diazepam and alphaxalone

diazepam has been researched along with alphaxalone in 34 studies

Research

Studies (34)

TimeframeStudies, this research(%)All Research%
pre-19908 (23.53)18.7374
1990's9 (26.47)18.2507
2000's4 (11.76)29.6817
2010's12 (35.29)24.3611
2020's1 (2.94)2.80

Authors

AuthorsStudies
Bertrand, PP; Galligan, JJ1
Kokka, N; Olsen, RW; Sapp, DW; Witte, U1
Elliott, RC1
Barbi, S; Beccia, F; Ferraro, M; Pala, F; Sabato, AF1
Amakata, Y; Amenomori, Y; Hirano, H; Matsumoto, T; Sumikawa, K1
Christensen, SE; Elsass, P; Klauber, PV; Lunding, M; Stibolt, O1
Biggio, G; Concas, A; Dazzi, L; Maciocco, E; Mascia, MP; Santoro, G1
Barker, JL; Cruciani, RA; Lange, GD; Mahan, LC; Smallwood, VV; Valeyev, AY1
Biggio, G; Ghiani, CA; Maciocco, E; Sanna, E; Serra, M; Tuligi, G1
Deutsch, SI; Koetzner, L; Mastropaolo, J; Riggs, RL1
Amato, F; Biggio, G; Deserra, T; Motzo, C; Murgia, A; Sanna, E1
Greenfield, LJ; Macdonald, RL; Neelands, TR; Turner, RS; Zhang, J1
Chen, CL; Chiu, TH; Yang, YR1
Cagetti, E; Liang, J; Olsen, RW; Spigelman, I1
Hansen, SL; Sánchez, C; Sperling, BB1
Asproni, B; Biggio, G; Busonero, F; Cerri, R; Maciocco, E; Mascia, MP; Pau, A; Sanna, E; Talani, G1
France, CP; Javors, MA; McMahon, LR1
Alibhai, HI; Armitage-Chan, E; Brodbelt, DC; Jimenez-Lozano, A; Psatha, E1
D'Hulst, C; De Deyn, PP; Heulens, I; Kooy, RF; Van Dam, D1
Chambers, JP; Gieseg, M; Mitchinson, SL; Singh, PM; Walsh, VP1
Akk, G; Eaton, MM; Li, P; Steinbach, JH1
Bertrán de Lis, BT; Santos González, M; Tendillo Cortijo, FJ1
Bridges, J; Gieseg, M; Hon, H; Walsh, V1
del Álamo, AM; Mandsager, RE; Payton, ME; Riebold, TW1
Higashi, T; Nakashima, K; Okumura, A; Sato, T; Yoshizawa, K1
Akk, G; Cao, LQ; Chakrabarti, S; Evers, AS; Germann, AL; Mennerick, S; Montana, MC; Shin, DJ; Wozniak, DF; Yuede, CM1
Ambros, B; Duke-Novakovski, T; Gaunt, MC; Taylor, SM1
Italiano, M; Robinson, R1
Hampton, CE; Mandsager, RE; Riebold, TW1
Berry, MJ; Dyson, RM; Gray, CL; Pacharinsak, C; Sixtus, RP1
Maksay, G1
Iversen, LL; Wong, EH1
Clements-Jewery, S; Hunt, P1
Kofman, O; Myslobodsky, MS1

Trials

8 trial(s) available for diazepam and alphaxalone

ArticleYear
A clinical neuropsychological study of the postoperative course after three types of anaesthesia.
    Acta anaesthesiologica Scandinavica, 1982, Volume: 26, Issue:2

    Topics: Adult; Aged; Alfaxalone Alfadolone Mixture; Anesthetics; Clinical Trials as Topic; Cognition Disorders; Diazepam; Double-Blind Method; Female; Fentanyl; Humans; Male; Middle Aged; Mood Disorders; Postoperative Period; Pregnanediones; Thiopental

1982
Clinical efficacy and cardiorespiratory effects of alfaxalone, or diazepam/fentanyl for induction of anaesthesia in dogs that are a poor anaesthetic risk.
    Veterinary anaesthesia and analgesia, 2011, Volume: 38, Issue:1

    Topics: Anesthesia; Anesthetics, Intravenous; Animals; Blood Pressure; Body Temperature; Diazepam; Dog Diseases; Dogs; Drug Therapy, Combination; Female; Fentanyl; Heart Rate; Male; Preanesthetic Medication; Pregnanediones; Respiration

2011
A comparison of two different ketamine and diazepam combinations with an alphaxalone and medetomidine combination for induction of anaesthesia in sheep.
    New Zealand veterinary journal, 2012, Volume: 60, Issue:2

    Topics: Anesthesia Recovery Period; Anesthesia, General; Anesthetics, Dissociative; Animals; Diazepam; Drug Therapy, Combination; Hypnotics and Sedatives; Ketamine; Medetomidine; Pregnanediones; Sheep

2012
Effects of intramuscular alfaxalone alone or in combination with diazepam in swine.
    Veterinary anaesthesia and analgesia, 2013, Volume: 40, Issue:4

    Topics: Anesthetics; Animals; Diazepam; Drug Therapy, Combination; Hypnotics and Sedatives; Injections, Intramuscular; Pregnanediones; Swine

2013
A comparison of anaesthetic recoveries in cats following induction with either alfaxalone or ketamine and diazepam.
    New Zealand veterinary journal, 2014, Volume: 62, Issue:3

    Topics: Anesthesia Recovery Period; Anesthetics; Animals; Cats; Diazepam; Female; Hysterectomy; Ketamine; Ovariectomy; Pregnanediones

2014
Evaluation of intravenous administration of alfaxalone, propofol, and ketamine-diazepam for anesthesia in alpacas.
    Veterinary anaesthesia and analgesia, 2015, Volume: 42, Issue:1

    Topics: Anesthesia; Anesthetics; Animals; Camelids, New World; Diazepam; Drug Therapy, Combination; Female; Injections, Intravenous; Ketamine; Male; Pregnanediones; Propofol

2015
Effect of benzodiazepines on the dose of alfaxalone needed for endotracheal intubation in healthy dogs.
    Veterinary anaesthesia and analgesia, 2018, Volume: 45, Issue:6

    Topics: Adjuvants, Anesthesia; Anesthetics; Animals; Diazepam; Dogs; Dose-Response Relationship, Drug; Intubation, Intratracheal; Midazolam; Pregnanediones; Prospective Studies; Single-Blind Method

2018
Recovery characteristics of dogs following anesthesia induced with tiletamine-zolazepam, alfaxalone, ketamine-diazepam, or propofol and maintained with isoflurane.
    Journal of the American Veterinary Medical Association, 2019, 06-15, Volume: 254, Issue:12

    Topics: Anesthesia; Animals; Cross-Over Studies; Diazepam; Dogs; Heart Rate; Isoflurane; Ketamine; Pregnanediones; Propofol; Prospective Studies; Reproducibility of Results; Retrospective Studies; Tiletamine; Zolazepam

2019

Other Studies

26 other study(ies) available for diazepam and alphaxalone

ArticleYear
Alfaxalone, pentobarbital and diazepam potentiate gamma-aminobutyric acid-induced depolarizations in single myenteric neurons of guinea pig intestine.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:2

    Topics: Anesthetics; Animals; Diazepam; Drug Synergism; gamma-Aminobutyric Acid; Guinea Pigs; Hydrocortisone; Intestines; Male; Membrane Potentials; Muscimol; Pentobarbital; Pregnanediones; Receptors, GABA-A

1992
Sex differences in sensitivity to pentylenetetrazol but not in GABAA receptor binding.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 43, Issue:2

    Topics: Anesthetics; Animals; Anticonvulsants; Autoradiography; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Diazepam; Electroshock; Ethanol; Female; Flunitrazepam; Male; Muscimol; Orchiectomy; Ovariectomy; Pentylenetetrazole; Pregnanediones; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Seizures; Sex Characteristics

1992
The action of intravenous anaesthetic and central depressant drugs on the contractures elicited by tetraethylammonium in the chick biventer cervicis muscle.
    General pharmacology, 1985, Volume: 16, Issue:6

    Topics: Alfaxalone Alfadolone Mixture; Anesthetics; Animals; Central Nervous System Depressants; Chickens; Chloralose; Diazepam; Drug Synergism; Ethanol; Etomidate; In Vitro Techniques; Methohexital; Muscle Contraction; Neck Muscles; Paraldehyde; Pregnanediones; Propanidid; Tetraethylammonium; Tetraethylammonium Compounds; Thiopental; Urethane

1985
The effect of five drugs in coma doses on neurotransmitter amino acids in the brains of guinea pigs.
    Resuscitation, 1983, Volume: 10, Issue:4

    Topics: Amino Acids; Animals; Brain; Brain Chemistry; Central Nervous System Agents; Central Nervous System Depressants; Diazepam; Flunitrazepam; Guinea Pigs; Neurotransmitter Agents; Phenobarbital; Phenytoin; Pregnanediones

1983
Selective actions of intravenous anesthetics on nicotinic- and muscarinic-receptor-mediated responses of the dog adrenal medulla.
    Anesthesiology, 1983, Volume: 59, Issue:5

    Topics: Adrenal Medulla; Anesthetics; Animals; Catecholamines; Diazepam; Dogs; In Vitro Techniques; Ketamine; Pregnanediones; Receptors, Muscarinic; Receptors, Nicotinic; Thiopental

1983
Effects of propofol, pentobarbital and alphaxalone on t-[35S]butylbicyclophosphorothionate binding in rat cerebral cortex.
    European journal of pharmacology, 1994, Apr-15, Volume: 267, Issue:2

    Topics: Anesthetics; Animals; Bicuculline; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Diazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Ion Channel Gating; Male; Membranes; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Sulfur Radioisotopes

1994
Characterization of the gamma-aminobutyric acidA receptor-channel complex composed of alpha 1 beta 2 and alpha 1 beta 3 subunits from rat brain.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:2

    Topics: Animals; Brain; Chlorides; CHO Cells; Cricetinae; Diazepam; gamma-Aminobutyric Acid; Membrane Potentials; Pentobarbital; Pregnanediones; Rats; Receptors, GABA-A; Transfection

1993
Biochemical evaluations of the effects of loreclezole and propofol on the GABAA receptor in rat brain.
    Biochemical pharmacology, 1996, Jun-14, Volume: 51, Issue:11

    Topics: Anesthetics; Animals; Anticonvulsants; Brain; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Male; Muscimol; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sulfur Radioisotopes; Triazoles; Tritium

1996
Selective cyclodextrin inhibition of alfaxolone-induced ataxia.
    The Journal of pharmacy and pharmacology, 1996, Volume: 48, Issue:5

    Topics: Animals; Ataxia; Cyclodextrins; Diazepam; Dose-Response Relationship, Drug; Ethanol; Male; Mice; Pharmaceutical Vehicles; Plant Oils; Pregnanediones; Propylene Glycols; Solvents

1996
Expression of native GABAA receptors in Xenopus oocytes injected with rat brain synaptosomes.
    Journal of neurochemistry, 1996, Volume: 67, Issue:5

    Topics: Anesthetics; Animals; Brain; Cell Membrane; Chloride Channels; Chlorides; Diazepam; Female; GABA Antagonists; gamma-Aminobutyric Acid; Membrane Potentials; Oocytes; Picrotoxin; Pregnanediones; Pyridazines; Rats; Receptors, GABA-A; Synaptosomes; Xenopus laevis; Zinc Compounds

1996
GABAA receptor pharmacology and subtype mRNA expression in human neuronal NT2-N cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Jul-01, Volume: 18, Issue:13

    Topics: Anticonvulsants; Bicuculline; Carbolines; Convulsants; Diazepam; Diuretics; DNA Primers; Furosemide; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Hypnotics and Sedatives; Lanthanum; Neurons; Patch-Clamp Techniques; Pentobarbital; Phenobarbital; Picrotoxin; Polymerase Chain Reaction; Pregnanediones; Pregnenolone; Pyridines; Receptors, GABA-A; RNA, Messenger; Teratocarcinoma; Triazoles; Tumor Cells, Cultured; Zinc; Zolpidem

1998
Activation of rat locus coeruleus neuron GABA(A) receptors by propofol and its potentiation by pentobarbital or alphaxalone.
    European journal of pharmacology, 1999, Dec-15, Volume: 386, Issue:2-3

    Topics: Anesthetics; Anesthetics, Intravenous; Animals; Baclofen; Barium Compounds; Bicuculline; Chlorides; Diazepam; Drug Synergism; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Ionophores; Locus Coeruleus; Male; Neurons; Pentobarbital; Picrotoxin; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Zinc Compounds

1999
Withdrawal from chronic intermittent ethanol treatment changes subunit composition, reduces synaptic function, and decreases behavioral responses to positive allosteric modulators of GABAA receptors.
    Molecular pharmacology, 2003, Volume: 63, Issue:1

    Topics: Affinity Labels; Alcoholism; Allosteric Regulation; Anesthetics; Animals; Anxiety; Azides; Benzodiazepines; Benzodiazepinones; Binding Sites; Diazepam; Electrophysiology; Ethanol; GABA Modulators; Hippocampus; Hypnosis; Immunoblotting; Kinetics; Male; Maze Learning; Neurons; Pregnanediones; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Reverse Transcriptase Polymerase Chain Reaction; Sleep

2003
Anticonvulsant and antiepileptogenic effects of GABAA receptor ligands in pentylenetetrazole-kindled mice.
    Progress in neuro-psychopharmacology & biological psychiatry, 2004, Volume: 28, Issue:1

    Topics: Animals; Anticonvulsants; Bicuculline; Convulsants; Dehydroepiandrosterone Sulfate; Diazepam; Dose-Response Relationship, Drug; Epilepsy; Flumazenil; GABA Agonists; GABA Antagonists; GABA Modulators; Isoxazoles; Kindling, Neurologic; Ligands; Mice; Pentylenetetrazole; Pregnanediones; Receptors, GABA-A

2004
Ethyl 2-(4-bromophenyl)-1-(2,4-dichlorophenyl)-1H-4-imidazolecarboxylate is a novel positive modulator of GABAA receptors.
    European journal of pharmacology, 2005, Jun-15, Volume: 516, Issue:3

    Topics: Animals; Binding, Competitive; Cell Membrane; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Etomidate; Female; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Glycine; Humans; Hydrocarbons, Halogenated; Imidazoles; Male; Membrane Potentials; Oocytes; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Glycine; Receptors, Serotonin, 5-HT3; Serotonin; Tritium; Xenopus laevis

2005
Changes in relative potency among positive GABA(A) receptor modulators upon discontinuation of chronic benzodiazepine treatment in rhesus monkeys.
    Psychopharmacology, 2007, Volume: 192, Issue:1

    Topics: Animals; Behavior, Animal; Benzodiazepines; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Female; Flumazenil; GABA Modulators; Lorazepam; Macaca mulatta; Male; Midazolam; Pentobarbital; Pregnanediones; Pregnanolone; Receptors, GABA-A; Substance Withdrawal Syndrome

2007
Pharmacological treatment of fragile X syndrome with GABAergic drugs in a knockout mouse model.
    Behavioural brain research, 2012, Apr-01, Volume: 229, Issue:1

    Topics: Analysis of Variance; Anesthetics; Animals; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Epilepsy, Reflex; Fragile X Mental Retardation Protein; Fragile X Syndrome; GABA Modulators; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Pregnanediones; Psychomotor Performance; Rotarod Performance Test

2012
The benzodiazepine diazepam potentiates responses of α1β2γ2L γ-aminobutyric acid type A receptors activated by either γ-aminobutyric acid or allosteric agonists.
    Anesthesiology, 2013, Volume: 118, Issue:6

    Topics: Anesthetics; Animals; Binding Sites; Diazepam; Drug Synergism; Etomidate; GABA Modulators; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Patch-Clamp Techniques; Pentobarbital; Pregnanediones; Rats; Receptors, GABA-A

2013
Role of allopregnanolone biosynthesis in acute stress-induced anxiety-like behaviors in mice.
    Synapse (New York, N.Y.), 2017, Volume: 71, Issue:8

    Topics: 5-alpha Reductase Inhibitors; Animals; Anxiety Disorders; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Finasteride; Freezing Reaction, Cataleptic; Male; Mice, Inbred C57BL; Muscle Relaxants, Central; Muscle Strength; Muscle Tonus; Pregnanediones; Pregnanolone; Restraint, Physical; Stress, Psychological

2017
Enhanced GABAergic actions resulting from the coapplication of the steroid 3α-hydroxy-5α-pregnane-11,20-dione (alfaxalone) with propofol or diazepam.
    Scientific reports, 2018, 07-09, Volume: 8, Issue:1

    Topics: Animals; Cells, Cultured; Diazepam; Drug Synergism; Inhibitory Postsynaptic Potentials; Locomotion; Male; Mice; Neurons; Oocysts; Patch-Clamp Techniques; Pregnanediones; Propofol; Rats; Receptors, GABA-A; Recombinant Proteins; Xenopus

2018
Effects of alfaxalone, thiopental, or propofol and diazepam on laryngeal motion in healthy dogs.
    The Canadian veterinary journal = La revue veterinaire canadienne, 2018, Volume: 59, Issue:7

    Topics: Anesthesia, General; Anesthetics; Animals; Arytenoid Cartilage; Diazepam; Dogs; Drug Combinations; Laryngoscopy; Pregnanediones; Propofol; Thiopental; Video Recording

2018
Differential effects of four intramuscular sedatives on cardiorespiratory stability in juvenile guinea pigs (Cavia porcellus).
    PloS one, 2021, Volume: 16, Issue:11

    Topics: Animals; Blood Pressure; Diazepam; Guinea Pigs; Heart Rate; Hypnotics and Sedatives; Injections, Intramuscular; Ketamine; Midazolam; Pregnanediones; Respiratory Rate

2021
GABAA receptor populations bind agonists and antagonists differentially and with opposite affinities.
    Journal of neurochemistry, 1988, Volume: 50, Issue:6

    Topics: Affinity Labels; Androstanes; Animals; Azasteroids; Brain; Diazepam; Diazonium Compounds; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscimol; Photochemistry; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sulfanilic Acids; Synaptic Membranes

1988
Modulation of [3H]diazepam binding in rat cortical membranes by GABAA agonists.
    Journal of neurochemistry, 1985, Volume: 44, Issue:4

    Topics: Androstanes; Animals; Azasteroids; Bicuculline; Cell Membrane; Cerebral Cortex; Diazepam; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Isonicotinic Acids; Isoxazoles; Muscimol; Piperidines; Rats; Receptors, GABA-A; Taurine

1985
A steroid derivative, R 5135, antagonizes the GABA/benzodiazepine receptor interaction.
    Neuropharmacology, 1981, Volume: 20, Issue:4

    Topics: Androstanes; Animals; Azasteroids; Chlorides; Diazepam; gamma-Aminobutyric Acid; Glycine; Male; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Steroids, Heterocyclic; Strychnine

1981
Regular and lasting neocortical spiking produced by systemic administration of a steroid derivative in the rat.
    Neuropharmacology, 1983, Volume: 22, Issue:2

    Topics: Action Potentials; Androstanes; Animals; Azasteroids; Behavior, Animal; Cerebral Cortex; Diazepam; Electroencephalography; Evoked Potentials, Visual; gamma-Aminobutyric Acid; Humans; Rats; Rats, Inbred Strains; Stereotyped Behavior; Steroids, Heterocyclic; Valproic Acid

1983