Page last updated: 2024-08-24

dexverapamil and lekoptin

dexverapamil has been researched along with lekoptin in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (66.67)29.6817
2010's2 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Pajeva, IK; Wiese, M1
Choi, SU; Kwon, MJ; Lee, BH; Lee, CO; Yi, KY; Yoo, SE1
Dansette, PM; Fontana, E; Poli, SM1
Baubichon-Cortay, H; Chang, XB; Di Pietro, A; Perrotton, T; Trompier, D1
Avdeef, A; Tam, KY1
Chen, G; Hu, N; Liu, H; Liu, L; Liu, X; Pan, X; Wang, G; Wang, X; Xie, L; Xie, S; Zhang, L1

Reviews

1 review(s) available for dexverapamil and lekoptin

ArticleYear
Cytochrome p450 enzymes mechanism based inhibitors: common sub-structures and reactivity.
    Current drug metabolism, 2005, Volume: 6, Issue:5

    Topics: Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Interactions; Enzyme Inhibitors; Humans; Isoenzymes; Structure-Activity Relationship; Terminology as Topic

2005

Other Studies

5 other study(ies) available for dexverapamil and lekoptin

ArticleYear
Pharmacophore model of drugs involved in P-glycoprotein multidrug resistance: explanation of structural variety (hypothesis).
    Journal of medicinal chemistry, 2002, Dec-19, Volume: 45, Issue:26

    Topics: Adenosine Triphosphatases; Algorithms; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Binding, Competitive; Caco-2 Cells; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluoresceins; Humans; Ligands; Models, Molecular; Molecular Structure; Quantitative Structure-Activity Relationship; Radioligand Assay; Rhodamine 123; Stereoisomerism; Verapamil; Vinblastine

2002
Differential effects of the optical isomers of KR30031 on cardiotoxicity and on multidrug resistance reversal activity.
    Anti-cancer drugs, 2003, Volume: 14, Issue:2

    Topics: Animals; Antineoplastic Agents; Aorta; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blood Pressure; Calcium Channel Blockers; Colorectal Neoplasms; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Humans; Isomerism; Male; Rats; Rats, Sprague-Dawley; Tumor Cells, Cultured; Uterine Neoplasms; Vasodilation; Ventricular Function, Left; Verapamil

2003
(R)- and (S)-verapamil differentially modulate the multidrug-resistant protein MRP1.
    The Journal of biological chemistry, 2007, Oct-26, Volume: 282, Issue:43

    Topics: Adenosine Triphosphatases; Animals; Cell Line; Cell Proliferation; Cell Survival; Cricetinae; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Fluoresceins; Fluorescent Dyes; Formazans; Glutathione; Inhibitory Concentration 50; Kidney; Leukotriene C4; Multidrug Resistance-Associated Proteins; Protein Conformation; Sodium Iodide; Spectrometry, Fluorescence; Stereoisomerism; Tetrazolium Salts; Transfection; Tryptophan; Verapamil

2007
How well can the Caco-2/Madin-Darby canine kidney models predict effective human jejunal permeability?
    Journal of medicinal chemistry, 2010, May-13, Volume: 53, Issue:9

    Topics: Animals; Disease Models, Animal; Dogs; Humans; Jejunal Diseases; Kidney Diseases; Models, Biological; Permeability; Porosity; Regression Analysis

2010
Opposite effect of diabetes mellitus induced by streptozotocin on oral and intravenous pharmacokinetics of verapamil in rats.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:3

    Topics: Administration, Oral; Animals; Antihypertensive Agents; Biological Availability; Calcium Channel Blockers; Cytochrome P-450 CYP3A; Diabetes Mellitus, Experimental; Half-Life; Injections, Intravenous; Intestine, Small; Male; Membrane Proteins; Metabolic Clearance Rate; Microsomes; Microsomes, Liver; Organ Specificity; Rats; Rats, Sprague-Dawley; Streptozocin; Verapamil

2011