diazepam and brotizolam

diazepam has been researched along with brotizolam in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-199012 (54.55)18.7374
1990's2 (9.09)18.2507
2000's6 (27.27)29.6817
2010's1 (4.55)24.3611
2020's1 (4.55)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Anzini, M; Brogi, S; Cappelli, A; Chemi, G; Di Capua, A; Di Cesare Mannelli, L; Garofalo, A; Ghelardini, C; Giorgi, G; Grande, F; Matucci, R; Paolino, M; Reale, A1
Ejlersen, E; Espersen, K; Krintel, JJ; Laub, M1
Nader, MA; Winger, G; Woods, JH; Woolverton, WL1
Koot, M; Van Duin, CT; Van Miert, AS1
Böke-Kuhn, K; Danneberg, PB; Hommer, D; Kuhn, FJ; Lehr, E; Paul, SM; Skolnick, P; Weber, KH1
Bechtel, WD; Ensinger, HA; Mierau, J1
Kuhn, FJ1
Böke-Kuhn, K; Danneberg, P; Lehr, E1
Bechtel, WD; Stockhaus, K1
Stockhaus, K1
Böke-Kuhn, K; Knappen, F1
Apfelbaum, M; Betoulle, D; Falcou, R; Seyrig, JA1
Shibata, K; Shibata, S; Ueki, S; Watanabe, S; Yamamoto, T1
Inagaki, C; Ishiko, J; Takaori, S1
Nicholson, AN; Pascoe, PA; Stone, BM1
Kishore, K; Saraf, MK; Sharma, A; Singh, M; Thomas, KM1
Katsura, M; Kurokawa, K; Ohkuma, S; Shibasaki, M; Tsujimura, A1
Elkobi, A; Jacobson-Pick, S; Richter-Levin, G; Rosenblum, K; Vander, S1
Kamei, C; Nishino, T; Takechi, K; Takeuchi, T1

Trials

2 trial(s) available for diazepam and brotizolam

ArticleYear
Sublingual premedication with brotizolam.
    Acta anaesthesiologica Scandinavica, 1992, Volume: 36, Issue:8

    Topics: Administration, Oral; Administration, Sublingual; Adult; Anesthesia, General; Anxiety; Azepines; Diazepam; Double-Blind Method; Female; Humans; Hypnotics and Sedatives; Middle Aged; Patient Satisfaction; Placebos; Preanesthetic Medication; Reaction Time

1992
Studies on sleep and performance with a triazolo-1, 4-thienodiazepine (brotizolam).
    British journal of clinical pharmacology, 1980, Volume: 10, Issue:1

    Topics: Adolescent; Adult; Azepines; Diazepam; Half-Life; Humans; Hypnotics and Sedatives; Male; Motor Skills; Sleep; Sleep Stages; Sleep, REM; Task Performance and Analysis; Triazoles

1980

Other Studies

20 other study(ies) available for diazepam and brotizolam

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Design, synthesis and biological evaluation of 7-substituted 4-phenyl-6H-imidazo[1,5-a]thieno[3,2-f] [1,4]diazepines as safe anxiolytic agents.
    European journal of medicinal chemistry, 2020, Aug-15, Volume: 200

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Binding Sites; Drug Design; Locomotion; Memory Disorders; Mice; Molecular Docking Simulation; Rats; Receptors, GABA-A

2020
Discriminative and reinforcing effects of brotizolam in rhesus monkeys.
    Psychopharmacology, 1991, Volume: 103, Issue:2

    Topics: Animals; Avoidance Learning; Azepines; Conditioning, Operant; Diazepam; Discrimination, Psychological; Female; Macaca mulatta; Male; Methohexital; Pentobarbital; Reinforcement Schedule; Self Administration

1991
Appetite-modulating drugs in dwarf goats, with special emphasis on benzodiazepine-induced hyperphagia and its antagonism by flumazenil and RO 15-3505.
    Journal of veterinary pharmacology and therapeutics, 1989, Volume: 12, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Appetite Regulation; Azepines; Benzodiazepines; Benzodiazepinones; Body Weight; Diazepam; Female; Flumazenil; Goats; Hyperphagia; Ivermectin; Male; Midazolam; Time Factors

1989
Pharmacological and neurochemical properties of 1,4-diazepines with two annelated heterocycles ('hetrazepines').
    European journal of pharmacology, 1985, Feb-12, Volume: 109, Issue:1

    Topics: Action Potentials; Aggression; Animals; Anticonvulsants; Azepines; Behavior, Animal; Benzodiazepinones; Brain Chemistry; Carbolines; Cerebral Cortex; Conflict, Psychological; Diazepam; Flumazenil; Heterocyclic Compounds; Humans; Hypnotics and Sedatives; Male; Mice; Motor Activity; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sleep; Social Isolation; Wakefulness

1985
Biochemical studies with the new thienotriazolo-diazepine brotizolam.
    Arzneimittel-Forschung, 1986, Volume: 36, Issue:3A

    Topics: Animals; Azepines; Binding, Competitive; Biogenic Amines; Diazepam; Dopamine; Flunitrazepam; Homovanillic Acid; Hypnotics and Sedatives; In Vitro Techniques; Male; Rats; Receptors, Drug; Receptors, GABA-A; Synaptosomes

1986
Effects of brotizolam on the sleep-waking cycle of the cat.
    Arzneimittel-Forschung, 1986, Volume: 36, Issue:3A

    Topics: Animals; Azepines; Cats; Diazepam; Electrodes, Implanted; Electroencephalography; Female; Flurazepam; Hypnotics and Sedatives; Male; Nitrazepam; Sleep; Sleep, REM; Time Factors; Triazolam; Wakefulness

1986
Therapeutic safety studies of brotizolam in animals.
    Arzneimittel-Forschung, 1986, Volume: 36, Issue:3A

    Topics: Aggression; Animals; Azepines; Diazepam; Hypnotics and Sedatives; Mice; Pentylenetetrazole; Psychomotor Performance

1986
Physical dependence capacity of brotizolam in rhesus monkeys. 1st communication: primary dependence studies.
    Arzneimittel-Forschung, 1986, Volume: 36, Issue:3A

    Topics: Animals; Azepines; Diazepam; Hypnotics and Sedatives; Macaca mulatta; Motor Activity; Psychomotor Performance; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors

1986
Physical dependence capacity of brotizolam in rhesus monkeys. 2nd communication: primary dependence and barbital substitution.
    Arzneimittel-Forschung, 1986, Volume: 36, Issue:3A

    Topics: Animals; Azepines; Barbital; Barbiturates; Body Weight; Diazepam; Female; Hypnotics and Sedatives; Macaca mulatta; Male; Psychomotor Performance; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam

1986
Interactions of brotizolam and diazepam with some psychotropic drugs on motor performance in mice.
    Arzneimittel-Forschung, 1986, Volume: 36, Issue:3A

    Topics: Animals; Azepines; Desipramine; Diazepam; Drug Interactions; Ethanol; Female; Hexobarbital; Hypnotics and Sedatives; Mice; Psychomotor Performance; Psychotropic Drugs; Reflex; Time Factors

1986
Effects of a chronic administration of two benzodiazepines on food intake in rats given a highly palatable diet.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 25, Issue:4

    Topics: Adipose Tissue; Animals; Azepines; Body Weight; Diazepam; Feeding Behavior; Food Preferences; Male; Rats; Rats, Inbred Strains

1986
Behavioral effects of brotizolam, a new thienotriazolodiazepine derivative.
    Japanese journal of pharmacology, 1984, Volume: 35, Issue:3

    Topics: Aggression; Anesthesia; Animals; Anticonvulsants; Azepines; Behavior, Animal; Conflict, Psychological; Diazepam; Electroshock; Estazolam; Humans; Hypnotics and Sedatives; Male; Mice; Motor Activity; Nitrazepam; Olfactory Bulb; Pentylenetetrazole; Postural Balance; Raphe Nuclei; Rats; Rats, Inbred Strains; Thiopental

1984
Effects of diazepam, nitrazepam and brotizolam on dopamine turnover in the olfactory tubercle, nucleus accumbens and caudate nucleus of rats.
    Japanese journal of pharmacology, 1983, Volume: 33, Issue:3

    Topics: Animals; Azepines; Brain; Caudate Nucleus; Diazepam; Dopamine; Hypnotics and Sedatives; Male; Nitrazepam; Nucleus Accumbens; Rats; Rats, Inbred Strains

1983
Role of platelet activating factor in triazolobenzodiazepines-induced retrograde amnesia.
    Behavioural brain research, 2003, Jun-16, Volume: 142, Issue:1-2

    Topics: 1-Alkyl-2-acetylglycerophosphocholine Esterase; Amnesia, Anterograde; Amnesia, Retrograde; Animals; Anti-Anxiety Agents; Azepines; Diazepam; Diterpenes; Escape Reaction; Female; Flumazenil; Ginkgolides; Lactones; Learning; Male; Mice; Phospholipases A; Platelet Activating Factor; Platelet Membrane Glycoproteins; Reaction Time; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Receptors, GABA-A; Retention, Psychology; Triazolam

2003
Up-regulation of L-type high voltage-gated calcium channel subunits by sustained exposure to 1,4- and 1,5-benzodiazepines in cerebrocortical neurons.
    Journal of neurochemistry, 2007, Volume: 103, Issue:6

    Topics: Animals; Azepines; Benzodiazepines; Binding, Competitive; Calcium Channels; Calcium Channels, L-Type; Calcium Signaling; Cells, Cultured; Cerebral Cortex; Diazepam; Hypnotics and Sedatives; Mice; Neurons; Protein Subunits; Substance Withdrawal Syndrome; Up-Regulation

2007
Juvenile stress-induced alteration of maturation of the GABAA receptor alpha subunit in the rat.
    The international journal of neuropsychopharmacology, 2008, Volume: 11, Issue:7

    Topics: Aging; Amygdala; Animals; Anti-Anxiety Agents; Anxiety; Azepines; Behavior, Animal; Blotting, Western; Diazepam; Hippocampus; Indicators and Reagents; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Reflex, Startle; Stress, Psychological

2008
Evaluation of anxiolytic-like effects of some short-acting benzodiazepine hypnotics in mice.
    Journal of pharmacological sciences, 2008, Volume: 107, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Azepines; Benzodiazepines; Diazepam; Hypnotics and Sedatives; Lorazepam; Male; Maze Learning; Mice; Mice, Inbred ICR; Motor Activity; Triazolam

2008