desipramine and proadifen

desipramine has been researched along with proadifen in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-199025 (92.59)18.7374
1990's1 (3.70)18.2507
2000's0 (0.00)29.6817
2010's1 (3.70)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Jonsson, J1
Summers, RJ; Tillman, J1
Renyi, AL; Ross, SB1
Bellward, GD; Morgan, RG; Szombathy, VH1
Illing, HP; Kunke, S; Netter, KJ1
Carrara, C; Garattini, S; Jori, A; Paglialunga, S1
Jori, A; Pugliatti, C1
Bernardi, D; Jori, A1
Colson, SH; Tolson, WW; Umberger, EJ1
Bickel, MH1
Clark, B; Thompson, JW; Widdrington, G1
Juul, P; Sand, O1
Bellward, GD; Black, NB; Dayton, PG; O'Brien, L; Perel, JM1
Bertilsson, L; von Bahr, C1
Conney, AH; Levin, W; Welch, RM1
Nakazawa, K1
Bickel, MH; Minder, R1
Gillette, J; Hammer, W; Schumacher, H; Sjöqvist, F1
Gillette, J; Sjöqvist, F1
Burns, JJ; Conney, AH; Kuntzman, R; Lemberger, L1
Spencer, PS1
Jenner, P; Marsden, CD; Reavill, C1
Daniel, W; Maj, J; Rogóz, Z; Skuza, G; Sowińska, H1
Mehendale, HM; Ohmiya, Y1
Ishikawa, K; Sato, Y; Shibanoki, S; Sugahara, M1

Other Studies

27 other study(ies) available for desipramine and proadifen

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
On the aromatic hydroxylation of amphetamine in rat liver microsomes and perfused liver preparations: effects of long-term administration.
    Acta pharmacologica et toxicologica, 1977, Volume: 40, Issue:4

    Topics: Administration, Oral; Amphetamines; Animals; Carbon Monoxide; Cytochrome P-450 Enzyme System; Desipramine; Fenfluramine; Hydroxylation; Male; Microsomes, Liver; NADP; NADPH-Ferrihemoprotein Reductase; Perfusion; Phenobarbital; Proadifen; Rats; Rats, Inbred Strains; Time Factors

1977
Investigation of the role of calcium in the supersensitivity produced by cocaine in cat spleen strips.
    British journal of pharmacology, 1979, Volume: 65, Issue:4

    Topics: Angiotensin II; Animals; Calcium; Cats; Chlorpheniramine; Cocaine; Desipramine; Drug Interactions; Female; In Vitro Techniques; Male; Muscle Contraction; Norepinephrine; Oxymetazoline; Potassium; Proadifen; Spleen

1979
Tricyclic antidepressant agents. II. Effect of oral administration on the uptake of 3-H-noradrenaline and 14-C-5-hydroxytryptamine in slices of the midbrain-hypothalamus region of the rat.
    Acta pharmacologica et toxicologica, 1975, Volume: 36, Issue:Suppl 5

    Topics: Administration, Oral; Amitriptyline; Animals; Antidepressive Agents, Tricyclic; Biotransformation; Desipramine; Hypothalamus; Imipramine; Male; Mesencephalon; Norepinephrine; Proadifen; Rats; Serotonin; Time Factors

1975
The effects of pretreatment of mice with norethindrone on the metabolism of 14C-imipramine by the liver microsomal drug-metabolizing enzymes.
    Canadian journal of physiology and pharmacology, 1974, Volume: 52, Issue:1

    Topics: Animals; Carbon Radioisotopes; Chromatography, Thin Layer; Cobalt; Cytochrome c Group; Cytochrome Reductases; Dealkylation; Desipramine; Female; Hydrogen-Ion Concentration; Hydroxylation; Imipramine; Methylcholanthrene; Mice; Microsomes, Liver; NADP; Norethindrone; Oxides; Phenobarbital; Proadifen; Time Factors

1974
On the spectral intermediate at 440 nm formed during mixed function substrate oxidation.
    Biochemical pharmacology, 1974, Sep-15, Volume: 23, Issue:18

    Topics: Acetanilides; Aniline Compounds; Animals; Barbiturates; Cytochrome P-450 Enzyme System; Desipramine; Imipramine; In Vitro Techniques; Kinetics; Male; Metyrapone; Microsomes, Liver; Mixed Function Oxygenases; Morphinans; NAD; NADP; Oxidation-Reduction; Oxidoreductases; Oxygen Consumption; Pentobarbital; Proadifen; Protein Binding; Rats; Spectrophotometry, Ultraviolet

1974
Pharmacological studies on modaline sulphate (w 3207).
    The Journal of pharmacy and pharmacology, 1965, Volume: 17, Issue:11

    Topics: Antidepressive Agents; Desipramine; Dibenzylchlorethamine; Dihydroxyphenylalanine; Fever; Hydrazines; Isoproterenol; Monoamine Oxidase Inhibitors; Nortriptyline; Phentolamine; Proadifen; Propranolol; Reserpine; Sympatholytics; Tryptamines

1965
An interaction between the antidepressant drugs desipramine and modaline sulphate.
    The Journal of pharmacy and pharmacology, 1967, Volume: 19, Issue:12

    Topics: Animals; Behavior, Animal; Brain; Desipramine; In Vitro Techniques; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Proadifen; Rats; Tryptamines

1967
Brain desipramine level in relation to the anti-reserpine acitivity of imipramine.
    The Journal of pharmacy and pharmacology, 1968, Volume: 20, Issue:12

    Topics: Animals; Body Temperature; Cats; Desipramine; Female; Imipramine; Proadifen; Reserpine; Tetrabenazine

1968
The effects of some centrally acting drugs on the glucocorticoid induction of hepatic tyrosine transaminase.
    Life sciences, 1969, Nov-15, Volume: 8, Issue:22

    Topics: Adrenalectomy; Amitriptyline; Animals; Chlorpheniramine; Chlorpromazine; Desipramine; Diphenhydramine; Enzyme Induction; Female; Fluocinolone Acetonide; Fluorometholone; Glucocorticoids; Hydrocortisone; Imipramine; Liver; Male; Prednisone; Proadifen; Promazine; Promethazine; Rats; Reserpine; Sex Factors; Triflupromazine; Tyrosine Transaminase

1969
Liver metabolic reactions: tertiary amine N-dealkylation, tertiary amine N-oxidation, N-oxide reduction, and N-oxide N-dealkylation. I. Tricyclic tertiary amine drugs.
    Archives of biochemistry and biophysics, 1972, Volume: 148, Issue:1

    Topics: Amitriptyline; Animals; Carbon Isotopes; Carbon Monoxide; Chlorpromazine; Cyclic N-Oxides; Cytochromes; Dealkylation; Desipramine; Horses; Imipramine; Kinetics; Liver; Male; NADP; Organ Specificity; Oxidation-Reduction; Proadifen; Rats; Species Specificity; Subcellular Fractions; Swine; Tetrazolium Salts

1972
Analysis of the inhibition of pethidine N-demethylation by monoamine oxidase inhibitors and some other drugs with special reference to drug interactions in man.
    British journal of pharmacology, 1972, Volume: 44, Issue:1

    Topics: Amphetamine; Animals; Chlorpromazine; Desipramine; Drug Interactions; Histamine; Hydrazines; Hydrocortisone; Imipramine; Iproniazid; Male; Meperidine; Methylation; Microsomes, Liver; Monoamine Oxidase Inhibitors; Nialamide; Opipramol; Phenothiazines; Phenylhydrazines; Prednisolone; Proadifen; Promazine; Rats; Transferases

1972
Determination of guanethidine in sympathetic ganglia.
    Acta pharmacologica et toxicologica, 1973, Volume: 32, Issue:6

    Topics: Animals; Autoradiography; Cell Survival; Depression, Chemical; Desipramine; Fluorometry; Ganglia, Autonomic; Guanethidine; Half-Life; Male; Neurons; Proadifen; Rats; Reserpine; Stimulation, Chemical; Time Factors

1973
Imipramine and chlorpromazine in hepatic microsomal systems.
    Advances in biochemical psychopharmacology, 1974, Volume: 9, Issue:0

    Topics: Animals; Carbon Radioisotopes; Chlorpromazine; Chromatography, Thin Layer; Cobalt; Cytochrome P-450 Enzyme System; Cytochrome Reductases; Dealkylation; Desipramine; Dose-Response Relationship, Drug; Hydrogen-Ion Concentration; Hydroxylation; Imipramine; In Vitro Techniques; Kinetics; Male; Methylphenidate; Microsomes, Liver; Phenobarbital; Proadifen; Proteins; Spectrophotometry, Ultraviolet

1974
Hydroxylation and subsequent glucuronide conjugation of desmethylimipramine in rat liver microsomes.
    Xenobiotica; the fate of foreign compounds in biological systems, 1971, Volume: 1, Issue:3

    Topics: Animals; Cytochromes; Desipramine; Glucuronates; Hydroxylation; In Vitro Techniques; Kinetics; Male; Microsomes, Liver; Proadifen; Rats; Rats, Inbred Strains; Spectrum Analysis; Tritium; Uracil Nucleotides

1971
Effect of carbon tetrachloride and other inhibitors of drug metabolism on the metabolism and action of estradiol-17 beta and estrone in the rat.
    The Journal of pharmacology and experimental therapeutics, 1970, Volume: 173, Issue:2

    Topics: Alanine Transaminase; Animals; Carbon Tetrachloride; Desipramine; Estradiol; Estrone; Female; Microsomes, Liver; Organ Size; Proadifen; Rats; Tritium; Uterus

1970
Studies on the demethylation, hydroxylation and N-oxidation of imipramine in rat liver.
    Biochemical pharmacology, 1970, Volume: 19, Issue:4

    Topics: Amino Alcohols; Animals; Carbon Isotopes; Chlorides; Chromatography, Paper; Dealkylation; Desipramine; Ethylamines; Imipramine; Liver; Magnesium; Male; Metabolism; Methylation; Oxidation-Reduction; Oxides; Phenobarbital; Proadifen; Rats; Valerates

1970
Metabolism and biliary excretion of the lipophilic drug molecules, imipramine and desmethylimipramine in the rat. I. Experiments in vivo and with isolated perfused livers.
    Biochemical pharmacology, 1970, Volume: 19, Issue:8

    Topics: Alcohols; Animals; Benzyl Compounds; Bile; Bile Acids and Salts; Biliary Fistula; Chromatography, Thin Layer; Desipramine; Glucuronates; Imines; Imipramine; Injections, Intravenous; Intestine, Small; Kinetics; Laparotomy; Liver; Male; Perfusion; Phenobarbital; Proadifen; Rats; Time Factors

1970
[The effect of desmethylimipramine and other "anti-tremorine" drugs on the metabolism of tremorine and oxotremorine in rats and mice].
    Biochemical pharmacology, 1968, Volume: 17, Issue:6

    Topics: Animals; Body Temperature; Brain; Desipramine; Drug Synergism; Imipramine; Liver; Male; Malonates; Mice; Models, Biological; Proadifen; Pyrrolidines; Rats; Receptors, Drug; Species Specificity; Thermography; Tremor; Tremorine; Tritium

1968
Prolongation and potentiation of oxotremorine effects by desmethylimipramine an "anti-tremorine" drug.
    Life sciences, 1965, Volume: 4, Issue:10

    Topics: Animals; Atropine; Desipramine; Drug Synergism; Proadifen; Rats; Tremor; Tremorine

1965
Metabolism of tyramine to dopamine by liver microsomes.
    The Journal of pharmacology and experimental therapeutics, 1965, Volume: 150, Issue:2

    Topics: Animals; Carbon Isotopes; Chromatography, Paper; Desipramine; Dopamine; Enzymes; Guanidines; Hydrazines; In Vitro Techniques; Liver; Microsomes; Mixed Function Oxygenases; Proadifen; Rabbits; Radiometry; Tyramine

1965
The antagonism of oxotremorine effects in the mouse by thymoleptics.
    Life sciences, 1966, Volume: 5, Issue:11

    Topics: Amphetamine; Animals; Desipramine; Drug Antagonism; Imipramine; Male; Mice; Proadifen; Tremorine; Trihexyphenidyl

1966
Metabolite involvement in bromocriptine-induced circling behaviour in rodents.
    The Journal of pharmacy and pharmacology, 1980, Volume: 32, Issue:4

    Topics: Amphetamine; Animals; Apomorphine; Biotransformation; Bromocriptine; Desipramine; Female; Hydroxydopamines; Male; Medial Forebrain Bundle; Methyltyrosines; Mice; Motor Activity; Nomifensine; Paralysis; Proadifen; Rats; Receptors, Dopamine; Receptors, Neurotransmitter; Reserpine; Sleep; Zoxazolamine

1980
Influence of proadifen, an inhibitor of the metabolism of drugs, on the action of imipramine and desipramine in rats.
    Polish journal of pharmacology and pharmacy, 1981, Volume: 33, Issue:6

    Topics: Animals; Blepharoptosis; Desipramine; Hypothermia; Imipramine; Male; Motor Activity; Proadifen; Rats; Rats, Inbred Strains; Reserpine

1981
N-oxidation of imipramine by isolated perfused rat and rabbit lung.
    Life sciences, 1980, Apr-28, Volume: 26, Issue:17

    Topics: Animals; Cytosol; Desipramine; Imipramine; Lung; Male; Microsomes; Mitochondria; Oxidation-Reduction; Perfusion; Proadifen; Rabbits; Rats; Species Specificity; Subcellular Fractions

1980
Measurement and pharmacokinetic analysis of imipramine and its metabolite by brain microdialysis.
    British journal of pharmacology, 1994, Volume: 112, Issue:2

    Topics: Aminopyrine; Animals; Brain; Chromatography, High Pressure Liquid; Desipramine; Electrochemistry; Half-Life; Imipramine; Male; Microdialysis; Proadifen; Rats; Rats, Wistar

1994