapy; Stress, Psychological | 1978 |
Reduced diazepam binding following chronic benzodiazepine treatment.
Topics: Animals; Anti-Anxiety Agents; Brain; Diazepam; Flurazepam; Male; Rats; Synaptosomes; Time Factors | 1978 |
Oral-buccal dyskinesia symptoms associated with low-dose benzodiazepine treatment.
Topics: Anti-Anxiety Agents; Depression; Diazepam; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Flurazepam; Humans; Male; Middle Aged | 1978 |
Diazepam and flurazepam: effects on conditioned fear as measured with the potentiated startle paradigm.
Topics: Animals; Anti-Anxiety Agents; Conditioning, Operant; Diazepam; Fear; Flurazepam; Male; Rats; Reflex, Startle | 1979 |
Decreased 3H-diazepam binding is a specific response to chronic benzodiazepine treatment.
Topics: Animals; Anti-Anxiety Agents; Barbital; Brain; Depression, Chemical; Diazepam; Flurazepam; Kinetics; Male; Rats; Time Factors | 1979 |
Antagonism of benzodiazepine binding in rat and human brain by Antilirium.
Topics: Animals; Anti-Anxiety Agents; Brain; Depression, Chemical; Diazepam; Flurazepam; Humans; In Vitro Techniques; Kinetics; Physostigmine; Rats; Time Factors | 1979 |
Benzodiazepines alter acquisition and retention of an inhibitory avoidance response in mice.
Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Diazepam; Flurazepam; Lorazepam; Male; Memory; Mice; Retention, Psychology | 1979 |
Management of the geriatric patient in a general hospital. Psychotropic drugs and polypharmacy in elderly patients in a general hospital.
Topics: Aged; Antidepressive Agents, Tricyclic; Antiemetics; Antipsychotic Agents; Diazepam; Drug Therapy, Combination; Flurazepam; Hospitals, General; Humans; Mental Disorders; Middle Aged; Psychotropic Drugs | 1979 |
Drug-induced encephalopathy in patients on maintenance haemodialysis.
Topics: Aged; Anti-Anxiety Agents; Arthritis; Coronary Disease; Dementia; Diazepam; Flurazepam; Fractures, Bone; Humans; Kidney Failure, Chronic; Male; Middle Aged; Pain; Renal Dialysis | 1976 |
Neurophysiological effects of benzodiazepines on identified neurones.
Topics: Animals; Aplysia; Diazepam; Evoked Potentials; Flurazepam; Ganglia; Interneurons; Ion Channels; Neurons | 1977 |
Rational drug therapy of alcoholism with sedative hypnotic drugs! Is this possible?
Topics: Administration, Oral; Alcoholism; Antipsychotic Agents; Anxiety; Barbiturates; Community Mental Health Services; Diazepam; Drug Therapy, Combination; Drug Tolerance; Flurazepam; Humans; Hypnotics and Sedatives; Noise; Phenothiazines; Psychopharmacology; Secobarbital; Smoking; Substance Withdrawal Syndrome | 1975 |
The effect of various doses of minor tranquilizers on plasma corticosteroids in stressed rats.
Topics: Adrenal Cortex Hormones; Animals; Anti-Anxiety Agents; Chlordiazepoxide; Diazepam; Flurazepam; Male; Phenobarbital; Rats; Stimulation, Chemical; Stress, Physiological | 1975 |
The effects of three benzodiazepines and of meprobamate on the action of smooth muscle stimulants on the guinea-pig ileum.
Topics: Acetylcholine; Animals; Anti-Anxiety Agents; Chlordiazepoxide; Diazepam; Drug Interactions; Flurazepam; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Meprobamate; Muscle Contraction; Muscle, Smooth; Serotonin; Stimulation, Chemical | 1975 |
A guide to the use of hypnotic drugs.
Topics: Benzodiazepines; Chlordiazepoxide; Clorazepate Dipotassium; Diazepam; Drug Interactions; Flurazepam; Humans; Hypnotics and Sedatives; Sleep Wake Disorders; Substance-Related Disorders | 1979 |
Performance studies with diazepam and its hydroxylated metabolites.
Topics: Barbiturates; Diazepam; Flurazepam; Humans; Hydroxylation; Motor Skills; Oxazepam; Temazepam; Time Factors | 1979 |
The screening and quantitation of diazepam, flurazepam, chloridazepoxide, and their metabolites in blood and plasma by electron-capture gas chromatography and high pressure liquid chromatography.
Topics: Chlordiazepoxide; Chromatography, Gas; Chromatography, High Pressure Liquid; Diazepam; Flurazepam; Humans | 1979 |
The temporal dimensions of anticonvulsant action of some newer benzodiazepines against metrazol induced seizures in mice and rats.
Topics: Animals; Benzodiazepines; Clonazepam; Diazepam; Drug Evaluation, Preclinical; Ethosuximide; Female; Flurazepam; Male; Mice; Nitrazepam; Pentylenetetrazole; Phenobarbital; Seizures; Trimethadione | 1977 |
Central actions of benzodiazepines.
Topics: Animals; Benzodiazepines; Cerebellar Cortex; Diazepam; Flurazepam; gamma-Aminobutyric Acid; Glycine; Neural Inhibition; Rats; Spinal Cord | 1976 |
Reduction in potency of selective gamma-aminobutyric acidA agonists and diazepam in CA1 region of in vitro hippocampal slices from chronic flurazepam-treated rats.
Topics: Animals; Diazepam; Evoked Potentials; Flurazepam; gamma-Aminobutyric Acid; Hippocampus; Isonicotinic Acids; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1992 |
Determination of diazepam and nordazepam in milk and plasma in the presence of oxazepam and temazepam.
Topics: Chromatography, High Pressure Liquid; Diazepam; Flurazepam; Humans; Hydrogen-Ion Concentration; Milk, Human; Nordazepam; Oxazepam; Temazepam | 1991 |
Evaluation of experimental combined toxicity by use of dose-frequency curves: comparison with theoretical additivity as well as independence.
Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Drug Synergism; Drug Therapy, Combination; Ethanol; Flurazepam; Lethal Dose 50; Malathion; Male; Mice; Mice, Inbred Strains; Parathion; Phencyclidine; Reflex; Toxicology | 1990 |
Profound stress-induced alterations in flurazepam's antiseizure efficacy can be attenuated.
Topics: Animals; Carbolines; Clonazepam; Cold Temperature; Diazepam; Dose-Response Relationship, Drug; Electroshock; Flumazenil; Flurazepam; Male; Mice; Mice, Inbred Strains; Midazolam; Seizures; Stress, Psychological | 1990 |
Partial agonists of the benzodiazepine receptor: from animal data to results in patients.
Topics: Affinity Labels; Allosteric Site; Animals; Azides; Benzodiazepines; Benzodiazepinones; Chlordiazepoxide; Chlorides; Clonazepam; Diazepam; Drug Interactions; Ethanol; Flumazenil; Flurazepam; Humans; Ion Channels; Ligands; Models, Neurological; Neurons; Receptors, GABA-A | 1988 |
Regional GABA/benzodiazepine receptor/chloride channel coupling after acute and chronic benzodiazepine treatment.
Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Bicuculline; Brain; Chlorides; Diazepam; Flunitrazepam; Flurazepam; gamma-Aminobutyric Acid; Ion Channels; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stimulation, Chemical | 1989 |
Both systemic and local administration of benzodiazepine agonists inhibit the in vivo release of 5-HT from ventral hippocampus.
Topics: Animals; Benzodiazepines; Carbolines; Chromatography, High Pressure Liquid; Dialysis; Diazepam; Flumazenil; Flurazepam; Hippocampus; Hydroxyindoleacetic Acid; Ion Channels; Male; Muscimol; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin | 1989 |
Responses of substantia nigra pars reticulata neurons to benzodiazepine ligands after acute and prolonged diazepam exposure. I. Modulation of gamma-aminobutyric acid sensitivity.
Topics: Animals; Carbolines; Diazepam; Flumazenil; Flurazepam; gamma-Aminobutyric Acid; Ligands; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra | 1989 |
Combined medical and psychological treatment of postchemotherapy nausea and vomiting: a case study.
Topics: Acute Disease; Behavior Therapy; Combined Modality Therapy; Cytarabine; Diazepam; Flurazepam; Humans; Leukemia; Male; Middle Aged; Nausea; Vomiting | 1989 |
Reversal of antinociceptive effect of cholecystokinin by benzodiazepines and a benzodiazepine antagonist, Ro 15-1788.
Topics: Analgesics; Animals; Anti-Anxiety Agents; Benzodiazepinones; Chlordiazepoxide; Cholecystokinin; Diazepam; Flumazenil; Flurazepam; Male; Mice; Morphine; Naloxone; Pain; Sensory Thresholds; Time Factors | 1985 |
Psychotropic drugs in the elderly. Selection of the appropriate agent.
Topics: Age Factors; Aged; Antidepressive Agents; Antipsychotic Agents; Benzodiazepines; Chlordiazepoxide; Cimetidine; Diazepam; Flurazepam; Haloperidol; Humans; Kinetics; Lithium; Phenothiazines; Physostigmine; Psychotropic Drugs; Thiothixene; Trazodone | 1985 |
Inhibitory effect on 3H-diazepam binding and potentiating action on GABA of ethyl loflazepate, a new minor tranquilizer.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Diazepam; Drug Synergism; Flurazepam; gamma-Aminobutyric Acid; Guinea Pigs; Male; Purkinje Cells | 1985 |
Cholecystokinin antagonism by benzodiazepines in the food intake in mice.
Topics: Animals; Anti-Anxiety Agents; Chlordiazepoxide; Diazepam; Eating; Flurazepam; Injections, Intraperitoneal; Male; Mice; Naloxone; Sincalide; Subarachnoid Space | 1986 |
Evidence for a role of central type benzodiazepine receptors in the inhibition of the thyrotropin-releasing hormone-induced thyrotropin release from rat perifused pituitaries.
Topics: Animals; Anti-Anxiety Agents; Chlordiazepoxide; Diazepam; Flurazepam; In Vitro Techniques; Male; Midazolam; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains; Receptors, GABA-A; Thyrotropin; Thyrotropin-Releasing Hormone | 1986 |
Long-term benzodiazepine treatment reduces neuronal responsiveness to cholecystokinin: an electrophysiological study in the rat.
Topics: Acetylcholine; Animals; Anti-Anxiety Agents; Cholecystokinin; Diazepam; Electrophysiology; Flurazepam; Hippocampus; Iontophoresis; Male; Neurons; Pyramidal Tracts; Rats; Rats, Inbred Strains | 1988 |
Benzodiazepines inhibit human platelet activation: comparison of the mechanism of antiplatelet actions of flurazepam and diazepam.
Topics: Adenosine Diphosphate; Arachidonic Acid; Arachidonic Acids; Benzodiazepinones; Blood Platelets; Collagen; Cyclic AMP; Cyclic GMP; Diazepam; Epinephrine; Flumazenil; Flurazepam; Humans; Malondialdehyde; Platelet Aggregation; Prostaglandin Endoperoxides, Synthetic; Serotonin; Thrombin; Type C Phospholipases | 1985 |
Monoclonal antibodies to benzodiazepines.
Topics: Animals; Anti-Anxiety Agents; Antibodies, Monoclonal; Benzodiazepines; Benzodiazepinones; Diazepam; Flumazenil; Flunitrazepam; Flurazepam; Mice; Mice, Inbred BALB C; Receptors, GABA-A; Structure-Activity Relationship | 1985 |
Solubilization of peripheral benzodiazepine-binding sites from rat kidney.
Topics: Animals; Benzodiazepinones; Binding, Competitive; Carbolines; Chlordiazepoxide; Clonazepam; Diazepam; Digitonin; Flumazenil; Flurazepam; Guanidine; Guanidines; Hot Temperature; Isoquinolines; Kidney; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Solubility; Time Factors; Urea | 1985 |
Benzodiazepine receptor involvement in the control of receptive field size and responsiveness in primary somatosensory cortex.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Cats; Diazepam; Female; Flumazenil; Flurazepam; gamma-Aminobutyric Acid; Male; Midazolam; Neurons; Receptors, GABA-A; Sensory Thresholds; Somatosensory Cortex; Touch | 1986 |
Hypnotic specificity of benzodiazepines.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Brain; Cats; Diazepam; Electroencephalography; Flurazepam; Hypnotics and Sedatives; Receptors, GABA-A; Sleep | 1985 |
Modulation of GABA-gated chloride ion flux in rat brain by acute and chronic benzodiazepine administration.
Topics: Animals; Benzodiazepines; Brain; Chlorides; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flurazepam; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred Strains | 1988 |
The lateral vestibular nucleus is a site for the depressant action of benzodiazepines on the crossed extensor reflex.
Topics: Action Potentials; Animals; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flurazepam; Male; Microinjections; Neural Inhibition; Posture; Rats; Rats, Inbred Strains; Reflex; Vestibular Nuclei | 1988 |
Benzodiazepine enhancement of gamma-aminobutyric acid-mediated chloride ion flux in rat brain synaptoneurosomes.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Chlorides; Clonazepam; Diazepam; Drug Synergism; Flurazepam; gamma-Aminobutyric Acid; Male; Muscimol; Rats; Rats, Inbred Strains; Synaptosomes | 1988 |
[Electroencephalographic study of Sch 161 (quazepam), a new benzodiazepine hypnotic, in rats and rabbits].
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Electric Stimulation; Electroencephalography; Flurazepam; Hypnotics and Sedatives; Photic Stimulation; Rabbits; Rats; Reticular Formation; Sound | 1987 |
Withdrawal regimen for triazolam-dependent patients.
Topics: Diazepam; Flurazepam; Humans; Sleep Initiation and Maintenance Disorders; Substance Withdrawal Syndrome; Triazolam | 1986 |
Peptide derivatives as prodrugs.
Topics: Amino Acids; Animals; Bacteria; Biological Availability; Biological Transport, Active; Chlordiazepoxide; Diazepam; Flunitrazepam; Flurazepam; Humans; Kinetics; Nitrazepam; Papio; Rats | 1986 |
Effects of brotizolam on the sleep-waking cycle of the cat.
Topics: Animals; Azepines; Cats; Diazepam; Electrodes, Implanted; Electroencephalography; Female; Flurazepam; Hypnotics and Sedatives; Male; Nitrazepam; Sleep; Sleep, REM; Time Factors; Triazolam; Wakefulness | 1986 |
Blood pressure response to Ro15-1788, a benzodiazepine antagonist.
Topics: Animals; Benzodiazepinones; Blood Pressure; Cats; Convulsants; Diazepam; Drug Tolerance; Flumazenil; Flurazepam; Heart Rate; Humans; Substance-Related Disorders | 1985 |
Effects of adenosine uptake blockers and adenosine on evoked potentials of guinea-pig olfactory cortex.
Topics: Adenosine; Adenosine Deaminase; Animals; Diazepam; Dilazep; Dipyridamole; Evoked Potentials; Flurazepam; Guanosine; Guinea Pigs; Hexobendine; In Vitro Techniques; Limbic System; Olfactory Pathways; Thioinosine; Thionucleosides | 1986 |
Benzodiazepines for supplementing steroid anesthesia.
Topics: Anesthetics; Animals; Benzodiazepinones; Chlordiazepoxide; Diazepam; Drug Synergism; Flurazepam; Hydroxysteroids; Mice; Pregnanediones; Pregnanes; Steroids; Time Factors | 1974 |
Inhibitory and disinhibitory effects of nitrazepam, diazepam and flurazepam hydrochloride on delayed matching behaviour in monkeys (Macaca mulatta).
Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Flurazepam; Macaca mulatta; Male; Motor Activity; Nitrazepam; Time Factors | 1974 |
Influence of pH on the benzodiazepine-human serum albumin complex. Circular dichroism studies.
Topics: Benzazepines; Benzodiazepinones; Binding Sites; Chemical Phenomena; Chemistry; Chlordiazepoxide; Circular Dichroism; Diazepam; Flurazepam; Humans; Hydrogen-Ion Concentration; Kinetics; Nitrazepam; Osmolar Concentration; Oxazepam; Protein Binding; Serum Albumin | 1974 |
Quinazolines and 1,4-benzodiazepines. 69. 1-Vinyl-1,4-benzodiazepin-2-ones and 1-vinylquinazolin-2(1H)-ones.
Topics: Animals; Benzodiazepinones; Central Nervous System; Chlordiazepoxide; Depression, Chemical; Diazepam; Flurazepam; Lethal Dose 50; Mice; Pentylenetetrazole; Quinazolines; Seizures; Vinyl Compounds | 1974 |
The effect of benzodiazepines on the analgesic effect of morphine and sodium salicylate.
Topics: Analgesics; Animals; Benzazepines; Chlordiazepoxide; Diazepam; Drug Interactions; Female; Flurazepam; Male; Mice; Morphine; Nitrazepam; Quinones; Salicylates; Time Factors | 1973 |
[Flurazepam in depressive anxiety syndromes].
Topics: Adjustment Disorders; Adult; Aged; Anxiety; Anxiety Disorders; Benzodiazepinones; Depression; Diazepam; Female; Flurazepam; Humans; Hypochondriasis; Male; Middle Aged; Tranquilizing Agents | 1971 |
The benzodiazepine receptor and sleep.
Topics: Animals; Barbiturates; Benzodiazepines; Benzodiazepinones; Calcium; Carbolines; Diazepam; Flumazenil; Flurazepam; Humans; Motor Activity; Nifedipine; Phenobarbital; Pyrazoles; Rats; Receptors, GABA-A; Sleep; Synaptosomes | 1984 |
Benzodiazepine agonist-type activity of raubasine, a rauwolfia serpentina alkaloid.
Topics: Animals; Anticonvulsants; Benzodiazepinones; Binding, Competitive; Brain; Diazepam; Flumazenil; Flurazepam; In Vitro Techniques; Kinetics; Male; Mice; Rats; Receptors, GABA-A; Secologanin Tryptamine Alkaloids; Yohimbine | 1984 |
An integrated approach to iatrogenic drug abuse in a closed delivery system.
Topics: Adult; Aged; Anti-Anxiety Agents; Chlordiazepoxide; Diazepam; Doxepin; Drug and Narcotic Control; Drug Prescriptions; Female; Flurazepam; Germany, West; Hospitals, Military; Hospitals, Public; Humans; Iatrogenic Disease; Male; Medication Systems, Hospital; Meprobamate; Middle Aged; Oxazepam; Substance-Related Disorders; United States | 1980 |
Diazepam and flurazepam inhibit adenosine uptake by rat brain synaptosomes.
Topics: Adenosine; Animals; Brain; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Flurazepam; In Vitro Techniques; Male; Rats; Synaptosomes | 1980 |
Improving benzodiazepine prescribing in family practice through review and education.
Topics: Adolescent; Adult; Age Factors; Aged; Anti-Anxiety Agents; Chlordiazepoxide; Diazepam; Drug Prescriptions; Family Practice; Female; Flurazepam; Humans; Male; Middle Aged; Oxazepam | 1981 |
Routine quality evaluation of benzodiazepine drugs to USP-NF specifications.
Topics: Anti-Anxiety Agents; Chlordiazepoxide; Chromatography, Gas; Diazepam; Flurazepam; Pharmacopoeias as Topic; Quality Control; Tablets; United States | 1981 |
Choice of benzodiazepines.
Topics: Aged; Anti-Anxiety Agents; Anxiety; Chlordiazepoxide; Diazepam; Flurazepam; Half-Life; Humans; Liver Diseases; Lorazepam; Male; Sleep Initiation and Maintenance Disorders; Substance Withdrawal Syndrome | 1981 |
Benzodiazepines suppress the light response of retinal dopaminergic neurons in vivo.
Topics: Animals; Anti-Anxiety Agents; Diazepam; Dopamine; Flurazepam; Light; Male; Neurons; Rats; Rats, Inbred Strains; Retina | 1982 |
Benzodiazepines in clinical medicine: discussion.
Topics: Anti-Anxiety Agents; Diazepam; Flurazepam; Half-Life; Humans; Protein Binding; Substance Withdrawal Syndrome | 1981 |
Differential effects of benzodiazepines on EEG activity and hypnogenic mechanisms of the brain stem in cats.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Brain Stem; Cats; Decerebrate State; Diazepam; Electroencephalography; Flurazepam; Pentobarbital; Sleep | 1983 |
Withdrawal after substitution of a short-acting for a long-acting benzodiazepine.
Topics: Anti-Anxiety Agents; Anxiety; Chronic Disease; Delayed-Action Preparations; Diazepam; Flurazepam; Half-Life; Humans; Oxazepam; Sleep Initiation and Maintenance Disorders; Substance Withdrawal Syndrome; Temazepam | 1983 |
[Behavioral effects of ethyl loflazepate and its metabolites].
Topics: Aggression; Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Conflict, Psychological; Diazepam; Drug Synergism; Flurazepam; Humans; Lorazepam; Male; Mice; Motor Activity; Nitrazepam; Rats; Rats, Inbred Strains; Thiopental | 1983 |
Simulated car driving as a useful technique for the determination of residual effects and alcohol interaction after short- and long-acting benzodiazepines.
Topics: Anti-Anxiety Agents; Automobile Driving; Benzodiazepines; Diazepam; Double-Blind Method; Drug Interactions; Ethanol; Flurazepam; Heart Rate; Humans; Hypnotics and Sedatives; Lorazepam; Pindolol; Psychomotor Performance; Reaction Time | 1984 |
Differential effects of the benzodiazepine antagonist Ro 15-1788 after "general anaesthetic" doses of benzodiazepines in mice.
Topics: Anesthesia, General; Anesthetics; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Chlordiazepoxide; Convulsants; Diazepam; Flumazenil; Flurazepam; Male; Mice; Mice, Inbred Strains; Midazolam; Reflex | 1984 |
Depression following withdrawal from long-term benzodiazepine use: a report of four cases.
Topics: Adult; Anti-Anxiety Agents; Depressive Disorder; Diazepam; Female; Flurazepam; Humans; Lorazepam; Male; Medazepam; Middle Aged; Substance Withdrawal Syndrome | 1984 |
Chlordiazepoxide selectively potentiates GABA conductance of spinal cord and sensory neurons in cell culture.
Topics: Animals; Cells, Cultured; Chick Embryo; Chlordiazepoxide; Diazepam; Dose-Response Relationship, Drug; Flurazepam; gamma-Aminobutyric Acid; Neurons; Spinal Cord; Synaptic Transmission; Time Factors | 1981 |
Norharman inhibition of [3H]diazepam binding in mouse brain.
Topics: Alkaloids; Animals; Brain; Carbolines; Diazepam; Flurazepam; Harmine; In Vitro Techniques; Kinetics; Male; Mice; Receptors, Drug; Receptors, GABA-A | 1981 |
Benzodiazepine--specific and nonspecific tolerance following chronic flurazepam treatment.
Topics: Animals; Ataxia; Diazepam; Drug Tolerance; Ethanol; Flurazepam; Male; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Acute effects of drug administration and withdrawal on the benzodiazepine receptor.
Topics: Animals; Benzodiazepines; Cerebral Cortex; Clonazepam; Diazepam; Flurazepam; Humans; Lorazepam; Male; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Substance Withdrawal Syndrome | 1983 |
Benzodiazepine inhibition of adenosine uptake is not prevented by benzodiazepine antagonists.
Topics: Adenosine; Animals; Benzodiazepines; Benzodiazepinones; Brain; Diazepam; Flumazenil; Flurazepam; Hexobendine; In Vitro Techniques; Pyrazoles; Rats; Rats, Inbred Strains; Synaptosomes; Temperature | 1983 |
Studies on [3H]diazepam and [3H]ethyl-beta-carboline carboxylate binding to rat brain in vivo. I. Regional variations in displacement.
Topics: Animals; Benzodiazepinones; Brain; Carbolines; Convulsants; Diazepam; Flumazenil; Flurazepam; Indoles; Male; Rats; Rats, Inbred Strains; Tissue Distribution | 1983 |
Inhibition of adenosine accumulation by a CNS benzodiazepine antagonist (Ro 15-1788) and a peripheral benzodiazepine receptor ligand (Ro 05-4864).
Topics: Adenosine; Animals; Benzodiazepines; Benzodiazepinones; Central Nervous System; Diazepam; Flumazenil; Flurazepam; Hexobendine; Male; Rats; Synaptosomes; Time Factors | 1983 |
Attention tasks as skills performance measures of drug effects.
Topics: Accidents, Traffic; Attention; Automobile Driving; Behavior; Caffeine; Cannabis; Cognition; Diazepam; Diphenhydramine; Ethanol; Flurazepam; Humans; Perception; Psychomotor Performance; Reaction Time; Time Factors | 1984 |
Successful treatment of human non-24-hour sleep-wake syndrome.
Topics: Adult; Diazepam; Flurazepam; Humans; Male; Periodicity; Sleep Wake Disorders; Thyroxine; Vitamin B 12 | 1983 |
Withdrawal symptoms after long-term treatment with flurazepam.
Topics: Anxiety Disorders; Depressive Disorder; Diazepam; Flurazepam; Humans; Sleep Initiation and Maintenance Disorders; Substance Withdrawal Syndrome | 1984 |
Stimulus control by diazepam of behavior maintained under fixed-ratio stimulus-shock termination schedules in rats.
Topics: Animals; Behavior, Animal; Conditioning, Operant; Cyproheptadine; Diazepam; Discrimination, Psychological; Electroshock; Flurazepam; Male; Pentobarbital; Rats; Rats, Inbred F344; Reinforcement Schedule | 1984 |
Radioimmunoassay of benzodiazepines.
Topics: Benzodiazepines; Chlordiazepoxide; Clonazepam; Diazepam; Flurazepam; Humans; Microchemistry; Nitrazepam; Nordazepam; Oxazepam; Radioimmunoassay | 1982 |
Effects of benzodiazepines on single unit activity in the substantia nigra pars reticulata.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Bicuculline; Caffeine; Diazepam; Dose-Response Relationship, Drug; Electric Conductivity; Flumazenil; Flurazepam; Male; Neurons; Picrotoxin; Rats; Rats, Inbred Strains; Substantia Nigra; Theophylline | 1982 |
Alcohol withdrawal syndromes - prediction from detailed medical and drinking histories.
Topics: Adult; Aged; Alcohol Drinking; Alcohol Withdrawal Delirium; Alcoholism; Diazepam; Female; Flurazepam; Humans; Male; Middle Aged; Prognosis; Psychoses, Alcoholic | 1983 |
Pharmacological effects of flurazepam and diazepam on isolated canine arteries.
Topics: Animals; Aorta, Thoracic; Calcium; Coronary Vessels; Diazepam; Dogs; Female; Flurazepam; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Norepinephrine; Potassium | 1983 |
Benzodiazepine utilization in a family medicine residency program.
Topics: Adolescent; Adult; Aged; Benzodiazepines; Diazepam; Drug Utilization; Family Practice; Female; Flurazepam; Humans; Internship and Residency; Male; Middle Aged; North Dakota; Retrospective Studies; Sex Factors | 1982 |
Effects of flurazepam and diazepam in isolated guinea-pig taenia coli and longitudinal muscle.
Topics: Animals; Calcium; Cecum; Diazepam; Female; Flurazepam; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Potassium | 1982 |
Effects of physostigmine on benzodiazepine toxicity.
Topics: Animals; Benzodiazepines; Chlordiazepoxide; Diazepam; Electroencephalography; Flurazepam; Hemodynamics; Lethal Dose 50; Male; Mice; Physostigmine; Postural Balance; Rats; Rats, Inbred Strains; Reflex | 1981 |
Diazepam receptors on mouse astrocytes in primary cultures: displacement by pharmacologically active concentrations of benzodiazepines or barbiturates.
Topics: Animals; Astrocytes; Barbiturates; Benzodiazepines; Binding Sites; Binding, Competitive; Cells, Cultured; Clonazepam; Diazepam; Flurazepam; Mice; Pentobarbital; Phenobarbital; Receptors, Drug | 1980 |
Systematic review of the benzodiazepines. Guidelines for data sheets on diazepam, chlordiazepoxide, medazepam, clorazepate, lorazepam, oxazepam, temazepam, triazolam, nitrazepam, and flurazepam. Committee on the Review of Medicines.
Topics: Benzodiazepines; Chlordiazepoxide; Clorazepate Dipotassium; Diazepam; Flurazepam; Humans; Lorazepam; Medazepam; Nitrazepam; Oxazepam; Safety; Substance Withdrawal Syndrome; Substance-Related Disorders; Temazepam; Triazolam | 1980 |
[Does a rebound insomnia following benzodiazepine administration exist?].
Topics: Benzodiazepines; Diazepam; Flunitrazepam; Flurazepam; Humans; Nitrazepam; Sleep Initiation and Maintenance Disorders; Substance Withdrawal Syndrome; Triazolam | 1980 |
Effects of barbital or diazepam withdrawal on seizure thresholds to bicuculline, picrotoxin and flurazepam.
Topics: Animals; Barbital; Bicuculline; Convulsants; Diazepam; Flurazepam; Male; Picrotoxin; Rats; Rats, Sprague-Dawley; Seizures; Substance Withdrawal Syndrome | 1995 |
Regional changes in [3H]zolpidem binding to brain benzodiazepine receptors in flurazepam tolerant rat: comparison with changes in [3H]flunitrazepam binding.
Topics: Animals; Brain; Diazepam; Drug Tolerance; Flunitrazepam; Flurazepam; Male; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; RNA, Messenger; Tritium; Zolpidem | 1994 |
[Inhibitory effect of diazepam or flurazepam on pressor response induced by the stimulation of midbrain in the rabbit].
Topics: Animals; Blood Pressure; Diazepam; Flurazepam; Heart Rate; Medulla Oblongata; Mesencephalon; Pressoreceptors; Rabbits | 1993 |
Sleep and motor activity of community elderly who frequently use bedtime medications.
Topics: Aged; Circadian Rhythm; Diazepam; Drug Administration Schedule; Female; Flurazepam; Humans; Hypnotics and Sedatives; Male; Motor Activity; Sleep Initiation and Maintenance Disorders; Sleep Stages | 1994 |
Reduced expression of gamma-aminobutyric acid type A/benzodiazepine receptor gamma 2 and alpha 5 subunit mRNAs in brain regions of flurazepam-treated rats.
Topics: Alternative Splicing; Animals; Base Sequence; Cerebellum; Cerebral Cortex; Diazepam; DNA Primers; Flurazepam; Gene Expression; Hippocampus; Molecular Sequence Data; Rats; Receptors, GABA; RNA, Messenger | 1994 |
Tolerance to the effects of diazepam, clonazepam and bretazenil on GABA-stimulated Cl- influx in flurazepam tolerant rats.
Topics: Animals; Benzodiazepinones; Chloride Channels; Clonazepam; Diazepam; Drug Tolerance; Flurazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA | 1993 |
Behavioral approaches to polydipsia.
Topics: Adult; Behavior Therapy; Combined Modality Therapy; Diazepam; Female; Flurazepam; Humans; Male; Reinforcement, Psychology; Relaxation Therapy; Schizophrenia; Schizophrenic Psychology; Water Intoxication | 1993 |
Application of capillary electrophoresis to the simultaneous screening and quantitation of benzodiazepines.
Topics: Autoanalysis; Benzodiazepines; Bromazepam; Buffers; Diazepam; Electrophoresis, Capillary; Estazolam; Flurazepam; Humans; Hydrogen-Ion Concentration; Nitrazepam; Reproducibility of Results; Sensitivity and Specificity; Triazolam | 1996 |
Down-regulation of benzodiazepine binding to alpha 5 subunit-containing gamma-aminobutyric Acid(A) receptors in tolerant rat brain indicates particular involvement of the hippocampal CA1 region.
Topics: Alkynes; Animals; Anti-Anxiety Agents; Autoradiography; Benzodiazepines; Binding Sites; Brain; Diazepam; Down-Regulation; Drug Tolerance; Flunitrazepam; Flurazepam; GABA Modulators; Hippocampus; Imidazoles; Kinetics; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Tritium | 2000 |
Determination of partition coefficients of diazepam and flurazepam between phosphatidylcholine bilayer vesicles and water by second derivative spectrophotometric method.
Topics: Algorithms; Anti-Anxiety Agents; Buffers; Chemical Phenomena; Chemistry, Physical; Diazepam; Flurazepam; Hydrogen-Ion Concentration; Indicators and Reagents; Lipid Bilayers; Phosphatidylcholines; Spectrophotometry, Ultraviolet; Water | 2001 |
Effect of phosphatidylserine content on the partition coefficients of diazepam and flurazepam between phosphatidylcholine-phosphatidylserine bilayer of small unilamellar vesicles and water studied by second derivative spectrophotometry.
Topics: Diazepam; Flurazepam; Lipid Bilayers; Phosphatidylserines; Spectrophotometry; Water | 2002 |
Benzodiazepine modulation of partial agonist efficacy and spontaneously active GABA(A) receptors supports an allosteric model of modulation.
Topics: Allosteric Regulation; Animals; Benzodiazepines; Cells, Cultured; Chick Embryo; Computer Simulation; Diazepam; Dose-Response Relationship, Drug; Flurazepam; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; Mutagenesis, Site-Directed; Neurons; Pyrones; Receptors, GABA-A; Transfection | 2005 |
K+ channel TASK-1 knockout mice show enhanced sensitivities to ataxic and hypnotic effects of GABA(A) receptor ligands.
Topics: Animals; Anti-Anxiety Agents; Ataxia; Benzodiazepines; Brain; Diazepam; Female; Flurazepam; Hypnotics and Sedatives; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Nerve Tissue Proteins; Pentobarbital; Potassium Channels, Tandem Pore Domain; Propofol; Protein Kinase C; Receptors, GABA-A; Sex Factors; Spinal Cord | 2008 |