diazepam and alpidem

diazepam has been researched along with alpidem in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19902 (15.38)18.7374
1990's7 (53.85)18.2507
2000's1 (7.69)29.6817
2010's2 (15.38)24.3611
2020's1 (7.69)2.80

Authors

AuthorsStudies
Anzini, M; Basile, AS; Bruni, G; Cappelli, A; Giorgi, G; Langer, T; Romeo, MR; Vomero, S1
Alelyunas, YW; Bui, K; Empfield, JR; McCarthy, D; Pelosi-Kilby, L; Shen, C; Spreen, RC1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Costa, E; Puia, G; Seeburg, PH; Vicini, S1
Advenier, C; Candenas, ML; Devillier, P; Naline, E1
De Luca, C; De Medici, D; Massotti, M1
Biggio, G; Carcangiu, G; Concas, A; Mereu, G; Passino, N1
Arbilla, S; Langer, SZ1
Arbilla, S; Langer, SZ; Lista, A1
O'Hanlon, JF; Swijgman, HF; Uiterwijk, MM; van Veggel, LM; Vermeeren, A1
Morel, E; Perrault, G; Sanger, DJ; Zivkovic, B1
Betti, L; Bistocchi, M; Giannaccini, G; Gori, M; Lucacchini, A1
Baglini, E; Barresi, E; Costa, B; Da Pozzo, E; Da Settimo, F; Martini, C; Robello, M; Salerno, S; Taliani, S1

Reviews

2 review(s) available for diazepam and alpidem

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
An update into the medicinal chemistry of translocator protein (TSPO) ligands.
    European journal of medicinal chemistry, 2021, Jan-01, Volume: 209

    Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Anticonvulsants; Apoptosis; Benzimidazoles; Benzodiazepines; Cell Proliferation; Diazepam; Humans; Imidazoles; Membrane Potential, Mitochondrial; Mitochondria; Mitochondrial ADP, ATP Translocases; Mitochondrial Membranes; Mitochondrial Permeability Transition Pore; Oxidative Stress; Protein Binding; Pyridines; Quinolines; Receptors, GABA; Structure-Activity Relationship; Voltage-Dependent Anion Channels

2021

Trials

1 trial(s) available for diazepam and alpidem

ArticleYear
Anxiolytics' effects on the actual driving performance of patients and healthy volunteers in a standardized test. An integration of three studies.
    Neuropsychobiology, 1995, Volume: 31, Issue:2

    Topics: Anti-Anxiety Agents; Anxiety Disorders; Attention; Automobile Driving; Cross-Over Studies; Diazepam; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Humans; Imidazoles; Lorazepam; Middle Aged; Naphthyridines; Ondansetron; Piperazines; Psychomotor Performance; Pyridines; Sulfur Compounds

1995

Other Studies

10 other study(ies) available for diazepam and alpidem

ArticleYear
Molecular basis of peripheral vs central benzodiazepine receptor selectivity in a new class of peripheral benzodiazepine receptor ligands related to alpidem.
    Journal of medicinal chemistry, 1996, Oct-11, Volume: 39, Issue:21

    Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Cerebral Cortex; Drug Design; Flunitrazepam; Imidazoles; Isoquinolines; Models, Molecular; Protein Conformation; Pyridines; Rats; Receptors, GABA-A; Structure-Activity Relationship

1996
Experimental solubility profiling of marketed CNS drugs, exploring solubility limit of CNS discovery candidate.
    Bioorganic & medicinal chemistry letters, 2010, Dec-15, Volume: 20, Issue:24

    Topics: Central Nervous System Agents; Drug Evaluation, Preclinical; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Solubility

2010
Influence of recombinant gamma-aminobutyric acid-A receptor subunit composition on the action of allosteric modulators of gamma-aminobutyric acid-gated Cl- currents.
    Molecular pharmacology, 1991, Volume: 39, Issue:6

    Topics: Allosteric Regulation; Animals; Cells, Cultured; Chloride Channels; Diazepam; gamma-Aminobutyric Acid; Imidazoles; Membrane Proteins; Pyridines; Rats; Receptors, GABA-A; Recombinant Proteins

1991
Influence of diazepam, alpidem, zolpidem and zopiclone, on the response to adenosine of the guinea pig isolated trachea.
    Fundamental & clinical pharmacology, 1991, Volume: 5, Issue:1

    Topics: 2-Chloroadenosine; Adenosine; Animals; Anti-Anxiety Agents; Diazepam; Dipyridamole; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Histamine; Hypnotics and Sedatives; Imidazoles; Male; Muscle Contraction; Muscle, Smooth; Pyridines; Receptors, GABA-A; Trachea; Zolpidem

1991
Relative efficacies of benzodiazepine receptor agonists in affecting red nucleus electrical activity in rabbits.
    Psychopharmacology, 1990, Volume: 102, Issue:4

    Topics: Animals; Bicuculline; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; Imidazoles; Isoquinolines; Male; Pentylenetetrazole; Pyridazines; Pyridines; Rabbits; Receptors, GABA-A; Red Nucleus; Zolpidem

1990
Reduction of reticulata neuronal activity by zolpidem and alpidem, two imidazopyridines with high affinity for type I benzodiazepine receptors.
    European journal of pharmacology, 1990, Apr-25, Volume: 179, Issue:3

    Topics: Action Potentials; Animals; Anti-Anxiety Agents; Diazepam; Flumazenil; Hypnotics and Sedatives; Imidazoles; Male; Neurons; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reticular Formation; Zolpidem

1990
Limitations of the benzodiazepine receptor nomenclature: a proposal for a pharmacological classification as omega receptor subtypes.
    Fundamental & clinical pharmacology, 1988, Volume: 2, Issue:3

    Topics: Animals; Benzodiazepinones; Cerebellum; Diazepam; Imidazoles; Kidney; Pyridines; Rats; Receptors, GABA-A; Spinal Cord; Terminology as Topic; Zolpidem

1988
Modulation of the electrically evoked release of 5-[3H]hydroxytryptamine from rat cerebral cortex: effects of alpidem, CL 218872, and diazepam.
    Journal of neurochemistry, 1988, Volume: 51, Issue:5

    Topics: Animals; Benzodiazepines; Carbolines; Cerebral Cortex; Diazepam; Electric Stimulation; Flumazenil; gamma-Aminobutyric Acid; Imidazoles; Male; Monoamine Oxidase Inhibitors; Pargyline; Pyrazoles; Pyridazines; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin

1988
Repeated treatment with alpidem, a new anxiolytic, does not induce tolerance or physical dependence.
    Neuropharmacology, 1993, Volume: 32, Issue:9

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Bicuculline; Carbolines; Convulsants; Diazepam; Drug Tolerance; Flumazenil; Imidazoles; Isoniazid; Male; Mice; Pentylenetetrazole; Pyridines; Seizures; Substance Withdrawal Syndrome; Substance-Related Disorders

1993
[3H]Ro 15-1788 binding sites to brain membrane of the saltwater Mugil cephalus.
    Comparative biochemistry and physiology. Toxicology & pharmacology : CBP, 2001, Volume: 128, Issue:3

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Carbolines; Cell Membrane; Chlorides; Diazepam; Female; Fishes; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Imidazoles; Ionophores; Male; Pyridines; Receptors, GABA-A; Synaptosomes; Tritium; Zolpidem

2001