desipramine and agi-5198

desipramine has been researched along with agi-5198 in 2 studies

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gu, Y; Ma, T; Pusch, S; von Deimling, A; Xu, Y; Yang, L; Zha, X; Zhu, Q; Zou, F1
Gu, Y; Hua, J; Ma, T; Pusch, S; von Deimling, A; Xu, Y; Yang, L; Zha, X; Zhu, Q; Zou, F1

Other Studies

2 other study(ies) available for desipramine and agi-5198

ArticleYear
Design, synthesis and biological activity of 3-pyrazine-2-yl-oxazolidin-2-ones as novel, potent and selective inhibitors of mutant isocitrate dehydrogenase 1.
    Bioorganic & medicinal chemistry, 2017, 12-15, Volume: 25, Issue:24

    Topics: Cell Survival; Dose-Response Relationship, Drug; Drug Design; Enzyme Inhibitors; HEK293 Cells; Humans; Isocitrate Dehydrogenase; Molecular Docking Simulation; Molecular Structure; Mutation; Oxazolidinones; Pyrazines; Structure-Activity Relationship

2017
Identification of novel allosteric inhibitors of mutant isocitrate dehydrogenase 1 by cross docking-based virtual screening.
    Bioorganic & medicinal chemistry letters, 2018, 02-01, Volume: 28, Issue:3

    Topics: Allosteric Site; Blood-Brain Barrier; Brain Neoplasms; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Enzyme Inhibitors; Glioma; HEK293 Cells; Humans; Isocitrate Dehydrogenase; Molecular Docking Simulation; Molecular Structure; Mutation; Small Molecule Libraries; Structure-Activity Relationship

2018