Page last updated: 2024-09-03

des-enkephalin-gamma-endorphin and u-50488

des-enkephalin-gamma-endorphin has been researched along with u-50488 in 1 studies

Compound Research Comparison

Studies
(des-enkephalin-gamma-endorphin)
Trials
(des-enkephalin-gamma-endorphin)
Recent Studies (post-2010)
(des-enkephalin-gamma-endorphin)
Studies
(u-50488)
Trials
(u-50488)
Recent Studies (post-2010) (u-50488)
41601,6643209

Protein Interaction Comparison

ProteinTaxonomydes-enkephalin-gamma-endorphin (IC50)u-50488 (IC50)
Delta-type opioid receptorRattus norvegicus (Norway rat)2.15
Kappa-type opioid receptorMus musculus (house mouse)0.0027
Mu-type opioid receptorRattus norvegicus (Norway rat)2.15
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.7171
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.0958
Kappa-type opioid receptorHomo sapiens (human)0.0537

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Capasso, A1

Other Studies

1 other study(ies) available for des-enkephalin-gamma-endorphin and u-50488

ArticleYear
Beta-endorphin fragments DTgammaE and DEgammaE reduced morphine inhibition of electrically-induced contractions and opiate withdrawal.
    Medicinal chemistry (Shariqah (United Arab Emirates)), 2009, Volume: 5, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetylcholine; Animals; beta-Endorphin; Electric Stimulation; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Guinea Pigs; Ileum; In Vitro Techniques; Jejunum; Male; Morphine; Muscle Contraction; Muscle, Smooth; Naloxone; Oligopeptides; Peptide Fragments; Rabbits; Substance Withdrawal Syndrome

2009