Page last updated: 2024-08-23

dexetimide and pirenzepine

dexetimide has been researched along with pirenzepine in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19905 (71.43)18.7374
1990's1 (14.29)18.2507
2000's1 (14.29)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dannals, RF; Frost, JJ; Ravert, HT; Wagner, HN; Wilson, AA1
Kovacs, I; Roeske, WR; Varga, EV; Waite, SL; Yamamura, HI1
Elzinga, CR; Meurs, H; Roffel, AF; Zaagsma, J1
Beld, AJ; Klaassen, AB; Kuijpers, W; Rodrigues de Miranda, JF; Scheres, HM1
de Zeeuw, RA; in't Hout, WG; Roffel, AF; Zaagsma, J1
Gorissen, H; Laduron, PM; Leysen, JE1
Christopoulos, A; Lanzafame, A; Mitchelson, F1

Other Studies

7 other study(ies) available for dexetimide and pirenzepine

ArticleYear
Synthesis and biological evaluation of [125I]- and [123I]-4-iododexetimide, a potent muscarinic cholinergic receptor antagonist.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:5

    Topics: Animals; Dexetimide; Iodine Radioisotopes; Isotope Labeling; Male; Mice; Parasympatholytics; Piperidines; Receptors, Muscarinic; Tomography, Emission-Computed

1989
Pharmacological comparison of the cloned human and rat M2 muscarinic receptor genes expressed in the murine fibroblast (B82) cell line.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:2

    Topics: Amino Acid Sequence; Animals; Carbachol; Cloning, Molecular; Cyclic AMP; Humans; Mice; Molecular Sequence Data; Muscarinic Agonists; Muscarinic Antagonists; Phosphatidylinositols; Radioligand Assay; Rats; Receptors, Muscarinic; Sequence Alignment; Sequence Homology, Amino Acid; Signal Transduction; Species Specificity

1998
Allosteric interactions of three muscarine antagonists at bovine tracheal smooth muscle and cardiac M2 receptors.
    European journal of pharmacology, 1989, Mar-07, Volume: 172, Issue:1

    Topics: Animals; Cattle; Dexetimide; Diamines; Gallamine Triethiodide; Heart; In Vitro Techniques; Membrane Proteins; Muscle, Smooth; Parasympatholytics; Pirenzepine; Receptors, Muscarinic; Trachea

1989
Cholinergic receptors in the upper respiratory system of the rat.
    Archives of otolaryngology--head & neck surgery, 1986, Volume: 112, Issue:4

    Topics: Animals; Benzilates; Benzodiazepinones; Binding, Competitive; Dexetimide; Methacholine Chloride; Methacholine Compounds; Nasal Mucosa; Pirenzepine; Quaternary Ammonium Compounds; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1986
The M2 selective antagonist AF-DX 116 shows high affinity for muscarine receptors in bovine tracheal membranes.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:5

    Topics: Animals; Binding, Competitive; Cattle; Dexetimide; In Vitro Techniques; Membrane Proteins; Muscle, Smooth; Myocardium; Pirenzepine; Receptors, Muscarinic; Trachea

1987
Muscarinic receptor: multiple sites or unitary concept?
    Archives internationales de pharmacodynamie et de therapie, 1981, Volume: 249, Issue:2

    Topics: Animals; Atropine; Benzodiazepinones; Brain; Dexetimide; Dogs; Gastric Mucosa; In Vitro Techniques; Microsomes; Piperazines; Piperidines; Pirenzepine; Receptors, Cholinergic; Receptors, Muscarinic

1981
The allosteric interaction of otenzepad (AF-DX 116) at muscarinic M2 receptors in guinea pig atria.
    European journal of pharmacology, 2001, Mar-30, Volume: 416, Issue:3

    Topics: Acetylcholine; Allosteric Regulation; Animals; Atropine; Carbachol; Cardiotonic Agents; Dexetimide; Electric Stimulation; Female; Gallamine Triethiodide; Guinea Pigs; Heart Atria; In Vitro Techniques; Kinetics; Male; Muscarinic Antagonists; N-Methylscopolamine; Nicotinic Antagonists; Parasympatholytics; Phthalimides; Pirenzepine; Quaternary Ammonium Compounds; Radioligand Assay; Receptor, Muscarinic M2; Receptors, Muscarinic

2001