diazepam has been researched along with fluorobenzenes in 18 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (16.67) | 18.7374 |
1990's | 1 (5.56) | 18.2507 |
2000's | 11 (61.11) | 29.6817 |
2010's | 3 (16.67) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Duffy, EM; Jorgensen, WL | 1 |
Caron, G; Ermondi, G | 1 |
Abellán Guillén, A; Cordeiro, MN; Garrido Escudero, A; Morales Helguera, A; Pérez-Garrido, A | 1 |
Akatsu, M; Asami, Y; Inaba, S; Kitagawa, S; Otsuka, M; Yamamoto, H | 1 |
Asami, Y; Hirohashi, T; Inaba, S; Otsuka, M; Yamamoto, H | 1 |
Barnett, A; Fiedler, EP; Goldstein, J; Taber, RI | 1 |
Griebel, G; Perrault, G; Sanger, DJ | 1 |
Atack, JR; Bristow, L; Brown, N; Carling, RW; Castro, JL; Cook, G; Dawson, GR; Farrar, S; Ferris, P; Garrett, L; Howell, O; Macaulay, A; Marshall, G; McKernan, RM; Moore, KW; Myers, J; Ragan, CI; Reynolds, DS; Rosahl, TW; Street, LJ; Sur, C; Wafford, KA; Whiting, PJ | 1 |
Dawson, GR; McKernan, RM; Reynolds, DS | 1 |
Kiss, A; Mikkelsen, JD; Mirza, N; Søderman, A | 1 |
Groenink, L; Olivier, B; Oosting, R; Toth, M; Van Bogaert, M; van Oorschot, R | 1 |
Ahmadi, S; Brockhaus, J; Brune, K; Fritschy, JM; Hess, A; Hösl, K; Knabl, J; Möhler, H; Reinold, H; Rudolph, U; Sergejeva, M; Witschi, R; Zeilhofer, HU; Zeilhofer, UB | 1 |
Bostwick, R; Chen, T; Huston, J; Knappenberger, K; Liu, J; Norris, T; Wood, M | 1 |
Bundzikova, J; Hansen, HH; Kiss, A; Larsen, MH; Mikkelsen, JD | 1 |
Clifton, PG; Dixon, CI; Morris, HV; Nilsson, S; Stephens, DN | 1 |
Atack, JR; Cook, JM; Dawson, GR; Licata, SC; Platt, DM; Rowlett, JK; Rüedi-Bettschen, D; Van Linn, ML | 1 |
Atack, JR | 2 |
2 review(s) available for diazepam and fluorobenzenes
Article | Year |
---|---|
GABAA receptor subtype-selective modulators. II. α5-selective inverse agonists for cognition enhancement.
Topics: Animals; Benzodiazepines; Cognition; Diazepam; Female; Fluorobenzenes; GABA-A Receptor Agonists; Hippocampus; Humans; Isoxazoles; Male; Maze Learning; Memory; Mice; Nootropic Agents; Protein Isoforms; Pyridazines; Pyridines; Rats; Receptors, GABA-A; Structure-Activity Relationship; Substrate Specificity; Triazines; Triazoles | 2011 |
GABAA receptor subtype-selective modulators. I. α2/α3-selective agonists as non-sedating anxiolytics.
Topics: Animals; Anti-Anxiety Agents; Benzimidazoles; Benzodiazepines; Diazepam; Dogs; Fluorobenzenes; GABA-A Receptor Agonists; Humans; Hypnotics and Sedatives; Male; Mice; Mice, Transgenic; Protein Isoforms; Pyridazines; Pyridines; Rats; Receptors, GABA-A; Structure-Activity Relationship; Substrate Specificity; Triazoles | 2011 |
16 other study(ies) available for diazepam and fluorobenzenes
Article | Year |
---|---|
Prediction of drug solubility from Monte Carlo simulations.
Topics: Monte Carlo Method; Pharmaceutical Preparations; Solubility | 2000 |
Calculating virtual log P in the alkane/water system (log P(N)(alk)) and its derived parameters deltalog P(N)(oct-alk) and log D(pH)(alk).
Topics: 1-Octanol; Alkanes; Hydrogen-Ion Concentration; Least-Squares Analysis; Mathematics; Models, Chemical; Models, Molecular; Solvents; Water | 2005 |
Convenient QSAR model for predicting the complexation of structurally diverse compounds with beta-cyclodextrins.
Topics: beta-Cyclodextrins; Hydrophobic and Hydrophilic Interactions; Organic Chemicals; Quantitative Structure-Activity Relationship | 2009 |
The synthesis and pharmacology of a novel benzodiazepine derivative, 1-(beta-methylsulfonylethyl)-5-(o-fluorophenyl)-7-chloro-1,3-dihydro-2H-1,4-benzodiazepin-2-one (ID-622).
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Bemegride; Cats; Chlorprothixene; Diazepam; Drug Synergism; Electroencephalography; Electroshock; Female; Fluorobenzenes; Hexobarbital; Male; Mice; Motor Activity; Muscle Relaxants, Central; Rats; Reflex | 1975 |
The synthesis and pharmacology of a novel benzodiazepine derivative, 1-methyl-5-(o-fluorophenyl)-7-chloro-1,3-dihydro-2H-1,4-benzodiazepin-2-one(ID-540).
Topics: Aggression; Animals; Anti-Anxiety Agents; Behavior, Animal; Bemegride; Benzodiazepinones; Cats; Chlorprothixene; Diazepam; Drug Synergism; Electroencephalography; Electroshock; Female; Fluorobenzenes; Hexobarbital; Humans; Lethal Dose 50; Male; Mice; Motor Activity; Muscle Tonus; Olfactory Bulb; Pentylenetetrazole; Rats; Reflex; Seizures; Septum Pellucidum; Strychnine | 1974 |
The pharmacology of fletazepam a centrally-acting muscle relaxant.
Topics: Aggression; Animals; Anticonvulsants; Avoidance Learning; Benzazepines; Benzodiazepines; Cats; Diazepam; Dose-Response Relationship, Drug; Electroshock; Female; Fluorobenzenes; Humans; Male; Mice; Muscle Relaxants, Central; Muscle Rigidity; Pentylenetetrazole; Rats; Reflex; Seizures; Strychnine; Time Factors | 1974 |
A comparative study of the effects of selective and non-selective 5-HT2 receptor subtype antagonists in rat and mouse models of anxiety.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Diazepam; Drinking; Fluorobenzenes; Indoles; Male; Maze Learning; Mianserin; Mice; Mice, Inbred BALB C; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists | 1997 |
Sedative but not anxiolytic properties of benzodiazepines are mediated by the GABA(A) receptor alpha1 subtype.
Topics: Allosteric Site; Animals; Anti-Anxiety Agents; Anticonvulsants; Azides; Benzodiazepines; Binding, Competitive; Brain; Cell Line; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Fluorobenzenes; GABA-A Receptor Antagonists; Hypnotics and Sedatives; Ligands; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Motor Activity; Patch-Clamp Techniques; Receptors, GABA-A; Reflex, Startle; Triazoles | 2000 |
Anxiolytic-like action of diazepam: which GABA(A) receptor subtype is involved?
Topics: Animals; Anti-Anxiety Agents; Diazepam; Fluorobenzenes; Locomotion; Mice; Point Mutation; Rats; Receptors, GABA-A; Triazoles | 2001 |
Effects of benzodiazepines receptor agonists on the hypothalamic-pituitary-adrenocortical axis.
Topics: Adrenocorticotropic Hormone; Animals; Azabicyclo Compounds; Carbolines; Corticosterone; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Fluorobenzenes; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; Hypothalamo-Hypophyseal System; Male; Mice; Mice, Inbred Strains; Models, Biological; Paraventricular Hypothalamic Nucleus; Piperazines; Pituitary-Adrenal System; Proto-Oncogene Proteins c-fos; Pyridines; Radioimmunoassay; Receptors, GABA-A; Triazoles; Zolpidem | 2005 |
Effects of genetic background and null mutation of 5-HT1A receptors on basal and stress-induced body temperature: modulation by serotonergic and GABAA-ergic drugs.
Topics: Animals; Body Temperature; Body Temperature Regulation; Buspirone; Diazepam; Fever; Flumazenil; Fluorobenzenes; GABA Agonists; GABA Modulators; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Pyridines; Receptor, Serotonin, 5-HT1A; Receptors, GABA-A; Serotonin; Serotonin Agents; Serotonin Receptor Agonists; Stress, Psychological; Triazoles; Zolpidem | 2006 |
Reversal of pathological pain through specific spinal GABAA receptor subtypes.
Topics: Analgesics; Animals; Brain; Capsaicin; Chronic Disease; Diazepam; Disease Models, Animal; Fluorobenzenes; Formaldehyde; Ganglia, Spinal; Hot Temperature; Inflammation; Male; Mice; Neurons; Organ Specificity; Pain; Protein Isoforms; Protein Subunits; Rats; Rats, Wistar; Receptors, GABA-A; Spinal Cord; Triazoles | 2008 |
A high-throughput functional assay for characterization of gamma-aminobutyric acid(A) channel modulators using cryopreserved transiently transfected cells.
Topics: Carbolines; Cell Culture Techniques; Cell Line; Cell Membrane; Cryopreservation; Diazepam; DNA; Dose-Response Relationship, Drug; Drug Discovery; Flumazenil; Flunitrazepam; Fluorescent Dyes; Fluorobenzenes; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Membrane Potentials; Receptors, GABA-A; Reproducibility of Results; Spectrometry, Fluorescence; Transfection; Triazoles; Tritium | 2008 |
GABA regulates the rat hypothalamic-pituitary-adrenocortical axis via different GABA-A receptor alpha-subtypes.
Topics: Animals; Brain; Corticotropin-Releasing Hormone; Diazepam; Fluorobenzenes; GABA Agonists; GABA Modulators; gamma-Aminobutyric Acid; Hypothalamo-Hypophyseal System; Male; Neural Pathways; Paraventricular Hypothalamic Nucleus; Pituitary-Adrenal System; Protein Subunits; Proto-Oncogene Proteins c-fos; Pyridines; Random Allocation; Rats; Rats, Wistar; Receptors, GABA-A; Triazoles; Zolpidem | 2008 |
Alpha1- and alpha2-containing GABAA receptor modulation is not necessary for benzodiazepine-induced hyperphagia.
Topics: Analysis of Variance; Animals; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Energy Intake; Female; Fluorobenzenes; GABA Modulators; GABA-A Receptor Agonists; Hyperphagia; Male; Mice; Mice, Knockout; Midazolam; Random Allocation; Receptors, GABA-A; Triazoles | 2009 |
Discriminative stimulus effects of L-838,417 (7-tert-butyl-3-(2,5-difluoro-phenyl)-6-(2-methyl-2H-[1,2,4]triazol-3-ylmethoxy)-[1,2,4]triazolo[4,3-b]pyridazine): role of GABA(A) receptor subtypes.
Topics: Animals; Barbiturates; Carbolines; Catheterization; Central Nervous System Depressants; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Ethanol; Flumazenil; Fluorobenzenes; GABA Agonists; GABA Antagonists; GABA Modulators; Neuropsychological Tests; Pyridines; Receptors, GABA-A; Saimiri; Triazoles; Zolpidem | 2010 |