desipramine and prazosin

desipramine has been researched along with prazosin in 82 studies

Research

Studies (82)

TimeframeStudies, this research(%)All Research%
pre-199029 (35.37)18.7374
1990's19 (23.17)18.2507
2000's19 (23.17)29.6817
2010's13 (15.85)24.3611
2020's2 (2.44)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Andrews, PR; Craik, DJ; Martin, JL1
Topliss, JG; Yoshida, F1
Alvarez-Pedraglio, A; Colmenarejo, G; Lavandera, JL1
Bacsó, Z; Cianfriglia, M; Fenyvesi, F; Goda, K; Kappelmayer, J; Lustyik, G; Nagy, H; Szabó, G; Szilasi, M1
Nagashima, R; Nishikawa, T; Tobita, M1
Lombardo, F; Obach, RS; Waters, NJ1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Sun, Y; Yan, Z1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Du-Cuny, L; Mash, EA; Meuillet, EJ; Moses, S; Powis, G; Song, Z; Zhang, S1
Campillo, NE; Guerra, A; Páez, JA1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Sen, S; Sinha, N1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Bandyopadhyaya, A; Rajagopalan, DR; Rajagopalan, P; Rajagopalan, R1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Acevedo, O; Dasararaju, G; Devadasan, V; Halakova, D; Jayaprakash, V; Kovacikova, L; Mohd Siddique, MU; Mondal, SK; Prnova, MS; Shilkar, D; Stefek, M; Thakur, A; Yasmin, S1
Holmes, PH; Mounsey, A; Sutherland, IA1
Fukuda, H; Hirayama, T; Ono, H1
Di Bona, G; Finberg, JP; Lavian, G1
Cervo, L; Samanin, R1
Boura, AL; King, RG; Lau, WA1
Cai, B; Matsumoto, K; Ohta, H; Satoh, T; Watanabe, H1
Brunello, N; Galimberti, R; Racagni, G; Riva, M; Rovescalli, AC1
Lacroix, JS; Lundberg, JM1
Gonzales, RA; Moerschbaecher, JM; Mosaddeghi, M1
Broadley, KJ; Williamson, KL1
Katahira, K; Kohara, K; Kumahara, Y; Mikami, H; Ogihara, T; Ohde, H1
Tessel, RE; Yourick, DL1
Iuvone, PM; Johnson, RD; Minneman, KP1
Dodt, C; Gross, G; Hanft, G1
Chiu, A; Li, PP; Sibony, D; Warsh, JJ1
Bradley, L; Doggrell, SA1
Mogilnicka, E; Wedzony, K; Zazula, M1
Moulds, RF; Stevens, MJ1
Hjemdahl, P; Kahan, T1
Blaschke, D; Laakmann, G; Meissner, R; Schoen, HW; Weiss, A; Wittmann, M; Zygan, K1
Laakmann, G; Meissner, R; Schoen, HW; Weiss, A; Wittmann, M; Zygan, K1
Laakmann, G; Meissner, R; Mueller, OA; Schoen, HW; Stalla, GK; Weiss, A; Wittmann, M; Zygan, K1
Duman, R; Hewitt, L; Swann, AC1
Pulvirenti, L; Samanin, R1
Swann, AC1
Krueger, CG; Purdy, RE; Young, S1
Briley, MS; Langer, SZ; Wetzel, HW1
Hedler, L; Majewski, H; Starke, K1
Borsini, F; Nowakowska, E; Samanin, R1
Chang, RS; Kling, P; Lotti, VJ1
Aghajanian, GK; Gallager, DW; Menkes, DB1
Aghajanian, GK; Davis, M; Gallager, DW; Kehne, JH; Menkes, DB1
Górka, Z; Maj, J; Melzacka, M; Pilc, A; Rawłów, A1
Kengatharan, M; Mackay, D1
Kulkarni, SK; Sharma, A1
Fawcett, JP; Menkes, DB; Patel, PP1
Kurz, K; Starke, K; von Kügelgen, I1
al-Damluji, S; Catt, KJ; Krsmanovic, LZ1
Al-Damluji, S; Kopin, IJ1
Ball, WA; Gresch, PJ; Morrison, AR; Ross, RJ; Sanford, LD1
Dunn-Meynell, AA; Levin, BE; Yarlagadda, Y1
al-Damluji, S; Knutson, JR; Kopin, IJ; Krsmanovic, LZ; Porter, D1
Martin, JR1
Kleven, MS; Koek, W1
Dailey, JW; Jobe, PC; Steenbergen, JL; Yan, QS1
Kurz, T; Richardt, G; Schneider, I; Tölg, R1
Gerevich, Z; Lendvai, B; Santha, E1
Al-Damluji, S; Shen, WB1
Harkin, A; Kelly, JP; Leonard, BE; Morris, K; O'Donnell, JM1
Hopwood, SE; Stamford, JA1
Barrento, C; Lima, BS; Mota-Filipe, H; Pinto, R1
Cao, N; Haynes, JM; Ventura, S1
Aiso, S; Ito, M; Katada, M; Kawasaki, A; Matsuoka, M; Nishizawa, K; Terashita, K; Torii, K1
Huang, Y; O'Donnell, JM; Whisler, LR; Xiang, Y; Zhang, HT1
Gorzalka, BB; Hill, MN; Morrish, AC; Riebe, CJ1
Docherty, JR1
Bielecka, AM; Daniel, WA; Drzyzga, Ł; Kot, M; Obuchowicz, E; Paul-Samojedny, M; Prymus, A1
Amorim, AC; Antunes, E; Britto-Júnior, J; Campos, R; da Silva-Filho, WP; De Nucci, G; Fregonesi, A; Monica, FZ; Moraes, MEA; Moraes, MO1

Reviews

1 review(s) available for desipramine and prazosin

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

81 other study(ies) available for desipramine and prazosin

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Cheminformatic models to predict binding affinities to human serum albumin.
    Journal of medicinal chemistry, 2001, Dec-06, Volume: 44, Issue:25

    Topics: Adrenergic beta-Antagonists; Antidepressive Agents, Tricyclic; Chromatography, Affinity; Cyclooxygenase Inhibitors; Databases, Factual; Humans; Hydrophobic and Hydrophilic Interactions; Penicillins; Pharmaceutical Preparations; Protein Binding; Quantitative Structure-Activity Relationship; Reproducibility of Results; Serum Albumin; Steroids

2001
Distinct groups of multidrug resistance modulating agents are distinguished by competition of P-glycoprotein-specific antibodies.
    Biochemical and biophysical research communications, 2004, Mar-19, Volume: 315, Issue:4

    Topics: Adenosine Triphosphatases; Animals; Anti-Bacterial Agents; Antibodies, Monoclonal; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding, Competitive; Calcium Channel Blockers; Cyclosporine; Detergents; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Fluoresceins; Humans; Ivermectin; Mice; NIH 3T3 Cells; Substrate Specificity

2004
A discriminant model constructed by the support vector machine method for HERG potassium channel inhibitors.
    Bioorganic & medicinal chemistry letters, 2005, Jun-02, Volume: 15, Issue:11

    Topics: Animals; CHO Cells; Cricetinae; Discriminant Analysis; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Humans; Potassium Channel Blockers; Potassium Channels, Voltage-Gated

2005
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
First-principle, structure-based prediction of hepatic metabolic clearance values in human.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:4

    Topics: Computational Biology; Drug Discovery; Hepatocytes; Humans; Hydrogen-Ion Concentration; Liver; Metabolic Clearance Rate; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship; Sensitivity and Specificity; Software

2009
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Computational modeling of novel inhibitors targeting the Akt pleckstrin homology domain.
    Bioorganic & medicinal chemistry, 2009, Oct-01, Volume: 17, Issue:19

    Topics: Antineoplastic Agents; Blood Proteins; Caco-2 Cells; Cell Membrane Permeability; Computer Simulation; Drug Discovery; Drug Screening Assays, Antitumor; Humans; Models, Molecular; Phosphoproteins; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-akt; Quantitative Structure-Activity Relationship

2009
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Predicting hERG activities of compounds from their 3D structures: development and evaluation of a global descriptors based QSAR model.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:2

    Topics: Computer Simulation; Ether-A-Go-Go Potassium Channels; Humans; Molecular Structure; Organic Chemicals; Quantitative Structure-Activity Relationship

2011
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
    Bioorganic & medicinal chemistry letters, 2013, Mar-15, Volume: 23, Issue:6

    Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship

2013
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
The synthesis and comparative receptor binding affinities of novel, isomeric pyridoindolobenzazepine scaffolds.
    Bioorganic & medicinal chemistry letters, 2014, Jan-15, Volume: 24, Issue:2

    Topics: Benzodiazepinones; Isomerism; Protein Binding; Protein Structure, Tertiary; Receptors, Cell Surface

2014
Non-carboxylic acid inhibitors of aldose reductase based on N-substituted thiazolidinedione derivatives.
    European journal of medicinal chemistry, 2021, Nov-05, Volume: 223

    Topics: Aldehyde Reductase; Animals; Caco-2 Cells; Catalytic Domain; Dogs; Enzyme Inhibitors; Humans; Hypoglycemic Agents; Madin Darby Canine Kidney Cells; Male; Molecular Docking Simulation; Molecular Dynamics Simulation; Molecular Structure; Protein Binding; Rats, Wistar; Structure-Activity Relationship; Thiazolidinediones

2021
Transport of isometamidium (Samorin) by drug-resistant and drug-sensitive Trypanosoma congolense.
    Parasitology, 1992, Volume: 104 ( Pt 3)

    Topics: Animals; Biological Transport, Active; Desipramine; Drug Resistance; Glycerol; Hydrogen-Ion Concentration; Kinetics; Phenanthridines; Polysorbates; Prazosin; Salicylamides; Temperature; Trypanocidal Agents; Trypanosoma congolense; Verapamil

1992
Functional supersensitivity of alpha 1-adrenergic system in spinal ventral horn is due to absence of an uptake system and not to postsynaptic change.
    Brain research, 1991, Jan-25, Volume: 539, Issue:2

    Topics: Animals; Anterior Horn Cells; Biogenic Amines; Chromatography, High Pressure Liquid; Desipramine; Electric Stimulation; Electrochemistry; Hydroxydopamines; Isoproterenol; Male; Methoxamine; Norepinephrine; Oxidopamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1991
Inhibition of sympathetic nerve activity by acute administration of the tricyclic antidepressant desipramine.
    European journal of pharmacology, 1991, Mar-05, Volume: 194, Issue:2-3

    Topics: Animals; Blood Pressure; Desipramine; Drug Interactions; Heart Rate; Kidney; Male; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Splanchnic Nerves; Sympathetic Nervous System; Yohimbine

1991
Clonidine causes antidepressant-like effects in rats by activating alpha 2-adrenoceptors outside the locus coeruleus.
    European journal of pharmacology, 1991, Feb-14, Volume: 193, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Antidepressive Agents; Behavior, Animal; Clonidine; Desipramine; Dioxanes; Dose-Response Relationship, Drug; Drug Administration Schedule; Hydroxydopamines; Idazoxan; Locus Coeruleus; Male; Neurons; Norepinephrine; Oxidopamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1991
Methoxyphenamine inhibits basal and histamine-induced nasal congestion in anaesthetized rats.
    British journal of pharmacology, 1990, Volume: 101, Issue:2

    Topics: Airway Resistance; Animals; Desipramine; Ephedrine; Epinephrine; Histamine Antagonists; Male; Methamphetamine; Methoxamine; Nasal Decongestants; Pentobarbital; Prazosin; Rats; Rats, Inbred Strains; Tyramine

1990
Desipramine enhances isolation-induced aggressive behavior in mice.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:1

    Topics: Aggression; Animals; Clonidine; Desipramine; Imipramine; Male; Mice; Mice, Inbred Strains; Motor Activity; Phentolamine; Prazosin; Social Isolation; Yohimbine

1991
Age-related changes in rat serotonergic and adrenergic systems and in receptor responsiveness to subchronic desipramine treatment.
    Pharmacology & toxicology, 1988, Volume: 63, Issue:3

    Topics: Aging; Animals; Brain; Clonidine; Desipramine; Dihydroalprenolol; Hydroxyindoleacetic Acid; Imipramine; Ketanserin; Kinetics; Male; Paroxetine; Piperidines; Prazosin; Proteins; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Serotonin; Serotonin; Time Factors

1988
Sympathetic vascular control of the pig nasal mucosa: adrenoceptor mechanisms in blood flow and volume control.
    British journal of pharmacology, 1989, Volume: 97, Issue:4

    Topics: Animals; Antihypertensive Agents; Brimonidine Tartrate; Desipramine; Dioxanes; Electric Stimulation; Female; Idazoxan; Male; Nasal Mucosa; Norepinephrine; Oxymetazoline; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic; Regional Blood Flow; Rheology; Swine; Sympathetic Nervous System

1989
Effect of monoamine uptake inhibitors on norepinephrine-stimulated phosphatidylinositol hydrolysis in rat cortex.
    Biochemical pharmacology, 1989, Jan-15, Volume: 38, Issue:2

    Topics: Animals; Cerebral Cortex; Cocaine; Desipramine; Fluoxetine; In Vitro Techniques; Male; Neurotransmitter Uptake Inhibitors; Norepinephrine; Phosphatidylinositols; Prazosin; Rats; Receptors, Adrenergic, alpha

1989
Do both adrenaline and noradrenaline stimulate cardiac alpha-adrenoceptors to induce positive inotropy of rat atria?
    British journal of pharmacology, 1989, Volume: 98, Issue:2

    Topics: Animals; Cocaine; Desipramine; Dibenzylchlorethamine; Epinephrine; Haloperidol; Heart; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Norepinephrine; Pindolol; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Stimulation, Chemical; Timolol

1989
Direct vascular effects of 19-hydroxyandrostenedione.
    Methods and findings in experimental and clinical pharmacology, 1989, Volume: 11, Issue:4

    Topics: Aldosterone; Androstenedione; Animals; Desipramine; Dose-Response Relationship, Drug; Ear; Female; Hemodynamics; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Prazosin; Rabbits; Regional Blood Flow; Spironolactone; Vasoconstriction

1989
Mechanisms of phenylalanine-induced pressor effects in conscious rats.
    European journal of pharmacology, 1989, Jan-31, Volume: 160, Issue:2

    Topics: Animals; Biological Availability; Blood Pressure; Carbidopa; Desipramine; Dose-Response Relationship, Drug; Heart Rate; Male; Phenethylamines; Phenylalanine; Prazosin; Rats; Rats, Inbred Strains; Tyrosine; Valine

1989
Regulation of alpha-1 adrenergic receptor density and functional responsiveness in rat brain.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:3

    Topics: Animals; Benzylamines; Brain Chemistry; Cyclic AMP; Desipramine; Male; Norepinephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Reserpine; Yohimbine

1987
Effect of chronic lithium administration on adrenoceptor binding and adrenoceptor regulation in rat cerebral cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 337, Issue:3

    Topics: Animals; Cerebral Cortex; Desipramine; Dihydroalprenolol; Hydroxydopamines; In Vitro Techniques; Injections, Intraventricular; Lithium; Male; Oxidopamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Sympathectomy, Chemical; Yohimbine

1988
Assessment of rat brain alpha 1-adrenoceptor binding and activation of inositol phospholipid turnover following chronic imipramine treatment.
    Neurochemical research, 1988, Volume: 13, Issue:12

    Topics: Animals; Cerebral Cortex; Desipramine; Imipramine; In Vitro Techniques; Inositol Phosphates; Iodocyanopindolol; Norepinephrine; Pindolol; Prazosin; Radioligand Assay; Rats; Receptors, Adrenergic, alpha; Sugar Phosphates

1988
Modification by desipramine of the effects of alpha-adrenoceptor antagonists on the contractile responses of the trisected rat vas deferens.
    General pharmacology, 1985, Volume: 16, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Desipramine; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurotransmitter Uptake Inhibitors; Norepinephrine; Phentolamine; Prazosin; Rats; Rats, Inbred Strains; Vas Deferens; Yohimbine

1985
Functional supersensitivity to the alpha 1-adrenoceptor agonist after repeated treatment with antidepressant drugs is not conditioned by beta-down-regulation.
    Neuropharmacology, 1987, Volume: 26, Issue:10

    Topics: Adrenergic alpha-Agonists; Animals; Antidepressive Agents; Brain Chemistry; Desipramine; Dihydroalprenolol; Male; Maprotiline; Motor Activity; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1987
Factors determining alpha-adrenoceptor-mediated responses of human digital arteries and metacarpal veins.
    Clinical science (London, England : 1979), 1985, Volume: 68 Suppl 10

    Topics: Desipramine; Dose-Response Relationship, Drug; Fingers; Humans; Hydrocortisone; Metacarpus; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Prazosin; Propranolol; Quinazolines; Receptors, Adrenergic, alpha; Yohimbine

1985
Pre- and postjunctional alpha-adrenoceptor-mediated effects of prazosin, methoxamine and 6-fluoronoradrenaline in blood-perfused canine skeletal muscle in situ.
    European journal of pharmacology, 1987, Jan-06, Volume: 133, Issue:1

    Topics: Animals; Desipramine; Diclofenac; Dogs; Electric Stimulation; Female; Male; Methoxamine; Muscles; Norepinephrine; Perfusion; Prazosin; Prostaglandins; Receptors, Adrenergic, alpha; Vasoconstriction

1987
Effect of receptor blockers (methysergide, propranolol, phentolamine, yohimbine and prazosin) on desimipramine-induced pituitary hormone stimulation in humans--I. Growth hormone.
    Psychoneuroendocrinology, 1986, Volume: 11, Issue:4

    Topics: Adolescent; Adult; Blood Glucose; Blood Pressure; Carrier Proteins; Desipramine; Drug Interactions; Growth Hormone; Humans; Male; Methysergide; Phentolamine; Pituitary Hormones; Prazosin; Propranolol; Receptors, Drug; Receptors, Neurotransmitter; Time Factors; Yohimbine

1986
Effects of receptor blockers (methysergide, propranolol, phentolamine, yohimbine and prazosin) on desimipramine-induced pituitary hormone stimulation in humans--II. Prolactin.
    Psychoneuroendocrinology, 1986, Volume: 11, Issue:4

    Topics: Blood Glucose; Blood Pressure; Carrier Proteins; Desipramine; Drug Interactions; Heart Rate; Humans; Male; Methysergide; Phentolamine; Pituitary Hormones; Prazosin; Prolactin; Propranolol; Receptors, Drug; Receptors, Neurotransmitter; Time Factors; Yohimbine

1986
Effects of receptor blockers (methysergide, propranolol, phentolamine, yohimbine and prazosin) on desimipramine-induced pituitary hormone stimulation in humans--III. Hypothalamo-pituitary-adrenocortical axis.
    Psychoneuroendocrinology, 1986, Volume: 11, Issue:4

    Topics: Blood Glucose; Blood Pressure; Carrier Proteins; Desipramine; Drug Interactions; Heart Rate; Humans; Hypothalamo-Hypophyseal System; Male; Methysergide; Phentolamine; Pituitary Hormones; Pituitary-Adrenal System; Prazosin; Propranolol; Receptors, Drug; Receptors, Neurotransmitter; Yohimbine

1986
Desipramine binding: relationship to central and sympathetic noradrenergic activity.
    Journal of neurochemistry, 1985, Volume: 44, Issue:2

    Topics: Animals; Cerebral Cortex; Clonidine; Desipramine; Dextroamphetamine; Heart; Hydroxydopamines; Isoproterenol; Male; Muscles; Norepinephrine; Oxidopamine; Prazosin; Rats; Rats, Inbred Strains; Sympathetic Nervous System; Synapses

1985
Antagonism by dopamine, but not noradrenaline receptor blockers of the anti-immobility activity of desipramine after different treatment schedules in the rat.
    Pharmacological research communications, 1986, Volume: 18, Issue:1

    Topics: Animals; Desipramine; Dopamine; Male; Motor Activity; Norepinephrine; Phenoxybenzamine; Prazosin; Rats; Receptors, Adrenergic

1986
Caloric intake and Na+-K+-ATPase: differential regulation by alpha 1- and beta-noradrenergic receptors.
    The American journal of physiology, 1984, Volume: 247, Issue:3 Pt 2

    Topics: 4-Nitrophenylphosphatase; Adipose Tissue, Brown; Animals; Body Weight; Desipramine; Diet; Eating; Energy Intake; Fasting; Male; Ouabain; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Sodium-Potassium-Exchanging ATPase

1984
Evidence for nonclassical alpha adrenoceptor blockade by prazosin in isolated rabbit blood vessels.
    Life sciences, 1980, Dec-08, Volume: 27, Issue:23

    Topics: Adrenergic alpha-Antagonists; Animals; Arteries; Desipramine; Desoxycorticosterone; In Vitro Techniques; Norepinephrine; Prazosin; Quinazolines; Rabbits; Vasoconstriction; Veins

1980
3H-WB 4101 binding in the rat vas deferens. Effects of chronic treatments with desipramine and prazosin.
    Naunyn-Schmiedeberg's archives of pharmacology, 1981, Volume: 317, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Cell Membrane; Desipramine; Dioxanes; Dioxins; Male; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Vas Deferens

1981
Evidence for a physiological role of presynaptic alpha-adrenoceptors: modulation of noradrenaline release in the pithed rabbit.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 324, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Clonidine; Desipramine; Electric Stimulation; Epinephrine; Female; Guanethidine; Heart Rate; Male; Nordefrin; Norepinephrine; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Spinal Nerves; Yohimbine

1983
Effect of repeated treatment with desipramine in the behavioral "despair" test in rats: antagonism by "atypical" but not "classical" neuroleptics or antiadrenergic drugs.
    Life sciences, 1984, Mar-19, Volume: 34, Issue:12

    Topics: Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Butyrophenones; Chlorpromazine; Clonidine; Clozapine; Depressive Disorder; Desipramine; Dibenzazepines; Haloperidol; Humans; Male; Metoclopramide; Phentolamine; Prazosin; Propranolol; Rats; Sulpiride

1984
Pre- and postsynaptic adrenergic activation by norepinephrine reuptake inhibitors in the field-stimulated rat vas deferens.
    Life sciences, 1981, Aug-10, Volume: 29, Issue:6

    Topics: Amitriptyline; Animals; Chlorpromazine; Cocaine; Desipramine; Dibenzocycloheptenes; Dose-Response Relationship, Drug; Male; Norepinephrine; Prazosin; Protriptyline; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Vas Deferens; Yohimbine

1981
Chronic antidepressant treatment enhances agonist affinity of brain alpha 1-adrenoceptors.
    European journal of pharmacology, 1983, Jan-28, Volume: 87, Issue:1

    Topics: Amitriptyline; Animals; Antidepressive Agents; Binding, Competitive; Brain; Desipramine; Iprindole; Kinetics; Male; Phenylephrine; Prazosin; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Thalamus

1983
Functional supersensitivity of CNS alpha 1-adrenoceptors following chronic antidepressant treatment.
    Life sciences, 1983, Jul-11, Volume: 33, Issue:2

    Topics: Amitriptyline; Animals; Antidepressive Agents; Binding Sites; Desipramine; Hydroxydopamines; Iprindole; Male; Norepinephrine; Oxidopamine; Phenylephrine; Prazosin; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Reflex, Acoustic

1983
Chronic treatment with imipramine: further functional evidence for the enhanced noradrenergic transmission in flexor reflex activity.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 322, Issue:4

    Topics: Animals; Desipramine; Hindlimb; Imipramine; Male; Norepinephrine; Phenoxybenzamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Reflex; Spinal Cord; Synaptic Transmission

1983
pKI values of prazosin and idazoxan for receptors stimulated by neuronally released transmitter in the epididymal portion of rat isolated vas deferens.
    British journal of pharmacology, 1994, Volume: 111, Issue:1

    Topics: Adenosine Triphosphate; Animals; Binding, Competitive; Corticosterone; Desipramine; Dioxanes; Epididymis; Idazoxan; In Vitro Techniques; Male; Mathematics; Norepinephrine; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Vas Deferens

1994
On the characterization of dopamine-induced contractile response of rat anococcygeus muscle preparation.
    Indian journal of experimental biology, 1994, Volume: 32, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Azepines; Benzazepines; Desipramine; Dioxanes; Dopamine; Female; Haloperidol; Idazoxan; Male; Muscle Contraction; Prazosin; Rats; Receptors, Adrenergic; Receptors, Dopamine; Reserpine; Sulpiride; Yohimbine

1994
Antidepressant treatment and chemical sympathectomy fail to modulate alpha 1-adrenoceptor sensitivity in mouse eye.
    Neuropharmacology, 1993, Volume: 32, Issue:12

    Topics: Administration, Topical; Amitriptyline; Animals; Antidepressive Agents; Benzamides; Desipramine; Down-Regulation; Fluoxetine; Injections, Intraperitoneal; Male; Methoxamine; Mice; Moclobemide; Oxidopamine; Phentolamine; Phenylephrine; Prazosin; Pupil; Receptors, Adrenergic, alpha-1; Sympathectomy, Chemical; Time Factors

1993
Axon terminal P2-purinoceptors in feedback control of sympathetic transmitter release.
    Neuroscience, 1993, Volume: 56, Issue:2

    Topics: Adenosine Triphosphate; Animals; Axons; Desipramine; Drug Interactions; Feedback; GTP-Binding Proteins; Male; Mice; Nifedipine; Norepinephrine; Prazosin; Purinergic Antagonists; Receptors, Purinergic; Suramin; Sympathetic Nervous System; Triazines; Vas Deferens; Virulence Factors, Bordetella; Xanthines; Yohimbine

1993
High-affinity uptake of noradrenaline in postsynaptic neurones.
    British journal of pharmacology, 1993, Volume: 109, Issue:2

    Topics: Animals; Cell Membrane; Cells, Cultured; Desipramine; Female; Gonadotropin-Releasing Hormone; Hypothalamus; Iodine Radioisotopes; Kinetics; Methoxamine; Neurons; Norepinephrine; Oxidopamine; Prazosin; Pregnancy; Rats; Rats, Sprague-Dawley; Synapses

1993
Functional properties of the uptake of amines in immortalised peptidergic neurones (transport-P).
    British journal of pharmacology, 1996, Volume: 117, Issue:1

    Topics: Adrenergic Uptake Inhibitors; Amines; Anti-Bacterial Agents; Cell Line; Chloroquine; Desipramine; Hydrogen-Ion Concentration; Hypothalamus; Ionophores; Macrolides; Neurons; Norepinephrine; Prazosin; Proton-Translocating ATPases; Reserpine; Sodium; Sodium-Potassium-Exchanging ATPase; Steroids; Temperature; Vanadates

1996
REM sleep inhibition by desipramine: evidence for an alpha-1 adrenergic mechanism.
    Brain research, 1995, Dec-01, Volume: 701, Issue:1-2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Animals; Antihypertensive Agents; Cats; Desipramine; Female; Hydralazine; Prazosin; Propranolol; Sleep, REM

1995
Alpha 1-adrenoceptor blockade increases behavioral deficits in traumatic brain injury.
    Journal of neurotrauma, 1997, Volume: 14, Issue:1

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Behavior, Animal; Blood Pressure; Brain; Brain Injuries; Desipramine; Male; Norepinephrine; Prazosin; Rats; Rats, Sprague-Dawley; Somatosensory Cortex

1997
Visual detection of transport-P in peptidergic neurones.
    British journal of pharmacology, 1997, Volume: 120, Issue:5

    Topics: Adrenergic alpha-Antagonists; Amines; Animals; Biological Transport; Boron Compounds; Cell Line, Transformed; Desipramine; Fluorescent Dyes; Hypothalamus; Microscopy, Fluorescence; Neurons; Peptides; Prazosin; Rats; Receptors, Adrenergic, alpha-1; Spectrometry, Fluorescence

1997
DMPP-evoked increases in postganglionic sympathetic nerve activity and blood pressure occurs by two mechanisms in the rat.
    Journal of autonomic pharmacology, 1997, Volume: 17, Issue:4

    Topics: Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Blood Pressure; Desipramine; Dimethylphenylpiperazinium Iodide; Dose-Response Relationship, Drug; Ganglionic Stimulants; Male; Nicotinic Antagonists; Pentolinium Tartrate; Prazosin; Rats; Rats, Sprague-Dawley; Sympathetic Fibers, Postganglionic

1997
Discriminative stimulus properties of cocaine: enhancement by monoamine reuptake blockers.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:3

    Topics: Animals; Cocaine; Desipramine; Discrimination Learning; Dopamine; Dose-Response Relationship, Drug; Fluoxetine; Male; Neurotransmitter Uptake Inhibitors; Norepinephrine; Prazosin; Propranolol; Rats; Rats, Sprague-Dawley; Serotonin; Ventral Tegmental Area

1998
Anticonvulsant effect of enhancement of noradrenergic transmission in the superior colliculus in genetically epilepsy-prone rats (GEPRs): a microinjection study.
    Brain research, 1998, Jan-12, Volume: 780, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Anticonvulsants; Desipramine; Drug Interactions; Epilepsy; Female; Fluoxetine; Idazoxan; Methoxamine; Microinjections; Norepinephrine; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Superior Colliculi; Synaptic Transmission

1998
Alpha 1-adrenergic receptor-mediated increase in the mass of phosphatidic acid and 1,2-diacylglycerol in ischemic rat heart.
    Cardiovascular research, 1999, Volume: 42, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Analysis of Variance; Animals; Chromatography, Thin Layer; Desipramine; Diacylglycerol Kinase; Diglycerides; Estrenes; Male; Myocardial Ischemia; Myocardial Reperfusion; Myocardium; Norepinephrine; Perfusion; Phosphatidic Acids; Piperidines; Prazosin; Propranolol; Pyrrolidinones; Quinazolines; Quinazolinones; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Time Factors; Type C Phospholipases

1999
Low temperature prevents potentiation of norepinephrine release by phenylephrine.
    Neurochemistry international, 2001, Volume: 38, Issue:3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Calcium; Cell Membrane; Cold Temperature; Desipramine; Dose-Response Relationship, Drug; Electric Stimulation; Exocytosis; Extracellular Space; Guinea Pigs; In Vitro Techniques; Male; Norepinephrine; Phenylephrine; Prazosin; Vas Deferens

2001
Release of amines from acidified stores following accumulation by Transport-P.
    British journal of pharmacology, 2001, Volume: 132, Issue:4

    Topics: Antidepressive Agents; Biological Transport; Boron Compounds; Cells, Cultured; Chloroquine; Desipramine; Dose-Response Relationship, Drug; Hydrogen-Ion Concentration; Hypothalamus; Monensin; Prazosin; Temperature

2001
Modulation of MK-801-induced behaviour by noradrenergic agents in mice.
    Psychopharmacology, 2001, Mar-01, Volume: 154, Issue:2

    Topics: Adrenergic Agents; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Ataxia; Benzylamines; Clonidine; Desipramine; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Frontal Lobe; Male; Mesencephalon; Mice; Morpholines; Motor Activity; Norepinephrine; Prazosin; Reboxetine; Stereotyped Behavior

2001
Noradrenergic modulation of serotonin release in rat dorsal and median raphé nuclei via alpha(1) and alpha(2A) adrenoceptors.
    Neuropharmacology, 2001, Volume: 41, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Desipramine; Dexmedetomidine; Electric Stimulation; Electrophysiology; Imidazoles; In Vitro Techniques; Indoles; Isoindoles; Isoquinolines; Male; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Serotonin

2001
Phenylephrine induces endogenous noradrenaline release in the rat vas deferens through nitric oxide synthase pathway.
    Pharmacology & toxicology, 2003, Volume: 93, Issue:4

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Desipramine; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Norepinephrine; omega-N-Methylarginine; Phenylephrine; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Vas Deferens; Vasoconstrictor Agents

2003
Saw palmetto is an indirectly acting sympathomimetic in the rat-isolated prostate gland.
    The Prostate, 2006, Feb-01, Volume: 66, Issue:2

    Topics: Amphetamine; Animals; Cocaine; Desipramine; Electric Stimulation; Guanethidine; Male; Nifedipine; Phentolamine; Plant Extracts; Prazosin; Prostate; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Serenoa; Sympathomimetics; Tyramine; Urinary Bladder; Vas Deferens

2006
Antidepressant-like effect of Cordyceps sinensis in the mouse tail suspension test.
    Biological & pharmaceutical bulletin, 2007, Volume: 30, Issue:9

    Topics: 5-Hydroxytryptophan; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Antidepressive Agents; Antidepressive Agents, Second-Generation; Antidepressive Agents, Tricyclic; Behavior, Animal; Bupropion; Chromatography, Supercritical Fluid; Clorgyline; Cordyceps; Desipramine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Fluoxetine; Head Movements; Hindlimb Suspension; Male; Mice; Mice, Inbred C57BL; Monoamine Oxidase Inhibitors; Motor Activity; Prazosin; Serotonin Antagonists; Sulpiride; Water

2007
Postsynaptic alpha-2 adrenergic receptors are critical for the antidepressant-like effects of desipramine on behavior.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2009, Volume: 34, Issue:4

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Antidepressive Agents, Tricyclic; Depression; Desipramine; Idazoxan; Male; Mice; Mice, Knockout; Motor Activity; Prazosin; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Synapses

2009
Protracted cannabinoid administration elicits antidepressant behavioral responses in rats: role of gender and noradrenergic transmission.
    Physiology & behavior, 2009, Aug-04, Volume: 98, Issue:1-2

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Antidepressive Agents; Antidepressive Agents, Tricyclic; Behavior, Animal; Cannabinoids; Desipramine; Dronabinol; Female; Male; Norepinephrine; Piperidines; Prazosin; Propranolol; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Sex Characteristics; Substance Withdrawal Syndrome; Swimming; Synaptic Transmission

2009
Effects of desipramine on prazosin potency at α1A- and α1D-adrenoceptors in rat vas deferens: implications for the α1L-adrenoceptor subclassification.
    European journal of pharmacology, 2014, Dec-05, Volume: 744

    Topics: Animals; Cocaine; Desipramine; Male; Muscle Contraction; Norepinephrine; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Vas Deferens

2014
Desipramine administered chronically inhibits lipopolysaccharide-stimulated production of IL-1β in the brain and plasma of rats.
    Cytokine, 2016, Volume: 80

    Topics: Administration, Oral; Animals; Antidepressive Agents, Tricyclic; Antihypertensive Agents; Brain; Desipramine; Drug Administration Schedule; Hypothalamus; Interleukin-1beta; Lipopolysaccharides; Olfactory Bulb; Prazosin; Propranolol; Rats

2016
6-nitrodopamine is a major endogenous modulator of human vas deferens contractility.
    Andrology, 2022, Volume: 10, Issue:8

    Topics: Adrenergic Antagonists; Amitriptyline; Animals; Antidepressive Agents, Tricyclic; Carbamazepine; Chromatography, Liquid; Desipramine; Dopamine; Doxazosin; Epinephrine; Humans; Male; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide; Norepinephrine; Prazosin; Rats; Receptors, Adrenergic; Tamsulosin; Tandem Mass Spectrometry; Vas Deferens

2022