Page last updated: 2024-08-23

dexetimide and piperidines

dexetimide has been researched along with piperidines in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-199027 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Colpaert, FC; Lal, H; Niemegeers, C; Wauquier, A1
Bertram, U; Kasten, A; Lüllmann, H; Ziegler, A1
Schulze, F1
Binenfeld, Z; Deljac, V; Fajdetić, A; Wilhelm, K1
Janssen, PF; Laduron, PM1
Laduron, PM; Leysen, JE; Verwimp, M1
Reil, GH1
Amery, W; Kimya, S; Oei, TT; Zwanikken, GJ1
Fischer, VW1
Mitchelson, F; Reil, GH1
Lal, H; Niemegeers, CJ; Wauquier, A1
Niemegeers, CJ; Wauquier, A1
Gianutsos, G; Lal, H1
Gray, JA; Lüllmann, H; Mitchelson, F; Reil, GH1
Dannals, RF; Frost, JJ; Ravert, HT; Wagner, HN; Wilson, AA1
Dannals, RF; Långström, B; Ravert, HT; Wagner, HN; Wilson, AA1
De Roe, C; Laduron, PM; Luabeya, MK; Maloteaux, JM; Trouet, A1
Szobor, A1
Dobiásová, A; Faltus, F; Filip, V; Jirák, R; Karen, P; Posmurová, M; Skopová, J1
Laduron, P1
Beld, AJ; Huisman, GN; Rodrigues de Miranda, JF; van Ginneken, CA1
Gossuin, A; Laduron, P; Maloteaux, JM; Trouet, A1
Gorissen, H; Laduron, PM; Leysen, JE1
Lüllmann, H; Schmaus, H; Staemmler, C; Ziegler, A1
Lüllmann, H; Reil, GH; Timmermans, PB; Ziegler, A1
Alba, F; Mora, F; Vives, F1
Beld, AJ; Klok, EJ; Rodrigues de Miranda, JF1

Trials

2 trial(s) available for dexetimide and piperidines

ArticleYear
Safety and efficacy of prolonged treatment with Tremblex (dexetimide), an antiparkinsonian agent. A controlled study.
    Acta psychiatrica Belgica, 1976, Volume: 76, Issue:3

    Topics: Adult; Aged; Dexetimide; Drug Evaluation; Female; Humans; Middle Aged; Parkinson Disease; Piperidines; Time Factors

1976
[Fluspirilene in schizophrenia maintenance therapy and its interaction with dexetimide].
    Ceskoslovenska psychiatrie, 1985, Volume: 81, Issue:6

    Topics: Adult; Clinical Trials as Topic; Dexetimide; Drug Interactions; Drug Therapy, Combination; Female; Fluspirilene; Humans; Male; Middle Aged; Piperidines; Schizophrenia; Spiro Compounds

1985

Other Studies

25 other study(ies) available for dexetimide and piperidines

ArticleYear
Reversal by a central antiacetylcholine drug of pimozide-induced inhibition of mouse-jumping in amphetamine-dopa treated mice.
    The Journal of pharmacy and pharmacology, 1975, Volume: 27, Issue:7

    Topics: Acetylcholine; Amphetamine; Animals; Dexetimide; Levodopa; Male; Mice; Motor Activity; Pimozide; Piperidines; Time Factors

1975
Improved treatment of organophosphate intoxication by use of scopolamine or dexetimide.
    Experientia, 1977, Sep-15, Volume: 33, Issue:9

    Topics: Animals; Atropine; Dexetimide; Drug Therapy, Combination; Isoflurophate; Mice; Obidoxime Chloride; Organophosphorus Compounds; Oximes; Piperidines; Rabbits; Scopolamine

1977
[Effect of reduced gastrointestinal motility on the regulation of gastrointestinal flora and the pathogenesis of coli enterotoxinemia in market swine].
    Archiv fur experimentelle Veterinarmedizin, 1979, Volume: 33, Issue:2

    Topics: Animals; Bacteria; Dexetimide; Digestive System; Escherichia coli Infections; Gastrointestinal Motility; Opium; Piperidines; Species Specificity; Swine; Swine Diseases

1979
Protective effect of dexetimide and HI-6 in poisoning with highly toxic organophosphorus compounds.
    Arhiv za higijenu rada i toksikologiju, 1979, Volume: 30, Issue:2

    Topics: Animals; Antidotes; Atropine; Dexetimide; Male; Mice; Organophosphate Poisoning; Piperidines; Pyridinium Compounds; Rats

1979
Characterization and subcellular localization of brain muscarinic receptors labelled in vivo by [3H]dexetimide.
    Journal of neurochemistry, 1979, Volume: 33, Issue:6

    Topics: Animals; Brain; Cell Fractionation; Cerebellum; Cerebral Cortex; Corpus Striatum; Dexetimide; Hippocampus; Kinetics; Male; Medulla Oblongata; Piperidines; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Subcellular Fractions; Tissue Distribution

1979
Stereospecific in vitro binding of [3H]dexetimide to brain muscarinic receptors.
    Journal of neurochemistry, 1979, Volume: 32, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Corpus Striatum; Dexetimide; Kinetics; Male; Piperidines; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Stereoisomerism; Structure-Activity Relationship; Subcellular Fractions; Tissue Distribution

1979
Dependence of the transmembraneous penetration rate of an anticholinergic drug on the action potential frequency.
    Naunyn-Schmiedeberg's archives of pharmacology, 1977, Volume: 297 Suppl 1

    Topics: Action Potentials; Cell Membrane Permeability; Dexetimide; Humans; Membrane Lipids; Piperidines; Solubility

1977
[Experience with Benzetimide in the treatment of diarrheas of cattle and calves].
    DTW. Deutsche tierarztliche Wochenschrift, 1975, Mar-05, Volume: 82, Issue:3

    Topics: Animals; Cattle; Cattle Diseases; Dexetimide; Diarrhea; Drug Therapy, Combination; Enteritis; Female; Male; Piperidines

1975
Proceedings: Antimuscarinic action and tissue binding of the optical isomers of benzetimide.
    Naunyn-Schmiedeberg's archives of pharmacology, 1975, Volume: 287 Suppl

    Topics: Animals; Dexetimide; Guinea Pigs; Optical Rotation; Parasympatholytics; Piperidines; Stereoisomerism

1975
Differential antagonism by the antichlolinergic dexetimide of inhibitory effects of haloperidol and fentanyl on brain self-stimulation.
    Psychopharmacologia, 1975, Volume: 41, Issue:3

    Topics: Animals; Brain; Dexetimide; Dose-Response Relationship, Drug; Fentanyl; Haloperidol; Male; Piperidines; Rats; Self Stimulation

1975
The effects of dexetimide on pimozide-, haloperidol- and pipamperone-induced inhibition of brain self-stimulation in rats.
    Archives internationales de pharmacodynamie et de therapie, 1975, Volume: 217, Issue:2

    Topics: Animals; Brain; Butyrophenones; Depression, Chemical; Dexetimide; Drug Interactions; Electric Stimulation; Haloperidol; Isonipecotic Acids; Male; Pimozide; Piperidines; Rats; Self Stimulation; Tranquilizing Agents

1975
Alteration in the action of cholinergic and anti cholinergic drugs after chronic haloperidol: indirect evidence for cholinergic hyposensitivity.
    Life sciences, 1976, Mar-01, Volume: 18, Issue:5

    Topics: Acetylcholine; Amphetamines; Animals; Dexetimide; Dopamine; Haloperidol; Male; Motor Activity; Pentobarbital; Pilocarpine; Piperidines; Rats; Receptors, Cholinergic; Time Factors

1976
Stereoselective binding in cardiac tissue of the enatiomers of benzetimide, and antimuscarinic drug.
    British journal of pharmacology, 1976, Volume: 56, Issue:4

    Topics: Animals; Binding Sites; Dexetimide; Guinea Pigs; Heart; In Vitro Techniques; Myocardium; Piperidines; Stereoisomerism; Time Factors

1976
Synthesis and biological evaluation of [125I]- and [123I]-4-iododexetimide, a potent muscarinic cholinergic receptor antagonist.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:5

    Topics: Animals; Dexetimide; Iodine Radioisotopes; Isotope Labeling; Male; Mice; Parasympatholytics; Piperidines; Receptors, Muscarinic; Tomography, Emission-Computed

1989
Synthesis of radiotracers for studying muscarinic cholinergic receptors in the living human brain using positron emission tomography: [11C]dexetimide and [11C]levetimide.
    International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes, 1988, Volume: 39, Issue:4

    Topics: Brain; Carbon Radioisotopes; Dexetimide; Humans; Piperidines; Receptors, Muscarinic; Tomography, Emission-Computed

1988
Different subcellular localization of muscarinic and serotonin (S2) receptors in human, dog, and rat brain.
    Journal of neurochemistry, 1986, Volume: 46, Issue:2

    Topics: Adult; Aged; Animals; Brain; Brain Chemistry; Centrifugation, Density Gradient; Dexetimide; Dogs; Humans; Ketanserin; Mathematics; Microscopy, Electron; Middle Aged; Piperidines; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Receptors, Serotonin; Species Specificity; Subcellular Fractions

1986
Myasthenia gravis: control of drug-induced cholinergic symptoms with dexetimide.
    Therapia Hungarica (English edition), 1985, Volume: 33, Issue:3

    Topics: Adolescent; Adult; Aged; Dexetimide; Humans; Middle Aged; Muscular Diseases; Myasthenia Gravis; Parasympathomimetics; Piperidines; Respiratory Insufficiency

1985
Axonal flow of muscarinic receptors.
    Archives internationales de pharmacodynamie et de therapie, 1980, Volume: 244, Issue:2

    Topics: Animals; Axonal Transport; Dexetimide; Dogs; Piperidines; Receptors, Cholinergic; Receptors, Muscarinic; Spleen; Sympathetic Nervous System

1980
'Do abnormalities in agonist receptor-binding reflect the activation of the receptor?' An interpretation of the inhibition of 3H-dexetimide binding to the muscarinic receptor by a series of furtrethonium derivatives.
    European journal of respiratory diseases. Supplement, 1984, Volume: 135

    Topics: Animals; Binding, Competitive; Cattle; Dexetimide; Muscle, Smooth; Piperidines; Quaternary Ammonium Compounds; Receptors, Muscarinic; Trachea

1984
Differentiation between ligand trapping into intact cells and binding on muscarinic receptors.
    Biochimica et biophysica acta, 1984, May-22, Volume: 804, Issue:1

    Topics: Animals; Biological Transport; Cell Line; Cell Membrane; Dexetimide; Glioma; Ligands; Lysosomes; N-Methylscopolamine; Neuroblastoma; Piperidines; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Muscarinic; Scopolamine Derivatives

1984
Muscarinic receptor: multiple sites or unitary concept?
    Archives internationales de pharmacodynamie et de therapie, 1981, Volume: 249, Issue:2

    Topics: Animals; Atropine; Benzodiazepinones; Brain; Dexetimide; Dogs; Gastric Mucosa; In Vitro Techniques; Microsomes; Piperazines; Piperidines; Pirenzepine; Receptors, Cholinergic; Receptors, Muscarinic

1981
Comparison of atropine and dexetimide in treatment of intoxications by selected organophosphates.
    Acta pharmacologica et toxicologica, 1982, Volume: 50, Issue:3

    Topics: Animals; Atropine; Dexetimide; Diet; Guinea Pigs; Insecticides; Isoflurophate; Lethal Dose 50; Mice; Obidoxime Chloride; Organophosphate Poisoning; Organophosphorus Compounds; Paraoxon; Piperidines

1982
[The influence of the beat frequency on the time course of drug binding and pharmacological action of dexetimide in atrial muscle (author's transl)].
    Archiv der Pharmazie, 1980, Volume: 313, Issue:8

    Topics: Animals; Dexetimide; Guinea Pigs; Heart; Heart Rate; In Vitro Techniques; Myocardium; Piperidines; Time Factors

1980
Evidence for an involvement of acetylcholine in self-stimulation of the prefrontal cortex in the rat.
    Experientia, 1980, Oct-15, Volume: 36, Issue:10

    Topics: Acetylcholine; Animals; Cerebral Cortex; Dexetimide; Drinking Behavior; Electric Stimulation; Male; Motor Activity; Piperidines; Rats; Receptors, Muscarinic; Receptors, Nicotinic; Scopolamine; Self Stimulation

1980
Inhibition of [3H]dexetimide binding by a homologous series of methylfurthrethonium analogues at the peripheral muscarinic receptor.
    Biochemical and biophysical research communications, 1980, Nov-28, Volume: 97, Issue:2

    Topics: Animals; Binding, Competitive; Cattle; Cell Membrane; Dexetimide; Kinetics; Muscle, Smooth; Piperidines; Receptors, Cholinergic; Receptors, Muscarinic; Structure-Activity Relationship; Trachea

1980