diazepam and clonidine

diazepam has been researched along with clonidine in 192 studies

Research

Studies (192)

TimeframeStudies, this research(%)All Research%
pre-199078 (40.63)18.7374
1990's39 (20.31)18.2507
2000's30 (15.63)29.6817
2010's42 (21.88)24.3611
2020's3 (1.56)2.80

Authors

AuthorsStudies
Andrews, PR; Craik, DJ; Martin, JL1
Dalton, CR; Dudley, MW; Kane, JM; Kehne, JH; Ketteler, HJ; McCloskey, TC; Miller, FP; Ogden, AM; Senyah, Y; Staeger, MA1
Carrupt, PA; Crivori, P; Cruciani, G; Testa, B1
Topliss, JG; Yoshida, F1
Gao, F; Lombardo, F; Shalaeva, MY; Tupper, KA1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY2
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Baert, B; Beetens, J; Bodé, S; De Spiegeleer, B; Deconinck, E; Lambert, J; Slegers, G; Slodicka, M; Stoppie, P; Van Gele, M; Vander Heyden, Y1
Andricopulo, AD; Moda, TL; Montanari, CA1
Lombardo, F; Obach, RS; Waters, NJ1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Ahman, M; Holmén, AG; Wan, H1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Du-Cuny, L; Mash, EA; Meuillet, EJ; Moses, S; Powis, G; Song, Z; Zhang, S1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Choi, SS; Contrera, JF; Hastings, KL; Kruhlak, NL; Sancilio, LF; Weaver, JL; Willard, JM1
Campillo, NE; Guerra, A; Páez, JA1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Ahlin, G; Bergström, F; Bredberg, U; Fridén, M; Hammarlund-Udenaes, M; Rehngren, M; Wan, H1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Deng, Y; Li, Y; Liu, Q; Qiang, X; Sang, Z; Tan, Z; Xiao, G1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Deng, Y; Li, Y; Luo, L; Qiang, X; Tan, Z; Xiao, G1
Cao, Z; Deng, Y; Li, Y; Luo, L; Qiang, X; Sang, Z; Su, F; Xiao, G; Yang, X; Zheng, Y1
Ai, J; Deng, Y; Li, Y; Liu, Q; Luo, L; Qiang, X; Tan, Z; Xiao, G; Yang, X1
Cao, Z; Deng, Y; Li, Y; Luo, L; Qiang, X; Sang, Z; Su, F; Xiao, G; Xu, R; Yang, X; Zheng, Y1
Cao, Z; Deng, Y; Li, Y; Luo, L; Qiang, X; Tan, Z; Xu, R; Yang, X; Zheng, Y1
Cao, Z; Deng, Y; Li, Y; Luo, L; Qiang, X; Song, Q; Tan, Z; Xiao, G; Xu, R; Yang, X1
Bai, P; Leng, C; Li, X; Liu, W; Ma, Q; Pan, W; Sang, Z; Tan, Z; Wang, K; Xu, Q; Yang, Y; Yu, L1
Liu, W; Ma, Q; Pan, W; Sang, Z; Wang, K; Yu, L1
Han, X; Liu, W; Ma, Q; Sang, Z; Wang, H; Wang, K; Ye, M; Yu, L2
Dong, SN; Gong, Q; Li, J; Li, XK; Liu, WW; Mao, F; Tang, Y; Wang, H; Wang, TD; Xu, YX; Zhang, HY; Zhu, J1
Cao, Z; Deng, Y; Li, Y; Liu, H; Qiang, X; Song, Q; Tan, Z; Xu, R; Yang, J; Zhang, X1
Deng, Y; Li, Y; Liu, H; Song, Q; Tan, Z; Xiao, G; Xu, R; Yang, Z; Zhang, X; Zheng, Y1
Gong, Q; Li, J; Li, X; Liu, W; Mao, F; Qiu, X; Wang, H; Wang, W; Xu, Y; Zhang, H; Zhang, J; Zhu, J1
An, Q; Deng, Y; Liu, P; Luo, Y; Sang, Z; Tang, Y; Wang, T; Yang, T; Yang, Y; Zhang, T1
Cao, Z; Deng, Y; Li, Y; Liu, H; Qiang, X; Song, Q; Tan, Z; Tian, C; Yang, Z1
Deng, Y; He, Y; Li, W; Liu, H; Qiang, X; Song, Q; Tan, Z; Ye, C1
Liu, W; Sang, Z; Shi, J; Tan, Z; Wang, K1
Liu, W; Sang, Z; Shi, J; Tan, Z; Wang, K; Zhang, P1
Fan, X; Liu, W; Sang, Z; Shi, J; Wang, K; Yang, D; Zhang, P; Zhang, Z; Zhu, G1
Bai, P; Cheng, X; Cheng, Y; Lu, X; Sang, Z; Shi, J; Wang, K; Yang, J; Zhang, P; Zhang, Q; Zheng, C1
Dinnendahl, V; Gumulka, SW1
Walters, WA1
Canevari, A; Cugurra, F; Piredda, F1
Glover, V; Grant, E; Orton, D; Rose, FC; Sandler, M; Stevens, D; Wilkinson, M1
Ludin, HP1
Beshara, D; Levy, JM; Stoll, C1
Bolme, P; Fuxe, K1
Dorokhova, MI1
Poignant, JC; Rismondo, N1
Evans, RH; Long, SK; Siarey, RJ1
Buccafusco, JJ; Li, W1
Ishizuki, M; Yanagisawa, M1
Bhattacharya, A; Bose, S; Kumar, A; Kundra, P; Tandon, OP2
Devi, K; Hrishikeshavan, HJ; Munonyedi, US; Shanbhogue, RS1
Avrutskiĭ, MIa; Guseĭnov, TIu; Katkovskiĭ, DG; Musikhin, LV; Zhukov, VN1
Barone, D; Spignoli, G1
Asakura, N; Hamaya, Y; Harukuni, I; Nishikawa, T1
Hartmann, M; Seitz, W; Verner, L1
Dietz, V1
Holtzman, SG1
Pouttu, J; Rosenberg, PH; Scheinin, M; Tuominen, M1
Luo, ZP; Yang, XM; Zhou, JH5
Aley, KO; Kulkarni, SK1
Ferrari, F; Mangiafico, V; Monti, A; Tartoni, PG1
Baran, H; Hornykiewicz, O; Hörtnagl, H1
Jørum, E1
Carlsson, M; Eriksson, E; Nilsson, C; Söderpalm, B1
Kulkarni, SK; Kunchandy, J1
Dangoumau, L; Poncelet, M; Simon, P; Soubrié, P1
Costall, B; Kelly, ME; Naylor, RJ1
Chrousos, GP; Crawley, JN; Linnoila, M; Ninan, PT; Paul, SM; Pickar, D; Skolnick, P1
Green, AR; Johnson, P; Mountford, JA; Nimgaonkar, VL1
Baran, H; Hornykiewicz, O; Hörtnagl, H; Sapetschnig, G; Sperk, G1
Forster, P; Stone, TW1
Costa, LG; Murphy, SD1
Molyneux, S; Nutt, D1
Hao, W; Wei, H; Young, D1
Kulkarni, SK; Parale, MP1
Eisenhofer, G; Goldstein, DS; Keiser, HR; Kopin, IJ; Stull, R; Udelsman, R1
Spealman, RD; Wettstein, JG1
Mattila, M; Mattila, MJ; Seppala, T1
Bailey, C; Brewer, C; Rezae, H1
Calvillo, O; Ghignone, M; Noe, C; Quintin, L1
Bes, A; Eyssette, M; Pierrot-Deseilligny, E; Rohmer, F; Warter, JM1
Igarashi, S; Yamamura, H; Yanagita, T1
Kulkarni, GK; Kulkarni, SK; Parale, MP1
Ghignone, M; Orko, R; Pouttu, J; Rosenberg, PH1
Fukuda, H; Kato, F; Kato, K; Matsumoto, K; Miyamoto, M; Mori, T; Nakamura, T; Oka, J; Ono, H1
Lakić, N; Manev, H; Pericić, D1
Baiguerra, G; Kostowski, W; Valzelli, L1
Conrad, B; Meinck, HM1
Delwaide, PJ1
Caccia, MR; Mangoni, A1
Martin, JD1
Furukawa, T; Katsuragi, T; Ushijima, I1
Adams, MA; Hirst, M1
Handley, SL; Mithani, S1
Cooke, RG; Homeida, AM2
Galloway, MP; Roth, RH2
Jurna, I1
Doaré, L; Simon, P; Soubrié, P; Thiébot, MH1
Aloi, J; Insel, TR; Jimerson, DC; Ninan, PT; Paul, SM; Skolnick, P1
Decobert, M; Depoortere, H; Honoré, L1
Kulkarni, SK; Mehta, AK1
Emmett-Oglesby, MW; Lal, H; Lewis, MW; Spencer, DG1
Grilly, DM; Jacoby, D; Johnson, SK; LaRiccia, J; Minardo, R1
Hennies, OL1
Fryda-Kaurimsky, Z; Müller-Fassbender, H1
Johansson, G; Luostarinen, M; Virkkunen, P1
Medvedev, OS; Val'dman, AV1
McLellan, DL1
Pappas, BA; Walsh, P1
Conrad, B; Meinck, HM; Ricker, K1
Haertzen, CA; Henningfield, JE; Jasinski, DR; Johnson, RE; Makhzoumi, HM; Miyasato, K1
Trulson, ME; Trulson, VM1
Huupponen, R; Koulu, M; Pihlajamäki, K1
Charney, DS; Heninger, GR; Redmond, DE1
Metz, G; Nebel, B1
Inoue, K; Kasai, H; Kobayashi, M; Kohno, S; Murata, T; Nagasaka, Y; Ohata, K; Sakamoto, H1
Baum, T; Moran, RM; Sabin, C1
Bhavsar, VH; Dhumal, VR; Kelkar, VV1
Berge, KH; Strickland, RA1
Cheng, CH; Costall, B; Ge, J; Naylor, RJ1
Imaizumi, M; Machida, H; Miyazaki, S1
Evans, RH; Long, SK; Siarey, RJ; Tulp, MT1
Davis, C; Emre, M; Groves, L; Lataste, X1
Adinoff, B1
Fukuda, H; Iwata, N; Kozuka, M; Nakamura, T; Ono, H; Tanabe, M1
Doak, GJ; Duke, PC1
Friedman, LS; Mayo-Smith, MF; Saitz, R1
Coull, JT; Middleton, HC; Robbins, TW; Sahakian, BJ2
Coull, JT; Cowen, PJ; McShane, RH; Middleton, HC; Park, SB; Robbins, TW; Sahakian, BJ; Young, AH1
Asano, M; Maekawa, N; Mikawa, K; Nishina, K; Obara, H1
Abduljawad, KA; Bradshaw, CM; Langley, RW; Szabadi, E2
Berkovich, AN; Bulganin, AD; Kuznetsova, OIu; Mikhaĭlovich, VA1
Batra, YK; Bhardwaj, N; Ramesh, VJ1
Ikizler, Y; Koren, G; Selby, P; Theis, JG1
Horikawa, Y; Kagawa, T; Kondo, M; Obara, H; Ohnishi, H1
Ishizuka, I; Kakoi, H; Kawasaki, J; Kawazoe, T; Kodaka, M; Miyao, H; Okamoto, Y1
Broderick, PA1
Black, WD; Celly, CS; McDonell, WN; Young, SS1
Batra, YK; Bhardwaj, N; Jatti, K; Malhotra, S1
Bitsios, P; Bradshaw, CM; Szabadi, E1
Imai, Y; Kagawa, K; Kirita, T; Kishi, Y; Kita, T; Mammoto, T; Murakami, K; Sakai, T; Sugimura, M1
Farber, NB; Kim, SH; Olney, JW; Price, MT1
Arnsten, AF; Franowicz, JS1
Castro, JL; Ramirez, A; Ricci, D; Taira, CA1
Fujii, Y; Saitoh, Y; Tanaka, H; Toyooka, H1
Goodkin, DE; Kita, M1
Fujii, Y; Handa, F1
Kamanin, EI; Kasianov, AA; Mishunin, IuV; Reshed'ko, OA; Tikhonov, FG1
Cole, MJ; Jeffery, HE; Osborn, DA3
Mishunin, IuV1
Axelsson, K; Berggren, L; Dobrydnjov, I; Holmström, B; Samarütel, J1
Patel, DR; Soyode, O1
Honda, K; Inomata, S; Nakamura, T; Tanaka, E1
Abbate, M; Ferlazzo, E; Granata, F; Mazzù, I; Musolino, R; Narbone, MC1
Hall, DL; Rezvan, E; Tatakis, DN; Walters, JD1
Carvalho, HG; Modolo, NS; Nascimento, Jdos S; Santos, KP; Silva, RC1
Aisen, M; Ashwal, S; Delgado, MR; Fehlings, DL; Hirtz, D; McLaughlin, J; Morrison, LA; Shrader, MW; Tilton, A; Vargus-Adams, J1
Benecke, R; Patejdl, R1
Kuks, JB; Lapeyre, E; Meijler, WJ1
Delgado, MR; Tilton, A; Vargus-Adams, J1
Muck-Šeler, D; Pivac, N; Švob Štrac, D1
Zdziarski, P1
Bamford, A; Clarke, A; Crowe, BH; Hacohen, Y; Lim, M; Lin, JP; Pullaperuma, SP; Sancho-Shimizu, V; Tudor-Williams, G; Vincent, A1
Comi, G; Gold, R; Hartung, HP; Montalban, X; Otero-Romero, S; Sastre-Garriga, J; Soelberg Sørensen, P; Thompson, AJ; Vermersch, P1
Kouzouna, A; Lindsay, C; Pandyan, AD; Simcox, C1
Iyengar, AR; Pande, AH1
Barnes, E; Kaufmann, H; Norcliffe-Kaufmann, L; Palma, JA; Spalink, CL1
Fu, X; Li, J; Li, M; Ma, Q; Wang, C; Wang, Y; Wu, H; Yang, W1
Assam, PN; Chan, E; Cheok, C; de Souza, NN; Guo, S; Kandasami, G; Koh, PK; Lee, KM; Manning, V; Pangjaya, J; Sultana, R; Wijesinghe, R; Wong, KE; Yang, Y1
Amin, S; Basu, A; Cadwgan, J; Crowe, B; DeAlwis, Y; Devlin, A; Kumar, R; Lodh, R; Lumsden, DE; Lundy, CT; Mordekar, SR; Smith, M1
Davey, JG; Martin, J; Osborn, DA; Zankl, A2
Bengono Bengono, RS; Metogo, JM; Minkande, JZ; Ndikontar, R; Ngouatna, S; Ntock, FN; Tochie, JN1

Reviews

20 review(s) available for diazepam and clonidine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
[Spasticity: therapy of increased reflexes or movement disorder?].
    Der Nervenarzt, 1990, Volume: 61, Issue:10

    Topics: Baclofen; Clonidine; Combined Modality Therapy; Dantrolene; Diazepam; Glycine; Humans; Locomotion; Muscle Relaxants, Central; Muscle Spasticity; Muscle Tonus; Muscles; Phenothiazines; Reflex, Abnormal

1990
Drug effects on the EEG of various species of laboratory animals.
    Neuropsychobiology, 1983, Volume: 9, Issue:4

    Topics: 5-Hydroxytryptophan; Amantadine; Animals; Antihypertensive Agents; Azabicyclo Compounds; Brain; Cats; Chlormethiazole; Clonidine; Diazepam; Electroencephalography; Flunitrazepam; Guanabenz; Guanfacine; Guanidines; Imidazoles; Male; Nitrazepam; Pentobarbital; Phenylacetates; Piperazines; Piracetam; Rats; Sodium Oxybate; Yohimbine

1983
Comparative profile of tizanidine in the management of spasticity.
    Neurology, 1994, Volume: 44, Issue:11 Suppl 9

    Topics: Activities of Daily Living; Baclofen; Clonidine; Diazepam; Humans; Muscle Relaxants, Central; Muscle Spasticity; Muscle Tonus

1994
Current management of the neonatal abstinence syndrome: a critical analysis of the evidence.
    Biology of the neonate, 1997, Volume: 71, Issue:6

    Topics: Analgesics, Opioid; Anticonvulsants; Antipsychotic Agents; Chlorpromazine; Clinical Trials as Topic; Clonidine; Diazepam; Drug Therapy, Combination; Humans; Hypnotics and Sedatives; Infant, Newborn; MEDLINE; Methadone; Morphine; Neonatal Abstinence Syndrome; Opium; Parasympatholytics; Phenobarbital; Sympatholytics

1997
Drugs used to treat spasticity.
    Drugs, 2000, Volume: 59, Issue:3

    Topics: Baclofen; Clonidine; Dantrolene; Diazepam; Drug Administration Schedule; Humans; Muscle Relaxants, Central; Muscle Spasticity

2000
Sedatives for opiate withdrawal in newborn infants.
    The Cochrane database of systematic reviews, 2002, Issue:3

    Topics: Chlorpromazine; Clonidine; Diazepam; Humans; Hypnotics and Sedatives; Infant, Newborn; Neonatal Abstinence Syndrome; Opioid-Related Disorders; Phenobarbital; Randomized Controlled Trials as Topic

2002
Sedatives for opiate withdrawal in newborn infants.
    The Cochrane database of systematic reviews, 2005, Jul-20, Issue:3

    Topics: Chlorpromazine; Clonidine; Diazepam; Humans; Hypnotics and Sedatives; Infant, Newborn; Neonatal Abstinence Syndrome; Opioid-Related Disorders; Phenobarbital; Randomized Controlled Trials as Topic

2005
Pharmacologic interventions for reducing spasticity in cerebral palsy.
    Indian journal of pediatrics, 2005, Volume: 72, Issue:10

    Topics: Administration, Oral; Adrenergic alpha-Agonists; Age Factors; Anti-Infective Agents, Local; Baclofen; Botulinum Toxins; Cerebral Palsy; Child; Child, Preschool; Clonidine; Dantrolene; Diazepam; Ethanol; Humans; Infant; Injections, Intramuscular; Injections, Spinal; Muscle Relaxants, Central; Muscle Spasticity; Neuromuscular Agents; Phenol; Time Factors

2005
Practice parameter: pharmacologic treatment of spasticity in children and adolescents with cerebral palsy (an evidence-based review): report of the Quality Standards Subcommittee of the American Academy of Neurology and the Practice Committee of the Child
    Neurology, 2010, Jan-26, Volume: 74, Issue:4

    Topics: Adolescent; Botulinum Toxins, Type A; Cerebral Palsy; Child; Clonidine; Diazepam; Humans; Muscle Relaxants, Central; Muscle Spasticity; Neuromuscular Agents; Treatment Outcome

2010
[New therapies for spastic movement disorders].
    MMW Fortschritte der Medizin, 2009, Volume: 151 Suppl 3

    Topics: Administration, Oral; Baclofen; Botulinum Toxins, Type A; Cannabinoids; Clonidine; Diazepam; Humans; Injections, Intramuscular; Injections, Spinal; Movement Disorders; Muscle Relaxants, Central; Muscle Spasticity; Parasympatholytics; Physical Therapy Modalities; Tolperisone

2009
Spasticity: revisiting the role and the individual value of several pharmacological treatments.
    NeuroRehabilitation, 2010, Volume: 27, Issue:2

    Topics: Amines; Baclofen; Botulinum Toxins; Calcium Channel Blockers; Clonidine; Cyclohexanecarboxylic Acids; Dantrolene; Diazepam; Gabapentin; gamma-Aminobutyric Acid; Humans; Muscle Relaxants, Central; Muscle Spasticity; Recovery of Function; Treatment Outcome

2010
Sedatives for opiate withdrawal in newborn infants.
    The Cochrane database of systematic reviews, 2010, Oct-06, Issue:10

    Topics: Chlorpromazine; Clonidine; Diazepam; Humans; Hypnotics and Sedatives; Infant, Newborn; Narcotics; Neonatal Abstinence Syndrome; Opioid-Related Disorders; Phenobarbital; Randomized Controlled Trials as Topic

2010
Pharmacologic treatment of spasticity in children.
    Seminars in pediatric neurology, 2010, Volume: 17, Issue:4

    Topics: Age Factors; Baclofen; Botulinum Toxins; Child; Clonidine; Dantrolene; Diazepam; Humans; Injections, Spinal; Muscle Spasticity; Neuromuscular Agents

2010
Pharmacological management of spasticity in multiple sclerosis: Systematic review and consensus paper.
    Multiple sclerosis (Houndmills, Basingstoke, England), 2016, Volume: 22, Issue:11

    Topics: Amines; Analgesics; Baclofen; Cannabidiol; Clonidine; Cyclohexanecarboxylic Acids; Dantrolene; Diazepam; Dronabinol; Drug Combinations; Excitatory Amino Acid Antagonists; Gabapentin; gamma-Aminobutyric Acid; Humans; Injections, Spinal; Multiple Sclerosis; Muscle Relaxants, Central; Muscle Spasticity; Phenol

2016
Pharmacological interventions other than botulinum toxin for spasticity after stroke.
    The Cochrane database of systematic reviews, 2016, Oct-06, Volume: 10

    Topics: Baclofen; Botulinum Toxins, Type A; Clonidine; Diazepam; Humans; Muscle Relaxants, Central; Muscle Spasticity; Randomized Controlled Trials as Topic; Stroke; Tolperisone

2016
Organophosphate-Hydrolyzing Enzymes as First-Line of Defence Against Nerve Agent-Poisoning: Perspectives and the Road Ahead.
    The protein journal, 2016, Volume: 35, Issue:6

    Topics: Antidotes; Atropine; Chemical Warfare; Clonidine; Diazepam; Excitatory Amino Acid Antagonists; Humans; Hydrolases; Hydrolysis; Nerve Agents; Organophosphates; Oximes; Purinergic P1 Receptor Agonists; Pyridostigmine Bromide; Renal Dialysis

2016
A mixed treatment comparison on efficacy and safety of treatments for spasticity caused by multiple sclerosis: a systematic review and network meta-analysis.
    Clinical rehabilitation, 2018, Volume: 32, Issue:6

    Topics: Baclofen; Botulinum Toxins, Type A; Cannabinoids; Clonidine; Diazepam; Humans; Multiple Sclerosis; Muscle Relaxants, Central; Muscle Spasticity; Neuromuscular Agents; Transcutaneous Electric Nerve Stimulation

2018
Sedatives for opioid withdrawal in newborn infants.
    The Cochrane database of systematic reviews, 2021, 05-18, Volume: 5

    Topics: Bias; Chlorpromazine; Clonidine; Diazepam; Humans; Hypnotics and Sedatives; Infant, Newborn; Narcotics; Neonatal Abstinence Syndrome; Opioid-Related Disorders; Phenobarbital; Randomized Controlled Trials as Topic; Treatment Outcome

2021
Opioid treatment for opioid withdrawal in newborn infants.
    The Cochrane database of systematic reviews, 2021, 07-07, Volume: 7

    Topics: Buprenorphine; Chlorpromazine; Clonidine; Diazepam; Humans; Hypnotics and Sedatives; Infant, Newborn; Methadone; Morphine; Narcotics; Neonatal Abstinence Syndrome; Opioid-Related Disorders; Opium; Phenobarbital; Randomized Controlled Trials as Topic

2021

Trials

38 trial(s) available for diazepam and clonidine

ArticleYear
[The effect of DS 103--282, a new type of myotonolyticum, on the contractile mechanism in human skeletal muscle (author's transl)].
    Der Nervenarzt, 1977, Volume: 48, Issue:7

    Topics: Benzodiazepinones; Clinical Trials as Topic; Clonidine; Diazepam; Double-Blind Method; Humans; Muscle Contraction

1977
Oral clonidine premedication for elderly patients undergoing intraocular surgery.
    Acta anaesthesiologica Scandinavica, 1992, Volume: 36, Issue:2

    Topics: Administration, Oral; Aged; Anesthesia Recovery Period; Cataract Extraction; Clonidine; Diazepam; Double-Blind Method; Female; Hemodynamics; Humans; Intraocular Pressure; Male; Middle Aged; Preanesthetic Medication

1992
[Effects of epidural clonidine added to lidocaine solution upon the requirements of sedatives during epidural anesthesia].
    Masui. The Japanese journal of anesthesiology, 1991, Volume: 40, Issue:5

    Topics: Adult; Anesthesia, Epidural; Clonidine; Diazepam; Female; Humans; Hysterectomy; Injections, Intravenous; Lidocaine; Middle Aged; Thiamylal

1991
[Clonidine supplemented analgesia and sedation in prevention of postoperative delirium].
    Anasthesie, Intensivtherapie, Notfallmedizin, 1990, Volume: 25, Issue:4

    Topics: Adult; Aged; Alcohol Withdrawal Delirium; Anesthesia, General; Arousal; Clonidine; Critical Care; Diazepam; Drug Therapy, Combination; Esophageal Neoplasms; Female; Hemodynamics; Humans; Male; Middle Aged; Pirinitramide; Postoperative Complications; Prospective Studies

1990
Effects of oral clonidine premedication on concentrations of cortisol and monoamine neurotransmitters and their metabolites in cerebrospinal fluid and plasma.
    Acta anaesthesiologica Scandinavica, 1989, Volume: 33, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Administration, Oral; Adult; Anesthesia, Spinal; Clinical Trials as Topic; Clonidine; Diazepam; Double-Blind Method; Epinephrine; Humans; Hydrocortisone; Hydroxyindoleacetic Acid; Male; Methoxyhydroxyphenylglycol; Norepinephrine; Preanesthetic Medication; Random Allocation; Tryptophan

1989
Effect of clonidine on cigarette cessation and in the alleviation of withdrawal symptoms.
    British journal of addiction, 1988, Volume: 83, Issue:10

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Behavior Therapy; Clinical Trials as Topic; Clonidine; Combined Modality Therapy; Diazepam; Double-Blind Method; Female; Humans; Male; Middle Aged; Substance Withdrawal Syndrome; Tobacco Use Disorder

1988
Anxiogenic effect of yohimbine in healthy subjects: comparison with caffeine and antagonism by clonidine and diazepam.
    International clinical psychopharmacology, 1988, Volume: 3, Issue:3

    Topics: Adult; Anxiety; Arousal; Caffeine; Clonidine; Diazepam; Dose-Response Relationship, Drug; Double-Blind Method; Female; Growth Hormone; Humans; Hydrocortisone; Male; Panic; Prolactin; Yohimbine

1988
Anesthesia for ophthalmic surgery in the elderly: the effects of clonidine on intraocular pressure, perioperative hemodynamics, and anesthetic requirement.
    Anesthesiology, 1988, Volume: 68, Issue:5

    Topics: Anesthesia; Anesthesia, General; Anesthesia, Local; Animals; Clinical Trials as Topic; Clonidine; Diazepam; Double-Blind Method; Female; Hemodynamics; Humans; Intraocular Pressure; Intraoperative Period; Male; Middle Aged; Ophthalmologic Surgical Procedures; Preanesthetic Medication; Random Allocation

1988
A multi-centre, double-blind trial of tizanidine, a new antispastic agent, in spasticity associated with hemiplegia.
    Current medical research and opinion, 1988, Volume: 10, Issue:10

    Topics: Adolescent; Adult; Aged; Clinical Trials as Topic; Clonidine; Diazepam; Double-Blind Method; Female; Hemiplegia; Humans; Male; Middle Aged; Muscle Relaxants, Central; Muscle Spasticity; Random Allocation

1988
Effects of tizanidine in healthy volunteers: double-blind study compared with diazepam and a placebo.
    International journal of clinical pharmacology research, 1988, Volume: 8, Issue:2

    Topics: Adult; Blood Pressure; Clonidine; Diazepam; Double-Blind Method; Heart Rate; Humans; Male; Placebos; Substance-Related Disorders; Surveys and Questionnaires

1988
Effect of clonidine on haemodynamic responses to endotracheal intubation and on gastric acidity.
    Acta anaesthesiologica Scandinavica, 1987, Volume: 31, Issue:4

    Topics: Administration, Oral; Adolescent; Adult; Aged; Cimetidine; Clonidine; Diazepam; Female; Gastric Acid; Heart Rate; Hemodynamics; Humans; Intubation, Intratracheal; Male; Middle Aged; Preanesthetic Medication; Random Allocation

1987
A new skeletal muscle relaxant (DS 103-282) compared to diazepam in the treatment of muscle spasm of local origin.
    The Journal of international medical research, 1981, Volume: 9, Issue:1

    Topics: Adult; Aged; Back Pain; Clinical Trials as Topic; Clonidine; Diazepam; Double-Blind Method; Female; Humans; Male; Middle Aged; Muscle Relaxants, Central; Muscle Spasticity

1981
Tizanidine (DS 103-282) in the treatment of acute paravertebral muscle spasm: a controlled trial comparing tizanidine and diazepam.
    The Journal of international medical research, 1981, Volume: 9, Issue:6

    Topics: Acute Disease; Adult; Back Pain; Clinical Trials as Topic; Clonidine; Diazepam; Double-Blind Method; Female; Humans; Male; Middle Aged; Random Allocation; Spasm; Spinal Diseases; Time Factors

1981
Effect of the benzodiazepine derivative, diazepam, on the clonidine-stimulated human growth hormone secretion.
    The Journal of clinical endocrinology and metabolism, 1983, Volume: 56, Issue:6

    Topics: Adult; Clonidine; Diazepam; Growth Hormone; Humans; Infusions, Parenteral; Male; Pituitary Gland, Anterior; Stimulation, Chemical; Time Factors

1983
Double-blind study of alprazolam, diazepam, clonidine, and placebo in the alcohol withdrawal syndrome: preliminary findings.
    Alcoholism, clinical and experimental research, 1994, Volume: 18, Issue:4

    Topics: Adult; Alcohol Withdrawal Delirium; Alcoholism; Alprazolam; Blood Pressure; Clonidine; Diazepam; Double-Blind Method; Ethanol; Female; Heart Rate; Humans; Male; Middle Aged; Neurologic Examination; Receptors, GABA-A

1994
Recovery from pre-operative sedation with clonidine--brain stem auditory evoked response.
    Anaesthesia, 1994, Volume: 49, Issue:6

    Topics: Aged; Anesthesia Recovery Period; Anesthesia, Local; Blood Pressure; Clonidine; Diazepam; Double-Blind Method; Evoked Potentials, Auditory, Brain Stem; Female; Heart Rate; Humans; Male; Middle Aged; Ophthalmologic Surgical Procedures; Preanesthetic Medication; Time Factors

1994
Oral clonidine premedication attenuates the haemodynamic effects associated with ketamine anaesthetic induction in humans.
    Canadian journal of anaesthesia = Journal canadien d'anesthesie, 1993, Volume: 40, Issue:7

    Topics: Administration, Oral; Adult; Anesthesia, Intravenous; Blood Pressure; Clonidine; Diazepam; Double-Blind Method; Female; Hallucinations; Heart Rate; Hemodynamics; Humans; Ketamine; Male; Patient Satisfaction; Placebos; Preanesthetic Medication; Time Factors

1993
Contrasting effects of clonidine and diazepam on tests of working memory and planning.
    Psychopharmacology, 1995, Volume: 120, Issue:3

    Topics: Adult; Clonidine; Diazepam; Dose-Response Relationship, Drug; Double-Blind Method; Female; Health Planning; Humans; Male; Memory; Task Performance and Analysis; Volunteers

1995
Clonidine and diazepam have differential effects on tests of attention and learning.
    Psychopharmacology, 1995, Volume: 120, Issue:3

    Topics: Adult; Attention; Clonidine; Diazepam; Dose-Response Relationship, Drug; Female; Humans; Learning; Male; Placebo Effect; Task Performance and Analysis; Time Factors; Volunteers

1995
Differential effects of clonidine, haloperidol, diazepam and tryptophan depletion on focused attention and attentional search.
    Psychopharmacology, 1995, Volume: 121, Issue:2

    Topics: Adult; Attention; Clonidine; Diazepam; Haloperidol; Humans; Placebo Effect; Reaction Time; Tryptophan

1995
Oral clonidine premedication reduces vomiting in children after strabismus surgery.
    Canadian journal of anaesthesia = Journal canadien d'anesthesie, 1995, Volume: 42, Issue:11

    Topics: Administration, Oral; Adrenergic alpha-Agonists; Anesthesia, Inhalation; Anti-Inflammatory Agents, Non-Steroidal; Antiemetics; Child; Child, Preschool; Clonidine; Diazepam; Diclofenac; Double-Blind Method; Female; Humans; Incidence; Length of Stay; Male; Midazolam; Neuromuscular Nondepolarizing Agents; Pain, Postoperative; Placebos; Postoperative Complications; Preanesthetic Medication; Premedication; Prospective Studies; Strabismus; Vecuronium Bromide; Vomiting

1995
Effects of clonidine and diazepam on the acoustic startle response and on its inhibition by 'prepulses' in man.
    Journal of psychopharmacology (Oxford, England), 1997, Volume: 11, Issue:1

    Topics: Acoustic Stimulation; Adult; Blinking; Clonidine; Diazepam; Double-Blind Method; Electromyography; Flicker Fusion; Humans; Male; Oculomotor Muscles; Reaction Time; Reflex, Startle; Salivation

1997
[Clofelin in the anesthesiological support system for surgical operations].
    Khirurgiia, 1996, Issue:6

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Analgesia, Epidural; Analgesics; Anesthesia, General; Anesthetics, Combined; Anesthetics, General; Anesthetics, Intravenous; Clonidine; Diazepam; Female; Humans; Intraoperative Care; Male; Middle Aged; Pirinitramide; Postoperative Care; Surgical Procedures, Operative

1996
Comparative study of oral clonidine and diazepam as premedicants in children.
    International journal of clinical pharmacology and therapeutics, 1997, Volume: 35, Issue:5

    Topics: Adrenergic alpha-Agonists; Anti-Anxiety Agents; Blood Pressure; Child; Clonidine; Diazepam; Double-Blind Method; Female; Heart Rate; Humans; Male; Premedication

1997
[Influence of preanesthetic medication on the effect of a local anesthetic tape].
    Masui. The Japanese journal of anesthesiology, 1997, Volume: 46, Issue:9

    Topics: Adjuvants, Anesthesia; Administration, Topical; Adult; Aged; Anesthetics, Local; Anti-Anxiety Agents; Catheterization, Peripheral; Clonidine; Diazepam; Drug Interactions; Humans; Lidocaine; Middle Aged; Pain; Preanesthetic Medication; Sympatholytics

1997
[The effects of premedication on induction doses of propofol and hemodynamic responses during induction].
    Masui. The Japanese journal of anesthesiology, 1997, Volume: 46, Issue:10

    Topics: Adult; Atropine; Clonidine; Diazepam; Drug Interactions; Female; Hemodynamics; Humans; Hydroxyzine; Hypnotics and Sedatives; Male; Midazolam; Middle Aged; Preanesthetic Medication; Propofol

1997
Comparison of psychomotor functions and sedation following premedication with oral diazepam and clonidine in children.
    International journal of clinical pharmacology and therapeutics, 1998, Volume: 36, Issue:6

    Topics: Administration, Oral; Anti-Anxiety Agents; Child; Child, Preschool; Clonidine; Conscious Sedation; Diazepam; Double-Blind Method; Female; Humans; Intelligence; Intelligence Tests; Male; Premedication; Prospective Studies; Psychometrics; Psychomotor Performance; Sympatholytics

1998
The effects of clonidine on the fear-inhibited light reflex.
    Journal of psychopharmacology (Oxford, England), 1998, Volume: 12, Issue:2

    Topics: Adult; Anti-Anxiety Agents; Anxiety; Arousal; Clonidine; Diazepam; Double-Blind Method; Electroshock; Fear; Humans; Male; Neural Inhibition; Reflex, Pupillary; Sympatholytics

1998
The effects of preanesthetic oral clonidine on total requirement of propofol for general anesthesia.
    Journal of clinical anesthesia, 1998, Volume: 10, Issue:8

    Topics: Administration, Oral; Adult; Anesthesia, General; Anesthetics, Inhalation; Anesthetics, Intravenous; Anti-Anxiety Agents; Anxiety; Breast Neoplasms; Clonidine; Diazepam; Double-Blind Method; Drug Costs; Female; Fentanyl; Hemodynamics; Humans; Infusions, Intravenous; Intubation, Intratracheal; Lymph Node Excision; Mastectomy, Segmental; Middle Aged; Nitrous Oxide; Oxygen; Placebos; Preanesthetic Medication; Propofol

1998
Pretreatment with oral clonidine attenuates cardiovascular responses to tracheal extubation in children.
    Paediatric anaesthesia, 2000, Volume: 10, Issue:1

    Topics: Administration, Oral; Adrenergic alpha-Agonists; Anesthesia, General; Antiemetics; Antihypertensive Agents; Blood Pressure; Child; Child, Preschool; Clonidine; Diazepam; Double-Blind Method; Female; Heart Rate; Humans; Intubation, Intratracheal; Male; Postoperative Complications; Tachycardia

2000
The efficacy of oral clonidine premedication in the prevention of postoperative vomiting in children following strabismus surgery.
    Paediatric anaesthesia, 2001, Volume: 11, Issue:1

    Topics: Administration, Oral; Adrenergic alpha-Agonists; Anesthetics, Combined; Anesthetics, Inhalation; Anesthetics, Intravenous; Antiemetics; Child; Child, Preschool; Clonidine; Diazepam; Double-Blind Method; Female; Humans; Male; Nitrous Oxide; Postoperative Nausea and Vomiting; Preanesthetic Medication; Propofol; Prospective Studies; Strabismus

2001
[Potentiation of local anesthesia in endonasal surgery].
    Vestnik otorinolaringologii, 2001, Issue:1

    Topics: Adolescent; Adult; Analgesics; Anesthetics, Intravenous; Anesthetics, Local; Clonidine; Diazepam; Drug Synergism; Humans; Nasal Septum; Procaine

2001
Effects of clonidine and diazepam on prepulse inhibition of the acoustic startle response and the N1/P2 auditory evoked potential in man.
    Journal of psychopharmacology (Oxford, England), 2001, Volume: 15, Issue:4

    Topics: Acoustic Stimulation; Adolescent; Adrenergic alpha-Agonists; Adult; Affect; Anti-Anxiety Agents; Clonidine; Diazepam; Double-Blind Method; Electromyography; Evoked Potentials, Auditory; Hemodynamics; Humans; Male; Oculomotor Muscles; Reflex, Startle; Salivation

2001
Intrathecal and oral clonidine as prophylaxis for postoperative alcohol withdrawal syndrome: a randomized double-blinded study.
    Anesthesia and analgesia, 2004, Volume: 98, Issue:3

    Topics: Administration, Oral; Adrenergic alpha-Agonists; Aged; Alcoholism; Anesthesia; Central Nervous System Depressants; Clonidine; Diazepam; Double-Blind Method; Ethanol; Hemodynamics; Humans; Hypnotics and Sedatives; Injections, Spinal; Male; Middle Aged; Postoperative Complications; Psychomotor Agitation; Respiratory Mechanics; Substance Withdrawal Syndrome; Transurethral Resection of Prostate

2004
Oral clonidine pre-treatment and diazepam/meperidine sedation.
    Journal of dental research, 2006, Volume: 85, Issue:9

    Topics: Administration, Oral; Adrenergic alpha-Agonists; Adult; Analgesics, Opioid; Anesthesia, Dental; Anesthetics, Intravenous; Blood Pressure; Clonidine; Conscious Sedation; Cross-Over Studies; Diazepam; Electroencephalography; Female; Humans; Likelihood Functions; Male; Meperidine; Middle Aged; Preanesthetic Medication; Respiration; Statistics, Nonparametric; Surveys and Questionnaires

2006
Sedative and cardiovascular effects of midazolam and diazepam alone or combined with clonidine in patients undergoing hemodynamic studies for suspected coronary artery disease.
    Arquivos brasileiros de cardiologia, 2007, Volume: 89, Issue:6

    Topics: Adolescent; Adrenergic alpha-Agonists; Adult; Aged; Aged, 80 and over; Analysis of Variance; Blood Pressure; Cineangiography; Clonidine; Conscious Sedation; Coronary Disease; Diazepam; Double-Blind Method; Female; Heart Rate; Hemodynamics; Humans; Hypnotics and Sedatives; Male; Midazolam; Middle Aged; Monitoring, Physiologic; Prospective Studies

2007
Lofexidine versus diazepam for the treatment of opioid withdrawal syndrome: A double-blind randomized clinical trial in Singapore.
    Journal of substance abuse treatment, 2018, Volume: 91

    Topics: Adrenergic alpha-2 Receptor Agonists; Adult; Clonidine; Craving; Diazepam; Double-Blind Method; Female; Humans; Hypnotics and Sedatives; Male; Middle Aged; Opioid-Related Disorders; Pupil; Singapore; Substance Withdrawal Syndrome

2018
The efficacy and safety of an adapted opioid-free anesthesia regimen versus conventional general anesthesia in gynecological surgery for low-resource settings: a randomized pilot study.
    BMC anesthesiology, 2022, 10-24, Volume: 22, Issue:1

    Topics: Analgesics, Opioid; Anesthesia, General; Clonidine; Dexamethasone; Dexmedetomidine; Diazepam; Female; Fentanyl; Gynecologic Surgical Procedures; Humans; Isoflurane; Ketamine; Lidocaine; Magnesium Sulfate; Pain, Postoperative; Pilot Projects; Propofol; Rocuronium; Saline Solution

2022

Other Studies

134 other study(ies) available for diazepam and clonidine

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
5-Aryl-3-(alkylthio)-4H-1,2,4-triazoles as selective antagonists of strychnine-induced convulsions and potential antispastic agents.
    Journal of medicinal chemistry, 1994, Jan-07, Volume: 37, Issue:1

    Topics: Animals; Anticonvulsants; Cerebellum; Cerebral Cortex; Chlorides; Electroshock; Flumazenil; Male; Mice; Molecular Structure; Muscle Spasticity; Paralysis; Rats; Rats, Sprague-Dawley; Seizures; Structure-Activity Relationship; Strychnine; Triazoles

1994
Predicting blood-brain barrier permeation from three-dimensional molecular structure.
    Journal of medicinal chemistry, 2000, Jun-01, Volume: 43, Issue:11

    Topics: Blood-Brain Barrier; Databases, Factual; Models, Chemical; Molecular Conformation; Multivariate Analysis; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
ElogD(oct): a tool for lipophilicity determination in drug discovery. 2. Basic and neutral compounds.
    Journal of medicinal chemistry, 2001, Jul-19, Volume: 44, Issue:15

    Topics: 1-Octanol; Chromatography, High Pressure Liquid; Pharmaceutical Preparations; Solubility; Water

2001
Prediction of volume of distribution values in humans for neutral and basic drugs using physicochemical measurements and plasma protein binding data.
    Journal of medicinal chemistry, 2002, Jun-20, Volume: 45, Issue:13

    Topics: Blood Proteins; Chemical Phenomena; Chemistry, Physical; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding

2002
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Transdermal penetration behaviour of drugs: CART-clustering, QSPR and selection of model compounds.
    Bioorganic & medicinal chemistry, 2007, Nov-15, Volume: 15, Issue:22

    Topics: Anti-Inflammatory Agents; Cell Membrane Permeability; Cluster Analysis; Drug Evaluation, Preclinical; Humans; Models, Biological; Predictive Value of Tests; Quantitative Structure-Activity Relationship; Regression Analysis; Skin; Skin Absorption

2007
Hologram QSAR model for the prediction of human oral bioavailability.
    Bioorganic & medicinal chemistry, 2007, Dec-15, Volume: 15, Issue:24

    Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Relationship between brain tissue partitioning and microemulsion retention factors of CNS drugs.
    Journal of medicinal chemistry, 2009, Mar-26, Volume: 52, Issue:6

    Topics: Brain; Central Nervous System; Chromatography, Liquid; Emulsions; Mass Spectrometry

2009
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
Computational modeling of novel inhibitors targeting the Akt pleckstrin homology domain.
    Bioorganic & medicinal chemistry, 2009, Oct-01, Volume: 17, Issue:19

    Topics: Antineoplastic Agents; Blood Proteins; Caco-2 Cells; Cell Membrane Permeability; Computer Simulation; Drug Discovery; Drug Screening Assays, Antitumor; Humans; Models, Molecular; Phosphoproteins; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-akt; Quantitative Structure-Activity Relationship

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.
    Toxicology mechanisms and methods, 2008, Volume: 18, Issue:2-3

    Topics:

2008
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Measurement of unbound drug exposure in brain: modeling of pH partitioning explains diverging results between the brain slice and brain homogenate methods.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:3

    Topics: Animals; Biological Transport; Brain; Chemical Phenomena; Dialysis; Hydrogen-Ion Concentration; In Vitro Techniques; Lysosomes; Male; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Tissue Distribution

2011
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
Multifunctional scutellarin-rivastigmine hybrids with cholinergic, antioxidant, biometal chelating and neuroprotective properties for the treatment of Alzheimer's disease.
    Bioorganic & medicinal chemistry, 2015, Feb-15, Volume: 23, Issue:4

    Topics: Acetylcholinesterase; Alzheimer Disease; Animals; Antioxidants; Apigenin; Blood-Brain Barrier; Butyrylcholinesterase; Carbamates; Cell Line; Chelating Agents; Cholinesterase Inhibitors; Cognition; Glucuronates; Humans; Mice; Molecular Docking Simulation; Neuroprotective Agents; Rats

2015
Synthesis and evaluation of 4-hydroxyl aurone derivatives as multifunctional agents for the treatment of Alzheimer's disease.
    Bioorganic & medicinal chemistry, 2016, 05-15, Volume: 24, Issue:10

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Antioxidants; Benzofurans; Blood-Brain Barrier; Chelating Agents; Copper; Humans; Models, Molecular; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Peptide Fragments; Protein Aggregates; Swine

2016
Multitarget drug design strategy against Alzheimer's disease: Homoisoflavonoid Mannich base derivatives serve as acetylcholinesterase and monoamine oxidase B dual inhibitors with multifunctional properties.
    Bioorganic & medicinal chemistry, 2017, 01-15, Volume: 25, Issue:2

    Topics: Acetylcholinesterase; Alzheimer Disease; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Drug Design; Humans; Isoflavones; Mannich Bases; Molecular Docking Simulation; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Structure-Activity Relationship

2017
Aurone Mannich base derivatives as promising multifunctional agents with acetylcholinesterase inhibition, anti-β-amyloid aggragation and neuroprotective properties for the treatment of Alzheimer's disease.
    European journal of medicinal chemistry, 2017, Jan-27, Volume: 126

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Blood-Brain Barrier; Cholinesterase Inhibitors; Drug Design; Electrophorus; Humans; Mannich Bases; Neuroprotective Agents; PC12 Cells; Rats

2017
Design, synthesis and biological evaluation of 4'-aminochalcone-rivastigmine hybrids as multifunctional agents for the treatment of Alzheimer's disease.
    Bioorganic & medicinal chemistry, 2017, 02-01, Volume: 25, Issue:3

    Topics: Acetylcholinesterase; Alzheimer Disease; Animals; Blood-Brain Barrier; Chalcones; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Drug Design; Humans; Molecular Docking Simulation; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Rivastigmine; Structure-Activity Relationship; Swine

2017
DL-3-n-butylphthalide-Edaravone hybrids as novel dual inhibitors of amyloid-β aggregation and monoamine oxidases with high antioxidant potency for Alzheimer's therapy.
    Bioorganic & medicinal chemistry letters, 2017, 02-15, Volume: 27, Issue:4

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Antioxidants; Antipyrine; Benzofurans; Binding Sites; Blood-Brain Barrier; Edaravone; Humans; Hydrogen Bonding; Inhibitory Concentration 50; Molecular Docking Simulation; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Protein Binding; Protein Structure, Tertiary

2017
Multifunctional thioxanthone derivatives with acetylcholinesterase, monoamine oxidases and β-amyloid aggregation inhibitory activities as potential agents against Alzheimer's disease.
    Bioorganic & medicinal chemistry, 2017, 03-15, Volume: 25, Issue:6

    Topics: Acetylcholinesterase; Alzheimer Disease; Amyloid beta-Peptides; Cell Line; Cholinesterase Inhibitors; Humans; Kinetics; Models, Molecular; Monoamine Oxidase Inhibitors; Thioxanthenes; Xanthones

2017
Design, synthesis and evaluation of novel ferulic acid-O-alkylamine derivatives as potential multifunctional agents for the treatment of Alzheimer's disease.
    European journal of medicinal chemistry, 2017, Apr-21, Volume: 130

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Antioxidants; Blood-Brain Barrier; Butyrylcholinesterase; Cholinesterase Inhibitors; Coumaric Acids; Drug Design; Eels; Humans; Memory Disorders; Mice; PC12 Cells; Rats

2017
Design, synthesis and biological evaluation of 3,4-dihydro-2(1H)-quinoline-O-alkylamine derivatives as new multipotent cholinesterase/monoamine oxidase inhibitors for the treatment of Alzheimer's disease.
    Bioorganic & medicinal chemistry, 2017, 06-15, Volume: 25, Issue:12

    Topics: Acetylcholinesterase; Alzheimer Disease; Animals; Blood-Brain Barrier; Butyrylcholinesterase; Cholinesterase Inhibitors; Drug Design; Electrophorus; Humans; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quinolines; Swine

2017
Design, synthesis and biological evaluation of phthalimide-alkylamine derivatives as balanced multifunctional cholinesterase and monoamine oxidase-B inhibitors for the treatment of Alzheimer's disease.
    Bioorganic & medicinal chemistry letters, 2017, 11-15, Volume: 27, Issue:22

    Topics: Alzheimer Disease; Amines; Binding Sites; Blood-Brain Barrier; Cell Line, Tumor; Cell Survival; Cholinesterase Inhibitors; Cholinesterases; Drug Design; Humans; Inhibitory Concentration 50; Kinetics; Molecular Docking Simulation; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Phthalimides; Protein Structure, Tertiary; Structure-Activity Relationship

2017
Design, synthesis and biological evaluation of 2-acetyl-5-O-(amino-alkyl)phenol derivatives as multifunctional agents for the treatment of Alzheimer's disease.
    Bioorganic & medicinal chemistry letters, 2017, 11-15, Volume: 27, Issue:22

    Topics: Acetylcholinesterase; Alzheimer Disease; Animals; Antioxidants; Benzophenones; Binding Sites; Blood-Brain Barrier; Cell Survival; Cholinesterase Inhibitors; Drug Design; Humans; Hydrogen Peroxide; Inhibitory Concentration 50; Molecular Docking Simulation; Monoamine Oxidase; Neuroprotective Agents; PC12 Cells; Permeability; Phenols; Piperazines; Protein Structure, Tertiary; Rats; Structure-Activity Relationship

2017
Discovery of novel propargylamine-modified 4-aminoalkyl imidazole substituted pyrimidinylthiourea derivatives as multifunctional agents for the treatment of Alzheimer's disease.
    European journal of medicinal chemistry, 2018, Jan-01, Volume: 143

    Topics: Acetylcholinesterase; Alzheimer Disease; Animals; Butyrylcholinesterase; Cholinesterase Inhibitors; Cognitive Dysfunction; Dose-Response Relationship, Drug; Drug Discovery; Humans; Imidazoles; Mice; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Pargyline; Propylamines; Pyrimidines; Rats; Scopolamine; Structure-Activity Relationship; Thiourea

2018
Design, synthesis and evaluation of 4'-OH-flurbiprofen-chalcone hybrids as potential multifunctional agents for Alzheimer's disease treatment.
    Bioorganic & medicinal chemistry, 2018, 03-01, Volume: 26, Issue:5

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Antioxidants; Blood-Brain Barrier; Cell Line; Cell Survival; Chalcones; Chelating Agents; Copper; Drug Design; Flurbiprofen; Humans; Lipopolysaccharides; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Nitric Oxide; Peptide Fragments; Recombinant Proteins; Structure-Activity Relationship

2018
Multifunctional 5,6-dimethoxybenzo[d]isothiazol-3(2H)-one-N-alkylbenzylamine derivatives with acetylcholinesterase, monoamine oxidases and β-amyloid aggregation inhibitory activities as potential agents against Alzheimer's disease.
    Bioorganic & medicinal chemistry, 2018, 05-01, Volume: 26, Issue:8

    Topics: Acetylcholinesterase; Alzheimer Disease; Amyloid beta-Peptides; Antioxidants; Benzylamines; Blood-Brain Barrier; Cholinesterase Inhibitors; Drug Design; Humans; Kinetics; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Permeability; Protein Aggregates; Recombinant Proteins; Structure-Activity Relationship; Thiazoles

2018
Design, synthesis and evaluation of vilazodone-tacrine hybrids as multitarget-directed ligands against depression with cognitive impairment.
    Bioorganic & medicinal chemistry, 2018, 07-23, Volume: 26, Issue:12

    Topics: Acetylcholinesterase; Alzheimer Disease; Animals; Blood-Brain Barrier; Butyrylcholinesterase; Cholinesterase Inhibitors; Depression; Drug Design; Ligands; Mice; Permeability; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship; Tacrine; Vilazodone Hydrochloride

2018
Discovery of novel anti-tuberculosis agents with pyrrolo[1,2-a]quinoxaline-based scaffold.
    Bioorganic & medicinal chemistry letters, 2018, 06-15, Volume: 28, Issue:11

    Topics: Antineoplastic Agents; Antitubercular Agents; Cell Line, Tumor; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Drug Discovery; Drug Screening Assays, Antitumor; Humans; Microbial Sensitivity Tests; Molecular Structure; Mycobacterium tuberculosis; Pyrroles; Quinoxalines; Structure-Activity Relationship

2018
Discovery of novel 2,5-dihydroxyterephthalamide derivatives as multifunctional agents for the treatment of Alzheimer's disease.
    Bioorganic & medicinal chemistry, 2018, 12-15, Volume: 26, Issue:23-24

    Topics: Acetylcholinesterase; Alzheimer Disease; Amyloid beta-Peptides; Animals; Anti-Inflammatory Agents, Non-Steroidal; Antioxidants; Butyrylcholinesterase; Chelating Agents; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Drug Discovery; Humans; Models, Molecular; Molecular Structure; Peptide Fragments; Phthalimides; Protein Aggregates; Structure-Activity Relationship

2018
Discovery of 4'-OH-flurbiprofen Mannich base derivatives as potential Alzheimer's disease treatment with multiple inhibitory activities.
    Bioorganic & medicinal chemistry, 2019, 03-15, Volume: 27, Issue:6

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Antioxidants; Blood-Brain Barrier; Cell Line; Cholinesterase Inhibitors; Drug Design; Drug Discovery; Electrophorus; Flurbiprofen; Humans; Mannich Bases; Molecular Docking Simulation; Peptide Fragments; Protein Aggregates; Rats; Swine

2019
Design, synthesis, in-silico and biological evaluation of novel chalcone-O-carbamate derivatives as multifunctional agents for the treatment of Alzheimer's disease.
    European journal of medicinal chemistry, 2019, Sep-15, Volume: 178

    Topics: Acetylcholinesterase; Alzheimer Disease; Amyloid beta-Peptides; Animals; Blood-Brain Barrier; Butyrylcholinesterase; Chalcones; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Drug Design; Eels; Female; Horses; Humans; Male; Maze Learning; Mice; Mice, Inbred Strains; Models, Molecular; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Peptide Fragments; Protein Aggregates; Rats; Structure-Activity Relationship

2019
Design, synthesis, in-silico and biological evaluation of novel chalcone derivatives as multi-function agents for the treatment of Alzheimer's disease.
    European journal of medicinal chemistry, 2019, Oct-15, Volume: 180

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Butyrylcholinesterase; Chalcone; Cholinesterase Inhibitors; Drug Design; Eels; Horses; Humans; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Neuroprotective Agents; Peptide Fragments; Protein Aggregates

2019
The development of 2-acetylphenol-donepezil hybrids as multifunctional agents for the treatment of Alzheimer's disease.
    Bioorganic & medicinal chemistry letters, 2019, 10-01, Volume: 29, Issue:19

    Topics: Alzheimer Disease; Cholinesterase Inhibitors; Cholinesterases; Donepezil; Drug Design; Drug Development; Humans; Kinetics; Models, Molecular; Molecular Docking Simulation; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Structure-Activity Relationship

2019
Development of chalcone-O-alkylamine derivatives as multifunctional agents against Alzheimer's disease.
    European journal of medicinal chemistry, 2019, Dec-01, Volume: 183

    Topics: Acetylcholinesterase; Alzheimer Disease; Amyloid beta-Peptides; Animals; Antioxidants; Biological Transport; Blood-Brain Barrier; Butyrylcholinesterase; Chalcones; Chelating Agents; Cholinesterase Inhibitors; Coordination Complexes; Copper; Drug Design; Female; Humans; Male; Memory Disorders; Mice; Molecular Docking Simulation; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Neuroprotective Agents; Protein Binding; Scopolamine; Structure-Activity Relationship

2019
Stress-induced alterations of cyclic nucleotide levels in brain: effects of centrally acting drugs.
    Psychopharmacology, 1977, May-09, Volume: 52, Issue:3

    Topics: Aminooxyacetic Acid; Animals; Brain; Brain Chemistry; Chlorpromazine; Clonidine; Cyclic AMP; Cyclic GMP; Diazepam; Diphenhydramine; Haloperidol; Indomethacin; Male; Mice; Pentobarbital; Phentolamine; Propanolamines; Propranolol; Reserpine; Stress, Physiological

1977
Review: the significance and management of raised blood pressure in pregnancy.
    The Australian & New Zealand journal of obstetrics & gynaecology, 1979, Volume: 19, Issue:1

    Topics: Adrenergic beta-Antagonists; Adult; Antihypertensive Agents; Chlormethiazole; Clonidine; Diazepam; Diazoxide; Diuretics; Female; Heparin; Humans; Hydralazine; Hypertension; Methyldopa; Pregnancy; Pregnancy Complications, Cardiovascular

1979
[Detoxication of heroin addicts in the area of Genoa].
    La Clinica terapeutica, 1979, Dec-31, Volume: 91, Issue:6

    Topics: Adolescent; Adult; Amino Acids; Clonidine; Diazepam; Female; Fructose; Heroin Dependence; Humans; Male; Methadone; ortho-Aminobenzoates; Substance Withdrawal Syndrome; Sulpiride; Vitamins

1979
Transitory decrease in platelet monoamine-oxidase activity during migraine attacks.
    Lancet (London, England), 1977, Feb-19, Volume: 1, Issue:8008

    Topics: Adolescent; Adult; Aspirin; Blood Platelets; Blood Proteins; Child; Child, Preschool; Clonidine; Diazepam; Ergotamine; Female; Humans; Male; Middle Aged; Migraine Disorders; Monoamine Oxidase; Tyramine

1977
Roberts's syndrome and clonidine.
    Journal of medical genetics, 1979, Volume: 16, Issue:6

    Topics: Abnormalities, Drug-Induced; Abnormalities, Multiple; Cleft Lip; Cleft Palate; Clonidine; Diazepam; Ectromelia; Female; Humans; Hypertension; Infant, Newborn; Male; Maternal-Fetal Exchange; Pregnancy; Pregnancy Complications, Cardiovascular; Syndrome

1979
Possible involvement of GABA mechanisms in central cardiovascular and respiratory control. Studies on the interaction between diazepam, picrotoxin and clonidine.
    Medical biology, 1977, Volume: 55, Issue:6

    Topics: Aminobutyrates; Animals; Blood Pressure; Clonidine; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; gamma-Aminobutyric Acid; Heart Rate; Injections, Intraperitoneal; Injections, Intravenous; Injections, Intraventricular; Male; Picrotoxin; Rats; Respiration

1977
[Pharmacologic analysis of the cholinergic vasodilation in unanesthetized animals].
    Fiziologicheskii zhurnal SSSR imeni I. M. Sechenova, 1978, Volume: 64, Issue:7

    Topics: Animals; Blood Pressure; Cats; Cholinergic Fibers; Clonidine; Corpus Callosum; Diazepam; Hypothalamus; Iliac Artery; Norepinephrine; Reserpine; Vasodilation

1978
[Influence of the administration of psychopharmacological compounds on the take up time of an alimentary material in the hamster and a study of the associated behaviour (author's transl)].
    Psychopharmacologia, 1975, Jul-23, Volume: 43, Issue:1

    Topics: Animals; Apomorphine; Behavior, Animal; Chlorpromazine; Clonidine; Cricetinae; Dextroamphetamine; Diazepam; Feeding Behavior; Fenfluramine; Humans; Imipramine; Male; Meprobamate; Mesocricetus; Morphine; Motor Activity; Phenobarbital; Piribedil; Psychotropic Drugs; Stereotyped Behavior; Sulpiride; Time Factors

1975
The effect of centrally acting myorelaxants on NMDA receptor-mediated synaptic transmission in the immature rat spinal cord in vitro.
    British journal of pharmacology, 1992, Volume: 107, Issue:2

    Topics: Animals; Baclofen; Clonidine; Diazepam; In Vitro Techniques; Muscle Relaxants, Central; Rats; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Spinal Nerve Roots; Synaptic Transmission; Tetrodotoxin

1992
Effectiveness of alpha 2-adrenergic receptor stimulation in reducing the central toxicity following cholinesterase inhibition.
    Research communications in chemical pathology and pharmacology, 1992, Volume: 75, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Behavior, Animal; Cholinesterase Inhibitors; Clonidine; Diazepam; Dose-Response Relationship, Drug; Guanabenz; Guanfacine; Lethal Dose 50; Male; Motor Activity; Pyridostigmine Bromide; Rats; Rats, Inbred Strains; Soman

1992
Antinociceptive effects of tizanidine, diazepam and eperisone in isolated spinal cord-tail preparations of newborn rat.
    Pain, 1992, Volume: 48, Issue:1

    Topics: Analgesics; Animals; Animals, Newborn; Clonidine; Diazepam; Evoked Potentials; In Vitro Techniques; Muscle Relaxants, Central; Physical Stimulation; Propiophenones; Rats; Rats, Inbred Strains; Reflex; Spinal Cord; Spinal Nerve Roots; Tail; Time Factors

1992
Potentiation of poststartle activity by conditioned fear: effects of anxiolytic and anxiogenic drugs.
    Biological psychiatry, 1991, Apr-01, Volume: 29, Issue:7

    Topics: Animals; Anti-Anxiety Agents; Arousal; Buspirone; Clonidine; Conditioning, Classical; Diazepam; Dose-Response Relationship, Drug; Fear; Male; Rats; Rats, Inbred Strains; Reflex, Startle; Xylazine; Yohimbine

1991
[Effects of transcranial laser irradiation in near infrared range on antinociceptive reactions in mice after administration of diazepam, clopheline and morphine].
    Biulleten' eksperimental'noi biologii i meditsiny, 1991, Volume: 112, Issue:12

    Topics: Animals; Brain; Clonidine; Diazepam; Injections, Intraperitoneal; Lasers; Mice; Morphine; Pain Measurement

1991
Investigations on the binding properties of the nootropic agent pyroglutamic acid.
    Drugs under experimental and clinical research, 1990, Volume: 16, Issue:2

    Topics: Animals; Binding Sites; Brain; Calcium Channel Blockers; Chloride Channels; Clonidine; Diazepam; Dose-Response Relationship, Drug; Glutamates; Glutamic Acid; Guinea Pigs; Male; Membrane Proteins; Mianserin; Pyrrolidinones; Pyrrolidonecarboxylic Acid; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Amino Acid; Receptors, Cell Surface; Receptors, Cholinergic; Receptors, Dopamine; Receptors, GABA-A; Receptors, Glutamate; Receptors, Glycine; Receptors, Histamine; Receptors, Muscarinic; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Purinergic; Receptors, Serotonin; Stereoisomerism

1990
Discriminative stimulus properties of caffeine in the rat: noradrenergic mediation.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine; Adrenergic alpha-Antagonists; Animals; Apomorphine; Avoidance Learning; Caffeine; Clonidine; Diazepam; Discrimination Learning; Male; Norepinephrine; Pentobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Theobromine; Theophylline

1986
Behavioral evidence for the role of noradrenaline in the putative anxiogenic actions of the inverse benzodiazepine receptor agonist methyl-4-ethyl-6,7-dimethoxy-beta-carboline-3-carboxylate.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:1

    Topics: Animals; Carbolines; Chlorpromazine; Clonidine; Conditioning, Operant; Convulsants; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Male; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reference Values; Yohimbine

1989
[Effect of clonidine on the schedule-controlled performance action of two benzodiazepine receptor agonists].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1989, Volume: 24, Issue:1

    Topics: Animals; Bicuculline; Clonidine; Conditioning, Operant; Diazepam; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reinforcement Schedule; Yohimbine

1989
GABAergic agents and clonidine attenuate footshock-induced aggression in mice.
    Methods and findings in experimental and clinical pharmacology, 1989, Volume: 11, Issue:9

    Topics: Aggression; Animals; Baclofen; Clonidine; Diazepam; Electroshock; gamma-Aminobutyric Acid; Male; Mice; Reserpine

1989
Does anxiety underly imidazole-induced behavioural effects in the rat?
    Psychopharmacology, 1989, Volume: 99, Issue:3

    Topics: Animals; Anxiety; Arousal; Behavior, Animal; Blood Pressure; Clonidine; Diazepam; Emotions; Hemodynamics; Imidazoles; Male; Motor Activity; Rats; Rats, Inbred Strains; Social Behavior; Yohimbine

1989
Kainic acid-induced seizures: potentiation by alpha-methyl-p-tyrosine.
    Brain research, 1989, Aug-28, Volume: 495, Issue:2

    Topics: alpha-Methyltyrosine; Animals; Clonidine; Diazepam; Dopamine; Epilepsy; Kainic Acid; Male; Methyltyrosines; Neurons; Norepinephrine; Rats; Rats, Inbred Strains

1989
Noradrenergic mechanisms in mediation of stress-induced hyperalgesia in rats.
    Pain, 1988, Volume: 32, Issue:3

    Topics: Analgesia; Animals; Clonidine; Diazepam; Norepinephrine; Pain; Rats; Receptors, Adrenergic, alpha; Stress, Physiological; Vibration; Yohimbine

1988
[Effects of agonist and inverse agonist of central benzodiazepine receptors on discriminative yohimbine stimulation].
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1988, Volume: 9, Issue:6

    Topics: Animals; Carbolines; Clonidine; Convulsants; Diazepam; Discrimination Learning; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Yohimbine

1988
Does alprazolam, in contrast to diazepam, activate alpha 2-adrenoceptors involved in the regulation of rat growth hormone secretion?
    Life sciences, 1986, Apr-21, Volume: 38, Issue:16

    Topics: Adrenergic alpha-Antagonists; Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Clonidine; Diazepam; Dioxanes; Growth Hormone; Idazoxan; Kinetics; Male; Rats; Receptors, Adrenergic, alpha; Reserpine; Yohimbine

1986
Reversal by alpha-2 agonists of diazepam withdrawal hyperactivity in rats.
    Psychopharmacology, 1986, Volume: 90, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Azepines; Clonidine; Diazepam; Guanfacine; Guanidines; Male; Motor Activity; Phenylacetates; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome; Yohimbine

1986
Effects of neuroleptic drugs, clonidine and lithium on the expression of conditioned behavioral excitation in rats.
    Psychopharmacology, 1987, Volume: 92, Issue:3

    Topics: Animals; Antipsychotic Agents; Appetitive Behavior; Arousal; Clonidine; Conditioning, Classical; Diazepam; Dose-Response Relationship, Drug; Lithium; Male; Motor Activity; Rats; Rats, Inbred Strains

1987
The anxiolytic and anxiogenic actions of ethanol in a mouse model.
    The Journal of pharmacy and pharmacology, 1988, Volume: 40, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Body Weight; Clonidine; Diazepam; Drinking; Ethanol; Exploratory Behavior; Male; Mice; Substance Withdrawal Syndrome; Tiapamil Hydrochloride

1988
Behavioral evidence for the role of noradrenaline in putative anxiolytic and sedative effects of benzodiazepines.
    Psychopharmacology, 1988, Volume: 95, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Bicuculline; Clonidine; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Hypnotics and Sedatives; Male; Norepinephrine; Rats; Rats, Inbred Strains; Reinforcement Schedule; Yohimbine

1988
Neuropharmacological antagonism of the beta-carboline-induced "anxiety" response in rhesus monkeys.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1985, Volume: 5, Issue:2

    Topics: Adrenocorticotropic Hormone; Animals; Anxiety; Behavior, Animal; Blood Pressure; Carbolines; Clonidine; Cyproheptadine; Diazepam; Epinephrine; Heart Rate; Humans; Hydrocortisone; Indoles; Isoxazoles; Macaca mulatta; Male; Norepinephrine; Propranolol

1985
Some anticonvulsant drugs alter monoamine-mediated behaviour in mice in ways similar to electroconvulsive shock; implications for antidepressant therapy.
    British journal of pharmacology, 1985, Volume: 84, Issue:2

    Topics: 5-Hydroxytryptophan; Animals; Anticonvulsants; Antidepressive Agents; Apomorphine; Behavior, Animal; Biogenic Amines; Clonidine; Diazepam; Electroshock; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred C57BL; Motor Activity; Radioligand Assay; Receptors, Adrenergic, beta; Receptors, Serotonin; Valproic Acid

1985
Alpha 2-adrenoceptors modulate kainic acid-induced limbic seizures.
    European journal of pharmacology, 1985, Jul-17, Volume: 113, Issue:2

    Topics: Animals; Brain Chemistry; Clonidine; Diazepam; Haloperidol; Kainic Acid; Male; Metergoline; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Seizures

1985
Purine effects on (3H)-clonidine binding to rat brain.
    Biochemical pharmacology, 1986, May-15, Volume: 35, Issue:10

    Topics: Animals; Brain; Clonidine; Diazepam; In Vitro Techniques; Kinetics; Male; Phenylisopropyladenosine; Purines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tritium; Verapamil

1986
Interaction of the pesticide chlordimeform with adrenergic receptors in mouse brain: an in vitro study.
    Archives of toxicology, 1987, Volume: 59, Issue:5

    Topics: Amidines; Animals; Brain Chemistry; Chlorphenamidine; Clonidine; Diazepam; Dihydroalprenolol; Dioxanes; In Vitro Techniques; Kinetics; Male; Mice; Muscimol; Proteins; Quinuclidinyl Benzilate; Receptors, Adrenergic; Receptors, GABA-A

1987
Benzodiazepines, plasma MHPG and alpha-2-adrenoceptor function in man.
    International clinical psychopharmacology, 1987, Volume: 2, Issue:2

    Topics: Brain; Clonidine; Diazepam; Glycols; Humans; Male; Methoxyhydroxyphenylglycol; Psychomotor Performance; Receptors, Adrenergic; Substance Withdrawal Syndrome

1987
Clonidine--induced behavioural despair in mice: reversal by antidepressants.
    Psychopharmacology, 1986, Volume: 89, Issue:2

    Topics: Animals; Antidepressive Agents; Antidepressive Agents, Tricyclic; Azepines; Clonidine; Depression; Diazepam; Guanfacine; Guanidines; Lithium; Male; Phenylacetates; Rats; Rats, Inbred Strains; Tranylcypromine; Yohimbine

1986
Neuronal source of plasma dihydroxyphenylalanine.
    The Journal of clinical endocrinology and metabolism, 1987, Volume: 64, Issue:4

    Topics: Adolescent; Adrenalectomy; Adrenergic Fibers; Adult; Aged; alpha-Methyltyrosine; Anesthesia; Animals; Catecholamines; Clonidine; Diazepam; Dihydroxyphenylalanine; Dogs; Female; Humans; Isoproterenol; Macaca fascicularis; Male; Methyltyrosines; Middle Aged; Sympathectomy; Trimethaphan; Yohimbine

1987
Distinctive behavioral effects of the pyrazoloquinoline CGS 8216 in squirrel monkeys.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 29, Issue:4

    Topics: Animals; Behavior, Animal; Benzodiazepines; Clonidine; Diazepam; Flumazenil; Male; Pyrazoles; Saimiri

1988
[Potentiating effect of clonidine on the anxiolytic action of diazepam in a rat social interaction model of anxiety].
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1988, Volume: 9, Issue:2

    Topics: Animals; Anxiety; Behavior, Animal; Clonidine; Diazepam; Drug Synergism; Male; Rats

1988
Opioid withdrawal and naltrexone induction in 48-72 hours with minimal drop-out, using a modification of the naltrexone-clonidine technique.
    The British journal of psychiatry : the journal of mental science, 1988, Volume: 153

    Topics: Adolescent; Adult; Clonidine; Diazepam; Drug Administration Schedule; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Naltrexone; Narcotics; Substance Withdrawal Syndrome; Time Factors

1988
Clonidine in alcohol withdrawal: a clinical report.
    Methods and findings in experimental and clinical pharmacology, 1987, Volume: 9, Issue:10

    Topics: Adult; Alcoholism; Clonidine; Diazepam; Humans; Male; Substance Withdrawal Syndrome

1987
Effects of tizanidine, a centrally acting muscle relaxant, on motor systems.
    General pharmacology, 1986, Volume: 17, Issue:2

    Topics: Animals; Cerebral Cortex; Chlorpromazine; Clonidine; Decerebrate State; Diazepam; Male; Membranes; Motor Neurons; Muscle Relaxants, Central; Neuromuscular Junction; Neurons, Afferent; Rats; Rats, Inbred Strains; Reflex; Spinal Cord

1986
Mechanisms by which picrotoxin and a high dose of diazepam elevate plasma corticosterone level.
    Neuroendocrinology, 1986, Volume: 43, Issue:3

    Topics: Animals; Apomorphine; Atropine; Bicuculline; Clonidine; Corticosterone; Dexamethasone; Diazepam; Drug Interactions; Female; Haloperidol; Picrotoxin; Rats; Rats, Inbred Strains; Yohimbine

1986
Effect of chronic administration of alprazolam and adinazolam on clonidine- or apomorphine-induced aggression in laboratory rodents.
    Neuropharmacology, 1986, Volume: 25, Issue:7

    Topics: Aggression; Alprazolam; Animals; Anti-Anxiety Agents; Apomorphine; Benzodiazepines; Clonidine; Desipramine; Diazepam; Drug Interactions; Male; Mice; Rats; Rats, Inbred Strains

1986
Neuropharmacological investigations in the stiff-man syndrome.
    Journal of neurology, 1986, Volume: 233, Issue:6

    Topics: Adrenergic Fibers; Central Nervous System Diseases; Clonidine; Diazepam; Female; Humans; Methamphetamine; Muscle Rigidity; Reflex, Abnormal; Reserpine; Syndrome

1986
Electrophysiological analysis of the mode of action of muscle relaxants in spasticity.
    Annals of neurology, 1985, Volume: 17, Issue:1

    Topics: Baclofen; Clonidine; Diazepam; Electrophysiology; Ethanolamines; Female; Humans; Male; Middle Aged; Muscle Relaxants, Central; Muscle Spasticity

1985
Clonidine in essential tremor: preliminary observations from an open trial.
    Journal of neurology, 1985, Volume: 232, Issue:1

    Topics: Aged; Clonidine; Diazepam; Female; Handwriting; Humans; Levodopa; Male; Middle Aged; Piribedil; Tremor

1985
A critical survey of drugs used in the treatment of hypertensive crises of pregnancy.
    The Medical journal of Australia, 1974, Aug-17, Volume: 2, Issue:7

    Topics: Anesthesia, Conduction; Anesthesia, Obstetrical; Barbiturates; Chlormethiazole; Clonidine; Diazepam; Diazoxide; Diuretics; Eclampsia; Female; Ferricyanides; Humans; Hydralazine; Magnesium; Paraldehyde; Pentolinium Tartrate; Pre-Eclampsia; Pregnancy; Reserpine; Sodium Chloride Symporter Inhibitors; Trimethaphan; Veratrum Alkaloids

1974
Involvement of adenosine receptor activities in aggressive responses produced by clonidine in mice.
    Psychopharmacology, 1984, Volume: 83, Issue:4

    Topics: Adenosine; Aggression; Animals; Apomorphine; Bicuculline; Clonidine; Diazepam; Dipyridamole; Humans; Male; Mice; Receptors, Cell Surface; Receptors, Purinergic; Theophylline

1984
The ethanol withdrawal syndrome in the rat: effects of drug treatment on adrenal gland and urinary catecholamines.
    Substance and alcohol actions/misuse, 1982, Volume: 3, Issue:5

    Topics: Adrenal Glands; Alcohol Withdrawal Delirium; Animals; Catecholamines; Clonidine; Dexamethasone; Diazepam; Hexamethonium; Hexamethonium Compounds; Humans; Male; Propranolol; Psychoses, Alcoholic; Rats; Rats, Inbred Strains; Sympathetic Nervous System

1982
Effects of alpha-adrenoceptor agonists and antagonists in a maze-exploration model of 'fear'-motivated behaviour.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 327, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenocorticotropic Hormone; Amobarbital; Animals; Clonidine; Diazepam; Exploratory Behavior; Fear; Male; Models, Psychological; Picrotoxin; Prazosin; Rats

1984
Pharmacological aspects of metaldehyde poisoning in mice.
    Journal of veterinary pharmacology and therapeutics, 1982, Volume: 5, Issue:1

    Topics: Acetaldehyde; Animals; Brain; Clonidine; Diazepam; Female; Hydroxyindoleacetic Acid; Male; Mice; Mice, Inbred Strains; Molluscacides; Norepinephrine; Seizures; Serotonin

1982
Clonidine prevents methylxanthine stimulation of norepinephrine metabolism in rat brain.
    Journal of neurochemistry, 1983, Volume: 40, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Behavior, Animal; Brain; Cerebellum; Clonidine; Diazepam; Hippocampus; Kinetics; Male; Naloxone; Norepinephrine; Rats; Rats, Inbred Strains; Theophylline

1983
Neuropharmacology of 3-isobutylmethylxanthine: effects on central noradrenergic systems in vivo.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; 2-Chloroadenosine; Adenosine; Animals; Axons; Brain; Clonidine; Diazepam; Dihydroxyphenylalanine; Hydroxylation; Male; Methoxyhydroxyphenylglycol; Neurons; Norepinephrine; Rats; Rats, Inbred Strains; Stimulation, Chemical; Theophylline; Tyrosine 3-Monooxygenase; Yohimbine

1983
Pain-depressing agents and the spinal nociceptive system.
    Arzneimittel-Forschung, 1984, Volume: 34, Issue:9A

    Topics: Analgesics; Animals; Ceruletide; Clonidine; Diazepam; Endorphins; Humans; Morphine; Motor Neurons; Neurons, Afferent; Nociceptors; Pentobarbital; Receptors, GABA-A; Receptors, Opioid; Reflex; Sincalide; Spinal Cord; Substance P; Synapses

1984
Evidence against the involvement of a noradrenergic mechanism in the release by diazepam of novelty-induced hypophagia in rats.
    European journal of pharmacology, 1984, Apr-20, Volume: 100, Issue:2

    Topics: Animals; Anxiety; Clonidine; Diazepam; Drug Interactions; Eating; Guanfacine; Guanidines; Humans; Male; Mice; Norepinephrine; Phenylacetates; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Yohimbine

1984
A benzodiazepine receptor-mediated model of anxiety. Studies in nonhuman primates and clinical implications.
    Archives of general psychiatry, 1984, Volume: 41, Issue:8

    Topics: Animals; Anxiety Disorders; Behavior, Animal; Blood Pressure; Carbolines; Clonidine; Diazepam; Dose-Response Relationship, Drug; Heart Rate; Humans; Hydrocortisone; Indoles; Ligands; Macaca mulatta; Male; Methoxyhydroxyphenylglycol; Models, Biological; Motor Activity; Propranolol; Receptors, Cell Surface; Receptors, GABA-A; Time Factors

1984
Possible mechanism of digoxin-induced convulsions.
    Psychopharmacology, 1983, Volume: 79, Issue:2-3

    Topics: Animals; Calcium Chloride; Clonidine; Diazepam; Digoxin; Female; gamma-Aminobutyric Acid; Magnesium; Magnesium Chloride; Male; Phenytoin; Piracetam; Potassium Chloride; Rats; Rats, Inbred Strains; Seizures

1983
Bioassay of subjective effects associated with benzodiazepine withdrawal in animals: a novel direction in dependence research.
    NIDA research monograph, 1984, Volume: 49

    Topics: Animals; Benzodiazepinones; Biological Assay; Clonidine; Conditioning, Operant; Diazepam; Discrimination Learning; Flumazenil; Generalization, Stimulus; Humans; Male; Pentobarbital; Pentylenetetrazole; Rats; Substance Withdrawal Syndrome; Substance-Related Disorders

1984
How do tranquilizing agents selectively inhibit conditioned avoidance responding?
    Psychopharmacology, 1984, Volume: 84, Issue:2

    Topics: Animals; Avoidance Learning; Chlordiazepoxide; Clonidine; Conditioning, Operant; Diazepam; Male; Morphine; Rats; Rats, Inbred Strains; Reaction Time; Tranquilizing Agents

1984
Diazepam, alpha and beta neurotransmission modifying drugs and contrast media mortality in mice.
    Acta radiologica: diagnosis, 1984, Volume: 25, Issue:3

    Topics: Animals; Clonidine; Diatrizoate; Diatrizoate Meglumine; Diazepam; Drug Interactions; Female; Lethal Dose 50; Male; Metoprolol; Mice; Phentolamine; Prazosin; Propranolol; Sympatholytics; Sympathomimetics

1984
[Pharmacological analysis of the interactions of emotional-behavioral and hemodynamic reactions].
    Vestnik Akademii meditsinskikh nauk SSSR, 1984, Issue:4

    Topics: Animals; Blood Pressure; Cats; Clonidine; Diazepam; Humans; Motor Activity; Neurotensin; Pressoreceptors; Propranolol; Reflex; Stress, Psychological

1984
The drug treatment of spasticity.
    International rehabilitation medicine, 1983, Volume: 5, Issue:3

    Topics: Baclofen; Clonidine; Dantrolene; Diazepam; Humans; Muscle Spasticity; Parasympatholytics

1983
Behavioral comparison of pentylenetetrazol, clonidine, chlordiazepoxide and diazepam in infant rats.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:6

    Topics: Age Factors; Animals; Animals, Newborn; Behavior, Animal; Chlordiazepoxide; Clonidine; Diazepam; Motor Activity; Pentylenetetrazole; Rats; Rats, Inbred Strains; Seizures

1983
The stiff-man syndrome: new pathophysiological aspects from abnormal exteroceptive reflexes and the response to clomipramine, clonidine, and tizanidine.
    Journal of neurology, neurosurgery, and psychiatry, 1984, Volume: 47, Issue:3

    Topics: Adult; Brain Stem; Clomipramine; Clonidine; Diazepam; Electromyography; Female; Humans; Muscle Rigidity; Muscular Diseases; Physical Stimulation; Reflex, Abnormal; Spasm; Syndrome

1984
Progress report of the NIDA Addiction Research Center.
    NIDA research monograph, 1982, Volume: 41

    Topics: Analgesics; Buprenorphine; Chlordiazepoxide; Clonidine; Diazepam; Humans; Morphine; National Institutes of Health (U.S.); Substance Withdrawal Syndrome; Substance-Related Disorders; Tobacco Use Disorder; Tolmetin; United States

1982
Chloral hydrate anesthesia alters the responsiveness of dorsal raphe neurons to psychoactive drugs.
    Life sciences, 1983, Feb-28, Volume: 32, Issue:9

    Topics: Animals; Brain Stem; Cats; Chloral Hydrate; Clomipramine; Clonidine; Diazepam; Drug Interactions; Electrophysiology; Female; Lysergic Acid Diethylamide; Male; Neurons; Phenoxybenzamine; Psychotropic Drugs; Raphe Nuclei; Wakefulness

1983
Yohimbine induced anxiety and increased noradrenergic function in humans: effects of diazepam and clonidine.
    Life sciences, 1983, Jul-04, Volume: 33, Issue:1

    Topics: Adult; Anxiety; Autonomic Nervous System Diseases; Blood Pressure; Clonidine; Diazepam; Drug Interactions; Female; Humans; Kinetics; Male; Methoxyhydroxyphenylglycol; Middle Aged; Norepinephrine; Yohimbine

1983
[Clonidine in severe alcohol withdrawal delirium].
    Fortschritte der Medizin, 1983, Jul-14, Volume: 101, Issue:26

    Topics: Alcohol Withdrawal Delirium; Chlormethiazole; Clonidine; Diazepam; Haloperidol; Humans; Monitoring, Physiologic; Pneumonia; Psychoses, Alcoholic; Respiratory Insufficiency

1983
Anti-convulsant activity of diazepam and clonidine on metaldehyde-induced seizures in mice: effects on brain gamma-amino butyric acid concentrations and monoamine oxidase activity.
    Journal of veterinary pharmacology and therapeutics, 1982, Volume: 5, Issue:3

    Topics: Acetaldehyde; Animals; Brain Chemistry; Clonidine; Diazepam; Female; gamma-Aminobutyric Acid; Male; Mice; Monoamine Oxidase; Seizures

1982
[Pharmacological studies of guanabenz: effects of the central nervous system].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1982, Volume: 80, Issue:6

    Topics: Animals; Anticonvulsants; Avoidance Learning; Body Temperature; Brain; Chlorpromazine; Clonidine; Diazepam; Guanabenz; Guanidines; Male; Mice; Muscle Relaxants, Central; Psychomotor Performance; Rabbits; Rats; Rats, Inbred Strains; Sleep

1982
Comparison of hypotensive, orthostatic and sympathetic inhibitory actions of antihypertensive drugs in rats.
    Clinical and experimental hypertension, 1981, Volume: 3, Issue:2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Diazepam; Guanethidine; Heart Rate; Hydralazine; Hypotension; Male; Mecamylamine; Methyldopa; Minoxidil; Phentolamine; Posture; Prazosin; Propranolol; Rats; Reserpine; Sympathetic Nervous System

1981
The effect of some anti-epilepsy drugs on enhancement of the monoamine-mediated behavioural responses following the administration of electroconvulsive shocks to rats.
    European journal of pharmacology, 1981, Sep-11, Volume: 74, Issue:2-3

    Topics: Animals; Anticonvulsants; Apomorphine; Behavior, Animal; Carbamazepine; Clonidine; Diazepam; Dopamine; Electroshock; Lithium; Male; Norepinephrine; Phenytoin; Rats; Rats, Inbred Strains; Serotonin

1981
Management of alcohol withdrawal.
    Mayo Clinic proceedings, 1995, Volume: 70, Issue:12

    Topics: Adrenergic alpha-Agonists; Alcoholism; Anti-Anxiety Agents; Clonidine; Diazepam; Humans; Midazolam; Substance Withdrawal Syndrome

1995
The profiles of interaction of yohimbine with anxiolytic and putative anxiolytic agents to modify 5-HT release in the frontal cortex of freely-moving rats.
    British journal of pharmacology, 1993, Volume: 110, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Clonidine; Dialysis; Diazepam; Drug Interactions; Extracellular Space; Frontal Lobe; Hydroxyindoleacetic Acid; Male; Ondansetron; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Yohimbine

1993
Discriminative stimulus properties of diazepam and the novel anxiolytic agent 1-amino-5-bromouracil in rats.
    Arzneimittel-Forschung, 1994, Volume: 44, Issue:10

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Bromouracil; Clonidine; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Generalization, Stimulus; Imipramine; Male; Rats; Rats, Wistar

1994
The effects of central myorelaxants on synaptically-evoked primary afferent depolarization in the immature rat spinal cord in vitro.
    British journal of pharmacology, 1994, Volume: 111, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Adrenergic alpha-Agonists; Animals; Baclofen; Clonidine; Diazepam; Electric Stimulation; Evoked Potentials; Ganglia, Spinal; In Vitro Techniques; Muscle Relaxants, Central; Nerve Fibers; Neurons, Afferent; Rats; Receptors, Adrenergic, alpha-2; Spinal Cord; Synapses

1994
Local cerebral glucose utilization in rats with decerebrate rigidity and effects of centrally acting muscle relaxants, diazepam and tizanidine.
    Biological & pharmaceutical bulletin, 1993, Volume: 16, Issue:1

    Topics: Animals; Cerebellar Nuclei; Clonidine; Decerebrate State; Deoxyglucose; Diazepam; Glucose; Male; Muscle Relaxants, Central; Rats; Rats, Wistar; Vestibular Nuclei

1993
Alcohol withdrawal: a nationwide survey of inpatient treatment practices.
    Journal of general internal medicine, 1995, Volume: 10, Issue:9

    Topics: Adrenergic beta-Antagonists; Alcoholism; Barbiturates; Benzodiazepines; Chlordiazepoxide; Clonidine; Data Collection; Diazepam; Drug Administration Schedule; Hypnotics and Sedatives; Inpatients; Lorazepam; Oxazepam; Phenytoin; Substance Withdrawal Syndrome

1995
Alprazolam, diazepam, yohimbine, clonidine: in vivo CA1 hippocampal norepinephrine and serotonin release profiles under chloral hydrate anesthesia.
    Progress in neuro-psychopharmacology & biological psychiatry, 1997, Volume: 21, Issue:7

    Topics: Adrenergic alpha-Antagonists; Alprazolam; Anesthetics, Intravenous; Animals; Anti-Anxiety Agents; Anxiety; Chloral Hydrate; Clonidine; Diazepam; Hippocampus; Male; Microelectrodes; Rats; Rats, Sprague-Dawley; Serotonin; Time Factors; Yohimbine

1997
Cardiopulmonary effects of clonidine, diazepam and the peripheral alpha 2 adrenoceptor agonist ST-91 in conscious sheep.
    Journal of veterinary pharmacology and therapeutics, 1997, Volume: 20, Issue:6

    Topics: Adjuvants, Anesthesia; Adrenergic alpha-Agonists; Animals; Clonidine; Diazepam; Female; Hemodynamics; Hypoxia; Pulmonary Gas Exchange; Respiration; Sheep

1997
Excessive cerebrocortical release of acetylcholine induced by NMDA antagonists is reduced by GABAergic and alpha2-adrenergic agonists.
    Molecular psychiatry, 1999, Volume: 4, Issue:4

    Topics: Acetylcholine; Adrenergic alpha-Agonists; Animals; Cerebral Cortex; Clonidine; Diazepam; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Female; Ketamine; Microdialysis; Pentobarbital; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, GABA; Receptors, N-Methyl-D-Aspartate

1999
Treatment with the noradrenergic alpha-2 agonist clonidine, but not diazepam, improves spatial working memory in normal young rhesus monkeys.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1999, Volume: 21, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Behavior, Animal; Clonidine; Cognition; Diazepam; Dose-Response Relationship, Drug; Female; Hypnotics and Sedatives; Idazoxan; Macaca mulatta; Memory; Reaction Time; Receptors, Adrenergic, alpha-2; Reserpine; Space Perception

1999
Central benzodiazepine involvement in clonidine cardiovascular actions.
    Canadian journal of physiology and pharmacology, 1999, Volume: 77, Issue:11

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Atropine Derivatives; Blood Pressure; Carbolines; Cardiovascular Agents; Clonidine; Diazepam; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Heart Rate; Infusions, Intravenous; Injections, Intraventricular; Male; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, GABA-A; Stereotaxic Techniques; Time Factors; Yohimbine

1999
[A method for potentiation of local anesthesia for tooth removal and pulp extirpation].
    Stomatologiia, 2002, Volume: 81, Issue:4

    Topics: Adrenergic alpha-Agonists; Analgesics, Non-Narcotic; Anesthesia, Dental; Anesthesia, Local; Anti-Anxiety Agents; Clonidine; Dental Anxiety; Dental Pulp Devitalization; Diazepam; Drug Synergism; Drug Therapy, Combination; Humans; Preanesthetic Medication; Tooth Extraction

2002
Effects of premedication medicines on the formation of the CYP3A4-dependent metabolite of ropivacaine, 2', 6'-Pipecoloxylidide, on human liver microsomes in vitro.
    Basic & clinical pharmacology & toxicology, 2006, Volume: 98, Issue:2

    Topics: Amides; Anesthetics, Local; Bupivacaine; Cells, Cultured; Cimetidine; Clonidine; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Diazepam; Drug Interactions; Humans; Lidocaine; Microsomes, Liver; Midazolam; Premedication; Ropivacaine; Thiamylal; Vecuronium Bromide

2006
PRES: posterior or potentially reversible encephalopathy syndrome?
    Neurological sciences : official journal of the Italian Neurological Society and of the Italian Society of Clinical Neurophysiology, 2006, Volume: 27, Issue:3

    Topics: Adult; Anti-Inflammatory Agents; Anticonvulsants; Antihypertensive Agents; Brain; Brain Diseases; Clonidine; Dexamethasone; Diazepam; Diuretics, Osmotic; Eclampsia; Female; Humans; Magnesium Sulfate; Magnetic Resonance Imaging; Mannitol; Nifedipine; Pregnancy; Seizures

2006
The involvement of noradrenergic mechanisms in the suppressive effects of diazepam on the hypothalamic-pituitary-adrenal axis activity in female rats.
    Croatian medical journal, 2012, Volume: 53, Issue:3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic Neurons; Adrenocorticotropic Hormone; alpha-Methyltyrosine; Analysis of Variance; Animals; Antihypertensive Agents; Clonidine; Corticosterone; Diazepam; Disease Models, Animal; Enzyme Inhibitors; Female; Hypnotics and Sedatives; Rats; Rats, Wistar; Reserpine; Yohimbine

2012
A Case of Stiff Person Syndrome: Immunomodulatory Effect of Benzodiazepines: Successful Rituximab and Tizanidine Therapy.
    Medicine, 2015, Volume: 94, Issue:23

    Topics: Adult; Antibodies, Monoclonal, Murine-Derived; Benzodiazepines; Clonidine; Diazepam; Drug Therapy, Combination; Female; Glutamate Decarboxylase; Humans; Immunologic Factors; Muscle Relaxants, Central; Remission Induction; Rituximab; Stiff-Person Syndrome

2015
Pediatric Herpes Simplex Virus Encephalitis Complicated by N-Methyl-D-aspartate Receptor Antibody Encephalitis.
    Journal of the Pediatric Infectious Diseases Society, 2015, Volume: 4, Issue:2

    Topics: Acyclovir; Anti-N-Methyl-D-Aspartate Receptor Encephalitis; Antiviral Agents; Autoantibodies; Clonidine; Diazepam; Encephalitis, Herpes Simplex; Encephalomalacia; Female; Fever; Humans; Immunocompromised Host; Immunosuppression Therapy; Infant; Leukoencephalopathies; Movement Disorders; Neurological Rehabilitation; Pakistan; Paresis; Phenobarbital; Phenytoin; Plasmapheresis; Receptors, N-Methyl-D-Aspartate; Seizures; Trihexyphenidyl; United Kingdom; Valproic Acid

2015
Intranasal dexmedetomidine for adrenergic crisis in familial dysautonomia.
    Clinical autonomic research : official journal of the Clinical Autonomic Research Society, 2017, Volume: 27, Issue:4

    Topics: Administration, Intranasal; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adult; Anxiety; Autonomic Nervous System Diseases; Blood Pressure; Clonidine; Dexmedetomidine; Diazepam; Drug Resistance; Dysautonomia, Familial; Female; GABA Modulators; Heart Rate; Humans; Male; Pneumonia, Mycoplasma; Young Adult

2017
Pharmacological management of abnormal tone and movement in cerebral palsy.
    Archives of disease in childhood, 2019, Volume: 104, Issue:8

    Topics: Adolescent; Baclofen; Botulinum Toxins; Cerebral Palsy; Child; Child Health Services; Child, Preschool; Clonidine; Diazepam; Dystonia; Female; Humans; Infant; Male; Medical Records; Muscle Relaxants, Central; Muscle Spasticity; Prospective Studies; State Medicine; Trihexyphenidyl; United Kingdom

2019