Page last updated: 2024-09-04

desmethylcarvedilol and glyburide

desmethylcarvedilol has been researched along with glyburide in 1 studies

Compound Research Comparison

Studies
(desmethylcarvedilol)
Trials
(desmethylcarvedilol)
Recent Studies (post-2010)
(desmethylcarvedilol)
Studies
(glyburide)
Trials
(glyburide)
Recent Studies (post-2010) (glyburide)
5026,5546201,344

Protein Interaction Comparison

ProteinTaxonomydesmethylcarvedilol (IC50)glyburide (IC50)
ATP-binding cassette sub-family C member 9Homo sapiens (human)0.22
Bile salt export pumpRattus norvegicus (Norway rat)5.7
Bile salt export pumpHomo sapiens (human)5.5333
Cytochrome P450 2C9 Homo sapiens (human)1.602
ATP-binding cassette sub-family C member 8Homo sapiens (human)0.0043
ATP-sensitive inward rectifier potassium channel 11Homo sapiens (human)0.1121
NACHT, LRR and PYD domains-containing protein 3 Mus musculus (house mouse)10
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)1.8

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Coelho, EB; Della Pasqua, O; Lanchote, VL; Nardotto, GHB1

Other Studies

1 other study(ies) available for desmethylcarvedilol and glyburide

ArticleYear
Population pharmacokinetics of carvedilol enantiomers and their metabolites in healthy subjects and type-2 diabetes patients.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2017, Nov-15, Volume: 109S

    Topics: Adrenergic beta-Antagonists; Adult; Blood Glucose; Carbazoles; Carvedilol; Cytochrome P-450 CYP2C9; Cytochrome P-450 CYP2C9 Inhibitors; Cytochrome P-450 CYP2D6; Diabetes Mellitus, Type 2; Female; Glyburide; Healthy Volunteers; Humans; Hypoglycemic Agents; Male; Metformin; Middle Aged; Propanolamines; Stereoisomerism

2017