diazepam and alprazolam

diazepam has been researched along with alprazolam in 212 studies

Research

Studies (212)

TimeframeStudies, this research(%)All Research%
pre-199071 (33.49)18.7374
1990's56 (26.42)18.2507
2000's34 (16.04)29.6817
2010's37 (17.45)24.3611
2020's14 (6.60)2.80

Authors

AuthorsStudies
Gall, M; Hester, JB; Lahti, RA; Rudzik, AD1
Chidester, C; Duchamp, DJ; Gall, M; Lahti, RA; Rudzik, AD; Scahill, T1
Collins, RJ; Gall, M; Kamdar, BV1
Hester, JB; Von Voigtlander, P1
Walser, A; Zenchoff, G1
Evenson, GN; Hester, JB; VonVoigtlander, P1
Carrupt, PA; Crivori, P; Cruciani, G; Testa, B1
Topliss, JG; Yoshida, F1
Gao, F; Lombardo, F; Shalaeva, MY; Tupper, KA1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY2
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Abraham, MH; Acree, WE; Ibrahim, A1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Campillo, NE; Guerra, A; Páez, JA1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Alelyunas, YW; Bui, K; Empfield, JR; McCarthy, D; Pelosi-Kilby, L; Shen, C; Spreen, RC1
Ahlin, G; Bergström, F; Bredberg, U; Fridén, M; Hammarlund-Udenaes, M; Rehngren, M; Wan, H1
Artursson, P; Mateus, A; Matsson, P1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Ganeshpurkar, A; Gupta, SK; Gutti, G; Krishnamurthy, S; Kumar, D; Modi, G; Singh, SK1
Rai, SN; Shankar, S; Sharma, P; Shrivastava, SK; Singh, SP; Srivastava, P; Srivastava, RK; Tripathi, PN1
Carmona, AV; Kumari, S; Tiwari, AK; Trippier, PC1
Ahmed, T; Cook, JM; Golani, LK; Mondal, P; Pandey, KP; Rezvanian, S; Sharmin, D; Witkin, JM; Yeunus Mian, M1
Jaiswal, S; Raja Ayyannan, S; Tiwari, V; Uniyal, A1
Aamir Javed, M; Ikram, M; Jadoon, R; Mahnashi, MH; Rashid, U; Sadiq, A; Saeed Jan, M; Shahid, M1
Busto, UE; Kaplan, HL; Sellers, EM1
Loeffler, PM1
Cannizzaro, C; Cannizzaro, G; Flugy, A; Gagliano, M; Novara, V1
Cowley, DS; Greenblatt, DJ; Hommer, D; Kramer, GL; Petty, F; Roy-Byrne, PP1
Bouhours, P; Danjou, P; Hergueta, T; Lacomblez, L; Puech, AJ; Warot, D1
Ahrens, TN; Baumgartner, WA; Cutler, NR; Hill, VA; Sramek, JJ1
Cohen, MH; Johnston-Anderson, A; Krasnow, SH; Wadleigh, RG1
al-Tikriti, MS; Baldwin, RM; Innis, RB; Johnson, EW; Laruelle, MA; Malison, RT; Seibyl, JP; Sybirska, EH; Zimmermann, RC; Zoghbi, SS1
Franklin, SR; Tang, AH1
Coppola, A; Francis, E; Sheehan, DV; Sheehan, MF; Torres, A1
Boix, F; Escorihuela, RM; Fernández Teruel, A; Tobeña, A1
Altamura, M; Cannuscio, B; Covelli, V; Decandia, P; Jirillo, E; Maffione, AB; Munno, I1
Cannuscio, B; Covelli, V; Jirillo, E; Maffione, AB1
Cocores, J1
Boix, F; Escorihuela, RM; Fernández-Teruel, A; Tobena, A1
Biggio, G; Concas, A; Mascia, MP; Sanna, E; Santoro, V; Serra, M1
Apelt, S; Emrich, HM; Schmauss, C3
Burrows, GD; Judd, FK; Marriott, PF; Norman, TR1
Haefely, WE; Jenck, F; Martin, JR; Moreau, JL; Pieri, L; Schoch, P1
Bartel, PR; Becker, PJ; Blom, MW; de Sommers, K; Van der Meyden, CH1
Klerman, GL1
Cook, B; Garvey, MJ; Noyes, R; Suelzer, M1
Juergens, S1
Eckardt, MJ; Granger, A; Lane, E; Linnoila, M; Lister, R; Moss, H; Stapleton, JM1
Cook, B; Garvey, M; Noyes, R; Summers, R1
Kathol, RG; Lopez, AL; Noyes, R1
Anderson, BJ; Brown, TC; Exarchos, H; Lee, K1
Natelson, BH; Ottenweller, JE; Tapp, WN1
De Souza, EB; Grigoriadis, DE; Pearsall, D1
Engel, JA; Söderpalm, B1
Gastfriend, DR; Rosenbaum, JF1
Covington, EC; Rapport, DJ1
Grover, E; Natelson, BH; Ottenweller, JE; Tapp, WN1
Cook, B; Garvey, M; Noyes, R; Tollefson, G1
Caddeo, S; Ecari, U; Pariante, F1
Cowley, DS; Dager, SR; Dunner, DL; Roy-Byrne, PP; Vitaliano, P1
Engel, JA; Eriksson, E; Söderpalm, B1
Simson, PE; Weiss, JM1
Abernethy, DR; Greenblatt, DJ; Morse, DS; Shader, RI1
Davison, K; Farquharson, RG; Khan, MC; Majid, A2
Earley, B; Leonard, BE; O'Connor, WT1
Ciancio, SG1
Baker, RW; Zimmer, B; Zipursky, RB1
Bjornsson, TD; Ellinwood, EH; Heatherly, DG; Kilts, C; Nikaido, AM1
Aranko, K; Bordignon, D; Mattila, MJ1
Alderdice, MT; Marunycz, JD; Napoliello, MJ; Newton, RE1
Carlsson, M; Eriksson, E; Nilsson, C; Söderpalm, B1
Geller, AM; Lucki, I; Rickels, K1
Avery, DH; Dunner, DL; Hyde, TS; Ishiki, D; Wilson, LG1
Cowley, DS; Dager, SR; Dunner, DL1
Ellinwood, EH; Heatherly, DG; Nikaido, AM1
Bjornsson, TD; Ellinwood, EH; Heatherly, DG; Nikaido, AM1
Gallaher, EJ; Hollister, LE; Jacques, CJ1
Albeck, JH1
Coryell, W; Noyes, R1
Cole, JO; Orzack, MH1
Beake, B; Bird, M; Cole, JO; Dessain, E; Friedman, L; McEachern, J; Orzack, MH1
Cagiano, R; Cuomo, V; De Salvia, MA; Maselli, MA; Racagni, G; Renna, G1
Bell, J; Bickford-Wimer, PC; de la Garza, R; Egan, M; Freedman, R1
Hata, T; Itoh, E; Kawabata, A; Kita, T; Nishimura, Y1
Boix, F; Fernández Teruel, A; Tobeña, A1
Csernansky, JG; Hollister, LE; Lombrozo, L; Overall, JE; Riney, SJ1
Amsterdam, JD; Chung, HR; Csanalosi, IB; Hurowitz, AM; Kaplan, M; London, J; Rickels, K; Wiseman, K1
Patterson, WM1
Cagen, LM; Chesney, CM; Pifer, DD1
Batcha, KJ; Olson, SC; Votolato, NA1
Baiguerra, G; Kostowski, W; Valzelli, L1
Cohen, SA; Dement, WC; Seidel, WF; Wilson, L1
Aranko, K1
Maletzky, BM1
Cohn, JB1
Rickels, K1
Harris, DW; Sethy, VH2
Cohen, D; Csanalosi, I; Greisman, P; Harris, H; Rickels, K; Ross, HA; Werblowsky, J1
Hodges, DH; Sethy, VH2
Assenzo, JR; Shu, VS1
Annable, L; Chouinard, G; Fontaine, R; Labonte, A1
Brogden, RN; Dawson, GW; Jue, SG1
Elie, R; Lamontagne, Y1
Ator, NA; Brady, JV; Griffiths, RR; Lamb, RJ; Lukas, SE1
Greenblatt, DJ; Ochs, HR; Verburg-Ochs, B1
DeTurck, KH; Miller, J; Routzahn, BK; Vogel, WH1
Johnson, BW; Valvani, SC; Yalkowsky, SH1
Cooper, TB; Friedman, MJ; Harris, PQ; Stolk, JM1
Bonnet, MH; Kramer, M; Roth, T1
Aden, GC; Thein, SG1
Kolin, IS; Linet, OI1
Jenck, F; Martin, JR; Moreau, JL1
Frantik, E; Horváth, M; Kozená, L1
Cannizzaro, C; Cannizzaro, E; Cannizzaro, G; Gagliano, M; Mineo, A; Sabatino, M1
Needleman, SB; Porvaznik, M1
Cowley, DS; Greenblatt, DJ; Hommer, DW; Nemeroff, CB; Radant, A; Ritchie, JC; Roy-Byrne, PP1
Kulkarni, SK; Sharma, K1
Adinoff, B1
Busto, U; Kaplan, HL; Sellers, EM; Zawertailo, L1
Ciraulo, DA; DuPont, RL; Griffiths, RR; Kosten, TR; Romach, MK; Sellers, EM; Woody, GE1
Britton, K; Hauger, RL; Irwin, M1
Alburges, ME; Hunt, ME; Longlet, LL; Mahan, DR; Wamsley, JK1
Fulton, M; Petty, F; Rush, AJ; Trivedi, MH1
Griebel, G; Perrault, G; Sanger, DJ1
Burrows, GD; Cook, BL; Garvey, MJ; Judd, FK; Marriott, P; Norman, TR; Noyes, R; Reich, JH1
Mazurek, MF; Rosebush, PI1
Maletta, GJ1
Cannizzaro, C; Cannizzaro, E; Gagliano, M; Mangiapane, N1
Barnhill, JG; Ciraulo, AM; Ciraulo, DA; Greenblatt, DJ; Knapp, C; Sarid-Segal, O; Shader, RI1
Asahi, T; Kuribara, H1
Barros, HM; Manitiu, A; Miczek, KA; Vivian, JA1
Broderick, PA1
Cannizzaro, C; Cannizzaro, E; Gagliano, M; Mineo, A1
Berry, RA; Boezaart, AP; Laubscher, JJ; Nell, ML1
Covelli, V; Jirillo, E; Maffione, AB; Nacci, C; Tatò, E1
Matthews, J; Pollack, MH; Scott, EL1
Bourin, M; Hascoët, M1
Hemmersbach, P; Ragnar Norli, H; Rasmussen, KE; Reubsaet, KJ1
Atta-Politou, J; Dona, A; Koutselinis, A; Parissi-Poulou, M1
Adam, G; Cesura, AM; Dautzenberg, FM; Jenck, F; Kilpatrick, G; Kolczewski, S; Lundstrom, K; Martin, JR; Moreau, JL; Ouagazzal, AM; Poli, SM; Roever, S; Wichmann, J1
Gatti, JE1
Freeman, EW; Rickels, K1
Carlson, JN; Glick, SD; Haskew, R; Jerussi, TP; Maisonneuve, IM; Wacker, J1
Collins, DC; Lee, ML1
Lapierre, YD1
Bagaméri, A; Kulcsár, T; Lehoczky, O; Pulay, T; Sárosi, Z1
Beigh, A; Mir, B; Naqib, A1
Gomez, TH; Meisch, RA; Roache, JD1
Groenink, L; Maes, RA; Olivier, B; Oosting, RS; Pattij, T; van der Gugten, J1
Cannizzaro, C; Cannizzaro, E; Gagliano, M; Martire, M; Mineo, A; Provenzano, G; Steardo, L1
Alvi, SN; Khalid, S; Parimala, P; Rao, RN1
Isbister, GK; O'Regan, L; Sibbritt, D; Whyte, IM1
Bucior, J; Foltyn, W; Jastrzebska-Okoń, K; Kempiński, M; Knopik, J; Tomczyk, A; Ziółko, E1
Akiyoshi, J; Fujiki, M; Isogawa, K; Kobayashi, H; Kodama, K; Matsushita, H; Tanaka, Y; Tsutsumi, T1
Cottler, L; Inciardi, JA; Kurtz, SP; Surratt, HL1
Arias, JL; Conejo, NM; González-Pardo, H1
Dickson, SJ; Irving, RC1
Cook, JM; Duke, AN; Huang, S; Mattingly, BA; Platt, DM; Rowlett, JK; Yin, W1
Galetin, A; Hallifax, D; Houston, JB1
Kulvanich, P; Ongpipattanakul, B; Sila-on, W; Vardhanabhuti, N1
Mandrioli, R; Mercolini, L; Raggi, MA1
Arbanas, D; Arbanas, G; Dujam, K1
Jogani, V; Misra, A; Naik, S; Porecha, S; shah, T1
Dai, Z; Liang, X; Liu, W1
Chronister, CW; Goldberger, BA; Merves, ML1
Argyraki, M; Ekonomopoulou, MT; Iakovidou-Kritsi, Z; Polatoglou, E; Stephanidou-Stephanatou, J; Tsoleridis, CA1
Brown, RE; Fontana, M; Fraser, LM; Holmes, A; Hussin, A; Lederle, L; O'Leary, TP; Ramos, A; Whittaker, A1
Huemer, HP; Irschick, EU; Kitchen, M; Lassnig, C; Nowotny, N; Pavlic, M1
Carlezon, WA; Meloni, EG; Myers, KM; Rudolph, U; Smith, KS; Van't Veer, A1
Akritopoulou, K; Ekonomopoulou, MT; Iakovidou-Kritsi, Z; Mourelatos, C1
Chen, H; Shen, M; Xiang, P1
Buetler, J; Crestani, F; Koester, C; Masneuf, S1
Adams, JL; Blaschke, T; Dell, RM; Der, JS; Finkle, WD; Greenland, S; Ridgeway, G; VanRiper, KB; Wang, Z1
Amaral, VC; Campos, KF; Miguel, TT; Nunes-de-Souza, RL; Rico, JL1
Mendes-Gomes, J; Nunes-de-Souza, RL; Rico, JL; Rodgers, RJ; Sorregotti, T1
Krzek, J; Maślanka, A; Szlósarczyk, M; Wach, K; Żmudzki, P1
El Zahaf, NA; Salem Elhwuegi, A1
Arima, Y; Nagao, M; Namera, A; Shiraishi, H; Tajima, T; Torikoshi, A; Toubou, H1
Bertol, E; Boscolo Berto, R; Favretto, D; Mannaioni, G; Mari, F; Vaiano, F1
Christophersen, AS; Enger, A; Nordal, K; Vindenes, V; Øiestad, EL1
Gong, L; Guo, C; Jiang, S; Shi, F; Tan, H1
Manicke, NE; Zhang, C1
Tandeter, H1
Buckley, NA; Cairns, R; Pearson, SA; Schaffer, AL1
Holm, KM; Johansen, SS; Linnet, K; Skov, L1
Orlando, JM1
Bachs, L; Birdal, M; Bruun, LD; Høiseth, G; Karinen, R; Kjeldstadli, K; Middelkoop, G; Temte, V; Øiestad, E1
Aricescu, AR; Desai, R; Karia, D; Kotecha, A; Laverty, D; Malinauskas, T; Masiulis, S; Miller, KW; Pardon, E; Serna Martin, I; Steyaert, J; Uchański, T; Zivanov, J1
Aug, I; Bregin, A; Innos, J; Mazitov, T; Philips, MA; Vasar, E1
Amioka, E; Black, JC; Dargan, PI; Dart, RC; Haynes, CM; Hockenhull, J; Wood, DM1
Kościelniak, P; Majda, A; Mrochem, K; Świądro, M; Wietecha-Posłuszny, R1
Cherner, M; Grelotti, DJ; Heaton, RK; Letendre, S; Ma, Q; Saloner, R; Sundermann, EE; Tyree, G1
Falcon, M; Fernadez-Lopez, L; Luna, A; Mancini, R; Pellegrini, M; Rotolo, M1
Boy, D; Büttner, A; Kegler, R; Kolbe, V; Rentsch, D; Schmidt, B1
Apollonio, LG; Huestis, MA; Kaspar, CK; Lavins, ES; Michel, HM; Mitchell-Mata, CL; Sofalvi, S1
Johannsen, ML; Jørgensen, FS; Munkboel, CH; Styrishave, B1
Christophoridis, C; Fytianos, K; Kouinoglou, N; Lazaridis, N; Mitsika, EE; Zacharis, CK1
Araújo, JO; Bergamaschi, CC; de Andrade, NK; Guimarães, CC; Lopes, LC; Motta, RHL; Ramacciato, JC1
Adhikari, S; Barron, LP; Bhatnagar, A; Bowes, DA; Coronado-Apodaca, KG; Driver, EM; Halden, RU; Kumar, R; Martínez-Ruiz, M; McCall, KL; Melchor-Martínez, EM; Ng, KT; Oyervides-Muñoz, MA; Parra-Saldivar, R; Piper, BJ; Smith, T; Sosa-Hernandez, JE1
Andersson, L; Håkansson, A; Johnson, B; Walde, J1
Guo, D; Kossintseva, I; Zloty, DM1
Barbui, C; Bighelli, I; Caldwell, DM; Cipriani, A; Davies, SJ; Dawson, S; Dias, S; Furukawa, TA; Guaiana, G; Imai, H; Koesters, M; Meader, N; Pompoli, A; Robertson, L; Tajika, A1

Reviews

20 review(s) available for diazepam and alprazolam

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Amide Bond Bioisosteres: Strategies, Synthesis, and Successes.
    Journal of medicinal chemistry, 2020, 11-12, Volume: 63, Issue:21

    Topics: Amides; Carbamates; Click Chemistry; Drug Design; Pyridines; Structure-Activity Relationship; Triazoles; Urea

2020
Oral benzodiazepines and conscious sedation: a review.
    Journal of oral and maxillofacial surgery : official journal of the American Association of Oral and Maxillofacial Surgeons, 1992, Volume: 50, Issue:9

    Topics: Administration, Oral; Alprazolam; Ambulatory Surgical Procedures; Anti-Anxiety Agents; Conscious Sedation; Diazepam; Flurazepam; Humans; Lorazepam; Midazolam; Oxazepam; Premedication; Receptors, GABA-A; Temazepam; Triazolam

1992
Treatment of intractable dyspnea: clinical and ethical issues.
    Cancer investigation, 1992, Volume: 10, Issue:4

    Topics: Alprazolam; Codeine; Diazepam; Dyspnea; Ethics, Medical; Humans; Infusions, Intravenous; Morphine; Neoplasms; Promethazine; Randomized Controlled Trials as Topic

1992
Effects of benzodiazepines on the immune system.
    Acta neurologica, 1991, Volume: 13, Issue:5

    Topics: Alprazolam; Antibody Formation; Benzodiazepines; Diazepam; Humans; Immune System; Immunity, Cellular; Neuroimmunomodulation; Neuropeptides; Phagocytosis; Phobic Disorders; Psychotropic Drugs

1991
Short-acting versus long-acting benzodiazepines: discontinuation effects in panic disorders.
    Journal of psychiatric research, 1990, Volume: 24 Suppl 2

    Topics: Alprazolam; Anti-Anxiety Agents; Anxiety Disorders; Diazepam; Drug Administration Schedule; Humans; Panic; Risk Factors; Substance Withdrawal Syndrome

1990
Alprazolam and diazepam: addiction potential.
    Journal of substance abuse treatment, 1991, Volume: 8, Issue:1-2

    Topics: Alprazolam; Diazepam; Humans; Risk Factors; Substance Withdrawal Syndrome; Substance-Related Disorders

1991
Review of the side-effect profile of buspirone.
    The American journal of medicine, 1986, Mar-31, Volume: 80, Issue:3B

    Topics: Alprazolam; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Buspirone; Clinical Trials as Topic; Clorazepate Dipotassium; Diazepam; Dizziness; Double-Blind Method; Drug Evaluation; Fatigue; Headache; Humans; Lorazepam; Pyrimidines

1986
Withdrawal and detoxification from benzodiazepine dependence: a potential role for clonazepam.
    The Journal of clinical psychiatry, 1987, Volume: 48 Suppl

    Topics: Adolescent; Adult; Aged; Alprazolam; Anti-Anxiety Agents; Clonazepam; Diazepam; Drug Tolerance; Humans; Male; Middle Aged; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam

1987
Comparative study of the abuse liability of alprazolam, lorazepam, diazepam, methaqualone, and placebo.
    The International journal of the addictions, 1988, Volume: 23, Issue:5

    Topics: Adolescent; Adult; Alprazolam; Arousal; Diazepam; Euphoria; Female; Humans; Lorazepam; Male; Methaqualone; Risk Factors; Substance-Related Disorders

1988
Alprazolam: a review of its pharmacodynamic properties and efficacy in the treatment of anxiety and depression.
    Drugs, 1984, Volume: 27, Issue:2

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Antidepressive Agents; Anxiety Disorders; Benzodiazepines; Clinical Trials as Topic; Depressive Disorder; Diazepam; Humans; Imipramine; Kinetics

1984
Alprazolam and benzodiazepine dependence.
    The Journal of clinical psychiatry, 1993, Volume: 54 Suppl

    Topics: Adult; Alcoholism; Alprazolam; Benzodiazepines; Comorbidity; Diazepam; Female; Humans; Incidence; Male; Methadone; Middle Aged; Opioid-Related Disorders; Substance Abuse Detection; Substance-Related Disorders

1993
Benzodiazepines as antidepressants: does GABA play a role in depression?
    Biological psychiatry, 1995, Nov-01, Volume: 38, Issue:9

    Topics: Alprazolam; Antidepressive Agents; Benzodiazepines; Chlordiazepoxide; Depressive Disorder; Diazepam; GABA Modulators; gamma-Aminobutyric Acid; Humans; Treatment Outcome

1995
Stress, neuropsychiatric disorders and immunological effects exerted by benzodiazepines.
    Immunopharmacology and immunotoxicology, 1998, Volume: 20, Issue:2

    Topics: Adjuvants, Immunologic; Alprazolam; Animals; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Diazepam; Humans; Immune System; Immunosuppressive Agents; Stress, Physiological

1998
Alprazolam is relatively more toxic than other benzodiazepines in overdose.
    British journal of clinical pharmacology, 2004, Volume: 58, Issue:1

    Topics: Adolescent; Adult; Aged; Alprazolam; Anti-Anxiety Agents; Benzodiazepines; Critical Care; Diazepam; Drug Overdose; Humans; Length of Stay; Middle Aged

2004
Benzodiazepine metabolism: an analytical perspective.
    Current drug metabolism, 2008, Volume: 9, Issue:8

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Azepines; Benzodiazepines; Bromazepam; Chromatography, High Pressure Liquid; Diazepam; Humans; Lorazepam; Mass Spectrometry; Midazolam; Triazolam

2008
[The present study situation and application prospect of nail analysis for abused drugs].
    Fa yi xue za zhi, 2010, Volume: 26, Issue:5

    Topics: Alprazolam; Azabicyclo Compounds; Chromatography, High Pressure Liquid; Cocaine; Diazepam; Eszopiclone; Forensic Toxicology; Gas Chromatography-Mass Spectrometry; Hair; Humans; Illicit Drugs; Nails; Piperazines; Specimen Handling; Substance Abuse Detection

2010
Postmortem Brain and Blood Reference Concentrations of Alprazolam, Bromazepam, Chlordiazepoxide, Diazepam, and their Metabolites and a Review of the Literature.
    Journal of analytical toxicology, 2016, Volume: 40, Issue:7

    Topics: Alprazolam; Blood-Brain Barrier; Bromazepam; Chlordiazepoxide; Diazepam; Forensic Toxicology; Humans

2016
Effectiveness and safety of oral sedation in adult patients undergoing dental procedures: a systematic review.
    BMJ open, 2021, 01-25, Volume: 11, Issue:1

    Topics: Adult; Alprazolam; Anesthesia; Benzodiazepines; Diazepam; Humans; Midazolam

2021
Pharmacological treatments in panic disorder in adults: a network meta-analysis.
    The Cochrane database of systematic reviews, 2023, 11-28, Volume: 11

    Topics: Adult; Alprazolam; Antidepressive Agents; Antidepressive Agents, Tricyclic; Benzodiazepines; Clomipramine; Clonazepam; Desipramine; Diazepam; Fluoxetine; Humans; Network Meta-Analysis; Panic Disorder; Paroxetine; Reboxetine; Selective Serotonin Reuptake Inhibitors; Serotonin and Noradrenaline Reuptake Inhibitors; Venlafaxine Hydrochloride

2023

Trials

49 trial(s) available for diazepam and alprazolam

ArticleYear
Abuse liability of bretazenil and other partial agonists.
    Clinical neuropharmacology, 1992, Volume: 15 Suppl 1 Pt A

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Benzodiazepinones; Diazepam; Double-Blind Method; Humans; Male; Receptors, GABA-A; Substance-Related Disorders

1992
Effect of acute and chronic benzodiazepines on plasma GABA in anxious patients and controls.
    Psychopharmacology, 1992, Volume: 109, Issue:1-2

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Anxiety Disorders; Diazepam; gamma-Aminobutyric Acid; Humans; Middle Aged; Panic Disorder; Psychiatric Status Rating Scales

1992
Comparative study of the psychomotor and antistress effects of ritanserin, alprazolam and diazepam in healthy subjects: some trait anxiety-independent responses.
    International clinical psychopharmacology, 1992, Volume: 7, Issue:2

    Topics: Acoustic Stimulation; Adult; Alprazolam; Anxiety; Diazepam; Double-Blind Method; Feedback; Flicker Fusion; Humans; Male; Memory; Psychomotor Performance; Reaction Time; Ritanserin; Stress, Psychological

1992
Preference for alprazolam as opposed to diazepam in benzodiazepine-dependent psychiatric inpatients.
    Pharmacopsychiatry, 1990, Volume: 23, Issue:2

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Diazepam; Double-Blind Method; Female; Humans; Male; Middle Aged; Substance-Related Disorders

1990
Short-acting versus long-acting benzodiazepines: discontinuation effects in panic disorders.
    Journal of psychiatric research, 1990, Volume: 24 Suppl 2

    Topics: Alprazolam; Anti-Anxiety Agents; Anxiety Disorders; Diazepam; Drug Administration Schedule; Humans; Panic; Risk Factors; Substance Withdrawal Syndrome

1990
The effects of alprazolam, quazepam and diazepam on saccadic eye movements, parameters of psychomotor function and the EEG.
    Fundamental & clinical pharmacology, 1990, Volume: 4, Issue:6

    Topics: Administration, Oral; Adult; Affect; Alprazolam; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Electroencephalography; Flicker Fusion; Humans; Male; Psychomotor Performance; Saccades

1990
Controlled discontinuation of benzodiazepine treatment for patients with panic disorder.
    The American journal of psychiatry, 1991, Volume: 148, Issue:4

    Topics: Adult; Alprazolam; Anxiety Disorders; Diazepam; Double-Blind Method; Female; Half-Life; Humans; Male; Panic; Personality Inventory; Placebos; Psychiatric Status Rating Scales; Recurrence; Substance Withdrawal Syndrome

1991
Effects of single doses of alprazolam and diazepam, alone and in combination with ethanol, on psychomotor and cognitive performance and on autonomic nervous system reactivity in healthy volunteers.
    European journal of clinical pharmacology, 1990, Volume: 39, Issue:1

    Topics: Adult; Affect; Alprazolam; Anxiety; Autonomic Nervous System; Cognition; Diazepam; Drug Interactions; Ethanol; Female; Humans; Nordazepam; Norepinephrine; Psychomotor Performance

1990
Reduction in urinary free cortisol during benzodiazepine treatment of panic disorder.
    Psychoneuroendocrinology, 1990, Volume: 15, Issue:1

    Topics: Adult; Agoraphobia; Alprazolam; Benzodiazepines; Depression; Diazepam; Fear; Female; Humans; Hydrocortisone; Male; Middle Aged; Panic; Phobic Disorders

1990
Oral premedication in children: a comparison of chloral hydrate, diazepam, alprazolam, midazolam and placebo for day surgery.
    Anaesthesia and intensive care, 1990, Volume: 18, Issue:2

    Topics: Administration, Oral; Alprazolam; Ambulatory Surgical Procedures; Anesthesia Recovery Period; Attitude; Child Behavior; Child, Preschool; Chloral Hydrate; Diazepam; Double-Blind Method; Female; Humans; Infant; Male; Midazolam; Placebos; Preanesthetic Medication; Random Allocation; Time Factors

1990
Etizolam in the treatment of generalized anxiety disorder associated with depressive symptoms.
    Current medical research and opinion, 1989, Volume: 11, Issue:9

    Topics: Adult; Alprazolam; Anxiety Disorders; Consumer Behavior; Depression; Diazepam; Double-Blind Method; Female; Humans; Middle Aged; Randomized Controlled Trials as Topic; Tranquilizing Agents

1989
Relapse and rebound following discontinuation of benzodiazepine treatment of panic attacks: alprazolam versus diazepam.
    The American journal of psychiatry, 1989, Volume: 146, Issue:7

    Topics: Adult; Alprazolam; Anxiety; Diazepam; Double-Blind Method; Fear; Female; Humans; Male; Middle Aged; Panic; Placebos; Recurrence; Test Anxiety Scale; Time Factors

1989
Interaction of propoxyphene with diazepam, alprazolam and lorazepam.
    British journal of clinical pharmacology, 1985, Volume: 19, Issue:1

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Benzodiazepines; Dextropropoxyphene; Diazepam; Drug Interactions; Female; Half-Life; Humans; Kinetics; Lorazepam; Male; Metabolic Clearance Rate; Middle Aged

1985
A double-blind comparison of alprazolam, diazepam and placebo in the treatment of anxious out-patients.
    British journal of clinical pharmacology, 1985, Volume: 19 Suppl 1

    Topics: Adolescent; Adult; Alprazolam; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Humans; Male; Middle Aged; Psychiatric Status Rating Scales; Random Allocation; Time Factors

1985
Comparative pharmacokinetics and pharmacodynamics of lorazepam, alprazolam and diazepam.
    Psychopharmacology, 1985, Volume: 86, Issue:4

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Drug Tolerance; Humans; Kinetics; Lorazepam; Male; Psychomotor Performance; Receptors, GABA-A

1985
Psychomotor effects of alprazolam and diazepam during acute and subacute treatment, and during the follow-up phase.
    Acta pharmacologica et toxicologica, 1985, Volume: 56, Issue:5

    Topics: Adolescent; Adult; Alprazolam; Analysis of Variance; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Drug Tolerance; Female; Follow-Up Studies; Humans; Male; Psychomotor Performance; Receptors, GABA-A

1985
Review of the side-effect profile of buspirone.
    The American journal of medicine, 1986, Mar-31, Volume: 80, Issue:3B

    Topics: Alprazolam; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Buspirone; Clinical Trials as Topic; Clorazepate Dipotassium; Diazepam; Dizziness; Double-Blind Method; Drug Evaluation; Fatigue; Headache; Humans; Lorazepam; Pyrimidines

1986
Effect of alprazolam and diazepam on anxiety and panic attacks in panic disorder: a controlled study.
    The Journal of clinical psychiatry, 1986, Volume: 47, Issue:9

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Clinical Trials as Topic; Diazepam; Double-Blind Method; Fear; Female; Humans; Male; Panic; Placebos; Psychiatric Status Rating Scales

1986
Benzodiazepine pharmacodynamics: evidence for biophase rate limiting mechanisms.
    Psychopharmacology, 1987, Volume: 91, Issue:2

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Cognition; Diazepam; Humans; Lorazepam; Male; Psychomotor Performance

1987
Placebo response in panic disorder.
    The American journal of psychiatry, 1988, Volume: 145, Issue:9

    Topics: Adult; Agoraphobia; Alprazolam; Anxiety Disorders; Clinical Trials as Topic; Dexamethasone; Diazepam; Double-Blind Method; Fear; Female; Humans; Hydrocortisone; Male; Panic; Placebos; Psychiatric Status Rating Scales

1988
Potential for abuse of alprazolam.
    The American journal of psychiatry, 1988, Volume: 145, Issue:12

    Topics: Alprazolam; Clinical Trials as Topic; Diazepam; Double-Blind Method; Humans; Lorazepam; Methaqualone; Random Allocation; Substance-Related Disorders

1988
Comparative study of the abuse liability of alprazolam, lorazepam, diazepam, methaqualone, and placebo.
    The International journal of the addictions, 1988, Volume: 23, Issue:5

    Topics: Adolescent; Adult; Alprazolam; Arousal; Diazepam; Euphoria; Female; Humans; Lorazepam; Male; Methaqualone; Risk Factors; Substance-Related Disorders

1988
Double-blind comparison of alprazolam, diazepam, and placebo for the treatment of negative schizophrenic symptoms.
    Archives of general psychiatry, 1988, Volume: 45, Issue:7

    Topics: Adult; Alprazolam; Ambulatory Care; Clinical Trials as Topic; Diazepam; Double-Blind Method; Humans; Placebos; Psychiatric Status Rating Scales; Schizophrenia; Schizophrenic Psychology

1988
Alprazolam, diazepam, imipramine, and placebo in outpatients with major depression.
    Archives of general psychiatry, 1987, Volume: 44, Issue:10

    Topics: Adult; Alprazolam; Ambulatory Care; Clinical Trials as Topic; Depressive Disorder; Diazepam; Double-Blind Method; Female; Humans; Imipramine; Male; Personality Inventory; Placebos; Psychiatric Status Rating Scales

1987
Effects of alprazolam and diazepam on the daytime sleepiness of non-anxious subjects.
    Psychopharmacology, 1985, Volume: 87, Issue:2

    Topics: Adult; Alprazolam; Benzodiazepines; Diazepam; Electroencephalography; Electrooculography; Female; Humans; Male; Psychomotor Performance; Sleep; Sleep Stages; Time Factors

1985
Task-dependent development of cross-tolerance to psychomotor effects of lorazepam in man.
    Acta pharmacologica et toxicologica, 1985, Volume: 56, Issue:5

    Topics: Adult; Alprazolam; Benzodiazepines; Diazepam; Drug Tolerance; Female; Humans; Lorazepam; Male; Nitrazepam; Psychomotor Performance; Temazepam

1985
Anxiolytic efficacy of alprazolam compared to diazepam and placebo.
    The Journal of international medical research, 1980, Volume: 8, Issue:2

    Topics: Adolescent; Adult; Aged; Alprazolam; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Clinical Trials as Topic; Diazepam; Double-Blind Method; Humans; Middle Aged; Placebos; Psychiatric Status Rating Scales; Triazoles

1980
Multicenter double-blind efficacy and safety study comparing alprazolam, diazepam and placebo in clinically anxious patients.
    The Journal of clinical psychiatry, 1981, Volume: 42, Issue:9

    Topics: Adolescent; Adult; Aged; Alprazolam; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Clinical Trials as Topic; Diazepam; Double-Blind Method; Humans; Middle Aged; Placebos; Time Factors

1981
Recent advances in anxiolytic therapy.
    The Journal of clinical psychiatry, 1981, Volume: 42, Issue:11 Pt 2

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Buspirone; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Humans; Male; Pyrimidines; Random Allocation

1981
A controlled clinical trial of alprazolam for the treatment of anxiety.
    The American journal of psychiatry, 1983, Volume: 140, Issue:1

    Topics: Adult; Alprazolam; Ambulatory Care; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Humans; Male; Psychiatric Status Rating Scales

1983
Use of statistics in the analysis of side effect data from clinical trials of psychoactive agents.
    Progress in neuro-psychopharmacology & biological psychiatry, 1982, Volume: 6, Issue:4-6

    Topics: Alprazolam; Anti-Anxiety Agents; Benzodiazepines; Clinical Trials as Topic; Diazepam; Double-Blind Method; Humans; Imipramine; Psychotropic Drugs; Statistics as Topic

1982
A double blind comparison of alprazolam, diazepam and placebo in the treatment of anxious out-patients.
    Psychopharmacology, 1983, Volume: 80, Issue:4

    Topics: Adolescent; Adult; Alprazolam; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Humans; Male; Middle Aged; Psychiatric Status Rating Scales

1983
New concepts in benzodiazepine therapy: rebound anxiety and new indications for the more potent benzodiazepines.
    Progress in neuro-psychopharmacology & biological psychiatry, 1983, Volume: 7, Issue:4-6

    Topics: Alprazolam; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Bipolar Disorder; Bromazepam; Clinical Trials as Topic; Clonazepam; Diazepam; Humans; Panic; Receptors, Cell Surface; Receptors, GABA-A; Recurrence; Substance Withdrawal Syndrome

1983
Alprazolam: a review of its pharmacodynamic properties and efficacy in the treatment of anxiety and depression.
    Drugs, 1984, Volume: 27, Issue:2

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Antidepressive Agents; Anxiety Disorders; Benzodiazepines; Clinical Trials as Topic; Depressive Disorder; Diazepam; Humans; Imipramine; Kinetics

1984
Alprazolam and diazepam in the treatment of generalized anxiety.
    Journal of clinical psychopharmacology, 1984, Volume: 4, Issue:3

    Topics: Adult; Aged; Alprazolam; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Humans; Male; Middle Aged; Random Allocation

1984
A dose response study of the hypnotic effectiveness of alprazolam and diazepam in normal subjects.
    Psychopharmacology, 1981, Volume: 75, Issue:3

    Topics: Adolescent; Adult; Alprazolam; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Humans; Hypnotics and Sedatives; Male; Sleep; Sleep Stages; Sleep, REM; Time Factors

1981
Alprazolam compared to diazepam and placebo in the treatment of anxiety.
    The Journal of clinical psychiatry, 1980, Volume: 41, Issue:7

    Topics: Adolescent; Adult; Aged; Alprazolam; Anxiety; Benzodiazepines; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Humans; Male; Middle Aged; Placebos; Triazoles

1980
Double-blind comparison of alprazolam and diazepam for subchronic withdrawal from alcohol.
    The Journal of clinical psychiatry, 1981, Volume: 42, Issue:4

    Topics: Adolescent; Adult; Aged; Alcoholism; Alprazolam; Anxiety Disorders; Benzodiazepines; Clinical Trials as Topic; Diazepam; Dose-Response Relationship, Drug; Double-Blind Method; Female; Humans; Male; Middle Aged; Substance Withdrawal Syndrome

1981
Vigilance impairment after a single dose of benzodiazepines.
    Psychopharmacology, 1995, Volume: 119, Issue:1

    Topics: Acoustic Stimulation; Adult; Alprazolam; Arousal; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Double-Blind Method; Female; Humans; Male; Nitrazepam; Psychiatric Status Rating Scales; Time Factors

1995
Double-blind study of alprazolam, diazepam, clonidine, and placebo in the alcohol withdrawal syndrome: preliminary findings.
    Alcoholism, clinical and experimental research, 1994, Volume: 18, Issue:4

    Topics: Adult; Alcohol Withdrawal Delirium; Alcoholism; Alprazolam; Blood Pressure; Clonidine; Diazepam; Double-Blind Method; Ethanol; Female; Heart Rate; Humans; Male; Middle Aged; Neurologic Examination; Receptors, GABA-A

1994
Pharmacologic effects and abuse liability of bretazenil, diazepam, and alprazolam in humans.
    Clinical pharmacology and therapeutics, 1994, Volume: 55, Issue:4

    Topics: Adult; Alprazolam; Analysis of Variance; Benzodiazepinones; Diazepam; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Humans; Male; Memory; Middle Aged; Psychomotor Performance; Substance-Related Disorders

1994
Diazepam versus alprazolam for the treatment of panic disorder.
    The Journal of clinical psychiatry, 1996, Volume: 57, Issue:8

    Topics: Adult; Age of Onset; Alprazolam; Diazepam; Double-Blind Method; Drug Administration Schedule; Female; Humans; Logistic Models; Male; Panic Disorder; Personality Inventory; Placebos; Research Design; Severity of Illness Index; Treatment Outcome

1996
Alterations in pharmacodynamics of anxiolytics in abstinent alcoholic men: subjective responses, abuse liability, and electroencephalographic effects of alprazolam, diazepam, and buspirone.
    Journal of clinical pharmacology, 1997, Volume: 37, Issue:1

    Topics: Adult; Affect; Alcoholism; Alprazolam; Anti-Anxiety Agents; Buspirone; Diazepam; Electrocardiography; Humans; Male; Substance-Related Disorders

1997
Evaluation of anxiolysis and pain associated with combined peri- and retrobulbar eye block for cataract surgery.
    Journal of clinical anesthesia, 1998, Volume: 10, Issue:3

    Topics: Aged; Alprazolam; Anesthesia, Local; Anesthetics, Local; Anti-Anxiety Agents; Anxiety; Bromazepam; Bupivacaine; Cataract Extraction; Catheterization, Peripheral; Diazepam; Double-Blind Method; Eye; Humans; Injections; Lidocaine; Pain; Patient Satisfaction; Placebos; Preanesthetic Medication

1998
A modified simple and rapid reversed phase liquid chromatographic method for quantification of diazepam and nordiazepam in plasma.
    Journal of pharmaceutical and biomedical analysis, 1999, Volume: 20, Issue:1-2

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Calibration; Chromatography, High Pressure Liquid; Diazepam; Female; Humans; Hydrogen-Ion Concentration; Indicators and Reagents; Middle Aged; Nordazepam; Reference Standards; Reproducibility of Results; Solvents

1999
Prior benzodiazepine exposure and benzodiazepine treatment outcome.
    The Journal of clinical psychiatry, 2000, Volume: 61, Issue:6

    Topics: Alprazolam; Anxiety Disorders; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Female; Humans; Medical Records; Placebos; Premenstrual Syndrome; Prospective Studies; Severity of Illness Index; Substance Withdrawal Syndrome; Treatment Outcome

2000
A comparative evaluation of the effects of oral lorazepam, alprazolam and diazepam on venous admixture.
    The Journal of the Association of Physicians of India, 2002, Volume: 50

    Topics: Administration, Oral; Adult; Alprazolam; Blood Gas Analysis; Diazepam; Female; Humans; Hypnotics and Sedatives; Lorazepam; Male; Middle Aged; Preanesthetic Medication

2002
[Evaluation of the usefulness and effectiveness of anxiolytic therapies in neoplastic diseases].
    Polski merkuriusz lekarski : organ Polskiego Towarzystwa Lekarskiego, 2004, Volume: 16, Issue:96

    Topics: Adult; Aged; Alprazolam; Anti-Anxiety Agents; Antineoplastic Combined Chemotherapy Protocols; Anxiety; Depression; Diazepam; Female; Humans; Male; Middle Aged; Neoplasms; Psychiatric Status Rating Scales; Treatment Outcome

2004
Efficacy and Safety of Anxiolytics in Mohs Micrographic Surgery: A Randomized, Double-Blinded, Placebo-Controlled Trial.
    Dermatologic surgery : official publication for American Society for Dermatologic Surgery [et al.], 2023, 11-01, Volume: 49, Issue:11

    Topics: Alprazolam; Anti-Anxiety Agents; Anxiety; Diazepam; Double-Blind Method; Gabapentin; Humans; Lorazepam; Melatonin; Mohs Surgery; Pregabalin

2023

Other Studies

147 other study(ies) available for diazepam and alprazolam

ArticleYear
Synthesis and pharmacology of novel anxiolytic agents derived from 2-[(dialkylamino)methyl-4H-triazol-4-yl] benzophenones and related heterocyclic benzophenones.
    Journal of medicinal chemistry, 1976, Volume: 19, Issue:8

    Topics: Animals; Anti-Anxiety Agents; Benzophenones; Drug Synergism; Electroshock; Ethanol; Male; Mice; Nicotine; Pentylenetetrazole; Semicarbazides; Strychnine; Triazoles

1976
Novel anxiolytic agents derived from alpha-amino-alpha-phenyl-o-tolyl-4H-triazoles and -imidazoles.
    Journal of medicinal chemistry, 1978, Volume: 21, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Brain; Crystallography; Hypnotics and Sedatives; Imidazoles; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Mice; Models, Molecular; Molecular Conformation; Muscle Relaxation; Nicotine; Pentylenetetrazole; Rats; Seizures; Semicarbazides; Triazoles

1978
Pharmacology of some metabolites of triazolam, alprazolam, and diazepam prepared by a simple, one-step oxidation of benzodiazepines.
    Journal of medicinal chemistry, 1978, Volume: 21, Issue:12

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Diazepam; Hydroxylation; Male; Methods; Mice; Oxidation-Reduction; Triazolam; Triazoles

1978
6-Aryl-4H-s-triazolo[4,3-a][1,4]benzodiazepines. Influence of 1-substitution on pharmacological activity.
    Journal of medicinal chemistry, 1979, Volume: 22, Issue:11

    Topics: Animals; Anti-Anxiety Agents; Apomorphine; Benzodiazepines; Body Temperature; Dextroamphetamine; Male; Mice; Motor Activity; Structure-Activity Relationship

1979
Quinazolines and 1,4-benzodiazepines. 81. s-Triazolo[4,3-a][1,4]benzodiazepines by oxidative cyclization of hydrazones.
    Journal of medicinal chemistry, 1977, Volume: 20, Issue:12

    Topics: Animals; Benzodiazepines; Central Nervous System; Chemical Phenomena; Chemistry; Cyclization; Hydrazones; Mice; Oxidation-Reduction; Structure-Activity Relationship; Triazoles

1977
6-(Substituted-amino)-4H-s-triazolo[4,3-a][1,4]benzodiazepines and 4-(substituted-amino)-6H-s-triazolo[4,3-a][1,4]benzodiazepines with potential antianxiety activity.
    Journal of medicinal chemistry, 1980, Volume: 23, Issue:8

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Isomerism; Male; Mice; Models, Molecular; Triazoles

1980
Predicting blood-brain barrier permeation from three-dimensional molecular structure.
    Journal of medicinal chemistry, 2000, Jun-01, Volume: 43, Issue:11

    Topics: Blood-Brain Barrier; Databases, Factual; Models, Chemical; Molecular Conformation; Multivariate Analysis; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
ElogD(oct): a tool for lipophilicity determination in drug discovery. 2. Basic and neutral compounds.
    Journal of medicinal chemistry, 2001, Jul-19, Volume: 44, Issue:15

    Topics: 1-Octanol; Chromatography, High Pressure Liquid; Pharmaceutical Preparations; Solubility; Water

2001
Prediction of volume of distribution values in humans for neutral and basic drugs using physicochemical measurements and plasma protein binding data.
    Journal of medicinal chemistry, 2002, Jun-20, Volume: 45, Issue:13

    Topics: Blood Proteins; Chemical Phenomena; Chemistry, Physical; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding

2002
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Air to lung partition coefficients for volatile organic compounds and blood to lung partition coefficients for volatile organic compounds and drugs.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:3

    Topics: Air; Animals; Humans; Lung; Organic Chemicals; Probability; Rats; Tissue Distribution; Volatilization

2008
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Experimental solubility profiling of marketed CNS drugs, exploring solubility limit of CNS discovery candidate.
    Bioorganic & medicinal chemistry letters, 2010, Dec-15, Volume: 20, Issue:24

    Topics: Central Nervous System Agents; Drug Evaluation, Preclinical; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Solubility

2010
Measurement of unbound drug exposure in brain: modeling of pH partitioning explains diverging results between the brain slice and brain homogenate methods.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:3

    Topics: Animals; Biological Transport; Brain; Chemical Phenomena; Dialysis; Hydrogen-Ion Concentration; In Vitro Techniques; Lysosomes; Male; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Tissue Distribution

2011
A high-throughput cell-based method to predict the unbound drug fraction in the brain.
    Journal of medicinal chemistry, 2014, Apr-10, Volume: 57, Issue:7

    Topics: Animals; Brain; Dialysis; HEK293 Cells; High-Throughput Screening Assays; Humans; Pharmaceutical Preparations; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization

2014
Development of Piperazinediones as dual inhibitor for treatment of Alzheimer's disease.
    European journal of medicinal chemistry, 2018, Apr-25, Volume: 150

    Topics: Acetylcholinesterase; Alzheimer Disease; Butyrylcholinesterase; Diketopiperazines; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Matrix Metalloproteinase 2; Molecular Structure; Neuroprotective Agents; Structure-Activity Relationship

2018
Design and development of some phenyl benzoxazole derivatives as a potent acetylcholinesterase inhibitor with antioxidant property to enhance learning and memory.
    European journal of medicinal chemistry, 2019, Feb-01, Volume: 163

    Topics: Antioxidants; Benzoxazoles; Cholinesterase Inhibitors; Drug Design; Humans; Learning; Memory; Pharmacokinetics; Quantitative Structure-Activity Relationship

2019
Rationalizing the binding and α subtype selectivity of synthesized imidazodiazepines and benzodiazepines at GABAA receptors by using molecular docking studies.
    Bioorganic & medicinal chemistry letters, 2022, 04-15, Volume: 62

    Topics: Alprazolam; Benzodiazepines; Chlorine; Diazepam; gamma-Aminobutyric Acid; Ion Channels; Ligands; Molecular Docking Simulation; Receptors, GABA; Receptors, GABA-A

2022
Synthesis and evaluation of dual fatty acid amide hydrolase-monoacylglycerol lipase inhibition and antinociceptive activities of 4-methylsulfonylaniline-derived semicarbazones.
    Bioorganic & medicinal chemistry, 2022, 04-15, Volume: 60

    Topics: Amidohydrolases; Analgesics; Enzyme Inhibitors; Humans; Molecular Docking Simulation; Monoacylglycerol Lipases; Neuralgia; Semicarbazones

2022
Design, synthesis, in-vitro, in-vivo and ex-vivo pharmacology of thiazolidine-2,4-dione derivatives as selective and reversible monoamine oxidase-B inhibitors.
    Bioorganic & medicinal chemistry letters, 2022, 11-15, Volume: 76

    Topics: Hydrazones; Molecular Docking Simulation; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Structure-Activity Relationship; Thiazolidines

2022
Antidepressant and anxiolytic effects of alprazolam versus the conventional antidepressant desipramine and the anxiolytic diazepam in the forced swim test in rats.
    European journal of pharmacology, 1992, Apr-22, Volume: 214, Issue:2-3

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Antidepressive Agents; Buspirone; Depression; Desipramine; Diazepam; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Serotonin; Swimming

1992
Detection of benzodiazepines in human hair by radioimmunoassay.
    The Annals of pharmacotherapy, 1992, Volume: 26, Issue:4

    Topics: Adult; Alprazolam; Benzodiazepines; Diazepam; Female; Hair; Humans; Lorazepam; Male; Middle Aged; Radioimmunoassay

1992
SPECT imaging of the benzodiazepine receptor: feasibility of in vivo potency measurements from stepwise displacement curves.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1991, Volume: 32, Issue:9

    Topics: Alprazolam; Animals; Benzodiazepines; Brain; Brain Chemistry; Clonazepam; Diazepam; Female; Flumazenil; Injections, Intravenous; Macaca mulatta; Male; Papio; Receptors, GABA-A; Tomography, Emission-Computed, Single-Photon

1991
The discriminative stimulus effects of diazepam in rats at two training doses.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:3

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Buspirone; Carbolines; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Flumazenil; Male; Morphine; Pentobarbital; Pyrazoles; Pyridazines; Rats; Rats, Inbred Strains; Triazolam

1991
Snorting benzodiazepines.
    The American journal of drug and alcohol abuse, 1991, Volume: 17, Issue:4

    Topics: Administration, Intranasal; Adult; Alprazolam; Anti-Anxiety Agents; Arousal; Bipolar Disorder; Diazepam; Female; Humans; Male; Personality Disorders; Substance Withdrawal Syndrome; Substance-Related Disorders

1991
Handling-habituation prevents the effects of diazepam and alprazolam on brain serotonin levels in rats.
    Behavioural brain research, 1990, Jan-22, Volume: 36, Issue:3

    Topics: Alprazolam; Animals; Arousal; Brain; Cerebral Cortex; Diazepam; Habituation, Psychophysiologic; Handling, Psychological; Hippocampus; Hydroxyindoleacetic Acid; Hypothalamus; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Synaptic Transmission

1990
Alprazolam enhances the antibacterial activity exerted by normal human peripheral blood lymphocytes.
    Acta neurologica, 1991, Volume: 13, Issue:5

    Topics: Adjuvants, Immunologic; Adult; Alprazolam; Antibody-Dependent Cell Cytotoxicity; Cytotoxicity Tests, Immunologic; Diazepam; Female; Humans; Male; Salmonella typhi; Stimulation, Chemical; T-Lymphocyte Subsets

1991
Benzodiazepine withdrawal.
    The American journal of psychiatry, 1991, Volume: 148, Issue:11

    Topics: Alprazolam; Benzodiazepines; Diazepam; Humans; Substance Withdrawal Syndrome; Time Factors

1991
Effects of different handling-stimulation procedures and benzodiazepines on two-way active avoidance acquisition in rats.
    Pharmacological research, 1991, Volume: 24, Issue:3

    Topics: Alprazolam; Analysis of Variance; Animals; Anxiety; Avoidance Learning; Diazepam; Habituation, Psychophysiologic; Handling, Psychological; Male; Rats; Rats, Inbred Strains

1991
"Ex vivo" binding of 35S-TBPS as a tool to study the pharmacology of GABAA receptors.
    Advances in biochemical psychopharmacology, 1990, Volume: 46

    Topics: Alprazolam; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Convulsants; Diazepam; Drug Synergism; Ethanol; In Vitro Techniques; Isoniazid; Male; Protein Conformation; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological; Sulfur Radioisotopes; Valproic Acid

1990
Physical dependence induced in DBA/2J mice by benzodiazepine receptor full agonists, but not by the partial agonist Ro 16-6028.
    European journal of pharmacology, 1990, Nov-06, Volume: 190, Issue:1-2

    Topics: Administration, Oral; Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepinones; Diazepam; Drug Implants; Mice; Mice, Inbred DBA; Receptors, GABA-A; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam

1990
Panic disorder: strategies for long-term treatment.
    The Journal of clinical psychiatry, 1991, Volume: 52 Suppl

    Topics: Adolescent; Adult; Alprazolam; Anxiety Disorders; Diazepam; Female; Humans; Panic

1991
Reduction of gastrointestinal symptoms following treatment for panic disorder.
    Psychosomatics, 1990,Winter, Volume: 31, Issue:1

    Topics: Adult; Alprazolam; Anxiety Disorders; Colonic Diseases, Functional; Diazepam; Fear; Female; Gastrointestinal Diseases; Humans; Male; Middle Aged; Panic

1990
Effects of chronic alprazolam treatment on plasma concentrations of glucocorticoids, thyroid hormones, and testosterone in cardiomyopathic hamsters.
    Psychopharmacology, 1989, Volume: 98, Issue:3

    Topics: Alprazolam; Animals; Cardiomyopathies; Cricetinae; Diazepam; Glucocorticoids; Male; Testosterone; Thyroid Hormones

1989
Effects of chronic antidepressant and benzodiazepine treatment on corticotropin-releasing-factor receptors in rat brain and pituitary.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1989, Volume: 2, Issue:1

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Antidepressive Agents; Benzodiazepines; Brain; Desipramine; Diazepam; Imipramine; Male; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains; Receptors, Corticotropin-Releasing Hormone; Receptors, Neurotransmitter; Receptors, Serotonin

1989
Alpha 2-adrenoceptor antagonists potentiate the anticonflict and the rotarod impairing effects of benzodiazepines.
    Journal of neural transmission, 1989, Volume: 76, Issue:3

    Topics: Adrenergic alpha-Antagonists; Alprazolam; Animals; Anxiety; Diazepam; Dioxanes; Dioxins; Idazoxan; Male; Rats; Rats, Inbred Strains

1989
Adjunctive buspirone in benzodiazepine treatment of four patients with panic disorder.
    The American journal of psychiatry, 1989, Volume: 146, Issue:7

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Anxiety; Buspirone; Clonazepam; Diazepam; Drug Combinations; Fear; Female; Humans; Male; Middle Aged; Panic; Phobic Disorders

1989
Motor phenomena in benzodiazepine withdrawal.
    Hospital & community psychiatry, 1989, Volume: 40, Issue:12

    Topics: Aged; Alprazolam; Anti-Anxiety Agents; Diagnosis, Differential; Diazepam; Drug Therapy, Combination; Female; Humans; Muscle Rigidity; Sleep Initiation and Maintenance Disorders; Substance Withdrawal Syndrome; Triazolam; Urinary Incontinence

1989
Alprazolam but not diazepam protects hamsters with heart disease from the medical consequences of stress.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 33, Issue:3

    Topics: Alprazolam; Animals; Behavior, Animal; Cardiomyopathies; Cold Temperature; Cricetinae; Diazepam; Mesocricetus; Restraint, Physical; Stress, Physiological

1989
The relationship of panic disorder and its treatment outcome to 24-hour urinary MHPG levels.
    Psychiatry research, 1989, Volume: 30, Issue:1

    Topics: Adolescent; Adult; Aged; Alprazolam; Anxiety Disorders; Diazepam; Double-Blind Method; Fear; Glycols; Humans; Methoxyhydroxyphenylglycol; Middle Aged; Panic; Random Allocation

1989
Anticonflict and rotarod impairing effects of alprazolam and diazepam in rat after acute and subchronic administration.
    Progress in neuro-psychopharmacology & biological psychiatry, 1989, Volume: 13, Issue:1-2

    Topics: Alprazolam; Animals; Conflict, Psychological; Diazepam; Drug Administration Schedule; Injections, Intraperitoneal; Male; Motivation; Rats; Rats, Inbred Strains; Reference Values; Water Deprivation

1989
Peripheral, but not local or intracerebroventricular, administration of benzodiazepines attenuates evoked activity of locus coeruleus neurons.
    Brain research, 1989, Jun-26, Volume: 490, Issue:2

    Topics: Action Potentials; Alprazolam; Animals; Benzodiazepines; Chlordiazepoxide; Diazepam; Dose-Response Relationship, Drug; Injections, Intraventricular; Locus Coeruleus; Male; Rats; Rats, Inbred Strains

1989
Antidepressant properties of the triazolobenzodiazepines alprazolam and adinazolam: studies on the olfactory bulbectomized rat model of depression.
    British journal of clinical pharmacology, 1985, Volume: 19 Suppl 1

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Antidepressive Agents; Benzodiazepines; Biogenic Amines; Body Weight; Brain Chemistry; Choice Behavior; Depressive Disorder; Diazepam; Feeding Behavior; Humans; Male; Neurotransmitter Agents; Olfactory Bulb; Phenobarbital; Rats; Rats, Inbred Strains

1985
Drugs in dentistry. Agents for anxiety disorders.
    Dental management, 1985, Volume: 25, Issue:6

    Topics: Alprazolam; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Chlordiazepoxide; Clorazepate Dipotassium; Dental Care; Diazepam; Humans; Oxazepam

1985
Alprazolam withdrawal delirium unresponsive to diazepam: case report.
    The Journal of clinical psychiatry, 1985, Volume: 46, Issue:8

    Topics: Aged; Alprazolam; Anti-Anxiety Agents; Benzodiazepines; Delirium; Diazepam; Half-Life; Humans; Male; Receptors, GABA-A; Substance Withdrawal Syndrome

1985
Does alprazolam, in contrast to diazepam, activate alpha 2-adrenoceptors involved in the regulation of rat growth hormone secretion?
    Life sciences, 1986, Apr-21, Volume: 38, Issue:16

    Topics: Adrenergic alpha-Antagonists; Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Clonidine; Diazepam; Dioxanes; Growth Hormone; Idazoxan; Kinetics; Male; Rats; Receptors, Adrenergic, alpha; Reserpine; Yohimbine

1986
Chronic use of benzodiazepines and psychomotor and cognitive test performance.
    Psychopharmacology, 1986, Volume: 88, Issue:4

    Topics: Adult; Affect; Aged; Alprazolam; Anti-Anxiety Agents; Benzodiazepines; Clorazepate Dipotassium; Cognition Disorders; Diazepam; Female; Flicker Fusion; Humans; Lorazepam; Male; Memory Disorders; Middle Aged; Neuropsychological Tests; Psychomotor Disorders

1986
Biological markers in panic states: lactate-induced panic and mitral valve prolapse.
    Biological psychiatry, 1987, Volume: 22, Issue:3

    Topics: Adolescent; Adult; Aged; Agoraphobia; Alprazolam; Anti-Anxiety Agents; Anxiety Disorders; Creatinine; Diazepam; Double-Blind Method; Fear; Humans; Lactates; Lactic Acid; Methoxyhydroxyphenylglycol; Middle Aged; Mitral Valve Prolapse; Panic

1987
Comparative pharmacodynamics of benzodiazepines.
    Psychopharmacology series, 1987, Volume: 3

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Humans; Kinetics; Lorazepam; Male; Psychomotor Performance; Triazolam

1987
Alprazolam dependence in mice.
    Alcohol and drug research, 1987, Volume: 7, Issue:5-6

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Diazepam; Male; Mice; Models, Psychological; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors

1987
Preference for alprazolam over diazepam.
    The American journal of psychiatry, 1989, Volume: 146, Issue:3

    Topics: Alprazolam; Attitude; Diazepam; Humans; Risk Factors; Substance-Related Disorders

1989
Ultrasonic vocalization in response to unavoidable aversive stimuli in rats: effects of benzodiazepines.
    Life sciences, 1988, Volume: 43, Issue:6

    Topics: Alprazolam; Animals; Benzodiazepines; Desipramine; Diazepam; Electroshock; Flumazenil; Haloperidol; Male; Rats; Rats, Inbred Strains; Ultrasonics; Vocalization, Animal

1988
Increased central noradrenergic activity during benzodiazepine withdrawal: an electrophysiological study.
    Neuropharmacology, 1988, Volume: 27, Issue:11

    Topics: Action Potentials; Alprazolam; Animals; Cerebellum; Diazepam; Lorazepam; Norepinephrine; Purkinje Cells; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome

1988
The abnormal open-field behavior of SART-stressed rats and effects of some drugs on it.
    Japanese journal of pharmacology, 1988, Volume: 48, Issue:4

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepines; Chlorpromazine; Diazepam; Dibenzazepines; Imipramine; Male; Motor Activity; Polysaccharides; Rats; Rats, Inbred Strains; Stress, Physiological

1988
The anxiolytic action of benzodiazepines is not present in handling-habituated rats.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 31, Issue:3

    Topics: Alprazolam; Animals; Avoidance Learning; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Handling, Psychological; Male; Rats; Rats, Inbred Strains; Touch

1988
The seeking and liking potentials of alprazolam.
    The American journal of psychiatry, 1988, Volume: 145, Issue:1

    Topics: Adult; Alprazolam; Diazepam; Female; Humans; Male; Substance Withdrawal Syndrome; Substance-Related Disorders

1988
Triazolam withdrawal.
    The Journal of clinical psychiatry, 1988, Volume: 49, Issue:9

    Topics: Alprazolam; Diazepam; Drug Tolerance; Humans; Seizures; Substance Withdrawal Syndrome; Triazolam

1988
Triazolobenzodiazepines competitively inhibit the binding of platelet activating factor (PAF) to human platelets.
    Biochemical and biophysical research communications, 1987, Apr-14, Volume: 144, Issue:1

    Topics: Alprazolam; Binding, Competitive; Blood Platelets; Diazepam; Humans; In Vitro Techniques; Kinetics; Platelet Activating Factor; Platelet Aggregation; Triazolam

1987
Alprazolam withdrawal.
    Drug intelligence & clinical pharmacy, 1987, Volume: 21, Issue:9

    Topics: Adult; Alprazolam; Diazepam; Humans; Male; Substance Withdrawal Syndrome

1987
Effect of chronic administration of alprazolam and adinazolam on clonidine- or apomorphine-induced aggression in laboratory rodents.
    Neuropharmacology, 1986, Volume: 25, Issue:7

    Topics: Aggression; Alprazolam; Animals; Anti-Anxiety Agents; Apomorphine; Benzodiazepines; Clonidine; Desipramine; Diazepam; Drug Interactions; Male; Mice; Rats; Rats, Inbred Strains

1986
Determination of biological activity of alprazolam, triazolam and their metabolites.
    The Journal of pharmacy and pharmacology, 1982, Volume: 34, Issue:2

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Binding, Competitive; Brain; Diazepam; Flunitrazepam; Kinetics; Male; Membranes; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A; Triazolam

1982
Benzodiazepine receptor number after acute administration of alprazolam and diazepam.
    Research communications in chemical pathology and pharmacology, 1982, Volume: 35, Issue:2

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Binding, Competitive; Brain; Diazepam; Flunitrazepam; In Vitro Techniques; Kinetics; Male; Membranes; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A

1982
Alprazolam in a biochemical model of depression.
    Biochemical pharmacology, 1982, Oct-01, Volume: 31, Issue:19

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Depression; Diazepam; Disease Models, Animal; Drug Evaluation, Preclinical; Female; Humans; Imipramine; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Reserpine

1982
Benzodiazepines: drug discrimination and physiological dependence.
    NIDA research monograph, 1984, Volume: 49

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Bromazepam; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Generalization, Stimulus; Humans; Lorazepam; Papio; Pentobarbital; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam

1984
Role of beta-adrenergic receptors in the antidepressant activity of alprazolam.
    Research communications in chemical pathology and pharmacology, 1982, Volume: 36, Issue:2

    Topics: Alprazolam; Animals; Antidepressive Agents; Benzodiazepines; Diazepam; Dihydroalprenolol; Female; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Reserpine

1982
Propranolol interactions with diazepam, lorazepam, and alprazolam.
    Clinical pharmacology and therapeutics, 1984, Volume: 36, Issue:4

    Topics: Adolescent; Adult; Alprazolam; Benzodiazepines; Biotransformation; Chromatography, High Pressure Liquid; Diazepam; Drug Interactions; Female; Humans; Injections, Intravenous; Kinetics; Lorazepam; Male; Nordazepam; Propranolol

1984
Effects of psychoactive drugs on plasma catecholamines during stress in rats.
    Neuropharmacology, 1984, Volume: 23, Issue:9

    Topics: Alprazolam; Amphetamine; Animals; Benzodiazepines; Diazepam; Epinephrine; Humans; Male; Morphine; Norepinephrine; Pentobarbital; Psychotropic Drugs; Rats; Rats, Inbred Strains; Stress, Psychological; Time Factors

1984
In vitro method for detecting precipitation of parenteral formulations after injection.
    Journal of pharmaceutical sciences, 1983, Volume: 72, Issue:9

    Topics: Alprazolam; Benzodiazepines; Chemical Precipitation; Chemistry, Pharmaceutical; Diazepam; Injections; Solubility; Solutions

1983
Serum dopamine-beta-hydroxylase activity in depression and anxiety.
    Biological psychiatry, 1984, Volume: 19, Issue:4

    Topics: Adult; Aged; Alprazolam; Anxiety; Anxiety Disorders; Benzodiazepines; Depression; Depressive Disorder; Diazepam; Dopamine beta-Hydroxylase; Double-Blind Method; Female; Humans; Imipramine; Longitudinal Studies; Male; Middle Aged

1984
Precipitated withdrawal in squirrel monkeys after repeated daily oral administration of alprazolam, diazepam, flunitrazepam or oxazepam.
    Psychopharmacology, 1995, Volume: 118, Issue:3

    Topics: Administration, Oral; Alprazolam; Animals; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Drug Tolerance; Female; Flumazenil; Flunitrazepam; Male; Muscle Relaxation; Oxazepam; Saimiri; Sleep; Substance Withdrawal Syndrome; Substance-Related Disorders; Tremor

1995
Effects of desipramine and alprazolam on forced swimming behaviour of adult rats exposed to prenatal diazepam.
    European journal of pharmacology, 1995, Feb-06, Volume: 273, Issue:3

    Topics: Alprazolam; Animals; Behavior, Animal; Depression; Desipramine; Diazepam; Electroencephalography; Electrophysiology; Female; Hippocampus; Injections; Locus Coeruleus; Male; Motor Activity; Picrotoxin; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Wistar; Receptors, GABA; Swimming

1995
Identification of parent benzodiazepines by gas chromotography/mass spectroscopy (GC/MS) from urinary extracts treated with B-glucuronidase.
    Forensic science international, 1995, May-09, Volume: 73, Issue:1

    Topics: Alprazolam; Benzodiazepines; Chlordiazepoxide; Clonazepam; Diazepam; Gas Chromatography-Mass Spectrometry; Glucuronidase; Humans; Lorazepam; Oxazepam; Triazolam

1995
Benzodiazepine sensitivity in panic disorder: effects of chronic alprazolam treatment.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1995, Volume: 12, Issue:2

    Topics: Adult; Alprazolam; Diazepam; Dose-Response Relationship, Drug; Drug Tolerance; Female; Growth Hormone; Heart Rate; Humans; Hydrocortisone; Male; Memory, Short-Term; Panic Disorder; Receptors, GABA-A; Saccades

1995
Alprazolam modifies animal behaviour on elevated plus-maze.
    Indian journal of experimental biology, 1993, Volume: 31, Issue:11

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Diazepam; Learning; Mice; Mice, Inbred BALB C; Substance-Related Disorders

1993
Benzodiazepines antagonize central corticotropin releasing hormone-induced suppression of natural killer cell activity.
    Brain research, 1993, Dec-17, Volume: 631, Issue:1

    Topics: Alprazolam; Animals; Benzodiazepines; Brain; Corticotropin-Releasing Hormone; Diazepam; Injections, Intraventricular; Killer Cells, Natural; Male; Pituitary-Adrenal System; Rats; Rats, Wistar

1993
Characterization of the binding and comparison of the distribution of benzodiazepine receptors labeled with [3H]diazepam and [3H]alprazolam.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1993, Volume: 8, Issue:4

    Topics: Alprazolam; Animals; Autoradiography; Brain; Diazepam; In Vitro Techniques; Male; Radioligand Assay; Rats; Receptors, GABA-A; Tritium

1993
The use of the rat elevated plus-maze to discriminate between non-selective and BZ-1 (omega 1) selective, benzodiazepine receptor ligands.
    Psychopharmacology, 1996, Volume: 124, Issue:3

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Chlordiazepoxide; Diazepam; GABA-A Receptor Agonists; Male; Motor Activity; Rats; Rats, Sprague-Dawley

1996
Catatonia after benzodiazepine withdrawal.
    Journal of clinical psychopharmacology, 1996, Volume: 16, Issue:4

    Topics: Aged; Aged, 80 and over; Alprazolam; Anti-Anxiety Agents; Catatonia; Clonazepam; Diazepam; Female; Humans; Male; Middle Aged; Substance Withdrawal Syndrome

1996
Use of benzodiazepines in elderly patients.
    Mayo Clinic proceedings, 1996, Volume: 71, Issue:11

    Topics: Aged; Alprazolam; Anti-Anxiety Agents; Diazepam; Drug Utilization; Half-Life; Humans

1996
Behavioural responsiveness to picrotoxin and desipramine in adult rats prenatally exposed to different benzodiazepine receptor agonists.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1995, Volume: 5, Issue:4

    Topics: Adrenergic Uptake Inhibitors; Alprazolam; Animals; Behavior, Animal; Desipramine; Diazepam; Female; GABA Antagonists; GABA Modulators; GABA-A Receptor Agonists; Hypnotics and Sedatives; Male; Picrotoxin; Pregnancy; Prenatal Exposure Delayed Effects; Pyridines; Rats; Rats, Wistar; Seizures; Zolpidem

1995
Assessment of the anxiolytic and amnesic effects of three benzodiazepines, diazepam, alprazolam and triazolam, by conflict and non-matching to sample tests in mice.
    Nihon shinkei seishin yakurigaku zasshi = Japanese journal of psychopharmacology, 1997, Volume: 17, Issue:1

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Conflict, Psychological; Diazepam; Male; Maze Learning; Memory; Mice; Triazolam

1997
Ultrasonic vocalizations in rat pups: modulation at the gamma-aminobutyric acidA receptor complex and the neurosteroid recognition site.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 282, Issue:1

    Topics: Alprazolam; Animals; Diazepam; Female; Male; Muscimol; Pentobarbital; Pregnanolone; Rats; Receptors, GABA-A; Vocalization, Animal

1997
Alprazolam, diazepam, yohimbine, clonidine: in vivo CA1 hippocampal norepinephrine and serotonin release profiles under chloral hydrate anesthesia.
    Progress in neuro-psychopharmacology & biological psychiatry, 1997, Volume: 21, Issue:7

    Topics: Adrenergic alpha-Antagonists; Alprazolam; Anesthetics, Intravenous; Animals; Anti-Anxiety Agents; Anxiety; Chloral Hydrate; Clonidine; Diazepam; Hippocampus; Male; Microelectrodes; Rats; Rats, Sprague-Dawley; Serotonin; Time Factors; Yohimbine

1997
Locomotor and antidepressant-like effects of 5-HT(1A) agonist LY 228729 in prenatally benzodiazepine-exposed rats.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1998, Volume: 8, Issue:1

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Antidepressive Agents; Depressive Disorder; Diazepam; Ergolines; Female; Injections, Subcutaneous; Male; Motor Activity; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Sprague-Dawley; Serotonin Receptor Agonists; Stereotyped Behavior; Swimming

1998
Gabapentin as a potential treatment for anxiety disorders.
    The American journal of psychiatry, 1998, Volume: 155, Issue:7

    Topics: Acetates; Adult; Alprazolam; Amines; Anticonvulsants; Anxiety Disorders; Cyclohexanecarboxylic Acids; Diazepam; Drug Administration Schedule; Drug Therapy, Combination; Female; Fluoxetine; Gabapentin; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Panic Disorder; Phobic Disorders

1998
A new approach to the light/dark test procedure in mice.
    Pharmacology, biochemistry, and behavior, 1998, Volume: 60, Issue:3

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Behavior, Animal; Carbolines; Central Nervous System Stimulants; Diazepam; GABA Antagonists; Male; Mice; Mice, Inbred C57BL; Motor Activity

1998
Determination of benzodiazepines in human urine and plasma with solvent modified solid phase micro extraction and gas chromatography; rationalisation of method development using experimental design strategies.
    Journal of pharmaceutical and biomedical analysis, 1998, Volume: 18, Issue:4-5

    Topics: Alprazolam; Anti-Anxiety Agents; Benzodiazepines; Chromatography, Gas; Diazepam; Flunitrazepam; Humans; Hydrogen-Ion Concentration; Models, Chemical; Nordazepam; Oxazepam; Research Design

1998
A synthetic agonist at the orphanin FQ/nociceptin receptor ORL1: anxiolytic profile in the rat.
    Proceedings of the National Academy of Sciences of the United States of America, 2000, Apr-25, Volume: 97, Issue:9

    Topics: Acoustic Stimulation; Alprazolam; Animals; Anti-Anxiety Agents; Cognition; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Electroshock; Epilepsy; Fear; Humans; Imidazoles; Male; Maze Learning; Nociceptin Receptor; Pain; Pentylenetetrazole; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Recombinant Proteins; Reflex, Startle; Seizures; Self Stimulation; Spiro Compounds

2000
Oral sedation allows for comfort and amnesia during office surgery.
    Annals of plastic surgery, 2000, Volume: 44, Issue:5

    Topics: Acetaminophen; Adult; Alprazolam; Ambulatory Surgical Procedures; Amnesia; Analgesics, Non-Narcotic; Analgesics, Opioid; Anesthetics, Local; Anti-Anxiety Agents; Antibiotic Prophylaxis; Conscious Sedation; Diazepam; Epinephrine; Female; Humans; Hydrocodone; Lidocaine; Male; Plastic Surgery Procedures; Treatment Outcome; Vasoconstrictor Agents

2000
Sedative and anxiolytic effects of zopiclone's enantiomers and metabolite.
    European journal of pharmacology, 2001, Volume: 415, Issue:2-3

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Anticonvulsants; Anxiety; Azabicyclo Compounds; Diazepam; Dose-Response Relationship, Drug; Electroshock; Hypnotics and Sedatives; Isomerism; Male; Motor Activity; Motor Skills; Piperazines; Rats; Rats, Long-Evans; Seizures

2001
Electrospray ionization gas-phase electrophoresis under ambient conditions and it's potential or high-speed separations.
    Fresenius' journal of analytical chemistry, 2001, Volume: 369, Issue:3-4

    Topics: Alprazolam; Anti-Anxiety Agents; Combinatorial Chemistry Techniques; Diazepam; Electrophoresis; Equipment Design; Herbicides; Nitrazepam; Oxazepam; Prazepam; Time Factors; Triazines

2001
What are the issues surrounding long-term benzodiazepine treatment for generalized anxiety disorder.
    Journal of psychiatry & neuroscience : JPN, 1998, Volume: 23, Issue:1

    Topics: Adult; Alprazolam; Anxiety Disorders; Benzodiazepines; Diazepam; Drug Administration Schedule; Female; Humans

1998
[Does the addition of an anxiolytic drug improve the anti-emetic effectiveness of the steroid and granisetron combination in the prophylaxis of cisplatin-induced vomiting?].
    Orvosi hetilap, 2001, Aug-05, Volume: 142, Issue:31

    Topics: Alprazolam; Anti-Anxiety Agents; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Cisplatin; Dexamethasone; Diazepam; Droperidol; Drug Administration Schedule; Drug Therapy, Combination; Female; Genital Neoplasms, Female; Granisetron; Humans; Meprobamate; Middle Aged; Treatment Outcome; Vomiting

2001
Orally delivered alprazolam, diazepam, and triazolam as reinforcers in rhesus monkeys.
    Psychopharmacology, 2002, Volume: 161, Issue:1

    Topics: Administration, Oral; Alprazolam; Animals; Anti-Anxiety Agents; Diazepam; Macaca mulatta; Male; Reinforcement, Psychology; Self Administration; Triazolam

2002
GABA(A)-benzodiazepine receptor complex sensitivity in 5-HT(1A) receptor knockout mice on a 129/Sv background.
    European journal of pharmacology, 2002, Jun-28, Volume: 447, Issue:1

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Diazepam; Ethanol; Fever; Flumazenil; GABA Antagonists; Hypnotics and Sedatives; Male; Maze Learning; Mice; Mice, Knockout; Pentylenetetrazole; Phenobarbital; Receptors, GABA-A; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Reflex; Species Specificity; Stress, Physiological

2002
Prenatal exposure to diazepam and alprazolam, but not to zolpidem, affects behavioural stress reactivity in handling-naïve and handling-habituated adult male rat progeny.
    Brain research, 2002, Oct-25, Volume: 953, Issue:1-2

    Topics: Age Factors; Alprazolam; Animals; Anti-Anxiety Agents; Behavior, Animal; Convulsants; Diazepam; Exploratory Behavior; Female; GABA Agonists; Habituation, Psychophysiologic; Handling, Psychological; Male; Picrotoxin; Pregnancy; Prenatal Exposure Delayed Effects; Pyridines; Rats; Rats, Wistar; Reflex; Reflex, Startle; Stress, Physiological; Swimming; Zolpidem

2002
Detection of the adulteration of traditional alcoholic beverages by the separation and determination of alprazolam, chloralhydrate and diazepam using reversed-phase high-performance liquid chromatography.
    Analytical sciences : the international journal of the Japan Society for Analytical Chemistry, 2004, Volume: 20, Issue:2

    Topics: Alcoholic Beverages; Alprazolam; Chloral Hydrate; Chromatography, High Pressure Liquid; Diazepam; Reference Standards; Sensitivity and Specificity

2004
Anxiolytic suppression of repetitive transcranial magnetic stimulation-induced anxiety in the rats.
    Progress in neuro-psychopharmacology & biological psychiatry, 2005, Volume: 29, Issue:5

    Topics: Acoustic Stimulation; Alprazolam; Animals; Anti-Anxiety Agents; Anxiety; Buspirone; Diazepam; Electromagnetic Fields; Male; Motor Activity; Rats; Rats, Wistar

2005
Prescription drug abuse among ecstasy users in Miami.
    Journal of addictive diseases, 2005, Volume: 24, Issue:4

    Topics: Adolescent; Adult; Alprazolam; Catchment Area, Health; Diazepam; Drug Prescriptions; Ethnicity; Female; Florida; Humans; Hydrocodone; Male; N-Methyl-3,4-methylenedioxyamphetamine; Oxycodone; Substance-Related Disorders; Surveys and Questionnaires

2005
Oxidative metabolism of limbic structures after acute administration of diazepam, alprazolam and zolpidem.
    Progress in neuro-psychopharmacology & biological psychiatry, 2006, Aug-30, Volume: 30, Issue:6

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Brain Chemistry; Diazepam; Electron Transport Complex IV; Emotions; GABA Modulators; Hypnotics and Sedatives; Immunohistochemistry; Limbic System; Male; Motor Activity; Neurons; Oxidation-Reduction; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Zolpidem

2006
The detection of sedatives in hair and nail samples using tandem LC-MS-MS.
    Forensic science international, 2007, Feb-14, Volume: 166, Issue:1

    Topics: Adult; Aged; Aged, 80 and over; Alprazolam; Azabicyclo Compounds; Benzodiazepines; Chromatography, Liquid; Clobazam; Clonazepam; Diazepam; Female; Forensic Pathology; Hair; Humans; Hypnotics and Sedatives; Male; Mass Spectrometry; Midazolam; Middle Aged; Nails; Oxazepam; Piperazines; Predictive Value of Tests; Rape; Temazepam; Triazolam

2007
Enhanced sucrose pellet consumption induced by benzodiazepine-type drugs in squirrel monkeys: role of GABAA receptor subtypes.
    Psychopharmacology, 2006, Volume: 187, Issue:3

    Topics: Alprazolam; Animals; Benzodiazepines; Diazepam; Flumazenil; Male; Pyridines; Receptors, GABA-A; Saimiri; Sucrose; Zolpidem

2006
Prediction of metabolic clearance using fresh human hepatocytes: comparison with cryopreserved hepatocytes and hepatic microsomes for five benzodiazepines.
    Xenobiotica; the fate of foreign compounds in biological systems, 2008, Volume: 38, Issue:4

    Topics: Alprazolam; Benzodiazepines; Cell Survival; Cells, Cultured; Cryopreservation; Cytochrome P-450 CYP3A; Diazepam; Flunitrazepam; Hepatocytes; Humans; Metabolic Clearance Rate; Microsomes, Liver; Midazolam; Substrate Specificity; Triazolam

2008
Influence of incorporation methods on partitioning behavior of lipophilic drugs into various phases of a parenteral lipid emulsion.
    AAPS PharmSciTech, 2008, Volume: 9, Issue:2

    Topics: Alprazolam; Benzodiazepines; Chemistry, Pharmaceutical; Clonazepam; Diazepam; Drug Carriers; Drug Compounding; Fat Emulsions, Intravenous; Hydrogen-Ion Concentration; Lorazepam; Molecular Structure; Particle Size; Phospholipids; Solubility; Soybean Oil; Technology, Pharmaceutical; Ultracentrifugation

2008
Adverse effects of benzodiazepines in psychiatric outpatients.
    Psychiatria Danubina, 2009, Volume: 21, Issue:1

    Topics: Adult; Alprazolam; Ambulatory Care; Anti-Anxiety Agents; Benzodiazepines; Croatia; Diazepam; Drug Therapy, Combination; Drug Utilization; Female; Humans; Hypnotics and Sedatives; Male; Mental Disorders; Patient Compliance; Surveys and Questionnaires

2009
Microemulsion based intranasal delivery system for treatment of insomnia.
    Drug delivery, 2009, Volume: 16, Issue:3

    Topics: Administration, Intranasal; Alprazolam; Animals; Diazepam; Disease Models, Animal; Drug Compounding; Drug Delivery Systems; Humans; Lorazepam; Male; Rats; Rats, Sprague-Dawley; Sleep; Sleep Initiation and Maintenance Disorders

2009
[Simultaneous determination of 5 sedative hypnotics in human plasma by reversed phase high-performance liquid chromatography].
    Zhong nan da xue xue bao. Yi xue ban = Journal of Central South University. Medical sciences, 2009, Volume: 34, Issue:7

    Topics: Alprazolam; Chromatography, High Pressure Liquid; Diazepam; Estazolam; Humans; Hypnotics and Sedatives; Nitrazepam; Oxazepam

2009
Quantitation of benzodiazepines in blood and urine using gas chromatography-mass spectrometry (GC-MS).
    Methods in molecular biology (Clifton, N.J.), 2010, Volume: 603

    Topics: Alprazolam; Benzodiazepines; Diazepam; Gas Chromatography-Mass Spectrometry; Humans; Lorazepam; Nordazepam; Oxazepam; Solid Phase Extraction; Triazolam

2010
Cytogenetic activity of newly synthesized 1,5-benzodiazepines in normal human lymphocyte cultures.
    Genetic testing and molecular biomarkers, 2010, Volume: 14, Issue:3

    Topics: Adult; Alprazolam; Benzodiazepines; Cell Proliferation; Cells, Cultured; Cytogenetic Analysis; Diazepam; Humans; Lorazepam; Lymphocytes; Mitotic Index; Sister Chromatid Exchange

2010
Measuring anxiety- and locomotion-related behaviours in mice: a new way of using old tests.
    Psychopharmacology, 2010, Volume: 211, Issue:1

    Topics: Adaptation, Ocular; Alprazolam; Analysis of Variance; Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Female; Locomotion; Male; Maze Learning; Mice; Mice, Inbred Strains; Species Specificity; Weights and Measures

2010
Diazepam leads to enhanced severity of orthopoxvirus infection and immune suppression.
    Vaccine, 2010, Aug-31, Volume: 28, Issue:38

    Topics: Alprazolam; Animals; Antibodies, Viral; Antibody Formation; Apoptosis; Body Weight; Cell Proliferation; Cells, Cultured; Cowpox virus; Diazepam; Female; Humans; Immune Tolerance; Mice; Mice, Inbred BALB C; Poxviridae Infections; Spleen; Vaccinia virus

2010
Reduction of fear-potentiated startle by benzodiazepines in C57BL/6J mice.
    Psychopharmacology, 2011, Volume: 213, Issue:4

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Chlordiazepoxide; Diazepam; Dose-Response Relationship, Drug; Fear; GABA Modulators; Male; Mice; Mice, Inbred C57BL; Receptors, GABA-A; Reflex, Startle

2011
A comparative study on the cytogenetic activity of three benzodiazepines in vitro.
    Genetic testing and molecular biomarkers, 2011, Volume: 15, Issue:6

    Topics: Adult; Alprazolam; Benzodiazepines; Cells, Cultured; Chromosome Aberrations; Diazepam; DNA Damage; DNA Repair; Humans; Lorazepam; Lymphocytes; Mutagens; Sister Chromatid Exchange

2011
Role of α1- and α2-GABA(A) receptors in mediating the respiratory changes associated with benzodiazepine sedation.
    British journal of pharmacology, 2012, Volume: 166, Issue:1

    Topics: Alprazolam; Animals; Diazepam; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Hypnotics and Sedatives; Injections, Intraperitoneal; Mice; Mice, Mutant Strains; Plethysmography, Whole Body; Point Mutation; Receptors, GABA-A; Respiration; Time Factors

2012
Risk of fractures requiring hospitalization after an initial prescription for zolpidem, alprazolam, lorazepam, or diazepam in older adults.
    Journal of the American Geriatrics Society, 2011, Volume: 59, Issue:10

    Topics: Aged; Aged, 80 and over; Alprazolam; Causality; Cohort Studies; Cross-Sectional Studies; Diazepam; Female; Fractures, Bone; Health Surveys; Hip Fractures; Hospitalization; Humans; Hypnotics and Sedatives; Joint Dislocations; Lorazepam; Male; Odds Ratio; Pyridines; Retrospective Studies; Risk; Statistics as Topic; Zolpidem

2011
Ethopharmacological evaluation of the rat exposure test: a prey-predator interaction test.
    Behavioural brain research, 2013, Mar-01, Volume: 240

    Topics: Adrenergic alpha-2 Receptor Antagonists; Alprazolam; Animals; Anti-Anxiety Agents; Antidepressive Agents; Caffeine; Central Nervous System Stimulants; Diazepam; Escape Reaction; Factor Analysis, Statistical; Fluoxetine; Food Chain; Imipramine; Male; Mice; Motor Activity; Posture; Predatory Behavior; Rats; Rats, Long-Evans; Time Factors; Yohimbine

2013
Ethopharmacological analysis of the open elevated plus-maze in mice.
    Behavioural brain research, 2013, Jun-01, Volume: 246

    Topics: Adrenergic alpha-2 Receptor Antagonists; Alprazolam; Animals; Anti-Anxiety Agents; Antidepressive Agents, Second-Generation; Convulsants; Corticosterone; Diazepam; Factor Analysis, Statistical; Fluoxetine; Male; Maze Learning; Mice; Pentylenetetrazole; Statistics, Nonparametric; Yohimbine

2013
Dependence of the kinetic and thermodynamic parameters on hydrophilic-lipophilic character of alprazolam, clonazepam, diazepam, doxepin and haloperidol in alkaline environment.
    International journal of pharmaceutics, 2013, Oct-15, Volume: 455, Issue:1-2

    Topics: Alprazolam; Clonazepam; Diazepam; Doxepin; Drug Stability; Haloperidol; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kinetics; Thermodynamics

2013
The effect of GABAmimetics on the duration of immobility in the forced swim test in albino mice.
    The Libyan journal of medicine, 2014, Volume: 9, Issue:1

    Topics: Alprazolam; Animals; Depression; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; GABA Modulators; gamma-Aminobutyric Acid; Hypokinesia; Imipramine; Injections, Intraperitoneal; Male; Mice; Motor Activity; Pyridines; Stress, Psychological; Swimming; Time Factors; Vigabatrin; Zolpidem

2014
[Cross-reactivity of Instant-View M-1 for detection of benzodiazepine-related drugs and their metabolites in urine].
    Chudoku kenkyu : Chudoku Kenkyukai jun kikanshi = The Japanese journal of toxicology, 2014, Volume: 27, Issue:1

    Topics: Alprazolam; Benzodiazepines; Biomarkers; Cross Reactions; Diazepam; Humans; Immunoassay; Nitrazepam; Reagent Kits, Diagnostic; Sensitivity and Specificity; Structure-Activity Relationship; Substance Abuse Detection; Triazolam

2014
A mixed MDPV and benzodiazepine intoxication in a chronic drug abuser: determination of MDPV metabolites by LC-HRMS and discussion of the case.
    Forensic science international, 2014, Volume: 243

    Topics: Adult; Alprazolam; Benzodiazepines; Benzodioxoles; Chlordiazepoxide; Chromatography, Liquid; Diazepam; Humans; Hypnotics and Sedatives; Male; Mass Spectrometry; Nordazepam; Oxazepam; Psychotropic Drugs; Pyrrolidines; Substance-Related Disorders; Synthetic Cathinone; Temazepam

2014
Detection Times of Diazepam, Clonazepam, and Alprazolam in Oral Fluid Collected From Patients Admitted to Detoxification, After High and Repeated Drug Intake.
    Therapeutic drug monitoring, 2015, Volume: 37, Issue:4

    Topics: Adult; Alprazolam; Chromatography, High Pressure Liquid; Clonazepam; Diazepam; Female; Humans; Male; Middle Aged; Saliva; Substance Abuse Detection; Substance-Related Disorders; Tandem Mass Spectrometry; Time Factors; Young Adult

2015
Development of an ultra-high-performance liquid chromatography coupled to high-resolution quadrupole-Orbitrap mass spectrometry method for the rapid detection and confirmation of illegal adulterated sedative-hypnotics in dietary supplements.
    Food additives & contaminants. Part A, Chemistry, analysis, control, exposure & risk assessment, 2015, Volume: 32, Issue:10

    Topics: Alprazolam; Chromatography, High Pressure Liquid; Clonazepam; Diazepam; Dietary Supplements; Drug Contamination; Food Safety; Humans; Hypnotics and Sedatives; Limit of Detection; Reproducibility of Results; Tandem Mass Spectrometry

2015
Development of a Paper Spray Mass Spectrometry Cartridge with Integrated Solid Phase Extraction for Bioanalysis.
    Analytical chemistry, 2015, Jun-16, Volume: 87, Issue:12

    Topics: Alprazolam; Animals; Atenolol; Carbamazepine; Cattle; Diazepam; Mass Spectrometry; Paper; Solid Phase Extraction; Sulfamethazine

2015
Hypothesis: A single dose of an anxiolitic may prevent unnecessary visits to the emergency room during blood pressure elevations.
    Medical hypotheses, 2016, Volume: 88

    Topics: Aged; Alprazolam; Anti-Anxiety Agents; Antihypertensive Agents; Autonomic Nervous System Diseases; Blood Pressure; Blood Pressure Determination; Calcium Channel Blockers; Captopril; Diazepam; Emergency Medicine; Emergency Service, Hospital; Humans; Hypertension; Models, Theoretical; Risk

2016
Interrupted Time Series Analysis of the Effect of Rescheduling Alprazolam in Australia: Taking Control of Prescription Drug Use.
    JAMA internal medicine, 2016, 08-01, Volume: 176, Issue:8

    Topics: Adult; Aged; Alprazolam; Antidepressive Agents; Antipsychotic Agents; Australia; Benzodiazepines; Diazepam; Drug and Narcotic Control; Drug Substitution; Female; Humans; Hypnotics and Sedatives; Interrupted Time Series Analysis; Male; Middle Aged; Oxazepam; Practice Patterns, Physicians'

2016
Animal Behavior Case of the Month.
    Journal of the American Veterinary Medical Association, 2017, 11-01, Volume: 251, Issue:9

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Antidepressive Agents, Second-Generation; Behavior, Animal; Diazepam; Dog Diseases; Dogs; Fear; Fluoxetine; Gabapentin; Male; Noise; Paroxetine; Phobic Disorders

2017
An Experimental Study of Diazepam and Alprazolam Kinetics in Urine and Oral Fluid Following Single Oral Doses.
    Journal of analytical toxicology, 2019, Mar-01, Volume: 43, Issue:2

    Topics: Administration, Oral; Adult; Alprazolam; Diazepam; Female; Healthy Volunteers; Humans; Kinetics; Male; Saliva; Time Factors; Young Adult

2019
GABA
    Nature, 2019, Volume: 565, Issue:7740

    Topics: Allosteric Regulation; Alprazolam; Benzodiazepines; Bicuculline; Binding, Competitive; Cryoelectron Microscopy; Diazepam; GABA Modulators; Humans; Ligands; Models, Molecular; Nanostructures; Picrotoxin; Receptors, GABA-A; Signal Transduction

2019
Increased sensitivity to psychostimulants and GABAergic drugs in Lsamp-deficient mice.
    Pharmacology, biochemistry, and behavior, 2019, Volume: 183

    Topics: Alprazolam; Animals; Behavior, Animal; Cell Adhesion Molecules, Neuronal; Central Nervous System Depressants; Central Nervous System Stimulants; Cocaine; Diazepam; Disease Models, Animal; Dizocilpine Maleate; Ethanol; Female; GABA Modulators; Gene Knockout Techniques; GPI-Linked Proteins; Locomotion; Male; Maze Learning; Mice; Mice, Knockout; Morphine; Neuroprotective Agents; Phenotype; Receptors, GABA-A

2019
Nonmedical use of alprazolam in the UK: Results from a nationally representative survey.
    British journal of clinical pharmacology, 2019, Volume: 85, Issue:8

    Topics: Adolescent; Adult; Age Factors; Aged; Alprazolam; Central Nervous System Stimulants; Child; Cross-Sectional Studies; Diazepam; Female; Humans; Male; Middle Aged; Motivation; Prescription Drug Misuse; Prevalence; Surveys and Questionnaires; United Kingdom; Young Adult

2019
Dried blood spots sampling in case samples deprived of hematocrit level information - Investigation and calculation strategy.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2019, Aug-15, Volume: 1124

    Topics: Alprazolam; Bone Marrow; Diazepam; Dried Blood Spot Testing; Hematocrit; Humans; Psychotropic Drugs

2019
Benzodiazepine Use Is Associated With an Increased Risk of Neurocognitive Impairment in People Living With HIV.
    Journal of acquired immune deficiency syndromes (1999), 2019, 12-15, Volume: 82, Issue:5

    Topics: Adult; Aged; Alprazolam; Benzodiazepines; Cross-Sectional Studies; Diazepam; Executive Function; Female; HIV Infections; Humans; Lorazepam; Male; Memory, Short-Term; Mental Recall; Mental Status and Dementia Tests; Middle Aged; Motor Skills; Neurocognitive Disorders; Propensity Score; Retrospective Studies; Self Report; Young Adult

2019
Postmortem Analysis of Benzodiazepines in Human Bone by Gas Chromatography-Mass Spectrometry.
    Journal of analytical toxicology, 2021, Jan-21, Volume: 44, Issue:9

    Topics: Alprazolam; Autopsy; Benzodiazepines; Chromatography, Liquid; Clonazepam; Diazepam; Forensic Toxicology; Gas Chromatography-Mass Spectrometry; Humans; Liquid-Liquid Extraction; Lorazepam; Nordazepam; Oxazepam; Tandem Mass Spectrometry

2021
The adulterated XANAX pill: a fatal intoxication with etizolam and caffeine.
    International journal of legal medicine, 2020, Volume: 134, Issue:5

    Topics: Alprazolam; Caffeine; Counterfeit Drugs; Diazepam; Fatal Outcome; Humans; Male; Middle Aged

2020
Development and Validation of an LC-MS-MS Method for the Detection of 40 Benzodiazepines and Three Z-Drugs in Blood and Urine by Solid-Phase Extraction.
    Journal of analytical toxicology, 2020, Oct-12, Volume: 44, Issue:7

    Topics: Alprazolam; Azabicyclo Compounds; Benzodiazepines; Chromatography, Liquid; Diazepam; Forensic Toxicology; Humans; Hypnotics and Sedatives; Limit of Detection; Piperazines; Sleep Aids, Pharmaceutical; Solid Phase Extraction; Substance Abuse Detection; Tandem Mass Spectrometry; Zolpidem

2020
Is the unique benzodiazepine structure interacting with CYP enzymes to affect steroid synthesis in vitro?
    The Journal of steroid biochemistry and molecular biology, 2021, Volume: 205

    Topics: Adrenal Cortex Hormones; Adrenal Glands; Alprazolam; Androgens; Benzodiazepines; Diazepam; Endocrine Disruptors; Humans; Molecular Docking Simulation; Oxazepam; Receptors, Androgen; Receptors, GABA-A; Steroid 17-alpha-Hydroxylase; Steroid 21-Hydroxylase; Steroids

2021
Optimized Photo-Fenton degradation of psychoactive pharmaceuticals alprazolam and diazepam using a chemometric approach-Structure and toxicity of transformation products.
    Journal of hazardous materials, 2021, 02-05, Volume: 403

    Topics: Alprazolam; Diazepam; Hydrogen Peroxide; Oxidation-Reduction; Pharmaceutical Preparations; Tandem Mass Spectrometry; Water Pollutants, Chemical

2021
Occurrence of Z-drugs, benzodiazepines, and ketamine in wastewater in the United States and Mexico during the Covid-19 pandemic.
    The Science of the total environment, 2023, Jan-20, Volume: 857, Issue:Pt 2

    Topics: Alprazolam; Benzodiazepines; Clonazepam; COVID-19; Diazepam; Humans; Ketamine; Lorazepam; Mexico; Nordazepam; Pandemics; Tandem Mass Spectrometry; Temazepam; United States; Wastewater; Zolpidem

2023
Drug prescriptions preceding opioid-related deaths-a register study in forensic autopsy patients.
    PloS one, 2023, Volume: 18, Issue:5

    Topics: Alprazolam; Analgesics, Opioid; Autopsy; Diazepam; Drug Overdose; Drug Prescriptions; Humans; Opioid-Related Disorders; Prescriptions; Retrospective Studies; Substance-Related Disorders

2023