desipramine and trifluoperazine

desipramine has been researched along with trifluoperazine in 38 studies

Research

Studies (38)

TimeframeStudies, this research(%)All Research%
pre-199026 (68.42)18.7374
1990's3 (7.89)18.2507
2000's3 (7.89)29.6817
2010's6 (15.79)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baldy, WJ; Davis, CB; DiStefano, DL; Elgin, RJ; Fedde, CL; Kesslick, JM; Martin, GE; Mathiasen, JR; Scott, MK; Shank, RP1
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Chiang, GH; Unger, SH1
Strassburg, CP; Tukey, RH1
Duffy, EM; Jorgensen, WL1
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ1
Ekins, S; Williams, AJ; Xu, JJ1
Chen, M; Fang, H; Liu, Z; Shi, Q; Tong, W; Vijay, V1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Løvstad, RA1
Lin, HL; Marks, MJ; Medzihradsky, F1
Aghajanian, GK; Bunney, BS2
Henry, BW; Overall, JE; Woodward, JA1
Kiryon, C; Miki, A; Nakayama, T; Ohsawa, K; Tanabe, K1
Davis, JM; Janicak, PG; Javaid, JI; Pandey, GN1
Comaty, J; Davis, JM; Faull, K; Janicak, P; Javaid, JI; Sharma, R1
Davis, JM; Javaid, JI; Maiorano, M1
Frisk-Holmberg, M; van der Kleijn, E1
Blacker, KH; Donlon, PT1
Tuomisto, J1
Green, AL1
Furlong, FW; Luby, ED1
Garriott, JC; Stolman, A1
Oates, JA; Shand, DG1
Foxwell, MH; Funderburk, WH; Hakala, MW1
Roux, JT; Wolpowitz, B1
Milner, G1
Schechter, MD1
Cardinal, JA; Hill, AG; Midha, KK; Verbeeck, RK1
Edström, A; Ekström, P; Kanje, M1
Dinsdale, HB; Nag, S; Raymond, JJ; Robertson, DM1
Wakade, AR; Wakade, TD1
Barrington, M; Majewski, H1
Graham, BG; Sattely-Miller, EA; Schiffman, SS; Suggs, MS1

Reviews

3 review(s) available for desipramine and trifluoperazine

ArticleYear
Human UDP-glucuronosyltransferases: metabolism, expression, and disease.
    Annual review of pharmacology and toxicology, 2000, Volume: 40

    Topics: Autoimmunity; Chromosome Mapping; Glucuronides; Glucuronosyltransferase; Humans; Hyperbilirubinemia; Neoplasms; Steroids; Terminology as Topic

2000
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Electrophysiological studies of dopamine- innervated cells in the frontal cortex.
    Advances in biochemical psychopharmacology, 1977, Volume: 16

    Topics: Animals; Benztropine; Cerebral Cortex; Desipramine; Dopamine; Drug Interactions; Electrophysiology; Hippocampus; Histocytochemistry; Horseradish Peroxidase; Iontophoresis; Neural Pathways; Norepinephrine; Rats; Trifluoperazine

1977

Trials

1 trial(s) available for desipramine and trifluoperazine

ArticleYear
Lithium in the control of mania.
    International journal of neuropsychiatry, 1967, Volume: 3, Issue:4

    Topics: Adult; Amitriptyline; Bipolar Disorder; Chlorpromazine; Clinical Trials as Topic; Desipramine; Female; Humans; Imipramine; Lithium; Male; Middle Aged; Nortriptyline; Thioridazine; Tranylcypromine; Trifluoperazine

1967

Other Studies

34 other study(ies) available for desipramine and trifluoperazine

ArticleYear
Activity of aromatic substituted phenylpiperazines lacking affinity for dopamine binding sites in a preclinical test of antipsychotic efficacy.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:5

    Topics: Animals; Antipsychotic Agents; Avoidance Learning; Dose-Response Relationship, Drug; Piperazines; Rats; Receptors, Dopamine; Receptors, Serotonin; Structure-Activity Relationship

1989
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Octanol-physiological buffer distribution coefficients of lipophilic amines by reversed-phase high-performance liquid chromatography and their correlation with biological activity.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:3

    Topics: Amines; Animals; Buffers; Chromatography, High Pressure Liquid; Histamine Release; Lipid Metabolism; Octanols; Protein Binding; Rats; Serum Albumin, Bovine; Sodium-Potassium-Exchanging ATPase; Solubility; Structure-Activity Relationship

1981
Prediction of drug solubility from Monte Carlo simulations.
    Bioorganic & medicinal chemistry letters, 2000, Jun-05, Volume: 10, Issue:11

    Topics: Monte Carlo Method; Pharmaceutical Preparations; Solubility

2000
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Developing structure-activity relationships for the prediction of hepatotoxicity.
    Chemical research in toxicology, 2010, Jul-19, Volume: 23, Issue:7

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes

2010
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
FDA-approved drug labeling for the study of drug-induced liver injury.
    Drug discovery today, 2011, Volume: 16, Issue:15-16

    Topics: Animals; Benchmarking; Biomarkers, Pharmacological; Chemical and Drug Induced Liver Injury; Drug Design; Drug Labeling; Drug-Related Side Effects and Adverse Reactions; Humans; Pharmaceutical Preparations; Reproducibility of Results; United States; United States Food and Drug Administration

2011
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Effect of centrally active drugs on dopamine oxidation by rat brain catecholamine oxidase.
    Experientia, 1979, Dec-15, Volume: 35, Issue:12

    Topics: Animals; Antipsychotic Agents; Brain; Chlorpromazine; Desipramine; Dopamine; Dopamine beta-Hydroxylase; Female; Haloperidol; Imipramine; Kinetics; Promazine; Rats; Thioridazine; Trifluoperazine; Trifluperidol

1979
Drug inhibitable ecta-ATPase in leukocytes.
    Life sciences, 1975, May-01, Volume: 16, Issue:9

    Topics: Adenosine Triphosphatases; Animals; Calcium; Cations, Divalent; Cations, Monovalent; Desipramine; Dinitrophenols; Enzyme Inhibitors; Kinetics; Leukocytes; Male; Nortriptyline; Oligomycins; Ouabain; Potassium; Rats; Sodium; Sulfhydryl Reagents; Thioridazine; Trifluoperazine

1975
Dopamine and norepinephrine innervated cells in the rat prefrontal cortex: pharmacological differentiation using microiontophoretic techniques.
    Life sciences, 1976, Dec-01, Volume: 19, Issue:11

    Topics: Action Potentials; Animals; Benztropine; Brain Mapping; Cerebral Cortex; Desipramine; Dopamine; Drug Synergism; Hippocampus; Male; Norepinephrine; Olfactory Bulb; Rats; Trifluoperazine

1976
Patterns of symptom change in anxious depressed outpatients treated with different drugs.
    Diseases of the nervous system, 1975, Volume: 36, Issue:3

    Topics: Amitriptyline; Antidepressive Agents; Anxiety; Chlordiazepoxide; Chlorpromazine; Depression; Desipramine; Diazepam; Drug Combinations; Fluphenazine; Humans; Imipramine; Mental Disorders; Nortriptyline; Perphenazine; Thioridazine; Thiothixene; Tranquilizing Agents; Trifluoperazine

1975
Plasmodium chabaudi: association of reversal of chloroquine resistance with increased accumulation of chloroquine in resistant parasites.
    Experimental parasitology, 1992, Volume: 74, Issue:2

    Topics: Animals; Antidepressive Agents, Tricyclic; Calcium Channel Blockers; Chloroquine; Chlorpromazine; Chromatography, High Pressure Liquid; Desipramine; Drug Resistance; Erythrocytes; Female; Imipramine; Malaria; Mice; Mice, Inbred ICR; Plasmodium chabaudi; Trifluoperazine

1992
Increased 3H-clonidine binding in the platelets of patients with depressive and schizophrenic disorders.
    Psychiatry research, 1989, Volume: 28, Issue:1

    Topics: Bipolar Disorder; Blood Platelets; Clonidine; Depressive Disorder; Desipramine; Humans; Imidazoline Receptors; Lithium; Psychiatric Status Rating Scales; Receptors, Adrenergic, alpha; Receptors, Adrenergic, alpha-2; Schizophrenia; Trifluoperazine

1989
Plasma and CSF HVA before and after pharmacological treatment.
    Psychiatry research, 1989, Volume: 28, Issue:1

    Topics: Adult; Brain; Desipramine; Female; Homovanillic Acid; Humans; Lithium; Male; Psychiatric Status Rating Scales; Psychotic Disorders; Psychotropic Drugs; Receptors, Dopamine; Schizophrenia; Schizophrenic Psychology; Trifluoperazine

1989
Uptake and/or binding of tricyclic antidepressants in human red cells.
    Life sciences, 1985, May-06, Volume: 36, Issue:18

    Topics: Buffers; Cations, Monovalent; Desipramine; Erythrocyte Membrane; Erythrocytes; Haloperidol; Humans; Hydrogen-Ion Concentration; Imipramine; In Vitro Techniques; Kinetics; Orosomucoid; Osmolar Concentration; Plasma; Protein Binding; Serum Albumin; Trifluoperazine

1985
The relationship between the lipophilic nature of tricyclic neuroleptics and antidepressants, and histamine release.
    European journal of pharmacology, 1972, Volume: 18, Issue:2

    Topics: Amitriptyline; Animals; Antidepressive Agents; Cell Membrane Permeability; Chemical Phenomena; Chemistry; Chlorpromazine; Chlorprothixene; Clopenthixol; Desipramine; Fluphenazine; Histamine Release; Imipramine; Kinetics; Male; Mast Cells; Methotrimeprazine; Nortriptyline; Perphenazine; Phenothiazines; Prochlorperazine; Promazine; Promethazine; Rats; Solvents; Structure-Activity Relationship; Thioridazine; Tranquilizing Agents; Trifluoperazine

1972
Stages of schizophrenic decompensation and reintegration.
    The Journal of nervous and mental disease, 1973, Volume: 157, Issue:3

    Topics: Adult; Affect; Aggression; Antipsychotic Agents; Anxiety; Depression; Desipramine; Fear; Female; Fluphenazine; Hostility; Humans; Male; Middle Aged; Schizophrenia; Thioridazine; Trifluoperazine

1973
A new modification for studying 5-HT uptake by blood platelets: a re-evaluation of tricyclic antidepressants as uptake inhibitors.
    The Journal of pharmacy and pharmacology, 1974, Volume: 26, Issue:2

    Topics: Amitriptyline; Animals; Blood Platelets; Carbon Radioisotopes; Chlorpromazine; Desipramine; Dibenzazepines; Doxepin; Imipramine; In Vitro Techniques; Kinetics; Models, Biological; Nortriptyline; Promazine; Rabbits; Serotonin; Synaptosomes; Temperature; Trifluoperazine; Triflupromazine

1974
Ionization constants and water solubilities of some aminoalkylphenothiazine tranquillizers and related compounds.
    The Journal of pharmacy and pharmacology, 1967, Volume: 19, Issue:1

    Topics: Amitriptyline; Chemical Phenomena; Chemistry; Chlorpromazine; Desipramine; Hydrogen-Ion Concentration; Imipramine; Perphenazine; Phenothiazines; Prochlorperazine; Promethazine; Solubility; Thioridazine; Tranquilizing Agents; Trifluoperazine; Water

1967
Detection of some psychotherapeutic drugs and their metabolites in urine.
    Clinical toxicology, 1971, Volume: 4, Issue:2

    Topics: Amitriptyline; Amphetamine; Analgesics; Antidepressive Agents; Chlordiazepoxide; Chlorpromazine; Chromatography, Thin Layer; Desipramine; Diazepam; Fluphenazine; Haloperidol; Humans; Imipramine; Indicators and Reagents; Methadone; Perphenazine; Solvents; Thioridazine; Tranquilizing Agents; Trifluoperazine

1971
Metabolism of propranolol by rat liver microsomes and its inhibition by phenothiazine and tricyclic antidepressant drugs.
    Biochemical pharmacology, 1971, Volume: 20, Issue:7

    Topics: Amitriptyline; Animals; Antidepressive Agents; Chlorpromazine; Desipramine; Imipramine; Kinetics; Liver; Male; Metabolism; Microsomes, Liver; NAD; NADP; Nitrogen; Nortriptyline; Perphenazine; Phenothiazines; Prochlorperazine; Promazine; Promethazine; Propranolol; Rats; Subcellular Fractions; Trifluoperazine; Triflupromazine

1971
Effects of psychotherapeutic drugs on hypothalamic- induced hissing in cats.
    Neuropharmacology, 1970, Volume: 9, Issue:1

    Topics: Amitriptyline; Animals; Cats; Chlordiazepoxide; Chlorpromazine; Desipramine; Electric Stimulation; Female; Hypothalamus; Imipramine; Injections, Intraperitoneal; Male; Pentobarbital; Perphenazine; Tranquilizing Agents; Trifluoperazine; Vocalization, Animal

1970
[Parenteral treatment of depressive diseases].
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1970, Oct-10, Volume: 44, Issue:40

    Topics: Antidepressive Agents; Bipolar Disorder; Dementia; Depression; Depressive Disorder, Major; Desipramine; Diazepam; Drug Synergism; Humans; Infusions, Parenteral; Neurotic Disorders; Schizophrenia; Trifluoperazine

1970
The effect of antidepressants and "tranquilizers" on the response of mice to ethanol.
    British journal of pharmacology, 1968, Volume: 34, Issue:2

    Topics: Accidents, Traffic; Amitriptyline; Animals; Antidepressive Agents; Chlorpromazine; Coma; Desipramine; Diazepam; Dibenzazepines; Drug Synergism; Ethanol; Humans; Imipramine; Methylphenidate; Mice; Nortriptyline; Phenelzine; Phenobarbital; Reflex; Substance-Related Disorders; Thioridazine; Tranquilizing Agents; Trifluoperazine

1968
Effect of neuroleptics and tricyclic antidepressants upon d-amphetamine discrimination.
    Pharmacology, biochemistry, and behavior, 1980, Volume: 12, Issue:1

    Topics: Animals; Antidepressive Agents, Tricyclic; Antipsychotic Agents; Chlorpromazine; Clozapine; Desipramine; Dextroamphetamine; Discrimination, Psychological; Dose-Response Relationship, Drug; Fluphenazine; Haloperidol; Imipramine; Male; Nortriptyline; Promethazine; Rats; Sodium Chloride; Thioridazine; Trifluoperazine

1980
Binding of phenothiazine neuroleptics to plasma proteins.
    Biochemical pharmacology, 1983, Sep-01, Volume: 32, Issue:17

    Topics: Antipsychotic Agents; Blood Proteins; Chlorpromazine; Desipramine; Humans; Kinetics; Perphenazine; Propranolol; Protein Binding; Salicylates; Salicylic Acid; Structure-Activity Relationship; Trifluoperazine; Tritium

1983
Effects of phenothiazines and dibenzazepines on axonal transport and microtubule assembly in vitro.
    Acta physiologica Scandinavica, 1982, Volume: 116, Issue:2

    Topics: Adenosine Triphosphate; Amitriptyline; Animals; Axonal Transport; Chlorpromazine; Desipramine; Dibenzazepines; Lofepramine; Microtubules; Phenothiazines; Phosphocreatine; Rana pipiens; Rana temporaria; Sciatic Nerve; Thioridazine; Trifluoperazine

1982
Pharmacological modification of blood-brain barrier permeability following a cold lesion.
    The Canadian journal of neurological sciences. Le journal canadien des sciences neurologiques, 1984, Volume: 11, Issue:4

    Topics: Animals; Blood-Brain Barrier; Brain Injuries; Cerebrovascular Circulation; Cold Temperature; Desipramine; Female; Imidazoles; Psychotropic Drugs; Rats; Rats, Inbred Strains; Thioridazine; Trifluoperazine

1984
Effects of desipramine, trifluoperazine and other inhibitors of calmodulin on the secretion of catecholamines from the adrenal medulla and postganglionic sympathetic nerves of the salivary gland.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 325, Issue:4

    Topics: Acetylcholine; Adrenal Medulla; Animals; Calcium; Calmodulin; Catecholamines; Desipramine; Electric Stimulation; Imipramine; In Vitro Techniques; Male; Norepinephrine; Perfusion; Rats; Salivary Glands; Splanchnic Nerves; Trifluoperazine

1984
Trifluoperazine and calmidazolium have multiple actions on the release of noradrenaline from sympathetic nerves of mouse atria.
    Naunyn-Schmiedeberg's archives of pharmacology, 1994, Volume: 349, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Atropine; Calmodulin; Desipramine; Electric Stimulation; Enterochromaffin Cells; Heart; Heart Atria; Imidazoles; In Vitro Techniques; Male; Mice; Myocardium; Norepinephrine; Phentolamine; Sympathetic Nervous System; Trifluoperazine

1994
Effect of psychotropic drugs on taste responses in young and elderly persons.
    Annals of the New York Academy of Sciences, 1998, Nov-30, Volume: 855

    Topics: Adult; Aged; Aging; Amitriptyline; Clomipramine; Desipramine; Doxepin; Female; Humans; Imipramine; Male; Psychotropic Drugs; Taste; Trifluoperazine

1998