Page last updated: 2024-08-22

deuterium and cgp 74588

deuterium has been researched along with cgp 74588 in 1 studies

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aichholz, R; Blasco, F; Manley, PW; Mestan, J1

Other Studies

1 other study(ies) available for deuterium and cgp 74588

ArticleYear
The kinetic deuterium isotope effect as applied to metabolic deactivation of imatinib to the des-methyl metabolite, CGP74588.
    Bioorganic & medicinal chemistry, 2013, Jun-01, Volume: 21, Issue:11

    Topics: Administration, Intravenous; Administration, Oral; Animals; Antineoplastic Agents; Benzamides; Biotransformation; Deuterium; Humans; Hydrogen; Imatinib Mesylate; Male; Microsomes, Liver; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Rats

2013
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